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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
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15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 178 / 315
Lactobacillus casei Approved DB16541
biotech | CAS: 68333-14-2

Deskripsi belum tersedia.

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biotech

Lactobacillus is a common bacteria found in the gut with Lactobacillus coryniformis K8 being originally isolated from artisan goat cheese.

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biotech

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small molecule

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Kategori:
Probiotics
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biotech

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biotech

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biotech

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biotech

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*Lactobacillus plantarum* is a member of Lactobacillus, or lactic acid bacteria, that it is widely used in the food industry as a microbial starter and probiotic microorganism. It is considered to be one of versatile species that carry out fermentative and me…

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biotech

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small molecule | CAS: 96-82-2

Deskripsi belum tersedia.

Kategori:
CarbohydratesOligosaccharidesPolysaccharides
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Lactoferrin DB16555
biotech | CAS: 151186-19-5

Lactoferrin is under investigation in clinical trial NCT03748043 (The Effectiveness of Lactoferrin in Treatment of Iron Deficiency Anemia in Children With Chronic Tonsillitis).

Kategori:
Amino Acids, Peptides, and ProteinsAnimal Proteins, DietaryAnti-Infective Agents +22
Target Protein:
Tryptase alpha/beta-1
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Lactuca sativa whole Approved DB15604
biotech

Lactuca sativa whole allergenic extract is used in allergenic testing.

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Lactulose Approved DB00581
small molecule | CAS: 4618-18-2

Lactulose is a synthetic disaccharide derivative of lactose that is most commonly used as a laxative agent despite also being formally indicated to serve as an adjunct therapy in treating portal-systemic encephalopathy (PSE).[FDA Label,L6199,L6202] Despite be…

Kategori:
Acidifying ActivityAlimentary Tract and MetabolismAmmonia Detoxicants +8
Target Protein:
Evolved beta-galactosidase subunit alpha
Waktu ParuhThe data regarding …
Vol. DistribusiNegligible amounts …
KlirensNegligible amounts …
Genetik -
Lacutamab DB15322
biotech | CAS: 2187368-16-5

Lacutamab is under investigation in clinical trial NCT02593045 (Study of IPH4102 in Patients With Relapsed/Refractory Cutaneous T-cell Lymphomas (CTCL)).

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Ladarixin DB16212
small molecule | CAS: 849776-05-2

Ladarixin is under investigation in clinical trial NCT04628481 (A Study of Oral Ladarixin in New-onset Type 1 Diabetes and a Low Residual ?-Cell Function).

Kategori:
AmidesReceptors, Interleukin-8A, antagonists & inhibitorsSulfones +1
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Lademirsen DB17611
biotech | CAS: 1404019-95-9

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biotech | CAS: 1629760-29-7

Ladiratuzumab vedotin is under investigation in clinical trial NCT01969643 (A Safety Study of SGN-LIV1A in Breast Cancer Patients).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Ladostigil DB16213
small molecule | CAS: 209394-27-4

Ladostigil is under investigation in clinical trial NCT01429623 (A 3 Year Study to Evaluate the Safety and Efficacy of Low Dose Ladostigil in Patients With Mild Cognitive Impairment).

Kategori:
IndenesMonoamine Oxidase A Inhibitors for interaction with Monoamine Oxidase A substrates
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] AAcetylcholinesterase
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Laevulinic Acid DB02239
small molecule | CAS: 123-76-2

Deskripsi belum tersedia.

Target Protein:
Delta-aminolevulinic acid dehydratase
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Lafutidine DB12770
small molecule | CAS: 118288-08-7

Lafutidine has been investigated in Peptic Ulcer, Community-acquired Pneumonia, and Gastroesophageal Reflux Disease (GERD).

Kategori:
AcetatesAcids, AcyclicAlimentary Tract and Metabolism +10
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biotech

Lagerstroemia indica whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Lamb Approved DB10537
biotech

Lamb allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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small molecule

Deskripsi belum tersedia.

