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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 173 / 236
biotech | CAS: 2376210-48-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Patiromer Approved DB09263
small molecule | CAS: 1260643-52-4

Patiromer is a powder for suspension in water for oral administration, approved in the U.S. as Veltassa in October, 2015. Patiromer is supplied as patiromer sorbitex calcium which consists of the active moiety, patiromer, a non-absorbed potassium-binding poly…

Kategori:
Cation Exchange ResinsCompounds used in a research, industrial, or household settingMacromolecular Substances +3
Target Protein:
Potassium
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Patisiran Approved DB14582
biotech | CAS: 1420706-45-1

Patisiran is a first in class short interfering RNA for the treatment of patients with polyneuropathy caused by hereditary transthyretin-mediated amyloidosis [L4220]. It is marketed as Onpattro which is formulated as patisiran within a liposome envelope for b…

Kategori:
Antisense Elements (Genetics)Compounds used in a research, industrial, or household settingDecreased RNA Integrity +12
Target Protein:
Transthyretin mRNA
Waktu ParuhPatisiran has a ter…
Vol. DistribusiThe steady state vo…
KlirensThe total body clea…
Genetik -
Patritumab DB12090
biotech | CAS: 1262787-83-6

Patritumab has been used in trials studying the treatment of LUNG CANCER, Solid Tumors, Neoplasms by Site, Head and Neck Neoplasms, and Non-small Cell Lung Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Patupilone DB03010
small molecule | CAS: 152044-54-7

Epothilone B is a 16-membered macrolide that mimics the biological effects of taxol.

Kategori:
Anti-Bacterial AgentsAntimitotic AgentsAntineoplastic Agents +9
Target Protein:
Tubulin beta chainTubulin beta-1 chainTubulin beta-4B chain +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pavinetant DB11692
small molecule | CAS: 941690-55-7

Pavinetant has been used in trials studying the basic science and treatment of Safety and Schizophrenia.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingQuinolines +3
Target Protein:
Neuromedin-K receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paxalisib DB15186
small molecule | CAS: 1382979-44-3

GDC-0084 is under investigation in clinical trial NCT03696355 (Study of GDC-0084 in Pediatric Patients With Newly Diagnosed Diffuse Intrinsic Pontine Glioma or Diffuse Midline Gliomas).

Kategori:
Enzyme Inhibitors
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pazopanib Approved DB06589
small molecule | CAS: 444731-52-6

Pazopanib is a small molecule inhibitor of multiple protein tyrosine kinases with potential antineoplastic activity. It is developed by GlaxoSmithKline and was FDA approved on October 19, 2009.

Kategori:
AmidesAngiogenesis InhibitorsAntineoplastic Agents +36
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +7
Gen Terkait:
UGT1A1 HCP5
Waktu Paruh35 hours. Oral abso…
Vol. DistribusiVd steady state, IV…
KlirensCL, cancer patient,…
Genetik 2 Varian
Pazufloxacin DB11774
small molecule | CAS: 127045-41-4

Pazufloxacin is under investigation in clinical trial NCT02592096 (Pazufloxacin Mesilate Ear Drops Clinical Trial Protocol).

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA topoisomerase 4 subunit A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PB-722 DB18447
biotech

PB-722 is a long-acting glucagon receptor agonist.[L48260]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PB127 DB06208
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBCAR20A DB17189
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PBCAR269A DB17188
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
PBR-06 F-18 DB17020
small molecule | CAS: 1003581-94-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBT-1033 DB05565
small molecule | CAS: 747408-78-2

Deskripsi belum tersedia.

Target Protein:
Microtubule-associated protein tau
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PBT-434 Approved DB16965
small molecule | CAS: 1232840-87-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PCI-27483 DB13000
small molecule | CAS: 871266-63-6

PCI-27483 has been used in trials studying the treatment of Pancreatic Cancer, Ductal Adrenocarcinoma, and Exocrine Pancreatic Cancer.

