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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 177 / 252
Norclozapine DB05766
small molecule | CAS: 6104-71-8

ACP-104, or N-desmethylclozapine, is the major metabolite of clozapine, and is being developed by ACADIA as a novel, stand-alone therapy for schizophrenia. It combines an atypical antipsychotic efficacy profile with the added potential benefit of enhanced cog…

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +4
Target Protein:
Muscarinic acetylcholine receptor M1D(2) dopamine receptorD(3) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Nordazepam DB14028
small molecule | CAS: 1088-11-5

An intermediate in the metabolism of DIAZEPAM to OXAZEPAM. It may have actions similar to those of diazepam.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +15
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
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Genetik -
Norelgestromin Approved DB06713
small molecule | CAS: 53016-31-2

Norelgestromin is a drug used in contraception. Norelgestromin is the active progestin responsible for the progestational activity that occurs in women after application of ORTHO EVRA patch.

Kategori:
Adrenal Cortex HormonesAminesCombination Contraceptives (with Estrogen and derivatives) +17
Target Protein:
Progesterone receptorAlbuminAndrogen receptor
Waktu Paruh-
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Norepinephrine Approved DB00368
small molecule | CAS: 51-41-2

Precursor of epinephrine that is secreted by the adrenal medulla and is a widespread central and autonomic neurotransmitter. Norepinephrine is the principal transmitter of most postganglionic sympathetic fibers and of the diffuse projection system in the brai…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +34
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +9
Waktu Paruh-
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Norethandrolone DB12787
small molecule | CAS: 52-78-8

Norethandrolone is under investigation in clinical trial NCT00700544 (Treatment Outcome in Elderly Patients).

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +9
Waktu Paruh-
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Genetik -
small molecule | CAS: 3836-23-5

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norethisterone Approved DB00717
small molecule | CAS: 68-22-4

Norethisterone, also known as norethindrone, is a synthetic progestational hormone belonging to the 19-nortestosterone-derived class of progestins.[A10367] It is further classified as a second-generation progestin, along with [levonorgestrel] and its derivati…

Kategori:
Adrenal Cortex HormonesAnti-Gonadotropin-Releasing HormonesCombination Contraceptives (with Estrogen and derivatives) +34
Target Protein:
Progesterone receptorAndrogen receptorGlucocorticoid receptor
Waktu ParuhThe half-life of no…
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
Norethynodrel Approved DB09371
small molecule | CAS: 68-23-5

A synthetic progestational hormone with actions and uses similar to those of PROGESTERONE. It has been used in the treatment of functional uterine bleeding and endometriosis. As a contraceptive, it has usually been administered in combination with MESTRANOL.

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +18
Target Protein:
Estrogen receptorAndrogen receptorSex hormone-binding globulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norfenefrine DB13378
small molecule | CAS: 536-21-0

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +14
Waktu Paruh-
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Norfloxacin Approved DB01059
small molecule | CAS: 70458-96-7

A synthetic fluoroquinolone (fluoroquinolones) with broad-spectrum antibacterial activity against most gram-negative and gram-positive bacteria. Norfloxacin inhibits bacterial DNA gyrase.

Kategori:
4-QuinolonesAgents Causing Muscle ToxicityAnti-Bacterial Agents +24
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA topoisomerase 4 subunit A +4
Waktu Paruh3-4 hours
Vol. Distribusi-
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Genetik -
Norgestimate Approved DB00957
small molecule | CAS: 35189-28-7

Norgestimate was first described in the literature in 1977.[A191068] It was developed by Ortho Pharmaceutical Corporation as part of an effort to develop new hormonal contraceptives with reduced adverse effects.[A191068] It is commonly formulated with [ethiny…

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +27
Target Protein:
Progesterone receptorEstrogen receptorAndrogen receptor
Waktu ParuhNorgestimate is rap…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Norgestomet DB11440
small molecule | CAS: 25092-41-5

Norgestomet, also known as 11?-methyl-17-hydroxy-19-norprogesterone acetate, is a steroidal progestin used in veterinary medicine to control estrus and ovulation in cattle.

Kategori:
Fused-Ring CompoundsPregnanesPregnenes +2
Waktu Paruh-
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Norgestrel Approved DB09389
small molecule | CAS: 6533-00-2

Norgestrel is synthetic steroidal progestin that is used in combination with ethinyl estradiol for oral contraception. Norgestrel is composed of a racemic mixture of two stereoisomers, dextronorgestrel and levonorgestrel. However, only the levorotary enantio…

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +20
Target Protein:
Progesterone receptor3-oxo-5-alpha-steroid 4-dehydrogenase 1Androgen receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Norgestrienone DB13563
small molecule | CAS: 848-21-5

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +13
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Norleucine DB15458
small molecule | CAS: 327-57-1

Norleucine is under investigation in clinical trial NCT00081952 (Amino Acid Therapy for Hot Flashes in Postmenopausal Women).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAminocaproates
Target Protein:
Hepatocyte nuclear factor 1-alpha
Waktu Paruh-
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Normethadone Approved DB11609
small molecule | CAS: 467-85-6

Normethadone is used as an opioid antitussive in combination with [DB11610]. It is marketed in Canada by Valeant under the tradename Cophylac.