Target Protein:
Camphor 5-monooxygenase
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small molecule

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Target Protein:
Azurin
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Lamivudine Approved DB00709
small molecule | CAS: 134678-17-4

A reverse transcriptase inhibitor and zalcitabine analog in which a sulfur atom replaces the 3' carbon of the pentose ring. It is used to treat Human Immunodeficiency Virus Type 1 (HIV-1) and hepatitis B (HBV).

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +26
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseHDNA +1
Waktu Paruh5 to 7 hours (healt…
Vol. DistribusiApparent volume of …
Klirens* Renal clearance =…
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Lamotrigine Approved DB00555
small molecule | CAS: 84057-84-1

Lamotrigine is an antiepileptic drug belonging in the phenyltriazine class. It is used in the treatment of both epilepsy and as a mood stabilizer in bipolar disorder. Lamotrigine is the first medication since lithium granted Food and Drug Administration (FDA)…

Kategori:
Agents causing hyperkalemiaAgents producing tachycardiaAnti-epileptic Agent +31
Target Protein:
Voltage-dependent R-type calcium channel subunit alpha-1ESodium channel protein type 11 subunit alphaVoltage-gated sodium channel alpha subunit +15
Waktu ParuhThe average elimina…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent p…
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Lampalizumab DB11826
biotech | CAS: 1278466-20-8

Lampalizumab has been used in trials studying the treatment of Geographic Atrophy.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +9
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Lanabecestat DB14814
small molecule | CAS: 1383982-64-6

Lanabecestat is under investigation in clinical trial NCT03499041 (A Study of LY3314814 in Participants With Liver Impairment).

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biotech | CAS: 1939139-26-0

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Lanadelumab Approved DB14597
biotech | CAS: 1426055-14-2

Lanadelumab, also known as DX-2930, is a human IgG1 monoclonal antibody designed for subcutaneous self-injection.[L4538] It is a fully human immunoglobulin, k-light-chain made in recombinant Chinese Hamster Ovary cells.[L4537] It has been granted priority rev…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Plasma kallikrein
Waktu ParuhLanadelumab has a h…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
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Lanatoside C DB13467
small molecule | CAS: 17575-22-3

Deskripsi belum tersedia.

Kategori:
CarbohydratesCardanolidesCardenolides +6
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Lancovutide DB05029
small molecule | CAS: 1391-36-2

Lancovutide, a peptide antibiotic, is in clinical development for the treatment of cystic fibrosis. Lancovutide is a 19-amino-acid tetracyclic peptide produced by Streptoverticillium cinnamoneus and is closely related to cinnamycin (Ro09-0198). It belongs to …

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Landiolol Approved DB12212
small molecule | CAS: 133242-30-5

Landiolol is a rapid-acting beta-blocker used for rapid ventricular rate control.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +11
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Landipirdine DB16214
small molecule | CAS: 1000308-25-7

Landipirdine is under investigation in clinical trial NCT02258152 (SYN120 Study to Evaluate Its Safety, Tolerability and Efficacy in Parkinson's Disease Dementia (SYNAPSE)).

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT2 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 65-hydroxytryptamine receptor 2A
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Landogrozumab DB11862
biotech | CAS: 1391726-30-9

Landogrozumab has been used in trials studying the treatment of Advanced Cancer, Muscular Atrophy, and Pancreatic Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Lanicemine DB11889
small molecule | CAS: 153322-05-5

Lanicemine has been used in trials studying the treatment and basic science of Depression, Major Depressive Disorder, and Treatment Resistant Major Depressive Disorder.

Kategori:
AminesAntidepressive AgentsCentral Nervous System Depressants +2
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Lanifibranor DB14801
small molecule | CAS: 927961-18-0

Lanifibranor is under investigation in clinical trial NCT03008070 (Phase 2b Study in NASH to Assess IVA337).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +2
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor deltaPeroxisome proliferator-activated receptor gamma
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Lanimostim DB06559
small molecule | CAS: 117276-75-2

Deskripsi belum tersedia.

