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13591

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10177 (74.9%)
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7625 (56.1%)
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104 (0.8%)
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13591 (100.0%)

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Halaman 176 / 272
Mitumomab DB06462
biotech | CAS: 216503-58-1

Mitumomab, an anti-BEC-2 monoclonal antibody derived from mice, was previously studied to treat small cell lung carcinoma in combination with BCG vaccination.

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MIV-701 DB05736
small molecule

MIV-701 is a selective, potent inhibitor of the protease Cathepsin K. It is developed for the treatment of osteoporosis.

Target Protein:
Cathepsin K
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MIV-711 DB15599
small molecule

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsAntineoplastic AgentsAntirheumatic Agents
Target Protein:
Cathepsin K
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Mivacurium Approved DB01226
small molecule | CAS: 133814-19-4

Mivacurium is a bisbenzylisoquinolinium based neuromuscular blocker or muscle relaxant. It binds competitively to cholinergic receptors on the motor end-plate to antagonize the action of acetylcholine, resulting in a block of neuromuscular transmission.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCentral Nervous System Depressants +13
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +1
Waktu ParuhThe mean eliminatio…
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Mivavotinib DB16849
small molecule | CAS: 1312691-33-0

Deskripsi belum tersedia.

Target Protein:
Receptor-type tyrosine-protein kinase FLT3Tyrosine-protein kinase SYK
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Mivelsiran DB19003
biotech | CAS: 2572991-83-2

Mivelsiran is under investigation in clinical trial NCT06393712 (A Phase 2 Trial of ALN-APP in Patients With Cerebral Amyloid Angiopathy).

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Mizagliflozin DB19036
small molecule | CAS: 666843-10-3

Mizagliflozin is under investigation in clinical trial NCT05721729 (Effect of Mizagliflozin Repeat Dosing on Adverse Events and Postprandial Glucose Excursions).

Kategori:
CarbohydratesGlycosides
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Mizolastine Approved DB12523
small molecule | CAS: 108612-45-9

Mizolastine is under investigation in clinical trial NCT01928316 (A Bioequivalence Study of Domestic (Made in China) and Imported Mizolastine Tablets in Healthy Volunteers).

Kategori:
Antihistamines for Systemic UseCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +9
Target Protein:
Histamine H1 receptor
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MK-0354 DB05939
small molecule | CAS: 851776-28-8

MK-0354, is an orally administered drug candidate under development by Merck for the treatment of atherosclerosis and related disorders. It targets G protein-coupled receptor, or GPCR, that have the potential to regulate plasma lipid profiles, including HDL, …

Target Protein:
Hydroxycarboxylic acid receptor 2G-protein coupled estrogen receptor 1
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MK-0482 DB17453
biotech

MK-0482 is a novel humanized IgG4 monoclonal antibody targeting the immunoglobulin-like transcript (ILT) 3.

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MK-0533 DB15242
small molecule | CAS: 668455-28-5

MK-0533 is under investigation in clinical trial NCT00543959 (Efficacy and Tolerability of MK0533 in Patients With Type 2 Diabetes (0533-005)).

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MK-0557 DB12168
small molecule | CAS: 328232-95-7

MK0557 has been investigated for the treatment of Schizophrenia and Paranoid Schizophrenia.

Kategori:
Cycloparaffins
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MK-0686 DB12563
small molecule | CAS: 578727-68-1

MK0686 has been used in trials studying the treatment of Osteoarthritis, Pain, Postoperative, and Neuralgia, Postherpetic.

Kategori:
AcetatesAcids, AcyclicAcids, Carbocyclic +2
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MK-0731 DB08037
small molecule | CAS: 845256-65-7

MK-0731 is a kinesin spindle protein inhibitor and antineoplastic agent.

Target Protein:
Kinesin-like protein KIF11
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MK-0736 DB15209
small molecule | CAS: 719272-79-4

MK-0736 is under investigation in clinical trial NCT00679055 (A Study of How MK-0736 Affects Arterial Plaque (0736-006)(TERMINATED)).

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MK-0767 DB12055
small molecule | CAS: 934017-32-0

MK0767 has been used in trials studying the treatment of Dyslipidemia, Diabetes Mellitus, Type 2 Diabetes Mellitus, Diabetes Mellitus, Type 2, and Diabetes Mellitus, Type II, among others.

