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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 176 / 282
Melphalan flufenamide Approved DB16627
small molecule | CAS: 380449-51-4

Melphalan flufenamide, also known as melflufen or J1, is a prodrug of [melphalan].[A230123,L32173] Melphalan flufenamide is more readily uptaken by cells than melphalan, and is cleaved to the active metabolite by aminopeptidases.[A230123] _In vitro_ models sh…

Kategori:
Alkylating ActivityAlkylating DrugsAmino Acids +12
Target Protein:
DNA
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Melrilimab DB16373
biotech | CAS: 2222865-46-3

Melrilimab is under investigation in clinical trial NCT03207243 (Efficacy and Safety Study of GSK3772847 in Subjects With Moderately Severe Asthma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEM 1003 DB05547
small molecule

MEM 10003 was under investigation in clinical trial NCT00257673 (Safety and Efficacy of MEM 1003 Versus Placebo in Patients With Mild to Moderate Alzheimer's Disease) for the treatment of Alzheimer's Disease.

Waktu Paruh-
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MEM136 DB17321
biotech

Deskripsi belum tersedia.

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Genetik -
Memantine Approved DB01043
small molecule | CAS: 19982-08-2

Initially approved by the FDA in 2013, memantine is an N-methyl-D-aspartate (NMDA) receptor antagonist used in the management of Alzheimer's Disease (AD). It is different from many other Alzheimer's Disease medications, as it works by a different mechanism t…

Kategori:
Anti-Dementia DrugsAnti-Dyskinesia AgentsAnti-Parkinson Drugs +20
Target Protein:
Glutamate (NMDA) receptor5-hydroxytryptamine receptor 3ANeuronal acetylcholine receptor subunit alpha-7 +3
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThis drug is cleare…
Genetik -
Menadiol diphosphate Approved DB14650
small molecule | CAS: 84-98-0

Deskripsi belum tersedia.

Kategori:
DiterpenesNaphthalenesNaphthoquinones +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menadione Approved DB00170
small molecule | CAS: 58-27-5

A synthetic naphthoquinone without the isoprenoid side chain and biological activity, but can be converted to active vitamin K2, menaquinone, after alkylation in vivo.

Kategori:
Antifibrinolytic AgentsBlood and Blood Forming OrgansCoagulants +45
Target Protein:
Aldehyde oxidaseVitamin K-dependent gamma-carboxylaseVitamin K epoxide reductase complex subunit 1 +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menaquinone DB15381
small molecule | CAS: 1182-68-9

Menaquinone is under investigation in clinical trial NCT01533441 (Vitamin K2 Intervention in Patients With Vitamin K Antagonists).

Kategori:
CoagulantsDiet, Food, and NutritionDiterpenes +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menaquinone 6 DB14936
small molecule | CAS: 84-81-1

Menaquinone 6 is under investigation in clinical trial NCT01194778 (Comparison of Efficacy of Different Dosages Vitamin K2).

Kategori:
CoagulantsDiet, Food, and NutritionDiterpenes +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menaquinone 7 DB13075
small molecule | CAS: 2124-57-4

Menaquinone 7 is under investigation in clinical trial NCT00402974 (The Effect of Vitamin K Supplementation on Osteocalcin Carboxylation in Healthy Children).

Kategori:
CoagulantsDiterpenesHematologic Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menatetrenone DB12148
small molecule | CAS: 863-61-6

Menatetrenone has been used in trials studying the treatment of Diabetes, Osteoporosis, Prediabetic State, and Hepatocellular Carcinoma.

Kategori:
CoagulantsDiterpenesDrugs Affecting Bone Structure and Mineralization +12
Target Protein:
Cruzipain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menglytate DB15983
small molecule | CAS: 579-94-2

Deskripsi belum tersedia.

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biotech

Meningococcal (groups A, C, Y and W-135) oligosaccharide diphtheria CRM197 conjugate vaccine is used to prevent invasive meningococcal disease, which is caused by bacteria _Neisseria meningitidis_ entering the bloodstream and invading the blood-brain barrier …

Kategori:
Diphtheria VaccinesMeningococcal VaccinesVaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menotropins Approved DB00032
biotech | CAS: 9002-68-0

Menotropins contains follicle stimulating hormone (FSH) and luteinizing hormone (LH) purified from the urine of postmenopausal women. It is used as a fertility medication that is injected either subcutaneously or intramuscularly. It is composed of LH with 2 …

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsComplex Mixtures +14
Target Protein:
Follicle-stimulating hormone receptorLutropin-choriogonadotropic hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menthol Approved DB14123
small molecule | CAS: 1490-04-6

Deskripsi belum tersedia.

Kategori:
AlcoholsAntipruriticsCyclohexane Monoterpenes +9
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menthone DB15920
small molecule | CAS: 89-80-5

Deskripsi belum tersedia.

Kategori:
AlcoholsCyclohexane MonoterpenesCyclohexanes +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menthyl salicylate Approved DB11201
small molecule | CAS: 89-46-3

Menthyl salicylate is an ester of menthol and salicylic acid [L2808]. This product is used to treat minor aches and pains of the muscles/joints (e.g., arthritis, backache, sprains) [L2810].

