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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 175 / 236
Pentafluoropropane Approved DB13117
small molecule | CAS: 460-73-1

Pentafluoropropane is under investigation in clinical trial NCT01673061 (Vapocoolant Spray for Numbing Small Boils Before Incision and Drainage).

Kategori:
Hydrocarbons, FluorinatedHydrocarbons, Halogenated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentaglobin DB15865
biotech | CAS: 97794-27-9

Pentaglobin, also known as IgM-enriched immunoglobulin, falls under a group of polyclonal immunoglobulin preparations.[A220173] It is comprised of [immunoglobulin G (IgG)](https://www.drugbank.ca/drugs/DB00028) and immunoglobulin A (IgA) while also being enri…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pentaglyme DB02580
small molecule | CAS: 1191-87-3

Deskripsi belum tersedia.

Target Protein:
Profilin-2Restriction endonuclease R.BpuJICytochrome c-552 +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentamidine Approved DB00738
small molecule | CAS: 100-33-4

Antiprotozoal agent effective in trypanosomiasis, leishmaniasis, and some fungal infections; used in treatment of pneumocystis pneumonia in HIV-infected patients. It may cause diabetes mellitus, central nervous system damage, and other toxic effects.

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAgents causing hyperkalemiaAmidines +20
Target Protein:
Tryptase alpha/beta-1tRNA (cytosine(38)-C(5))-methyltransferaseDNA
Waktu Paruh9.1-13.2 hours
Vol. Distribusi-
Klirens-
Genetik -
Pentamycin DB13571
small molecule | CAS: 6834-98-6

Deskripsi belum tersedia.

Kategori:
AlkenesAntifungal AgentsGenito Urinary System and Sex Hormones +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentapiperium DB19383
small molecule | CAS: 26372-86-1

Deskripsi belum tersedia.

Waktu Paruh-
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Pentastarch Approved DB09111
small molecule | CAS: 9005-27-0

Pentastarch is an artificial colloid (hydroxyethyl starch derivative). Pentastarch is characterized by presenting five hydroxyethyl groups, which signifies an approximate 50% hydroxyethylation. It is sold under the name Pentaspan by Bristol-Myers Squibb and i…

Kategori:
Blood SubstitutesCarbohydratesCompounds used in a research, industrial, or household setting +9
Waktu Paruh~2.5 hours.
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22537-51-5

Pentavalent Antimony has been investigated for the treatment of Cutaneous Leishmaniasis.

Waktu Paruh-
Vol. Distribusi-
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Pentazocine Approved DB00652
small molecule | CAS: 359-83-1

The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97)

Kategori:
Adjuvants, AnesthesiaAgents that reduce seizure thresholdAlkaloids +20
Target Protein:
Sigma non-opioid intracellular receptor 1Mu-type opioid receptorKappa-type opioid receptor
Waktu Paruh2 to 3 hours
Vol. Distribusi-
Klirens-
Genetik -
Pentetic acid Approved DB14007
small molecule | CAS: 67-43-6

Pentetic acid, also known as diethylenetriaminepentaacetic acid (DTPA), is a synthetic polyamino carboxylic acid with eight coordinate bond forming sites that can sequester metal ions and form highly stable DTPA-metal ion complexes. DTPA, along with its calci…

Kategori:
AcetatesAcids, AcyclicAmines +10
Target Protein:
Transuranium elements
Waktu ParuhIn preclinical stud…
Vol. DistribusiThe volume of distr…
KlirensPentetic acid prese…
Genetik -
Pentetrazol DB13415
small molecule | CAS: 54-95-5

Pentetrazol, also known as pentylenetetrazole, is a gamma-aminobutyric acid type A (GABA<sub>A</sub>) receptor antagonist that was approved by the FDA until 1982.[A254437]

Kategori:
AzepinesCentral Nervous System AgentsCentral Nervous System Stimulants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penthienate DB13695
small molecule | CAS: 22064-27-3

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAmines +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentifylline DB13634
small molecule | CAS: 1028-33-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsCytochrome P-450 CYP1A2 SubstratesCytochrome P-450 Substrates +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentobarbital Approved DB00312
small molecule | CAS: 76-74-4

