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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 179 / 315
small molecule | CAS: 131926-99-3

Deskripsi belum tersedia.

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesBenzimidazolesHeterocyclic Compounds, Fused-Ring +3
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small molecule | CAS: 16096-89-2

Deskripsi belum tersedia.

Kategori:
Metal cationsPhosphate BinderPhosphate Chelating Activity
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Lapachone DB11948
small molecule | CAS: 4707-32-8

Lapachone has been used in trials studying the treatment of Cancer, Carcinoma, Advanced Solid Tumors, Head and Neck Neoplasms, and Carcinoma, Squamous Cell.

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiviral Agents +6
Target Protein:
DNA topoisomerase 1Retinol-binding protein 3
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Lapaquistat DB16215
small molecule | CAS: 189059-71-0

Lapaquistat is under investigation in clinical trial NCT00256178 (Efficacy of Lapaquistat Acetate and Simvastatin in Subjects With Primary Dyslipidemia.).

Kategori:
AzepinesFarnesyl-Diphosphate Farnesyltransferase, antagonists & inhibitors
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Lapatinib Approved DB01259
small molecule | CAS: 231277-92-2

Lapatinib is an anti-cancer drug developed by GlaxoSmithKline (GSK) as a treatment for solid tumours such as breast and lung cancer. It was approved by the FDA on March 13, 2007, for use in patients with advanced metastatic breast cancer in conjunction with t…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +22
Target Protein:
Epidermal growth factor receptorEukaryotic elongation factor 2 kinaseReceptor tyrosine-protein kinase erbB-2
Gen Terkait:
HLA-DQA1 HLA-DRB1 HLA-DQB1 +1
Waktu ParuhSingle-dose termina…
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Genetik 4 Varian
Lapuleucel-t DB19117
biotech | CAS: 845680-07-1

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesVaccines
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Lapyrium Approved DB09376
small molecule | CAS: 109260-82-4

Lapyrium is a quaternary ammonium cation used as a surfactant, antistatic agent, and biocide in various cosmetic products [A19426]. It is commonly found formulated as lapyrium chloride.

Kategori:
Pyridines
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Laquinimod DB06685
small molecule | CAS: 248281-84-7

Laquinimod is an immunomodulator developed by Active Biotech and produced by Teva Pharmaceutical Industries. It is currently under development in phase III trials for treatment of multiple sclerosis as an oral therapy, like fingolimod. It has been shown to re…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +3
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +3
Waktu Paruh-
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Larazotide DB05645
small molecule | CAS: 258818-34-7

An octapeptide inhibitor of paracellular permeability whose structure is derived from a protein (zonula occludens toxin) secreted by Vibrio cholerae for treatment of Coeliac disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Haptoglobin
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Larcaviximab DB17775
biotech | CAS: 1792982-56-9

Deskripsi belum tersedia.

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Largemouth bass Approved DB10976
biotech

Largemouth bass allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Larix occidentalis pollen Approved DB10914
biotech

Larix occidentalis pollen is the pollen of the Larix occidentalis plant. Larix occidentalis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Larix sibirica wood Approved DB14289
biotech

Larix sibirica wood is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Laromustine DB05817
small molecule | CAS: 173424-77-6

VNP40101M is a novel alkylating agent that has been used in trials studying the treatment of Leukemia, Lymphoma, Lung Cancer, Small Intestine Cancer, and Myelodysplastic Syndromes, among others.

Kategori:
AmidesSulfonesSulfur Compounds
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Laronidase Approved DB00090
biotech | CAS: 210589-09-6

Human recombinant alpha-L-iduronidase, 628 residues (mature form), produced by recombinant DNAtechnology in a Chinese hamster ovary cell line. Laronidase is a glycoprotein with a molecular weight of approximately 83 kD. The predicted amino acid sequence of th…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +4
Target Protein:
Iduronic acid
Waktu Paruh1.5-3.6 hrs
Vol. Distribusi-
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Laropiprant Approved DB11629
small molecule | CAS: 571170-77-9

Laropiprant is an ingredient in the EMA-withdrawn product Pelzont.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Prostaglandin E2 receptor EP2 subtype3-hydroxy-3-methylglutaryl-coenzyme A reductaseThromboxane A2 receptor +4
Waktu Paruh-
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Genetik -
Larotaxel DB12984
small molecule | CAS: 156294-36-9

