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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 177 / 282
Mesdopetam DB16229
small molecule | CAS: 1403894-72-3

Mesdopetam is under investigation in clinical trial NCT04435431 (A Clinical Study of Mesdopetam in Patients With Parkinson's Disease Experiencing Levodopa Induced Dyskinesia).

Kategori:
AminesBenzene DerivativesDopamine Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 147-73-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesoheme DB02577
small molecule

The color-furnishing portion of hemoglobin. It is found free in tissues and as the prosthetic group in many hemeproteins.

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingPigments, Biological +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesoridazine Approved DB00933
small molecule | CAS: 5588-33-0

A phenothiazine antipsychotic with effects similar to chlorpromazine.

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +23
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A
Waktu Paruh24 to 48 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 208465-21-8

Mesosulfuron-methyl is under investigation in clinical trial NCT01118117 (A Multi-center Clinical Trial of the Misago™ Self-Expanding Stent System for Superficial Femoral Artery).

Kategori:
AmidesSulfonesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesterolone DB13587
small molecule | CAS: 1424-00-6

Mesterolone is a synthetic anabolic-androgenic steroid (AAS) and derivative of dihydrotestosterone (DHT). It is inactivated by 3?-hydroxysteroid dehydrogenase in skeleta muscules so it is considered a weak androgen. It is not a substrate for aromatase so it i…

Kategori:
5-Androstanon (3) DerivativesAnabolic AgentsAndrogens +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mestranol Approved DB01357
small molecule | CAS: 72-33-3

The 3-methyl ether of ethinyl estradiol. It must be demethylated to be biologically active. It is used as the estrogen component of many combination ORAL contraceptives.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +25
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metabutethamine DB13578
small molecule | CAS: 4439-25-2

Deskripsi belum tersedia.

Kategori:
AnestheticsAnesthetics, LocalEsters of Aminobenzoic Acid +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metacavir DB19084
small molecule | CAS: 120503-45-9

Metacavir is under investigation in clinical trial NCT02965859 (The Safety and Dose-range Study of Metacavir Enteric-coated Capsules in Patients With Chronic Hepatitis B).

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metamfetamine Approved DB01577
small molecule | CAS: 537-46-2

Metamfetamine (methamphetamine) is a psychostimulant and sympathomimetic drug, and a member of the amphetamine group of sympathomimetic amines. Methamphetamine can induce effects such as euphoria, increased alertness and energy, and enhanced self-esteem. It i…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +33
Target Protein:
D(2) dopamine receptorAlpha-1B adrenergic receptorSodium-dependent dopamine transporter +10
Gen Terkait:
PICK1
Waktu ParuhThe biological half…
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Metamizole Approved DB04817
small molecule | CAS: 50567-35-6

Metamizole (dipyrone) is a pyrazolone derivative that belongs to the group of nonacid nonopioids. It is considered a potent analgesic and antipyretic with favourable gastrointestinal tolerability.[A251885] Metamizole was formerly marketed in the US as Dimetho…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAminopyrine +16
Target Protein:
Prostaglandin G/H synthase 1
Waktu Paruh_In vitro_, the hal…
Vol. DistribusiMetamizole is quick…
KlirensThe clearance of 4-…
Genetik -
Metandienone DB13586
small molecule | CAS: 72-63-9

Metandienone is an orally active anabolic androgenic steroid. It was introduced to the market in the 1960s but later discontinued and withdrawn from the market. Although it is prohibited in and outside competition by the World Anti-Doping Agency, metandienone…

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat-labile enterotoxin B chainCholera enterotoxin subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metaraminol Approved DB00610
small molecule | CAS: 54-49-9

An adrenergic agonist that acts predominantly at alpha adrenergic receptors and also stimulates the release of norepinephrine. It has been used primarily as a vasoconstrictor in the treatment of hypotension.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +17
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metavert DB17306
small molecule | CAS: 1841125-91-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metelimumab DB18695
biotech | CAS: 272780-74-2

Metelimumab (CAT-192) is a monoclonal antibody targeted against transforming growth factor (TGF) beta-1.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metenkefalin DB12668
small molecule | CAS: 58569-55-4

Metenkefalin is an endogenous opioid and beta-endorphin.[A203225] It has been shown to reduce chromosomal abberations in patients with multiple sclerosis.[A203210] Metenkefalin, along with [tridecactide], are under investigation as an immunomodulatory therap…

Kategori:
Amino Acids, Peptides, and ProteinsEnkephalin, MethionineEnkephalins +9
Target Protein:
Delta-type opioid receptorMu-type opioid receptor
Waktu ParuhThe half life of me…
Vol. Distribusi-
Klirens-
Genetik -
Metergoline Approved DB13520
small molecule | CAS: 17692-51-2