A short-acting barbiturate that is effective as a sedative and hypnotic (but not as an anti-anxiety) agent and is usually given orally. It is prescribed more frequently for sleep induction than for sedation but, like similar agents, may lose its effectiveness…

Kategori:
Adjuvants, AnesthesiaAnticholinergic AgentsAnticonvulsants +23
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +10
Waktu Paruh5 to 50 hours (dose…
Vol. Distribusi-
Klirens-
Genetik -
Pentosan polysulfate Approved DB00686
small molecule | CAS: 37300-21-3

Pentosan polysulfate is a sulfated pentosyl polysaccharide with heparin-like properties.

Kategori:
AnticoagulantsAntivaricose TherapyCarbohydrates +12
Target Protein:
Fibroblast growth factor 2Fibroblast growth factor 1Fibroblast growth factor 4
Waktu Paruh4.8 hours
Vol. Distribusi-
Klirens-
Genetik -
Pentoxifylline Approved DB00806
small molecule | CAS: 6493-05-6

Pentoxifylline (PTX) is a synthetic dimethylxanthine derivative that modulates the rheological properties of blood and also has both anti-oxidant and anti-inflammatory properties.[A226415, L30300] Although originally developed to treat intermittent claudicati…

Kategori:
AlkaloidsAntioxidantsAntiplatelet agents +23
Target Protein:
Adenosine receptor A2aTumor necrosis factorPhosphodiesterase enzymes +2
Waktu ParuhOverall, pentoxifyl…
Vol. DistribusiPentoxifylline has …
KlirensPentoxifylline give…
Genetik -
Pentoxyverine Approved DB11186
small molecule | CAS: 77-23-6

Pentoxyverine, also referred to as carbetapentane, is a non-opioid central acting antitussive with antimuscarinic, anticonvulsant [A32717], and local anesthetic properties. It is an active ingredient in over-the-counter cough suppressants in combination with …

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +2
Target Protein:
Sigma non-opioid intracellular receptor 1Voltage-gated inwardly rectifying potassium channel KCNH2Voltage-gated sodium channel alpha subunit +2
Waktu ParuhThe half-life is 2.…
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peoniflorin DB16288
small molecule | CAS: 23180-57-6

Peoniflorin is under investigation in clinical trial NCT02878863 (Paeoniflorin Combination of Hepatoprotective Drugs Versus Hepatoprotective Drugs Only for Auto-immune Hepatitis).

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +8
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PEP0101 DB18572
biotech

PEP0101 is a nanocomplex consisting of elastin-like polypeptides and a small interfering RNA (siRNA) designed to down-regulate the expression of EVI1 oncogene in cancer cells.

Waktu Paruh-
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Pepinemab DB15155
biotech | CAS: 2097151-87-4

Pepinemab is under investigation in clinical trial NCT03769155 (VX15/2503 With or Without Ipilimumab and/or Nivolumab in Patients With Resectable Stage IIIB-D Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peppermint oil Approved DB11198
biotech | CAS: 8006-90-4

Extracted from the stem, leaves, and flowers of _Mentha piperita_ L. plant, peppermint oil (Mentha piperita) is a popular essential oil used in aromatherapy for both external and internal use. Mentha piperita is a hybrid of spearmint (Mentha spicata) and wate…

Kategori:
Alimentary Tract and MetabolismAngiospermsAntiemetics +31
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Pepsin Approved DB13198
biotech | CAS: 9001-75-6

Pepsin is a potent enzyme in gastric juice that digests proteins such as those in meat, eggs, seeds, and dairy products [L2358]. Studies on gastric digestion from 1820-1840 led to the discovery of pepsin as the substance which, in the presence of stomach a…

Kategori:
Alimentary Tract and MetabolismAspartic Acid EndopeptidasesAspartic Acid Proteases +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 118997-30-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal HormonesHormones +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 123583-37-9

Peptide YY (3-36), a synthetic human PYY 3-36, is a compound being evaluated for the treatment of obesity. It reduces appetite and increases satiety in obese patients.