Kategori:
AmidesAmidinesAmino Acids +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PCLX-001 DB15567
small molecule | CAS: 1215011-08-7

PCLX-001 is a first-in-kind N-Myristoyltransferase (NMT) inhibitor being developed by [Pacylex Pharmaceuticals](https://pacylex.com). Current studies have shown that PCLX-001 works differently than other known cancer drugs and has high activity and positive r…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PCO-371 DB14946
small molecule | CAS: 1613373-33-3

PCO-371 is under investigation in clinical trial NCT02475616 (A Single Ascending Dose Study of PCO371 in Healthy Volunteers).

Kategori:
Imidazoles
Target Protein:
Parathyroid hormone/parathyroid hormone-related peptide receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PCS-499 DB15122
small molecule | CAS: 1268605-91-9

PCS-499 is under investigation in clinical trial NCT01487109 (A Phase 2 Study to Evaluate the Safety and Efficacy of CTP-499 in Type 2 Diabetic Nephropathy Patients).

Kategori:
DeuteriumHeterocyclic Compounds, Fused-RingPurines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD-168393 DB07662
small molecule | CAS: 194423-15-9

PD-168393 is an epidermal growth factor receptor inhibitor.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD-169316 DB17040
small molecule | CAS: 152121-53-4

PD-169316 is a p38 MAP kinase inhibitor.[A253062]

Kategori:
Enzyme Inhibitors
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD-173952 DB17041
small molecule | CAS: 305820-75-1

PD-173952 is a potent Myt1 kinase inhibitor.[A253067]

Kategori:
Oxazines
Target Protein:
Platelet-derived growth factor receptor alphaProto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase Lck +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD-217014 DB12493
small molecule | CAS: 444088-20-4

PD-217,014 has been used in trials studying the treatment of Pain and Irritable Bowel Syndrome.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD-98059 DB17042
small molecule | CAS: 167869-21-8

PD-98059 is an inhibitor of MAP-kinase kinase activation.[A253072]

Kategori:
BenzopyransCalcium-Calmodulin-Dependent Protein Kinases, antagonists & inhibitorsChromones +4
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1Dual specificity mitogen-activated protein kinase kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD150606 DB02570
small molecule

Deskripsi belum tersedia.

Kategori:
Acids, Acyclic
Target Protein:
Calpain small subunit 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD173955 DB02567
small molecule

Deskripsi belum tersedia.

Kategori:
PyridinesTyrosine Kinase Inhibitors
Target Protein:
Platelet-derived growth factor receptor alphaTyrosine-protein kinase LckProto-oncogene tyrosine-protein kinase Src +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PDPSC18 DB05167
biotech

PDPSC18 is therapeutic DNA vaccine designed to fight chronic infections with the Hepatitis B virus, entering phase I clinical trials.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peanut oil Approved DB13964
biotech | CAS: 8002-03-7

Peanut oil is derived from _Arachis hypogaea_ which can be found in South America, Mexico, and Centro America. The kernels are consumed roasted but a large percentage is used for the production of vegetable oil. The peanut oil represents about 45-52% of the k…

Kategori:
Basic Ointments and ProtectantsBiological ProductsDetergents +8
Waktu ParuhThe exact pharmacok…
Vol. DistribusiThe exact pharmacok…
KlirensThe exact pharmacok…
Genetik -
biotech | CAS: 2408734-39-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pecavaptan DB16279
small molecule | CAS: 1914998-56-3

Pecavaptan is under investigation in clinical trial NCT03901729 (A Trial to Study BAY1753011 in Patients With Congestive Heart Failure).

Target Protein:
Vasopressin V1a receptorVasopressin V2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pecilocin DB13459
small molecule | CAS: 19504-77-9

Deskripsi belum tersedia.