Kategori:
Sulfur Compounds
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MK-0773 DB16244
small molecule | CAS: 606101-58-0

MK-0773 is under investigation in clinical trial NCT00529659 (A Study of the Safety and Efficacy of MK-0773 in Women With Sarcopenia (Loss of Muscle Mass)(mk-0773-005)).

Kategori:
Fused-Ring CompoundsSteroids
Target Protein:
Androgen receptor
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MK-0777 DB12238
small molecule | CAS: 252977-51-8

MK-0777 has been used in trials studying the treatment of Schizophrenia, Anxiety Disorder, and Generalized Anxiety Disorder.

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MK-0812 DB11990
small molecule | CAS: 624733-88-6

MK0812 has been used in trials studying the treatment of Relapsing-Remitting Multiple Sclerosis.

Target Protein:
C-C chemokine receptor type 2
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MK-0873 DB13029
small molecule | CAS: 500355-52-2

MK-0873 has been used in trials studying the treatment of Rheumatoid Arthritis.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPhosphodiesterase 4 Inhibitors +1
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4D
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MK-0893 DB12044
small molecule

MK0893 has been used in trials studying the treatment of Type 2 Diabetes Mellitus and Diabetes Mellitus, Type 2.

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +1
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MK-1064 DB15028
small molecule | CAS: 1207253-08-4

MK-1064 is under investigation in clinical trial NCT02549014 (A Single Dose Study of the Safety, Pharmacokinetics and Pharmacodynamics of MK-1064 (MK-1064-001)).

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MK-1454 DB14721
small molecule

A synthetic cyclic dinucleotide (CDN) and agonist of stimulator of interferon genes protein (STING), with potential immunoactivating and antineoplastic activities. Upon intratumoral (IT) administration, STING agonist MK-1454 binds to STING and activates the S…

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MK-1496 DB12763
small molecule | CAS: 1037254-47-9

MK-1496 has been used in trials studying the treatment of Neoplasms and Malignant.

Target Protein:
Serine/threonine-protein kinase PLK1
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MK-2206 DB16828
small molecule | CAS: 1032349-93-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Ubiquitin-conjugating enzyme E2 TRAC-gamma serine/threonine-protein kinase
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MK-2748 DB15371
small molecule | CAS: 1193902-95-2

MK-2748 is under investigation in clinical trial NCT01593735 (A Multiple Dose Study to Evaluate the Safety and Efficacy of MK-2748 in Hepatitis C-Infected Participants (MK-2748-002 AM1)).

Kategori:
Sulfur Compounds
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MK-3207 DB12424
small molecule | CAS: 957118-49-9

Mk3207 has been used in trials studying the treatment of Migraine and Migraine Disorders.

Kategori:
Receptors, Calcitonin Gene-Related Peptide, antagonists & inhibitors
Target Protein:
Calcitonin gene-related peptide type 1 receptor
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MK-3577 DB14957
small molecule | CAS: 1019112-29-8

MK-3577 is under investigation in clinical trial NCT00868790 (A Study of the Safety and Efficacy of MK-3577 in Participants With Type 2 Diabetes Mellitus (MK-3577-009)).

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MK-4541 DB17016
small molecule | CAS: 796885-38-6

MK-4541 is a 4-azasteroid and a selective androgen receptor modulator (SARM). MK-4541 acts as a dual selective SARM and is both a potent androgen receptor antagonist and a 5?-reductase inhibitor.[A252687]

Kategori:
Acids, AcyclicFused-Ring CompoundsSteroids
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MK-4721 DB05933
biotech

MK-4721 is a fully human monoclonal antibody directed to Agensys’ proprietary target Prostate Stem Cell Antigen (PSCA), an antigen expressed at significant levels on tumor cells from the majority of patients with all stages of prostate, pancreatic and bladder…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Prostate stem cell antigen
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MK-4830 DB17454
biotech

MK-4830 is a monoclonal antibody that targets the myeloid-specific immunoglobulin-like transcript (ILT) 4 receptor.

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MK-4965 DB08460
small molecule | CAS: 920035-77-4

MK-4965 is an HIV-1 reverse transcriptase inhibitor.

Kategori:
HIV Reverse Transcriptase, antagonists & inhibitors
Target Protein:
Gag-Pol polyprotein
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MK-5108 DB12556
small molecule | CAS: 1010085-13-8

MK-5108 has been used in trials studying the treatment of Cancer, Neoplasms, Tumors.