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal HormonesHormones +3
Target Protein:
Neuropeptide Y receptor type 2Neuropeptide Y receptor type 1Neuropeptide Y receptor type 5 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peptide-T DB19279
small molecule | CAS: 106362-32-7

Peptide-T is under investigation in clinical trial NCT00000392 (Phase II Study of the Efficacy of Peptide T in Hiv-positive Individuals With Cognitive Impairment.).

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peracetic acid DB14556
small molecule | CAS: 79-21-0

A liquid that functions as a strong oxidizing agent. It has an acrid odor and is used as a disinfectant.

Kategori:
AcetatesAcids, AcyclicAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peramivir Approved DB06614
small molecule | CAS: 330600-85-6

Peramivir is an antiviral agent developed by Biocryst Pharmaceuticals to treat influenza A/B. The development of peramivir has been supported by the US Department of Health and Human Services as part of the government's effort to prepare for a flu pandemic. B…

Kategori:
AmidinesAnti-Infective AgentsAntiinfectives for Systemic Use +6
Target Protein:
NeuraminidaseNeuraminidaseNeuraminidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perampanel Approved DB08883
small molecule | CAS: 380917-97-5

Perampanel is a noncompetitive AMPA glutamate receptor antagonist. It is marketed under the name Fycompa™ and is indicated as an adjunct in patients over 12 years old for the treatment of partial-onset seizures that may or may not occur with generalized seizu…

Kategori:
AMPA Receptor AntagonistsAnticonvulsantsCentral Nervous System Depressants +23
Target Protein:
Glutamate receptor 2Glutamate receptor 3Glutamate receptor 4 +1
Waktu ParuhPerampanel has a lo…
Vol. DistribusiThe volume of distr…
KlirensIn healthy patients…
Genetik -
Perazine Approved DB12710
small molecule | CAS: 84-97-9

Perazine has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders, among others.

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +12
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perboric acid Approved DB13235
small molecule | CAS: 14034-78-7

Perboric acid is mainly found in its salt form of sodium perborate and it can be found as a monohydrate or tetrahydrate.[A33037] It is one of the peroxy acid salts with very wide functionalities in industrial settings.[F66] Perboric acid in the form of sodium…

Kategori:
AcidsAlimentary Tract and MetabolismAnions +7
Waktu ParuhAs perboric acid an…
Vol. DistribusiAs perboric acid an…
KlirensAs perboric acid an…
Genetik -
Perchlorate DB03138
small molecule | CAS: 14797-73-0

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicChlorine Compounds
Target Protein:
Protein ArsC
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perenostobart DB18602
biotech | CAS: 2643331-31-9

Perenostobart is an alpha-CD39 IgG4 monoclonal antibody.

Waktu Paruh-
Vol. Distribusi-
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Peresolimab DB18874
biotech | CAS: 2411580-63-5

Peresolimab is under investigation in clinical trial NCT04634253 (A Study of LY3462817 in Participants With Rheumatoid Arthritis).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Perflenapent DB11625
small molecule | CAS: 678-26-2

Dodecafluoropentane is also known as perfluoropentane or perflenapent.

Kategori:
AlkanesCompounds used in a research, industrial, or household settingContrast Media +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perflubron DB05791
small molecule | CAS: 423-55-2

Perflubron (Oxygent) is being developed as an intravascular oxygen carrier designed to augment oxygen delivery in surgical patients.

Kategori:
Anti-Obesity AgentsCompounds used in a research, industrial, or household settingContrast Media +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 84808-64-0

Oxycyte has been used in trials studying the treatment of Traumatic Brain Injury.

Kategori:
Hydrocarbons, FluorinatedHydrocarbons, Halogenated
Waktu Paruh-
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Perfluorohexyloctane Approved DB17823
small molecule | CAS: 133331-77-8

Perfluorohexyloctane is a semifluorinated alkane that contains six perfluorinated carbon atoms and eight hydrogenated carbon atoms.[L46491] It is an inert, slightly amphiphilic compound.[A259746] Because it is a completely non-aqueous liquid, microbial growth…

Kategori:
Hydrocarbons, FluorinatedHydrocarbons, HalogenatedOphthalmic Solutions +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perfluorooctane DB15997
small molecule | CAS: 307-34-6

Deskripsi belum tersedia.

