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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 175 / 282
Mebrofenin Approved DB15779
small molecule | CAS: 78266-06-5

Deskripsi belum tersedia.

Kategori:
AminesAmino AcidsAmino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebutamate Approved DB06797
small molecule | CAS: 64-55-1

Mebutamate is a sedative and anxiolytic drug with anti-hypertensive (blood pressure lowering) effects comparable to those of other barbiturates but is only around 1/3rd the potency of secobarbital as a sedative. Side effects include dizziness and headaches.

Kategori:
Anti-Anxiety AgentsCarbamatesCentral Nervous System Depressants +2
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mecamylamine Approved DB00657
small molecule | CAS: 60-40-2

A nicotinic antagonist that is well absorbed from the gastrointestinal tract and crosses the blood-brain barrier. Mecamylamine has been used as a ganglionic blocker in treating hypertension, but, like most ganglionic blockers, is more often used now as a rese…

Kategori:
Agents that produce neuromuscular block (indirect)Antiadrenergic Agents, Ganglion-BlockingAnticholinergic Agents +15
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Neuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit alpha-4 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1570067-55-8

Mecapegfilgrastim is under investigation in clinical trial NCT05463601 (Mecapegfilgrastim for the Prevention of Dalpiciclib -Induced Neutropenia in Advanced Breast Cancer).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mecasermin Approved DB01277
biotech | CAS: 68562-41-4

Mecasermin contains recombinant-DNA-engineered human insulin-like growth factor-1 (rhIGF-1)[FDA Label]. IGF-1 consists of 70 amino acids in a single chain with three intramolecular disulfide bridges and a molecular weight of 7649 daltons. The amino acid seque…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesBiological Factors +15
Target Protein:
Insulin-like growth factor 1 receptorInsulin-like growth factor-binding protein 3Insulin receptor +1
Waktu ParuhMean half life of 5…
Vol. Distribusi* 0.257 ± 0.073 L/k…
KlirensClearance of Mecase…
Genetik -
Mecasermin rinfabate Approved DB14751
biotech | CAS: 478166-15-3

Mecasermin rinfabate is approved for severe primary insulin-like growth factor (IGF) deficiency or in patients with GH gene deletion who have developed antibodies to growth hormone (GH)[A176020]. Mecasermin rinfabate is similar to [DB01277] in that both drugs…

Kategori:
Anterior Pituitary Lobe Hormones and AnaloguesPituitary and Hypothalamic Hormones and AnaloguesSomatropin and Somatropin Agonists +1
Target Protein:
Insulin-like growth factor 1 receptorInsulin receptorCation-independent mannose-6-phosphate receptor
Waktu ParuhHalf life ranges fr…
Vol. DistribusiApproximately 1000m…
KlirensClearance ranges fr…
Genetik -
biotech | CAS: 2460400-64-8

Mecbotamab vedotin is an anti-Axl humanized monoclonal antibody conjugated to monomethyl auristatin E using a cleavable linker (CAB-Axl-ADC).[A255212]

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Mechlorethamine Approved DB00888
small molecule | CAS: 51-75-2

A vesicant and necrotizing irritant destructive to mucous membranes, mechlorethamine is an alkylating drug. It was formerly used as a war gas. The hydrochloride is used as an antineoplastic in Hodgkin's disease and lymphomas. It causes severe gastrointestinal…

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +16
Target Protein:
DNA
Waktu Paruh15 minutes
Vol. Distribusi-
Klirens-
Genetik -
Meclinertant DB06455
small molecule | CAS: 146362-70-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Neurotensin, antagonists & inhibitors
Target Protein:
Neurotensin receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meclocycline DB13092
small molecule | CAS: 2013-58-3

Meclocycline is under investigation in clinical trial NCT00385515 (Efficacy of SNX-1012 in the Treatment of Oral Mucositis) [L797].

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Topical UseAnti-Bacterial Agents +5
Target Protein:
30S ribosomal protein S7
Waktu ParuhHalf life estimated…
Vol. DistribusiEstimated Vd of 121…
Klirens-
Genetik -
Meclofenamic acid Approved DB00939
small molecule | CAS: 644-62-2

A non-steroidal anti-inflammatory agent with antipyretic and antigranulation activities. It also inhibits prostaglandin biosynthesis.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +25
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Polyunsaturated fatty acid 5-lipoxygenase +2
Waktu ParuhIn a study in 10 he…
Vol. Distribusi* 9.1 to 43.2 L
Klirens* Oral cl=206 mL/min
Genetik -
Mecobalamin Approved DB03614
small molecule | CAS: 13422-55-4

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCorrinoids +4
Target Protein:
Methionine synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medazepam DB13437
small molecule | CAS: 2898-12-6

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsAnticonvulsantsBenzazepines +17
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medetomidine DB11428
small molecule | CAS: 86347-14-0

Medetomidine is a synthetic compound used as a surgical anesthetic and analgesic. It is normally found as its hydrochloride salt, medetomidine hydrochloride. Medetomidine is an intravenously available alpha-2 adrenergic agonist. The drug has been developed by…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +12
Target Protein:
Alpha-2A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI-491 DB17859
biotech

MEDI-491 is a recombinant human parvovirus B19 vaccine composed of the VP1 and VP2 capsid proteins.