Kategori:
Anti-Inflammatory AgentsAnti-Inflammatory Agents, Non-Steroidal
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepartricin DB13633
small molecule | CAS: 11121-32-7

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAlkenesAnti-Bacterial Agents +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepenzolate Approved DB04843
small molecule | CAS: 25990-43-6

Mepenzolate is a post-ganglionic parasympathetic inhibitor. It decreases gastric acid and pepsin secretion and suppresses spontaneous contractions of the colon. Mepenzolate diminishes gastric acid and pepsin secretion. Mepenzolate also suppresses spontaneous …

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +7
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meperidine Approved DB00454
small molecule | CAS: 57-42-1

A narcotic analgesic that can be used for the relief of most types of moderate to severe pain, including postoperative pain and the pain of labor. Prolonged use may lead to dependence of the morphine type; withdrawal symptoms appear more rapidly than with mor…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents that reduce seizure threshold +34
Target Protein:
Kappa-type opioid receptorGlutamate receptor ionotropic, NMDA 1Glutamate receptor ionotropic, NMDA 2B +9
Waktu ParuhInitial distributio…
Vol. DistribusiMeperidine crosses …
Klirens-
Genetik -
Mephenesin Approved DB13583
small molecule | CAS: 59-47-2

Mephenesin is a synthetic cresol glyceryl ether which produces transient muscle relaxation and paralysis via central nervous system depression [A32760]. It first entered use in the 1950s.

Kategori:
AlcoholsCentral Nervous System AgentsCentral Nervous System Depressants +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 533-06-2

Deskripsi belum tersedia.

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Mephentermine Approved DB01365
small molecule | CAS: 100-92-5

A sympathomimetic agent with mainly indirect effects on adrenergic receptors. It is used to maintain blood pressure in hypotensive states, for example, following spinal anesthesia. Although the central stimulant effects of mephentermine are much less than tho…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +17
Target Protein:
Alpha adrenergic receptorD(2) dopamine receptorBeta adrenergic receptor
Waktu Paruh17 to 18 hours.
Vol. Distribusi-
Klirens-
Genetik -
Mephenytoin Approved DB00532
small molecule | CAS: 50-12-4

Mephenytoin is used for the treatment of refractory partial epilepsy. Mephenytoin is a solid. This compound belongs to the phenylhydantoins. These are heterocyclic aromatic compounds containing an imiazolidinedione moiety substituted by a phenyl group. Mephen…

Kategori:
Anti-epileptic AgentAnticonvulsantsCentral Nervous System Agents +17
Target Protein:
Sodium channel protein type 5 subunit alphaNuclear receptor subfamily 1 group I member 2
Gen Terkait:
CYP2C19 CYP2C19 CYP2C19
Waktu ParuhApproximately 7 hou…
Vol. Distribusi* 1.4 L/kg
Klirens-
Genetik 3 Varian
Mepindolol DB13530
small molecule | CAS: 23694-81-7

Mepindolol is a 2-methyl derivative of pindolol. It is a beta blocker.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +12
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepiprazole DB09197
small molecule | CAS: 20326-12-9

Mepiprazole is a minor tranquilizer with a phenylpiperazine structure. It is a pyrazolyl-alkyl-piperazine derivative. Mepiprazole mediates a weak inhibitory action on the uptake of 5-HT on hypothalamic neurons [A7816]. Mepiprazole is marketed in Spain for th…

Waktu Paruh-
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Mepivacaine Approved DB00961
small molecule | CAS: 96-88-8

A local anesthetic that is chemically related to bupivacaine but pharmacologically related to lidocaine. It is indicated for infiltration, nerve block, and epidural anesthesia. Mepivacaine is effective topically only in large doses and therefore should not be…

Kategori:
AmidesAnestheticsAnesthetics, Local +10
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu ParuhThe half-life of me…
Vol. Distribusi-
Klirens-
Genetik -
Mepolizumab Approved DB06612
biotech | CAS: 196078-29-2

Eosinophils are involved in inflammatory immune responses, and prolonged hypereosinophilia (typically defined as absolute eosinophil levels of 1500/mm<sup>3</sup> or more) is associated with a spectrum of diseases, including severe asthma, eosinophilic granul…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Interleukin-5
Waktu ParuhMepolizumab has a m…
Vol. DistribusiMepolizumab has a p…
KlirensMepolizumab has an …
Genetik -
MePPEP C-11 DB19280
small molecule | CAS: 1022083-25-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meprednisone Approved DB09383
small molecule | CAS: 1247-42-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCorticosteroids for Systemic Use +20
Target Protein:
Glucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1106-03-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Meprotixol DB13822
small molecule | CAS: 4295-63-0

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepyramine Approved DB06691
small molecule | CAS: 91-84-9

Mepyramine, or pyrilamine, targets the H1 receptor. It is a first generation antihistamine. However, it rapidly permeates the brain and so often causes drowsiness as a side effect. It has been found in over-the-counter combination products for colds and menst…

Kategori:
AminesAminopyridinesAnti-Allergic Agents +19
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mequitazine DB01071
small molecule | CAS: 29216-28-2