Kategori:
Acids, CarbocyclicCyclohexanesCycloparaffins +2
Target Protein:
Aurora kinase BAurora kinase A
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MK-6186 DB12999
small molecule | CAS: 1034474-19-5

MK6186 has been used in trials studying the treatment of HIV-1 Infection.

Target Protein:
Gag-Pol polyprotein
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MK-6325 DB15249
small molecule | CAS: 1263814-52-3

MK-6325 is under investigation in clinical trial NCT01329913 (Safety, Pharmacokinetics, and Pharmacodynamics of MK-6325 in Hepatitis C Virus (HCV) Infections (MK-6325-003)).

Target Protein:
Genome polyprotein
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MK-7288 DB17094
small molecule | CAS: 936626-07-2

Deskripsi belum tersedia.

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MK-7622 DB12897
small molecule | CAS: 1227923-29-6

MK-7622 has been used in trials studying the treatment of Alzheimer's Disease.

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MK-8189 DB19153
small molecule | CAS: 1424371-93-6

MK-8189 is under investigation in clinical trial NCT04624243 (Efficacy and Safety of MK-8189 in Participants With an Acute Episode of Schizophrenia (MK-8189-008)).

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MK-8245 DB13024
small molecule | CAS: 1030612-90-8

MK-8245 has been used in trials studying the treatment of Type 2 Diabetes Mellitus.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
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MK-8666 DB14937
small molecule | CAS: 1544739-75-4

MK-8666 is under investigation in clinical trial NCT01971554 (Safety, Tolerability, Pharmacodynamics, and Pharmacokinetics of MK-8666 in Participants With Type 2 Diabetes Mellitus (MK-8666-003)).

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MK-8719 DB16989
small molecule | CAS: 1382799-40-7

Deskripsi belum tersedia.

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MK-8776 DB11899
small molecule | CAS: 891494-63-6

Sch 900776 has been used in trials studying the treatment of Neoplasms, Hodgkin Disease, Adult Erythroleukemia, Lymphoma, Non-Hodgkin, and Myelogenous Leukemia, Acute, among others.

Target Protein:
Serine/threonine-protein kinase Chk1
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MK-8777 DB18904
small molecule | CAS: 1026791-61-6

MK-8777 is under investigation in clinical trial NCT00610649 (Trial to Determine the Maximum Tolerated Dose (MTD) Based on Safety and Tolerability, of Org 26576 in Participants With Major Depressive Disorder (174001/P05704/MK-8777-001)).

Kategori:
Isoxazoles
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MK-886 DB16739
small molecule | CAS: 118414-82-7

MK-886 is an experimental inhibitor of leukotriene synthesis.

Kategori:
Benzene DerivativesEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenaseArachidonate 5-lipoxygenase-activating protein
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MKC-1 DB05608
small molecule | CAS: 125313-92-0

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 2Cyclin-dependent kinase 1
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MKC1106-PP DB06030
small molecule

MKC1106-PP is a 3-component investigational vaccine made up of a DNA plasmid (pPRA-PSM) and 2 peptides E-PRA and E-PSM. The plasmid portion is a recombinant plasmid expressing segments of the 2 target antigens, PRAME and PSMA. MKC1106-PP was under investigati…

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MLN-977 DB05431
small molecule | CAS: 175212-04-1

MLN-977 is a small molecule compound that inhibits the production of leukotrienes, especially 5-lipoxygenase. It is developed by PharmaEngine to treat asthma and chronic obstructive pulmonary disease.

Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
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MLN0415 DB05183
small molecule

MLN0415 is a novel, small molecule IKK2 inhibitor, discovered by Millennium scientists. In preclinical studies, MLN0415 was shown to decrease NF-kB activation and down-regulate the expression of a number of inflammatory proteins. Because inflammatory proteins…

Target Protein:
Inhibitor of nuclear factor kappa-B kinase subunit beta
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MLN2222 DB06503
biotech

MLN2222 is a novel, proprietary recombinant protein that blocks both the C3 and C5 convertases, which are essential components of the complement activation pathway.

Target Protein:
Complement factor B
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MLN2704 DB06513
biotech

A Phase 1/2 trial (NCT00070837) evaluated the safety, dosage, and pharmacokinetics of MLN2704 in patients with metastatic androgen-independent prostate cancer.

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