Larotaxel has been used in trials studying the treatment of Cancer, Metastases, Breast Cancer, Breast Neoplasms, and Pancreatic Neoplasms, among others.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +1
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Larotrectinib Approved DB14723
small molecule | CAS: 1223403-58-4

Larotrectinib is an orally administered inhibitor of tropomyosin receptor kinase (Trk), a receptor tyrosine kinase activated by neurotrophins which is mutated in a variety of cancer cell types and plays an important role in tumor cell growth and survival.[L49…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +8
Target Protein:
High affinity nerve growth factor receptorBDNF/NT-3 growth factors receptorNT-3 growth factor receptor
Waktu ParuhIn healthy subjects…
Vol. DistribusiFollowing intraveno…
KlirensThe mean clearance …
Genetik -
Larsucosterol DB18079
small molecule | CAS: 884905-07-1

Deskripsi belum tersedia.

Kategori:
CholestanesCholestenesFused-Ring Compounds +5
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Lartesertib DB19045
small molecule | CAS: 2495096-26-7

Lartesertib is under investigation in clinical trial NCT06433219 (Tuvusertib Combined With Niraparib or Lartesertib in Participants With Epithelial Ovarian Cancer (Ddriver EOC 302)).

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biotech | CAS: 2425817-08-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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LAS-191954 DB17816
small molecule | CAS: 1403947-26-1

Deskripsi belum tersedia.

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Lasalocid DB11423
small molecule | CAS: 25999-31-9

Lasalocid is an agent that presents antibacterial and coccidiostat activities. It is produced by strains of _Streptomyces lasaliensis_.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +11
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Lasmiditan Approved DB11732
small molecule | CAS: 439239-90-4

Lasmiditan is an oral medication used in the termination of migraine headaches that was first approved for use in the United States in October 2019.[L9338,L9356] It was also approved by the European Commission on August 17, 2022.[L43997] Traditionally, the…

Kategori:
AmidesAnalgesicsAntidepressive Agents +17
Target Protein:
5-hydroxytryptamine receptor 1F
Waktu ParuhThe mean eliminatio…
Vol. DistribusiLasmiditan has been…
Klirens-
Genetik -
Lasofoxifene Approved DB06202
small molecule | CAS: 180916-16-9

Lasofoxifene is a non-steroidal 3rd generation selective estrogen receptor modulator (SERM) that selectively binds to both ER? and ER? with high affinity. It is a naphthalene derivative marketed for prevention and treatment of osteoporosis and for the treatme…

Kategori:
Genito Urinary System and Sex HormonesNaphthalenesSelective Estrogen Receptor Modulators +1
Target Protein:
Fusion glycoprotein F0Estrogen receptorEstrogen receptor beta +1
Waktu ParuhElimination half-li…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Latanoprost Approved DB00654
small molecule | CAS: 130209-82-4

Latanoprost is a prodrug analog of prostaglandin F2 alpha that is used to treat elevated intraocular pressure (IOP). It was initially approved by the FDA in 1998. Latanoprost is the first topical prostaglandin F2 alpha analog used for glaucoma treatment.[A184…

Kategori:
Antiglaucoma Preparations and MioticsAntihypertensive AgentsAutacoids +18
Target Protein:
Prostaglandin F2-alpha receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
Latanoprost acid Approved DB19360
small molecule | CAS: 41639-83-2

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +6
Waktu Paruh-
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Latanoprostene bunod Approved DB11660
small molecule | CAS: 860005-21-6

Latanoprostene Bunod has been used in trials studying the treatment of Glaucoma, Ocular Hypertension, Open-Angle Glaucoma, Open Angle Glaucoma, and Intraocular Pressure. As of November 2, 2017 the FDA approved Bausch + Lomb's Vyzulta (latanoprostene bunod …

Kategori:
Antiglaucoma Preparations and MioticsAutacoidsBiological Factors +12
Target Protein:
Prostaglandin F2-alpha receptor
Waktu ParuhThe half-life after…
Vol. DistribusiUnfortunately there…
KlirensSince latanoprost a…
Genetik -
Latiglutenase DB06326
biotech | CAS: 1360452-96-5

Deskripsi belum tersedia.

Kategori:
Celiac Disease, drug therapyEnzymesEnzymes and Coenzymes +1
Waktu Paruh-
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Genetik -
Latozinemab DB16978
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Latrepirdine DB11725
small molecule | CAS: 3613-73-8

Latrepirdine has been investigated for the treatment of Alzheimer's Disease and Huntington's Disease.

