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12560

Total database: 17430
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9109 (72.5%)
Target
6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 178 / 252
NUC B1000 DB05242
biotech

NUC B1000 is an expressed interfering RNA (eiRNA)- based product consisting of a plasmid DNA construct designed to produce four short interfering RNA (siRNA) molecules, formulated with a proprietary cationic-lipid delivery system. [F3910] eiRNA is an approach…

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NUC-7738 DB19148
small molecule | CAS: 2348493-39-8

NUC-7738 is under investigation in clinical trial NCT03829254 (A Safety, Pharmacokinetic and Clinical Activity Study of NUC-7738 in Patients With Advanced Solid Tumours and Lymphoma).

Kategori:
Benzene DerivativesHeterocyclic Compounds, Fused-Ring
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Nurulimab DB18946
biotech | CAS: 2168561-20-2

Nurulimab is under investigation in clinical trial NCT05732805 (A Clinical Study of BCD-217 (Nurulimab + Prolgolimab) Followed by Anti-pd-1 Compared to Anti-pd-1 Monotherapy as First-line Treatment in Subjects With Unresectable/metastatic Melanoma).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates
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Nusinersen Approved DB13161
small molecule | CAS: 1258984-36-9

An antisense oligonucleotide that induces survival motor neuron (SMN) protein expression, it was approved by the U.S. FDA in December, 2016 as Spinraza for the treatment of children and adults with spinal muscular atrophy (SMA). It is adminstrated as direct i…

Kategori:
Antisense OligonucleotidesIncreased Protein SynthesisMusculo-Skeletal System +4
Target Protein:
Survival motor neuron protein
Waktu ParuhThe mean terminal e…
Vol. DistribusiCSF: 0.4 L Plasma…
KlirensSlow clearance is o…
Genetik -
Nutlin-3 DB17039
small molecule | CAS: 548472-68-0

Nutlin-3 is a small molecule inhibitor that targets p53-Mdm2 interaction.[A253057]

Kategori:
Stereoisomerism
Target Protein:
Cellular tumor antigen p53
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Nutmeg oil DB15996
biotech | CAS: 8008-45-5

Deskripsi belum tersedia.

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Nuvaxovid Approved DB15810
biotech

SARS-CoV-2, the causative agent of COVID-19, relies on the interaction between its trimeric spike (S) glycoprotein and angiotensin-converting enzyme 2 (hACE2) expressed on host cells in order to establish a productive infection in humans.[A243789] Antibodies …

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
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biotech | CAS: 8046-97-7

Deskripsi belum tersedia.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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NV-07a DB05845
small molecule

NV-07a is topical skin repair compound protecting skin from sun-induced immunosuppression and UV-induced damage.

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NV-18 DB05886
small molecule

NV-18 is a product of the Novogen diphenolic synthetic analogue program that is creating drugs with diverse activities against specific types of cancer. Like phenoxodiol, NV-18 is broadly effective in the laboratory against almost all human cancer types, but …

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NV-354 DB18392
small molecule | CAS: 866465-21-6

Deskripsi belum tersedia.

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NV-5138 DB19180
small molecule | CAS: 2095886-80-7

NV-5138 is under investigation in clinical trial NCT06235905 (Open-label of SPN-820 in Adults With Major Depressive Disorder).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +1
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NV-52 DB05673
small molecule

NV-52 is an investigational synthetic flavonoid thromboxane synthase (TXS) inhibitor developed for the maintenance of remission in inflammatory bowel disease.

Target Protein:
Thromboxane-A synthase
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NVD-001 DB18459
biotech

Deskripsi belum tersedia.

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NVL-655 DB18682
small molecule

NVL-655 is an orally bioavailable, brain-penetrant anaplastic lymphoma kinase (ALK) inhibitor inhibitor being investigated for the treatment of non-small cell lung cancer.

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NVP-LEQ-506 DB12857
small molecule | CAS: 1204975-42-7

LEQ506 has been used in trials studying the treatment of Advanced Solid Tumors, Recurrent or Refractory Medulloblastoma, and Locally Advanced or Metastatic Basal Cell Carcinoma.

Target Protein:
Protein smoothened
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NVS antibody DB05312
small molecule

This drug has been developed using Medarex's UltiMAb Human Antibody Development System to treat autoimmune diseases.

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NX-1207 DB05493
small molecule

NX-1207 is an investigational new drug for BPH, whose chemical entity and mechanism of action remain undisclosed. Nymox Pharmaceutical Corporation recently completed studies of NX-1207 for treatment of benign prostatic hyperplasia (BPH).

Kategori:
Amino Acids, Peptides, and Proteins
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NXN-188 DB06096
small molecule

NXN-188 is a first-in-class, dual-action small molecule incorporating both neuronal nitric oxide synthase (nNOS) inhibition and 5-HT agonism that is being developed for the treatment of acute migraine.

