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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 176 / 252
Nitisinone Approved DB00348
small molecule | CAS: 104206-65-7

Nitisinone is a synthetic reversible inhibitor of 4-hydroxyphenylpyruvate dioxygenase. It is used in the treatment of hereditary tyrosinemia type 1. It is sold under the brand name Orfadin.

Kategori:
4-Hydroxyphenyl-Pyruvate Dioxygenase Inhibitor4-Hydroxyphenylpyruvate Dioxygenase, antagonists & inhibitorsAcids, Carbocyclic +12
Target Protein:
4-hydroxyphenylpyruvate dioxygenase
Waktu Paruh~54 hours
Vol. Distribusi-
Klirens-
Genetik -
Nitrate DB14049
small molecule | CAS: 14797-55-8

Deskripsi belum tersedia.

Kategori:
AnionsAntianginal AgentsElectrolytes +5
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitrazepam Approved DB01595
small molecule | CAS: 146-22-5

A benzodiazepine derivative used as an anticonvulsant and hypnotic.

Kategori:
Anti-Anxiety AgentsAnticonvulsantsBenzazepines +22
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site +1
Waktu Paruh15-38 hours (mean e…
Vol. Distribusi-
Klirens-
Genetik -
Nitrendipine Approved DB01054
small molecule | CAS: 39562-70-4

Nitrendipine is a calcium channel blocker with marked vasodilator action. It is an effective antihypertensive agent and differs from other calcium channel blockers in that it does not reduce glomerular filtration rate and is mildly natriuretic, rather than so…

Kategori:
ACE Inhibitors and Calcium Channel BlockersAgents causing hyperkalemiaAntiarrhythmic agents +21
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitric acid DB15995
small molecule | CAS: 7697-37-2

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicCompounds used in a research, industrial, or household setting +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitric Oxide Approved DB00435
small molecule | CAS: 10102-43-9

Nitric oxide or Nitrogen monoxide is a chemical compound with chemical formula NO. This gas is an important signaling molecule in the body of mammals including humans and is an extremely important intermediate in the chemical industry. It is also a toxic air …

Kategori:
Anti-Asthmatic AgentsAntioxidantsAutonomic Agents +30
Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1Guanylate cyclase soluble subunit alpha-2 +3
Waktu Paruh2–6 seconds
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 139-13-9

Nitrilotriacetic acid is a derivative of acetic acid, N(CH2COOH)3. It is a complexing (sequestering) agent that forms stable complexes with Zn2+. (From Miall's Dictionary of Chemistry, 5th ed.)

Kategori:
AcetatesAcids, AcyclicAmino Acids, Peptides, and Proteins +4
Target Protein:
Lactotransferrin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitrite Approved DB12529
small molecule | CAS: 14797-65-0

Nitrite is under investigation for the treatment of Heart Failure.

Kategori:
AnionsElectrolytesIons +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitroarginine DB04223
small molecule | CAS: 2149-70-4

An inhibitor of nitric oxide synthetase which has been shown to prevent glutamate toxicity. Nitroarginine has been experimentally tested for its ability to prevent ammonia toxicity and ammonia-induced alterations in brain energy and ammonia metabolites. (Neur…

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +3
Target Protein:
Nitric oxide synthase 1Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitroaspirin DB12445
small molecule | CAS: 175033-36-0

Nitroaspirin has been investigated for the treatment of Intermittent Claudication.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +19
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitrocefin DB11592
small molecule | CAS: 41906-86-9

Nitrocefin is a chromogenic cephalosporin substrate used to detect the presence of beta-lactamase enzymes, an important mediator of bacterial antibiotic resistance. While other detection methods exist, such as PCR, nitrocefin allows for rapid detection using …

Kategori:
Amidesbeta-LactamsCompounds used in a research, industrial, or household setting +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitrofural Approved DB00336
small molecule | CAS: 59-87-0

Nitrofural or nitrofurazone is a topical anti-infective agent effective against gram-negative and gram-positive bacteria. It is used for superficial wounds, burns, ulcers, and skin infections. Nitrofural has also been administered orally in the treatment of t…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Products, Insecticides and Repellents +15
Target Protein:
Glutathione reductase
Waktu Paruh5 hours
Vol. Distribusi-
Klirens-
Genetik -
Nitrofurantoin Approved DB00698
small molecule | CAS: 67-20-9

Nitrofurantoin is a nitrofuran antibiotic used to treat uncomplicated urinary tract infections.[L6856,L6859,L6862] Nitrofurantoin is converted by bacterial nitroreductases to electrophilic intermediates which inhibit the citric acid cycle as well as synthesis…

Kategori:
Agents causing hyperkalemiaAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
Probable pyruvate-flavodoxin oxidoreductaseOxygen-insensitive NADPH nitroreductase30S ribosomal protein S10
Waktu ParuhThe half life of ni…
Vol. DistribusiData regarding the …
KlirensThe clearance of ni…
Genetik -
Nitrogen Approved DB09152
small molecule | CAS: 7727-37-9

Nitrogen is a chemical element with symbol N and atomic number 7. At room temperature, it is a transparent, odorless diatomic gas. Liquid nitrogen is used principally in cryotherapy for removal of diseased skin. Liquid nitrogen helps in removal of skin lesi…

Kategori:
ElementsGasesMedical Gases +2
Waktu ParuhFor local use only.
Vol. DistribusiFor local use only.
KlirensFor local use only.
Genetik -
small molecule | CAS: 10025-85-1

Deskripsi belum tersedia.