Kategori:
Alzheimer DiseaseHeterocyclic Compounds, Fused-Ring
Target Protein:
5-hydroxytryptamine receptor 6Histamine H1 receptor
Waktu Paruh-
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Latrunculin A DB02621
small molecule | CAS: 76343-93-6

Latrunculin A is an actin binding macrolide purified from the red sea sponge Latrunculia magnifica. It is under investigation for the treatment of cancer. It disrupts actin polymerization, prevents mitotic spindle formation and thus cell replication.

Kategori:
PoriferaSulfur CompoundsThiazoles
Target Protein:
Actin, alpha skeletal muscleGelsolinIota toxin component Ia
Waktu Paruh-
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Latrunculin B DB08080
small molecule | CAS: 76343-94-7

Latrunculin B is a 14-membered macrolide attached to 2-thiazolidinone moiety, isolated from Red Sea sponge _Latrunculia magnifica_.

Kategori:
PoriferaSulfur CompoundsThiazoles
Target Protein:
Actin, alpha skeletal muscleMyocardin-related transcription factor AProtein spire homolog 2
Waktu Paruh-
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Lauric acid Approved DB03017
small molecule | CAS: 143-07-7

Lauric acid is an inexpensive, non-toxic and safe to handle compound often used in laboratory investigations of melting-point depression. Lauric acid is a solid at room temperature but melts easily in boiling water, so liquid lauric acid can be treated with v…

Kategori:
Fatty AcidsLipids
Target Protein:
Toll-like receptor 4LactotransferrinPhospholipase A2, membrane associated +18
Waktu Paruh-
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Laurocapram Approved DB17308
small molecule | CAS: 59227-89-3

Deskripsi belum tersedia.

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small molecule | CAS: 112-16-3

Deskripsi belum tersedia.

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Laurus nobilis Approved DB10670
biotech

Laurus nobilis allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
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Genetik -
small molecule | CAS: 16610-63-2

Deskripsi belum tersedia.

Target Protein:
Farnesyl pyrophosphate synthaseGeranylgeranyl pyrophosphate synthase
Waktu Paruh-
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Genetik -
small molecule | CAS: 27836-64-2

Deskripsi belum tersedia.

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small molecule | CAS: 683-10-3

Deskripsi belum tersedia.

Kategori:
AminesOnium CompoundsQuaternary Ammonium Compounds +1
Target Protein:
AppA protein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
LAVA-051 DB18395
biotech

LAVA-051 is a humanized V?9V?2-T cell-engaging bispecific antibody.

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Lavender oil Approved DB14566
biotech | CAS: 8000-28-0

Deskripsi belum tersedia.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +13
Waktu Paruh-
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Lavendustin A DB16768
small molecule | CAS: 125697-92-9

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesEnzyme InhibitorsTyrosine Kinase Inhibitors
Target Protein:
Epidermal growth factor receptorTyrosine-protein kinase Lck
Waktu Paruh-
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Lavendustin b DB16760
small molecule | CAS: 125697-91-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +5
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Lavoltidine DB12884
small molecule | CAS: 76956-02-0

Lavoltidine has been used in trials studying the diagnostic of Reflux, Gastroesophageal and Gastroesophageal Reflux Disease.

Kategori:
Gastric Acid Lowering AgentsHistamine AgentsHistamine Antagonists +2
Target Protein:
Histamine H2 receptor
Waktu Paruh-
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Lawsone DB04744
small molecule | CAS: 83-72-7

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsColoring Agents +10
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Genetik -
biotech

Lawsonia inermis leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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LAX-101 DB05301
small molecule | CAS: 909712-41-0

LAX-101 treats hungtington’s disease, not just the symptoms but the disease itself. The active molecule in LAX-101 is Eicosapentaenoic Acid (EPA). All molecules of EPA are identical. The molecules of EPA found in LAX-101 are identical to the molecules of EPA …

Target Protein:
Phospholipase D1Caspase-1
Waktu Paruh-
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Lazertinib Approved DB16216
small molecule | CAS: 1903008-80-9

Lazertinib is an oral, third-generation, epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI).[A264299, A264304] Lazertinib was first approved in South Korea on January 18, 2021, for the treatment of _EGFR_ T790M mutation-positive non-small…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +14
Target Protein:
Epidermal growth factor receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Lazuvapagon DB19046
small molecule | CAS: 2379889-71-9

Lazuvapagon is under investigation in clinical trial NCT03116191 (Trial of SK-1404 for Nocturia Due to Nocturnal Polyuria in Japanese Subjects).

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