Waktu Paruh-
Vol. Distribusi-
Klirens-
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MEDI-6469 DB15306
biotech | CAS: 1715924-11-0

MEDI-6469 is a monoclonal antibody under investigation in clinical trial NCT02205333 (A Phase 1b/2 Safety and Tolerability of MEDI6469 in Combination With Therapeutic Immune Agents or Monoclonal Antibodies).

Waktu Paruh-
Vol. Distribusi-
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MEDI3506 DB16473
biotech | CAS: 2376858-66-9

Tozorakimab (MEDI3506), developed by AstraZeneca, was investigated in multiple clinical trials to evaluate its safety, tolerability, efficacy, and pharmacokinetics across various conditions. These trials include NCT03096795 (completed; healthy participants, C…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Interleukin-33
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI6012 DB14833
biotech

Recombinant human lecithin:cholesterol acyltransferase is under investigation in clinical trial NCT03578809 (A Study to Evaluate the Safety and Efficacy of MEDI6012 in Acute ST Elevation Myocardial Infarction).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 84082-36-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Medical air Approved DB09337
small molecule | CAS: 132259-10-0

Medical air is supplied by a special air compressor to patient care areas using clean outside air.

Kategori:
Medical GasesOther Miscellaneous Therapeutic Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The use of the plant species _Cannabis sativa_ and _Cannabis indica_, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical conditions as a wave of legalization in North America has changed public …

Kategori:
Agents producing tachycardiaBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Inducers +51
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +38
Waktu ParuhThe half life of TH…
Vol. DistribusiAs a very lipophili…
KlirensOne study reported …
Genetik -
Medifoxamine Approved DB13219
small molecule | CAS: 32359-34-5

Medifoxamine was marketed as an atypical antidepressant, with anxiolyitc properties in France, Spain, and Morrocco in the 1990s but was later withdrawn from the market due to it causing cases of hepatotoxicity [L5461, A174976].

Kategori:
AminesAntidepressive AgentsCentral Nervous System Depressants +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medium-chain triglycerides Approved DB13959
small molecule | CAS: 438544-49-1

Medium-chain triglycerides (MCTs) are triglycerides made up of a glycerol backbone and three fatty acids with an aliphatic tail of six to 12 carbon atoms. MCTs are found in natural foods, such as coconut oil, palm kernel oil, and raw coconut meat. In the body…

Kategori:
LipidsOilsParenteral Nutrition Solutions +1
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of me…
Genetik -
Medrogestone Approved DB09124
small molecule | CAS: 977-79-7

Medrogestone (INN), also known as 6,17?-dimethyl-6-dehydroprogesterone, is a progestational agent derived from 17-methylprogesterone. It was conceived as an alternative for an orally effective contraceptive option.[A31526] It was developed by Ayerst, approved…

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +10
Target Protein:
Progesterone receptor
Waktu ParuhThe half-life of me…
Vol. Distribusi-
Klirens-
Genetik -
Medronic acid Approved DB14078
small molecule | CAS: 1984-15-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medroxyprogesterone acetate Approved DB00603
small molecule | CAS: 71-58-9

Medroxyprogesterone acetate (MPA) is a [progesterone] derivative that is more resistant to metabolism for improved pharmacokinetic properties.[A14848] MPA can be use to treat secondary amenorrhea, endometrial hyperplasia, abnormal uterine bleeding, osteoporos…

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +46
Target Protein:
Progesterone receptorEstrogen receptorATP-dependent translocase ABCB1 +1
Waktu ParuhOral medroxyprogest…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Medrysone Approved DB00253
small molecule | CAS: 2668-66-8

Medrysone is a corticosteroid used in ophthalmology.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +24
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mefenamic acid Approved DB00784
small molecule | CAS: 61-68-7

A non-steroidal anti-inflammatory agent with analgesic, anti-inflammatory, and antipyretic properties. It is an inhibitor of cyclooxygenase.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +37
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh2 hours
Vol. Distribusi* 1.06 L/kg [Normal…
Klirens* Oral cl=21.23 L/h…
Genetik -
Mefenorex DB13852
small molecule | CAS: 17243-57-1

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAlimentary Tract and Metabolism +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mefloquine Approved DB00358
small molecule | CAS: 53230-10-7

Malaria is a protozoan disease that places an enormous burden on human health in endemic areas around the world. The 2020 World Health Organization malaria report indicates a 60% decrease in the global malaria fatality rate between 2000 to 2019.[L30618] Despi…

Kategori:
Agents Causing Muscle ToxicityAgents that reduce seizure thresholdAminoquinolines +20
Target Protein:
Fe(II)-protoporphyrin IX80S ribosomal subunitAdenosine receptor A2a
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThe systemic cleara…
Genetik -
Mefruside DB13405
small molecule | CAS: 7195-27-9

Deskripsi belum tersedia.