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Laninamivir DB12791
small molecule | CAS: 203120-17-6

Laninamivir has been used in trials studying the treatment of Influenza.

Kategori:
Acids, AcyclicAmidinesAmino Sugars +11
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small molecule | CAS: 203120-46-1

Laninamivir octanoate has been used in trials studying the treatment of Asthma.

Kategori:
Acids, AcyclicAmidinesAmino Sugars +10
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Laniquidar DB12799
small molecule | CAS: 197509-46-9

Laniquidar has been used in trials studying the treatment of Breast Cancer.

Kategori:
Carbon RadioisotopesDrug Resistance, MultipleHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Phosphatidylcholine translocator ABCB4
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Lanolin Approved DB11112
small molecule | CAS: 8006-54-0

Lanolin is a yellow fat obtained from sheep's wool. It is used as an emollient, cosmetic, and pharmaceutic aid [L2580]. The US federal code of regulations states that lanolin in the concentration range of 12-50% may be included in over the counter skin ointme…

Kategori:
Basic Ointments and ProtectantsCompounds used in a research, industrial, or household settingCosmetics +3
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Lanolin alcohols Approved DB14181
small molecule | CAS: 8027-33-6

Lanolin alcohols are a complex combination of organic alcohols obtained by the hydrolysis of lanolin. It is administered as an ointment base with topical insulin and has shown to be antagonistic to wound healing. It is commonly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseStandardized Chemical Allergen
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Lanopepden DB11912
small molecule | CAS: 1152107-25-9

Lanopepden has been used in trials studying the treatment of Pneumonia, Infections, Bacterial, Skin Diseases, Infectious, and Skin Infections, Bacterial.

Kategori:
AminesAnti-Bacterial AgentsEnzyme Inhibitors +2
Target Protein:
Peptide deformylase
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Lanoteplase DB06245
biotech | CAS: 171870-23-8

Deskripsi belum tersedia.

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsBiological Factors +10
Target Protein:
Urokinase plasminogen activator surface receptorFibrinogen alpha chainKallikrein-1 +14
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Lanraplenib DB14770
small molecule | CAS: 1800046-95-0

Lanraplenib is under investigation in clinical trial NCT03285711 (Safety and Efficacy of Filgotinib and Lanraplenib in Adults With Lupus Membranous Nephropathy (LMN)).

Target Protein:
Tyrosine-protein kinase SYK
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Lanreotide Approved DB06791
small molecule | CAS: 108736-35-2

Lanreotide is a drug employed in the management of acromegaly (a hormonal condition caused by excess growth hormone) in addition to symptoms caused by neuroendocrine tumors, especially carcinoid syndrome. This drug is a long-acting analog of the drug somatost…

Kategori:
AcromegalyAmino Acids, Peptides, and ProteinsAntineoplastic Agents +22
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 5
Waktu ParuhHalf-life is approx…
Vol. DistribusiEstimated Volume of…
KlirensEstimated Clearance…
Genetik -
Lansoprazole Approved DB00448
small molecule | CAS: 103577-45-3

Lansoprazole marketed under the brand Prevacid, is a proton pump inhibitor (PPI) and is structurally classified as a substituted benzimidazole.[A177065] It reduces gastric acid secretion by targeting gastric H,K-ATPase pumps and is thus effective at promoting…

Kategori:
Acid ReducersAlimentary Tract and MetabolismAnti-Ulcer Agents +39
Target Protein:
Potassium-transporting ATPase alpha chain 1Microtubule-associated protein tau
Gen Terkait:
CYP2C19 CYP2C19 ABCB1
Waktu ParuhOne source reports …
Vol. DistribusiThe apparent volume…
KlirensThe reported cleara…
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