Mequitazine is a histamine H1 antagonist (antihistamine). It competes with histamine for the normal H1-receptor sites on effector cells of the gastrointestinal tract, blood vessels and respiratory tract. It provides effective, temporary relief of sneezing, wa…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseBronchodilator Agents +15
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meradimate Approved DB11096
small molecule | CAS: 134-09-8

Meradimate, before known as menthyl anthranilate, is used in a maximal concentration of 5% in different products as a UV filter.[T200] It is currently required to be named as meradimate in all FDA approved OTC products. Meradimate is approved by the FDA and H…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +2
Waktu ParuhAs meradimate is no…
Vol. DistribusiAs meradimate is no…
KlirensAs meradimate is no…
Genetik -
Merbromin DB13392
small molecule | CAS: 129-16-8

Mercurochrome is a trade name of merbromin commonly used as a topical first-aid antiseptic agent. It is an organomercuric disodium salt compound and a fluorescein that is available in many countries, except Switzerland, France, Germany, and the United States …

Kategori:
Antiseptics and DisinfectantsDermatologicalsFluoresceins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamase IMP-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mercaptoethanol DB03345
small molecule | CAS: 60-24-2

Deskripsi belum tersedia.

Kategori:
AlcoholsSulfhydryl CompoundsSulfur Compounds
Target Protein:
Lactoylglutathione lyaseFibroblast growth factor 2M-phase inducer phosphatase 2 +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mercaptopurine Approved DB01033
small molecule | CAS: 50-44-2

An antimetabolite antineoplastic agent with immunosuppressant properties. It interferes with nucleic acid synthesis by inhibiting purine metabolism and is used, usually in combination with other drugs, in the treatment of or in remission maintenance programs …

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +20
Target Protein:
Hypoxanthine-guanine phosphoribosyltransferaseInosine-5'-monophosphate dehydrogenase 1Amidophosphoribosyltransferase +1
Gen Terkait:
TPMT TPMT TPMT
Waktu ParuhTriphasic: 45 minut…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik 3 Varian
small molecule | CAS: 10124-48-8

Deskripsi belum tersedia.

Kategori:
Antiseptics and DisinfectantsChloridesChlorine Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7487-94-7

Mercury chloride (HgCl2) is a highly toxic compound that volatizes slightly at ordinary temperature and appreciably at 100 degrees C. It is corrosive to mucous membranes and used as a topical antiseptic and disinfectant. Mercuric chloride was used to disinfec…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntiseptics and Disinfectants +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mercuric iodide DB04445
small molecule | CAS: 7774-29-0

Deskripsi belum tersedia.

Kategori:
AnionsAntiseptics and DisinfectantsDermatologicals +4
Target Protein:
Sulfotransferase 2A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

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Merestinib DB12381
small molecule | CAS: 1206799-15-6

Merestinib has been used in trials studying the treatment of Cancer, Solid Tumor, Advanced cancer, ColoRectal Cancer, and Metastatic Cancer, among others.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-RingNicotinic Acids +3
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mericitabine DB12045
small molecule | CAS: 940908-79-2

Mericitabine has been investigated for the treatment of Hepatitis C, Chronic. Mericitabine is a polymerase inhibitor being developed for the treatment of chronic hepatitis C. Mericitabine is a prodrug of PSI-6130, which demonstrated excellent potency in p…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Merimepodib DB04862
small molecule | CAS: 198821-22-6

Merimepodib (VX-497) is a novel noncompetitive inhibitor of IMPDH. Merimepodib is orally bioavailable and inhibits the proliferation of primary human, mouse, rat, and dog lymphocytes at concentrations of approximately 100 nM.

Kategori:
Acids, AcyclicAmidesBenzene Derivatives +1
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meropenem Approved DB00760
small molecule | CAS: 96036-03-2

Meropenem is a broad-spectrum carbapenem antibiotic. It is active against Gram-positive and Gram-negative bacteria. Meropenem exerts its action by penetrating bacterial cells readily and interfering with the synthesis of vital cell wall components, which lead…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacB
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Merotocin DB12932
biotech | CAS: 1190083-57-8

Merotocin has been used in trials studying the treatment of Preterm Delivery.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mesalazine Approved DB00244
small molecule | CAS: 89-57-6

An anti-inflammatory agent, structurally related to the salicylates and non-steroidal anti-inflammatory drugs like acetylsalicylic acid, which is active in inflammatory bowel disease [A174022]. Although demonstrably effective in treating and maintaining remis…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAminosalicylate +13
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Polyunsaturated fatty acid 5-lipoxygenase +4
Waktu ParuhFor the delayed-rel…
Vol. DistribusiFor the extended-re…
KlirensThe mean (SD) renal…
Genetik -
Mescaline DB19083
small molecule | CAS: 54-04-6

Mescaline is under investigation in clinical trial NCT05933213 (Comparing Mescaline Sodium Enteric-coated Tablets vs Morte-mescaline in the Treatment of Adult Lupus Nephritis).

Kategori:
AlkaloidsAminesAntidepressive Agents +9
Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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