Target Protein:
Nitric oxide synthase 15-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1D
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Nylidrin Approved DB06152
small molecule | CAS: 447-41-6

Nylidrin, also known as _buphenine_ belongs to the category of drugs called _vasodilators_, which relax blood vessels and increase blood flow. Nylidrin is a peripheral vasodilator. Some studies show the evidence of improving cognitive impairment in selected i…

Kategori:
2-Amino-1-Phenylethanol DerivativesAdrenergic AgentsAdrenergic Agonists +29
Target Protein:
Interferon alpha/beta receptor 2Voltage-dependent T-type calcium channel subunit alpha-1I
Waktu ParuhDuration of action …
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Nystatin Approved DB00646
small molecule | CAS: 1400-61-9

Nystatin is a polyene antifungal drug that has broad-spectrum fungicidal and fungistatic activity against a number of yeasts and fungi, most notably _Candida_ species.[L10686] It is one of the most effective antifungal agents synthesized by bacteria, in this …

Kategori:
Alimentary Tract and MetabolismAnti-Infective AgentsAntidiarrheals, Intestinal Antiinflammatory/antiinfective Agents +17
Target Protein:
Ergosterol
Waktu Paruh-
Vol. DistribusiNystatin is not abs…
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NYX-2925 DB19149
small molecule | CAS: 2012536-16-0

NYX-2925 is under investigation in clinical trial NCT04146896 (Efficacy and Safety of NYX-2925 in Subjects With Neuropathic Pain Associated With Diabetic Peripheral Neuropathy (DPN)).

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small molecule

Deskripsi belum tersedia.

Target Protein:
Transaldolase B
Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
Poly [ADP-ribose] polymerase 1Exotoxin AElongation factor 2 +3
Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
Serine/threonine-protein kinase/endoribonuclease IRE1
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
N-succinylarginine dihydrolase
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small molecule

Deskripsi belum tersedia.

Target Protein:
ATP-dependent Clp protease proteolytic subunit
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small molecule

Deskripsi belum tersedia.

Target Protein:
Mitogen-activated protein kinase 14
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small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-secretase 1
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small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-secretase 1
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Vascular endothelial growth factor receptor 2
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Vascular endothelial growth factor receptor 2
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small molecule

Deskripsi belum tersedia.

Target Protein:
Carboxypeptidase A1
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small molecule | CAS: 5147-00-2

Deskripsi belum tersedia.

Target Protein:
Prostaglandin G/H synthase 1
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o-Bromophenol DB04586
small molecule | CAS: 95-56-7

Deskripsi belum tersedia.

Kategori:
Benzene Derivatives
Target Protein:
Thymidylate synthaseThymidylate synthase
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o-Cymen-5-ol DB15901
small molecule | CAS: 3228-02-2

Deskripsi belum tersedia.

Kategori:
Benzene Derivatives
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small molecule | CAS: 27415-09-4

Deskripsi belum tersedia.

Kategori:
Acids, Carbocyclic
Target Protein:
o-succinylbenzoate synthaseo-succinylbenzoate synthaseo-succinylbenzoate synthase
Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
Cyanovirin-N
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Oat Approved DB10546
biotech

Oat allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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OAV401 DB18254
biotech

Deskripsi belum tersedia.

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OBE101 DB05080
small molecule

OBE101 is a new weight loss drug developed by Obecure Ltd. It is a new formulation that is based on the vertigo medication, Betahistine. Obecure is repurposing betahistine, which is an H1 receptor agonist and partial H3 receptor antagonist for the treatment o…

Target Protein:
Histamine H1 receptorHistamine H3 receptor
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Obeldesivir DB18821
small molecule | CAS: 2647441-36-7

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
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Obeticholic acid Approved DB05990
small molecule | CAS: 459789-99-2

Primary biliary cirrhosis, or PBC, is a progressive and chronic condition that leads to hepatic injury often resulting in end-stage liver failure that requires liver transplantation.[A192786] Obeticholic acid is a farnesoid-X receptor (FXR) agonist used to…

Kategori:
Alimentary Tract and MetabolismBile Acid PreparationsBile acids and derivatives +14
Target Protein:
Bile acid receptor
Waktu ParuhThe biological half…
Vol. DistribusiThe volume of distr…
KlirensClearance informati…
Genetik -
Obexelimab DB15032
biotech | CAS: 1690307-05-1

Obexelimab is under investigation in clinical trial NCT02725515 (A Study of the Effect of XmAb®5871 in Patients With Systemic Lupus Erythematosus).

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OBI-3424 DB16057
small molecule | CAS: 2097713-68-1

OBI-3424 is under investigation in clinical trial NCT04315324 (Study to Test Akr1c3-activated Prodrug OBI-3424 (OBI-3424) in Patients With Relapsed/refractory T-cell Acute Lymphoblastic Leukemia (T-ALL)).

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OBI-888 DB18289
biotech | CAS: 2227156-40-1

Deskripsi belum tersedia.

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OBI-999 DB17356
biotech

Deskripsi belum tersedia.

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Obicetrapib DB14890
small molecule | CAS: 866399-87-3

Obicetrapib is under investigation in clinical trial NCT02241772 (A Study on the Effects of TA-8995 on Lp(a) in Subjects With Elevated Lp(a)).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Cholesteryl ester transfer protein
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Obidoxime DB13750
small molecule | CAS: 7683-36-5

Deskripsi belum tersedia.

Kategori:
AminesAntidotesCholinergic Agents +7
Target Protein:
Acetylcholinesterase
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Obiltoxaximab Approved DB05336
biotech | CAS: 1351337-07-9

Obiltoxaximab, an affinity-enhanced monoclonal antibody (Mab), is used for prevention and treatment of infection and death caused by anthrax toxin. Obiltoxaximab is a chimeric IgG1 kappa monoclonal antibody (mAb) that binds the PA component of B. anthracis to…

Kategori:
Amino Acids, Peptides, and ProteinsAnthrax Protective Antigen-directed AntibodyAnthrax Protective Antigen-directed Antibody Interactions +15
Target Protein:
Protective antigen
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