Kategori:
AnalgesicsAntitussive AgentsCentral Nervous System Agents +10
Waktu Paruh-
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Genetik -
small molecule | CAS: 156126-12-4

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Northern brown shrimp Approved DB15539
biotech

Northern brown shrimp allergenic extract is used in allergenic testing.

Waktu Paruh-
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Nortriptyline Approved DB00540
small molecule | CAS: 72-69-5

Nortriptyline hydrochloride, the active metabolite of [amitriptyline], is a tricyclic antidepressant (TCA).[L11878] It is used in the treatment of major depression and is also used off-label for chronic pain and other conditions.[L11881]

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +59
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +12
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +4
Waktu ParuhThe average plasma …
Vol. DistribusiThe apparent volume…
KlirensThe average plasma …
Genetik 7 Varian
Norvaline DB04185
small molecule | CAS: 6600-40-4

Norvaline is an isomer of the more common amino acid valine.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins
Target Protein:
Glycine amidinotransferase, mitochondrialOrnithine transcarbamylase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NOV-002 DB05393
small molecule

NOV-002, the lead compound acts as a chemoprotectant and an immunomodulator, in combination with chemotherapy. NOV-002 is approved and marketed in the Russian Fereration by Pharma BAM under the trade name Glutoxim. It has been administered to over 10,000 pati…

Kategori:
Amino Acids, Peptides, and ProteinsChlorine CompoundsNitrogen Compounds +3
Waktu Paruh-
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Genetik -
Novobiocin Approved DB01051
small molecule | CAS: 303-81-1

Novobiocin is an antibiotic compound derived from _Streptomyces niveus_. It has a chemical structure similar to coumarin. Novobiocin binds to DNA gyrase and blocks adenosine triphosphatase (ATPase) activity. (From Reynolds, Martindale The Extra Pharmacopoeia,…

Kategori:
AminocoumarinsAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA gyrase subunit B +1
Waktu Paruh6 hours
Vol. Distribusi-
Klirens-
Genetik -
Novolimus DB19085
small molecule | CAS: 151519-50-5

Novolimus is under investigation in clinical trial NCT04483791 (Dynamx Bioadaptor Hong Kong Registry).

Kategori:
LactonesPolyketides
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
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Genetik -
NOX-100 DB05799
small molecule

NOX-100 is the new nitric oxide (NO) neutralizing agent being developed by San Diego-based Medinox -- demonstrated its effectiveness and potential as a therapeutic to treat hemorrhagic shock. NOX-100 is the first in a series of proprietary NO neutralizing com…

Waktu Paruh-
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NOX-700 DB05464
small molecule

NOX-700, an new orally active dithiocarbamate-based nitric oxide (NO) blocking agent that is in development for the treatment of diabetes mellitus (type 2 diabetes). In animal studies, NOX-700 lowered serum glucose, improved glucose tolerance, and reduced the…

Kategori:
Acids, AcyclicCarbamatesSulfur Compounds
Target Protein:
Nuclear factor NF-kappa-B p100 subunitNuclear factor NF-kappa-B p105 subunit
Waktu Paruh-
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Klirens-
Genetik -
Noxytiolin Approved DB13838
small molecule | CAS: 15599-39-0

Local antibacterial that probably acts by releasing formaldehyde in aqueous solutions. It is used for THERAPEUTIC IRRIGATION of infected body cavities - bladder, peritoneum, etc. and as a spray for burns.

Kategori:
AmidesAnti-Infective AgentsAnti-Infective Agents, Local +5
Waktu Paruh-
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Genetik -
NP-50301 DB05662
small molecule

NP-50301 is an ophthalmic therapeutic eye drop treating post-menopausal Dry Eye Syndrome (DES). It is being developed by Nascent Pharmaceuticals. It is estimated that about 30% of postmenopausal women suffer symptoms of DES, which accounts for over 12 million…

Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NP-51 DB16995
small molecule | CAS: 66611-38-9

Deskripsi belum tersedia.