Kategori:
AnionsChlorine CompoundsElectrolytes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitroglycerin Approved DB00727
small molecule | CAS: 55-63-0

Nitroglycerin, also known as glyceryl trinitrate,[A180169] is an organic nitrate and a vasodilating agent [L38369] that was first discovered in 1847.[A249965] Originally used to dynamite, its antianginal effects were identified in the late 1860s after it prod…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAntianginal AgentsAntihypertensive Agents +14
Target Protein:
Epidermal growth factor receptorGuanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1 +1
Waktu ParuhFollowing intraveno…
Vol. DistribusiThe volume of distr…
KlirensThe estimated clear…
Genetik -
Nitroprusside Approved DB00325
small molecule | CAS: 15078-28-1

Nitroprusside serves as a source of nitric oxide, a potent peripheral vasodilator that affects both arterioles and venules (venules more than arterioles). Nitroprusside is often administered intravenously to patients who are experiencing a hypertensive emerge…

Kategori:
AnionsAntihypertensive AgentsArteriolar Smooth Muscle, Agents Acting On +20
Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1Atrial natriuretic peptide receptor 1
Waktu ParuhApproximately 2 min…
Vol. Distribusi-
Klirens-
Genetik -
Nitrosoethane DB02646
small molecule | CAS: 925-91-7

Deskripsi belum tersedia.

Target Protein:
Myoglobin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitroxoline DB01422
small molecule | CAS: 4008-48-4

Nitroxoline is a urinary antibacterial agent active against susceptible gram-positive and gram-negative organisms commonly found in urinary tract infections. It is a hydroxyquinoline derivative unrelated to other classes of drugs.[A179251] Nitroxoline is acti…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +5
Target Protein:
Methionine aminopeptidase 2Magnesium cationManganese cation
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nivatrotamab DB16654
biotech | CAS: 2278244-14-5

Nivatrotamab is under investigation in clinical trial NCT03860207 (Study of the Safety and Efficacy of Humanized 3F8 Bispecific Antibody (Hu3f8-bsab) in Patients With Relapsed/refractory Neuroblastoma, Osteosarcoma and Other Solid Tumor Cancers).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nivocasan DB12720
small molecule | CAS: 908253-63-4

Nivocasan has been used in trials studying the treatment of HCV Infection and Nonalcoholic Steatohepatitis.

Target Protein:
Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nivolumab Approved DB09035
biotech | CAS: 946414-94-4

Nivolumab is a fully human IgG4 antibody targeting the immune checkpoint programmed death receptor-1 (PD-1).[L12129] This antibody was produced entirely in mice and grafted onto human kappa and IgG4 Fc region with the mutation _S228P_ for additional stability…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntibodies +20
Target Protein:
Programmed cell death protein 1Programmed cell death 1 ligand 1
Waktu ParuhThe serum half life…
Vol. DistribusiThe volume of distr…
KlirensThe estimated clear…
Genetik -
Nizatidine Approved DB00585
small molecule | CAS: 76963-41-2

A histamine H2 receptor antagonist with low toxicity that inhibits gastric acid secretion. The drug is used for the treatment of duodenal ulcers.

Kategori:
Acid ReducersAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +13
Target Protein:
Histamine H2 receptor
Waktu Paruh1-2 hours
Vol. Distribusi* 0.8 to 1.5 L/kg
Klirens* 40-60 L/h * 7 – …
Genetik -
Nizofenone DB13546
small molecule | CAS: 54533-85-6

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsCardiovascular AgentsCentral Nervous System Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

These cells are prepared as universal off-the-shelf CAR-NK cells from cord blood with NKG2D-ACE2 proteins engineered as part of the CARs; the cell secretes IL-15 and GM-CSF. Chimeric antigen receptors (CARs) are artificial receptors consisting of an antibody-…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NKX101 DB18131
biotech

NKX101 is an investigational allogeneic chimeric antigen receptor (CAR)-natural killer cell therapy.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NLX-P101 DB05924
small molecule

NLX-P101, gene therapy is developed by Neurologix to treat Parkinson’s disease. The gene is glutamic acid decarboxylase (GAD), whose product synthesizes the major inhibitory neurotransmitter in the brain, (gamma)-aminobutyric acid (GABA), and targets the subt…

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NM-004 DB18066
small molecule | CAS: 402934-69-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NM-702 DB05505
small molecule

Nissan Chemical and Taisho have been jointly developing NM-702, a drug for the treatment of arteriosclerosis obliterans. M-702 is an orally active inhibitor of phosphodiesterase and thromboxane synthetase. In Japan, Phase 2 studies are being conducted for …

Target Protein:
Thromboxane-A synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NMD-670 DB18466
small molecule | CAS: 2354321-33-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NN344 DB05115
small molecule

NN344 is a neutral, soluble long-acting human insulin analogue with 24 hour coverage by once daily injection. NN344 has a very flat and predictable action profile. The product is intended for basal insulin treatment of diabetes mellitus.