Metergoline is an ergot-derived psychoactive drug that acts as a ligand for serotonin and dopamine receptors. Metergoline is an antagonist at various 5-HT receptor subtypes at a relatively low concentration and agonist at dopamine receptors.[A27181] Its use h…

Kategori:
Agents that produce hypertensionAlkaloidsAntidepressive Agents +18
Target Protein:
5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1E +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metformin Approved DB00331
small molecule | CAS: 657-24-9

Metformin is a biguanide antihyperglycemic agent and first-line pharmacotherapy used in the management of type II diabetes.[L12207,A176173] Metformin is considered an antihyperglycemic drug because it lowers blood glucose concentrations in type II diabete…

Kategori:
Alimentary Tract and MetabolismAmidinesBiguanides +11
Target Protein:
Multidrug and toxin extrusion protein 1Acetyl-CoA carboxylase 2Electron transfer flavoprotein-ubiquinone oxidoreductase, mitochondrial +2
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensRenal clearance is …
Genetik -
Metformin C-11 DB15181
small molecule

Metformin c-11 is under investigation in clinical trial NCT03122769 (Cardiac Uptake of Metformin, Visualized by Positron Emission Tomography).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 72156-70-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Methacholine Approved DB06709
small molecule | CAS: 55-92-5

Asthma is a complex condition associated with phenomena such as airway hyperresponsiveness (AHR), in which the smooth muscle in the airways (ASM) excessively contracts in response to stimuli, reducing pulmonary function and causing symptoms such as difficulty…

Kategori:
AminesAmmonium CompoundsAutonomic Agents +17
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methadone Approved DB00333
small molecule | CAS: 76-99-3

Methadone is a potent synthetic analgesic that works as a full µ-opioid receptor (MOR) agonist and N-methyl-d-aspartate (NMDA) receptor antagonist. As a full MOR agonist, methadone mimics the natural effects of the body's opioids, endorphins, and enkephalins …

Kategori:
AnalgesicsAnticholinergic AgentsAntidepressive Agents +50
Target Protein:
Mu-type opioid receptorNMDA receptorDelta-type opioid receptor +5
Waktu ParuhDue to interindivid…
Vol. DistribusiDue to interindivid…
KlirensDue to interindivid…
Genetik -
Methamidophos DB14972
small molecule | CAS: 10265-92-6

Methamidophos is under investigation in clinical trial NCT03223753 (Web-Based Physical Activity Intervention in Improving Long Term Health in Children and Adolescents With Newly Diagnosed Acute Lymphoblastic Leukemia in First Remission).

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methane DB15994
small molecule | CAS: 74-82-8

Deskripsi belum tersedia.

Kategori:
AlkanesHydrocarbons, Acyclic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 558-25-8

Methanesulfonyl Fluoride has been used in trials studying the treatment of Safety.

Kategori:
Cholinergic AgentsCholinesterase InhibitorsEnzyme Inhibitors +2
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methapyrilene DB04819
small molecule | CAS: 91-80-5

Methapyrilene, formerly marketed in many drug products, was shown to be a potent carcinogen. Manufacturers voluntarily withdrew methapyriline drug products from the market in May and June 1979.

Kategori:
AminesAminopyridinesAnti-Allergic Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methaqualone DB04833
small molecule | CAS: 72-44-6

Methaqualone is a sedative-hypnotic drug that is similar in effect to barbiturates, a general central nervous system depressant. The sedative-hypnotic activity was first noted by Indian researchers in the 1950s and in 1962 methaqualone itself was patented in …

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP3A Substrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methcathinone DB15339
small molecule | CAS: 5650-44-2

Methcathinone is under investigation in clinical trial NCT02617862 (PCI Imaging System in Pediatric Ophthalmology).

Kategori:
Ketones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methdilazine Approved DB00902
small molecule | CAS: 1982-37-2

Methdilazine is a phenothiazine compound with antihistaminic activity. It is used in the treatment of various dermatoses to relieve pruritus.

Kategori:
Agents that reduce seizure thresholdAntihistamines for Systemic UseHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methfuroxam DB16231
small molecule | CAS: 28730-17-8

Methfuroxam is under investigation in clinical trial NCT01213407 (Dendritic Cell Cancer Vaccine for High-grade Glioma).

Kategori:
AmidesAminesAniline Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactam-inducible penicillin-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 26403-67-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methimazole Approved DB00763
small molecule | CAS: 60-56-0

Methimazole is a thionamide antithyroid agent that inhibits the synthesis of thyroid hormones.[A184559,A184733,A184694] It was first introduced as an antithyroid agent in 1949[A184502] and is now commonly used in the management of hyperthyroidism, particularl…

Kategori:
Antithyroid agentsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +30
Target Protein:
Thyroid peroxidase
Waktu ParuhFollowing a single …
Vol. DistribusiThe apparent volume…
KlirensFollowing a single …
Genetik -
Methiodal DB13321
small molecule | CAS: 143-47-5

Deskripsi belum tersedia.