Kategori:
AmidesDiureticsLow-Ceiling Diuretics, Excl. Thiazides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mefuparib DB18248
small molecule | CAS: 1392502-82-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Megestrol Approved DB19378
small molecule | CAS: 3562-63-8

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +19
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Megestrol acetate Approved DB00351
small molecule | CAS: 595-33-5

17-Hydroxy-6-methylpregna-3,6-diene-3,20-dione. A progestational hormone used most commonly as the acetate ester. As the acetate, it is more potent than progesterone both as a progestagen and as an ovulation inhibitor. It has also been used in the palliative …

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +31
Target Protein:
Progesterone receptorGlucocorticoid receptor
Waktu Paruh34 hours
Vol. Distribusi-
Klirens-
Genetik -
Meglumine Approved DB09415
small molecule | CAS: 6284-40-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlcoholsAmino Sugars +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 133-51-7

Deskripsi belum tersedia.

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAlcoholsAmino Sugars +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meladrazine DB13272
small molecule | CAS: 13957-36-3

Deskripsi belum tersedia.

Kategori:
Drugs for Urinary Frequency and IncontinenceGenito Urinary System and Sex HormonesUrologicals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melagatran DB13616
small molecule | CAS: 159776-70-2

Deskripsi belum tersedia.

Kategori:
AminesAnticoagulantsAntithrombins +8
Target Protein:
ProthrombinPlasminogenSerine protease 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Melaleuca alternifolia leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Melanoma antigen recognized by T-cells 1 is under investigation in clinical trial NCT01748747 (Vaccine Therapy and Resiquimod in Treating Patients With Stage II-IV Melanoma That Has Been Removed By Surgery).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melarsomine DB11528
small molecule | CAS: 128470-15-5

Melarsomine is a trypanocidal agent marketed by Merial under the trade name Immiticide. It is the only FDA-approved treatment for adult heartworm infection in dogs, however, is is not approved for use in dogs with late-stage infection.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melarsoprol DB12864
small molecule | CAS: 494-79-1

Melarsoprol is under investigation in clinical trial NCT00330148 (Randomized Clinical Trial of Three Drug Combinations for Late-Stage Gambiense Human African Trypanosomiasis).

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melatonin Approved DB01065
small molecule | CAS: 73-31-4

Melatonin is a biogenic amine that is found in animals, plants and microbes. Aaron B. Lerner of Yale University is credited for naming the hormone and for defining its chemical structure in 1958. In mammals, melatonin is produced by the pineal gland. The pin…

Kategori:
AminesAntioxidantsBiogenic Amines +21
Target Protein:
Melatonin receptor type 1AMelatonin receptor type 1BRibosyldihydronicotinamide dehydrogenase [quinone] +7
Waktu Paruh35 to 50 minutes
Vol. Distribusi-
Klirens-
Genetik -
Meldonium DB13723
small molecule | CAS: 76144-81-5

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicCardiac TherapyCardiovascular Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melengestrol DB11529
small molecule | CAS: 5633-18-1

Melengestrol is a steroidal progestin and antineoplastic agent which was never marketed. An acylated derivative, melengestrol acetate, is used as a growth promoter in animals.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCorticosteroids for Systemic Use +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2919-66-6

A 6-methyl progesterone acetate with reported glucocorticoid activity and effect on estrus.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCytochrome P-450 CYP3A Inducers +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melitracen DB13384
small molecule | CAS: 5118-29-6

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meloxicam Approved DB00814
small molecule | CAS: 71125-38-7

Meloxicam is a nonsteroidal anti-inflammatory drug (NSAID) used to relieve various types of pain, including pain caused by musculoskeletal conditions, osteoarthritis, and rheumatoid arthritis.[A190189] With a longer half-life than most other NSAIDS, it is a f…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +28
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe half-life of me…
Vol. DistribusiThe volume of distr…
KlirensAfter an oral dose,…
Genetik -
Melperone DB09224
small molecule | CAS: 3575-80-2

Melperone is an atypical antipsychotic of the butyrophenone chemical class, making it structurally related to the typical antipsychotic haloperidol. Melperone has been used for a span of greater than 30 years in the European Union [L1316]. It has been well e…

Kategori:
Antiarrhythmic agentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +17
Target Protein:
D(2) dopamine receptor
Waktu ParuhApproximately 3-4 h…
Vol. Distribusi-
Klirens-
Genetik -
Melphalan Approved DB01042
small molecule | CAS: 148-82-3

Melphalan is a nitrogen mustard or bischloroethylamine type alkylating agent.[L40928] It was first synthesized in the early 1950s by substituting L-phenylalanine for the methyl group on nitrogen mustard.[A261150, A261155] Melphalan is used in the treatment of…

Kategori:
Alkylating ActivityAlkylating DrugsAmino Acids +17
Target Protein:
DNA
Waktu ParuhIn patients given a…
Vol. DistribusiThe volume of distr…
KlirensAverage total body …
Genetik -
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