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsCytochrome P-450 CYP1A2 Inducers +9
Target Protein:
Insulin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 357400-14-7

NNC-55-0396 is a T-type Ca(2+) channel inhibitor.[A253047]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NNI-351 DB18048
small molecule | CAS: 929607-23-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NNZ-2591 DB15601
small molecule | CAS: 847952-38-9

NNZ-2591 (cyclo-L-glycyl-L-2-allylproline)[A189390] is an investigational synthetic analog of cyclic glycine-proline (cGP), a breakdown product of human insulin-like growth factor 1 (IGF-1), that has been chemically modified to increase its half-life, stabili…

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPiperazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nofazinlimab DB18852
biotech | CAS: 2377845-98-0

Nofazinlimab is under investigation in clinical trial NCT04194775 (A Study of Nofazinlimab (CS1003) in Subjects With Advanced Hepatocellular Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nogapendekin alfa Approved DB18740
biotech | CAS: 1622189-43-8

Nogapendekin alfa is a human IL-15N72D variant. It is one of the active ingredients in Anktiva, a combination product also containing [inbakicept], where a single inbakicept is complexed with two nogapendekin alfa components.[L50592] This combination product …

Kategori:
Amino Acids, Peptides, and ProteinsInterleukin-15Proteins +2
Target Protein:
Interleukin-2 receptor subunit betaCytokine receptor common subunit gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nolasiban DB16259
small molecule | CAS: 1477482-19-1

Nolasiban is under investigation in clinical trial NCT03081208 (Phase 3 Placebo Controlled Study of Nolasiban to Improve Pregnancy Rates in Women Undergoing IVF/ICSI).

Kategori:
AminesHydroxylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 153050-21-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomacopan DB14991
biotech | CAS: 875125-19-2

Nomacopan is under investigation in clinical trial NCT03427060 (Coversin in PNH in Patients With Resistance to Eculizumab Due to Complement C5 Polymorphisms).

Kategori:
Recombinant Protein Inhibitor of Complement Factor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomegestrol Approved DB11636
small molecule | CAS: 58691-88-6

Nomegestrol is an ingredient in the EMA-authorised product Zoely.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomegestrol acetate Approved DB13981
small molecule | CAS: 58652-20-3

Nomegestrol acetate, also known as NOMAC, is a progestin used in oral contraceptives, menopausal hormone therapy, and for the treatment of gynecological disorders.

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +14
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomifensine Approved DB04821
small molecule | CAS: 24526-64-5

Nomifensine, formerly marketed as Merital capsules, was associated with an increased incidence of hemolytic anemia. The approved application holder removed Merital capsules from the market on January 23, 1986. FDA published a notice of its determination that …

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsDopamine Agents +8
Target Protein:
D(2) dopamine receptorSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomlabofusp DB17903
biotech | CAS: 2548202-05-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nonacog beta pegol Approved DB13933
biotech | CAS: 1175512-71-6

Nonacog beta pegol is a recombinant coagulation factor IX derivative. It is produced without animal-derived materials and with an attached 40kDa polyethylene glycol (PEG) molecule for peptide activation by a site-directed glycoPEGylation. Once activated, the …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +10
Target Protein:
Coagulation factor VIICoagulation factor VIIICoagulation factor X
Waktu ParuhThe mean half-life …
Vol. DistribusiThe volume of distr…
KlirensMean clearance in c…
Genetik -
Nonoxynol-9 Approved DB06804
small molecule | CAS: 26027-38-3

Nonoxynol-9 (N-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives. When present in the vagina during intercourse, they immobilize/inactivate/damage and/or kill sperms without eliciting systemic …

Kategori:
Adrenal Cortex HormonesAlcoholsAntispermatogenic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NOP-1A DB15208
small molecule | CAS: 1283095-70-4

NOP-1A is under investigation in clinical trial NCT01198197 (PET Brain and Whole Body Distribution Studies for Nociceptin/Orphanin FQ Peptide (NOP) Receptor Using [11C]NOP-1A).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
nor-NOHA DB02381
small molecule | CAS: 189302-40-7

N-Hydroxy-nor-L-arginine (nor-NOHA) is under investigation in clinical trial NCT02009527 (Arginase Inhibition in Ischemia-reperfusion Injury).

Target Protein:
Arginase-2, mitochondrialArginase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norbixin DB15201
small molecule | CAS: 542-40-5

Norbixin is under investigation in clinical trial NCT03820245 (Effect of Short-term Annatto Carotenoids Supplementation on Oxidative Stress Status in Healthy Individuals).

Kategori:
AlkenesBiological FactorsCyclohexanes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norcamphor DB03540
small molecule

Deskripsi belum tersedia.

Kategori:
Bridged-Ring Compounds
Target Protein:
Camphor 5-monooxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norclobazam DB17092
small molecule | CAS: 22316-55-8

Deskripsi belum tersedia.

Kategori:
AnticonvulsantsBenzazepinesCentral Nervous System Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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