Kategori:
AlkanesAlkanesulfonatesAlkanesulfonic Acids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methionine Approved DB00134
small molecule | CAS: 63-68-3

A sulfur containing essential amino acid that is important in many body functions. It is a chelating agent for heavy metals.

Kategori:
Amino AcidsAmino Acids, EssentialAmino Acids, Neutral +7
Target Protein:
Methionine synthase reductaseMethionine synthaseMethionine aminopeptidase 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methionine C-11 DB17147
small molecule | CAS: 60305-58-0

Deskripsi belum tersedia.

Kategori:
Diagnostic RadiopharmaceuticalsTumour Detection
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Methionine--tRNA ligaseMethionine aminopeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 15985-39-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 21752-32-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methocarbamol Approved DB00423
small molecule | CAS: 532-03-6

Methocarbamol was developed in the early 1950s as a treatment for muscle spasticity and the associated pain.[A178441,A178450] It is a guaiacol glyceryl ether.[A178450] Methocarbamol tablets and intramuscular injections are prescription medicines indicated …

Kategori:
Acids, AcyclicBenzene DerivativesCarbamates +14
Target Protein:
Carbonic anhydrase 1
Waktu ParuhThe elimination hal…
Vol. DistribusiVolume of distribut…
Klirens0.2-0.8L/h/kg.[L626…
Genetik -
Methohexital Approved DB00474
small molecule | CAS: 151-83-7

An intravenous anesthetic with a short duration of action that may be used for induction of anesthesia.

Kategori:
AnestheticsAnesthetics, GeneralAnesthetics, Intravenous +10
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh5.6 ± 2.7 mi…
Vol. Distribusi-
Klirens-
Genetik -
Methopterin DB16620
small molecule | CAS: 2410-93-7

Methopterin is thought to have effects on osteoclasts and to inhibit inflammatory bone destruction.[A229843]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methotrexate Approved DB00563
small molecule | CAS: 59-05-2

Methotrexate is a folate derivative that inhibits several enzymes responsible for nucleotide synthesis.[A180322] This inhibition leads to suppression of inflammation as well as prevention of cell division.[A180322] Because of these effects, methotrexate is of…

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAgents Causing Muscle Toxicity +42
Target Protein:
Thymidylate synthaseReduced folate transporterProton-coupled folate transporter +2
Gen Terkait:
ABCC2 MTHFR
Waktu ParuhThe half life of lo…
Vol. DistribusiThe volume of distr…
KlirensMethotrexate cleara…
Genetik 2 Varian
Methotrimeprazine Approved DB01403
small molecule | CAS: 60-99-1

A phenothiazine with pharmacological activity similar to that of both chlorpromazine and promethazine. It has the histamine-antagonist properties of the antihistamines together with central nervous system effects resembling those of chlorpromazine. (From Mart…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +46
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorD(1B) dopamine receptor +16
Waktu ParuhApproximately 20 ho…
Vol. Distribusi-
Klirens-
Genetik -
Methoxamine Approved DB00723
small molecule | CAS: 390-28-3

An alpha-adrenergic agonist that causes prolonged peripheral vasoconstriction. It has little if any direct effect on the central nervous system.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +19
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methoxsalen Approved DB00553
small molecule | CAS: 298-81-7

A naturally occurring furocoumarin compound found in several species of plants, including Psoralea corylifolia. It is a photoactive substance that forms DNA adducts in the presence of ultraviolet A irradiation.

Kategori:
AntipsoriaticsAntipsoriatics for Systemic UseAntipsoriatics for Topical Use +24
Target Protein:
DNACytochrome P450 2A6
Waktu ParuhApproximately 2 hou…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 180509-15-3

Methoxy arachidonyl fluorophosphonate, commonly referred as MAFP, is an irreversible active site-directed enzyme inhibitor that inhibits nearly all serine hydrolases and serine proteases. It inhibits phospholipase A2 and fatty acid amide hydrolase with specia…

Kategori:
EicosanoidsEnzyme InhibitorsFatty Acids +5
Target Protein:
Fatty-acid amide hydrolase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Pegylated agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 677324-53-7

Methoxy polyethylene glycol-epoetin beta is a chemically synthesised Erythropoiesis Stimulating Agent (ESA) with a longer half-life than erythropoietin. ESA is used to increase synthesis of red blood cells to treat chronic kidney disease associated anemia.

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsAntianemic Preparations +20
Target Protein:
Erythropoietin receptor
Waktu ParuhIn CKD patients on …
Vol. Distribusi~94.74 ml/kg
KlirensIn CKD patients on …
Genetik -
Menampilkan 8801–8850 dari 14063
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