Kategori:
Hydrocarbons, FluorinatedHydrocarbons, Halogenated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perflutren Approved DB00556
small molecule | CAS: 76-19-7

Perflutren, a diagnostic drug that is intended to be used for contrast enhancement during the indicated echocardiographic procedures, is comprised of lipid-coated microspheres filled with octafluoropropane(OFP) gas. When exposed to ultrasound waves, the micro…

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingContrast Media +10
Waktu ParuhThe mean half-life …
Vol. Distribusi-
Klirens-
Genetik -
Perfosfamide DB12727
small molecule | CAS: 62435-42-1

Perfosfamide has been used in trials studying the treatment of Lymphoma, Neuroblastoma, and Multiple Myeloma and Plasma Cell Neoplasm.

Kategori:
Hydrocarbons, HalogenatedMustard CompoundsNitrogen Mustard Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pergolide Approved DB01186
small molecule | CAS: 66104-22-1

Pergolide is a long-acting dopamine agonist approved in 1982 for the treatment of Parkinson’s Disease. It is an ergot derivative that acts on the dopamine D2 and D3, alpha2- and alpha1-adrenergic, and 5-hydroxytryptamine (5-HT) receptors. It was indicated as …

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-2 Receptor Agonists +24
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor +12
Waktu Paruh27 hours
Vol. Distribusi-
Klirens-
Genetik -
Perhexiline Approved DB01074
small molecule | CAS: 6621-47-2

Perhexiline is a coronary vasodilator used especially for angina of effort. It may cause neuropathy and hepatitis.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +18
Target Protein:
Carnitine O-palmitoyltransferase 1, liver isoformCarnitine O-palmitoyltransferase 1, muscle isoformCarnitine O-palmitoyltransferase 2, mitochondrial +1
Waktu ParuhVariable and non-li…
Vol. Distribusi-
Klirens-
Genetik -
Perifosine DB06641
small molecule | CAS: 157716-52-4

Perifosine is a novel alkylphospholipid with antiproliferative properties attributed to protein kinase B inhibition.

Kategori:
AminesOnium CompoundsQuaternary Ammonium Compounds +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformRAC-alpha serine/threonine-protein kinaseMitogen-activated protein kinase 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 18457-55-1

Perillyl alcohol is under investigation in clinical trial NCT02704858 (Safety and Efficacy Study in Recurrent Grade IV Glioma).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsPerilla +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perindopril Approved DB00790
small molecule | CAS: 82834-16-0

Perindopril is a nonsulfhydryl prodrug that belongs to the angiotensin-converting enzyme (ACE) inhibitor class of medications. It is rapidly metabolized in the liver to perindoprilat, its active metabolite, following oral administration. Perindoprilat is a po…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +18
Target Protein:
Angiotensin-converting enzymeSecreted frizzled-related protein 4
Waktu ParuhPerindopril, 1.2 ho…
Vol. Distribusi-
Klirens* 219 - 362 mL/min …
Genetik -
Periplaneta americana Approved DB10417
biotech

American cockroach allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perospirone DB08922
small molecule | CAS: 150915-41-6

Perospirone is an atypical or second-generation antipsychotic of the azapirone family that antagonizes serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist. Dainippon Sumitomo Pharma devel…

Kategori:
Antipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical])Central Nervous System Agents +13
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +3
Gen Terkait:
HTR1A
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean volume of …
KlirensApparent clearance …
Genetik 1 Varian
small molecule | CAS: 17528-28-8

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pertussis vaccine Approved DB15274
biotech

Pertussis vaccine is under investigation in clinical trial NCT01698346 (Pertussis (Tdap) Vaccination in Pregnancy).

Kategori:
Bacterial VaccinesBiological ProductsComplex Mixtures +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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