Kategori:
AminesEnzyme InhibitorsHydroxylamines
Target Protein:
Mitogen-activated protein kinase 8Mitogen-activated protein kinase 9Mitogen-activated protein kinase 10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NP-6A4 DB17599
biotech

NP-6A4 is a peptide designed to specifically bind and activate angiotensin II receptor type 2 (AT2R). It has an Orphan Drug designation from the FDA for pediatric cardiomyopathy.[A258523]

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NP-G2-044 DB14995
small molecule | CAS: 1807454-59-6

NP-G2-044 is under investigation in clinical trial NCT03199586 (Phase 1 Clinical Trial of Metastasis Inhibitor NP-G2-044 in Patients With Advanced or Metastatic Solid Tumors (Including Lymphoma)).

Kategori:
Heterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Fascin
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NPI 32101 DB05264
small molecule

NPI 32101 possesses both anti-inflammatory and broad spectrum antimicrobial activities. This combination of pharmacological properties may have additional therapeutic uses beyond dermatology.

Target Protein:
Cytokine receptor common subunit beta
Waktu Paruh-
Vol. Distribusi-
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NPS-2143 DB05695
small molecule | CAS: 284035-33-2

Deskripsi belum tersedia.

Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NPT520-34 DB17920
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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NRC-AN-019 DB17110
small molecule | CAS: 879507-25-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NRP-2945 DB18150
biotech

NRP-2945 is a 11-mer peptidomimetic.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NRP409 DB05235
small molecule

NRP409 is a triiodothyronine (T3) hormone, being investigated by New River Pharmaceuticals as a treatment for patients with primary hypothyroidism.

Target Protein:
Ketimine reductase mu-crystallinThyroid hormone receptor alpha
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NS-2359 DB05805
small molecule | CAS: 195875-68-4

NS2359 is a triple monoamine re-uptake inhibitor with a new, unique drug profile expected to yield important benefits compared to existing treatments of depression. Enhancing the function of the three neurotransmitters serotonin, noradrenalin and dopamine, NS…

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds +1
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS-3728 DB05835
small molecule | CAS: 265646-85-3

NS3728 is an orally active chloride channel blocker for the treatment of cancer.

Kategori:
AmidesAminesAnilides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS-398 DB14060
small molecule | CAS: 123653-11-2

NS-398 is a COX-2 inhibitor. It was developed as part of the mechanistic study of the cyclooxygenases.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +14
Target Protein:
Prostaglandin G/H synthase 2Cyclooxygenase 2
Waktu Paruh-
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Genetik -
NS-8593 DB16897
small molecule | CAS: 875755-39-8

Deskripsi belum tersedia.

Kategori:
AminesNaphthalenes
Waktu Paruh-
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NSC-663284 DB17038
small molecule | CAS: 383907-43-5

NSC-663284 is a potent quinolinedione Cdc25 phosphatase inhibitor.[A253052]

Kategori:
cdc25 Phosphatases, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
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NSI-189 DB16230
small molecule | CAS: 1270138-40-3

NSI-189 is under investigation in clinical trial NCT02695472 (Study of NSI-189 for Major Depressive Disorder).

Kategori:
AminesPyridines
Waktu Paruh-
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NSI-566 DB17954
biotech

NSI-566 is a stem cell therapy consisting of human spinal cord-derived neural stem cells. Developed by Seneca Biopharma, it is being investigated for the treatment of amyotrophic lateral sclerosis (ALS), stroke, and chronic spinal cord injury (cSCI).[L47097]

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NT 13 DB16953
small molecule | CAS: 117928-93-5

Deskripsi belum tersedia.

Waktu Paruh-
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NT-219 DB17490
small molecule | CAS: 1198078-60-2

Deskripsi belum tersedia.

Target Protein:
Insulin receptor substrate 2Insulin receptor substrate 1Signal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NTLA-2001 DB18525
biotech

NTLA-2001 is a clustered regularly interspaced short palindromic repeats CRISPR/ Cas9-based gene therapy consisting of a single guide RNA targeting the human TTR gene and a messenger RNA encoding Cas9.

Kategori:
Biomimetic MaterialsDrug CarriersMembranes, Artificial +6
Waktu Paruh-
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Genetik -
NTLA-2002 DB17597
biotech

NTLA-2002 is a lipid nanoparticle encapsulating single guide RNA (G012267) targeting the human KLKB1 gene and messenger RNA (mRNA000042) encoding Cas9. It is an investigational therapy designed to knock out the target gene kallikrein B1 (KLKB1) to reduce plas…

Waktu Paruh-
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Genetik -
NTP-42 DB18302
small molecule | CAS: 2055599-51-2

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
NTx-265 DB05649
biotech

NTx-265 is a combination of two currently marketed large molecules designed to stimulate the growth and differentiation of neural stem cells in adults who have suffered a stroke – the second leading cause of death worldwide. In May 2006, biotechnology company…

Waktu Paruh-
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NU1025 DB02690
small molecule | CAS: 90417-38-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Poly [ADP-ribose] polymerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 8801–8850 dari 12560
Sebelumnya Halaman 177 / 252 Berikutnya