Kategori:
Antifungal AgentsAntifungals for Dermatological UseAntifungals for Topical Use +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pectin Approved DB11158
biotech | CAS: 9000-69-5

Pectin is a heteropolysaccharide commercially derived from the cell wall of higher plants.[A32327] It is composed of partially methylated polygalacturonic acid units linked in the positions 1-4.[L1961] The carboxylic group of the constituents of pectin can ex…

Kategori:
Alimentary Tract and MetabolismAntidiarrheals, Intestinal Antiinflammatory/antiinfective AgentsBiological Products +15
Waktu ParuhPharmacokinetic stu…
Vol. DistribusiPharmacokinetic stu…
KlirensPharmacokinetic stu…
Genetik -
Pefcalcitol DB11786
small molecule | CAS: 381212-03-9

Pefcalcitol has been investigated for the basic science of Psoriasis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peficitinib DB11708
small molecule | CAS: 944118-01-8

Peficitinib has been used in trials studying the treatment and basic science of Psoriasis, Pharmacodynamics, Drug Interactions, Colitis, Ulcerative, and RHEUMATOID ARTHRITIS, among others.

Kategori:
Antineoplastic and Immunomodulating AgentsBridged-Ring CompoundsCycloparaffins +7
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pefloxacin Approved DB00487
small molecule | CAS: 70458-92-3

A synthetic broad-spectrum fluoroquinolone antibacterial agent active against most gram-negative and gram-positive bacteria.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-betaDNA topoisomerase 4 subunit ADNA gyrase subunit A +2
Waktu Paruh8.6 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
Pegademase Approved DB00061
biotech | CAS: 130167-68-9

Bovine adenosine deaminase derived from bovine intestine that has been extensively pegylated for extended serum half life.

Kategori:
Adjuvants, ImmunologicAminohydrolasesAntineoplastic and Immunomodulating Agents +7
Target Protein:
AdenosineGrowth factor receptor-bound protein 2
Waktu Paruhplasma adenosine de…
Vol. Distribusi-
Klirens-
Genetik -
Pegadricase DB15129
biotech | CAS: 1040753-26-1

Pegadricase is under investigation in clinical trial NCT01021241 (Safety and Efficacy Study of Intravenous Uricase-PEG 20).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegamotecan DB12842
small molecule | CAS: 581079-18-7

Pegamotecan has been used in trials studying the treatment of Cancer of Stomach, Sarcoma, Soft Tissue, and Gastroesophageal Cancer.

Kategori:
AlcoholsAlkaloidsCompounds used in a research, industrial, or household setting +5
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegapamodutide DB14817
biotech | CAS: 1492924-65-8

Pegapamodutide is under investigation in clinical trial NCT02188303 (A Study of LY2944876 in Healthy Japanese and Non-Japanese Participants).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegaptanib Approved DB04895
biotech | CAS: 222716-86-1

Pegaptanib is a polynucleotide aptamer. Pegatinib aids neovascular age-related macular degeneration by binding to VEGF which in order reduces angiogenesis and vessel permeability. Pegaptanib was granted FDA approval on 17 September 2004.[L17903]

Kategori:
Antineovascularisation AgentsCarbohydratesDrugs that are Mainly Renally Excreted +10
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhIn humans, after a …
Vol. DistribusiIt is distributed i…
Klirens-
Genetik -
Pegargiminase DB06592
small molecule | CAS: 1394129-74-8

Pegargiminase is an anticancer agent.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEnzymes +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegaspargase Approved DB00059
biotech | CAS: 130167-69-0

Pegaspargase is a conjugate of monomethoxypolyethylene glycol (mPEG) and L-asparaginase (L-asparagine amidohydrolase), an asparagine-specific enzyme that converts L-asparagine into aspartic acid and ammonia.[L44667] Asparagine is an amino acid that is vital f…

Kategori:
AlcoholsAmidohydrolasesAntineoplastic Agents +15
Target Protein:
L-asparagine
Waktu ParuhThe mean eliminatio…
Vol. DistribusiBased on a non-comp…
KlirensFor a single intram…
Genetik -
Pegcetacoplan Approved DB16694
biotech | CAS: 2019171-69-6

Pegcetacoplan is a complement inhibitor indicated in the treatment of paroxysmal nocturnal hemoglobinuria (PNH).[A235000,L34095] Prior to its FDA approval, patients with PNH were typically treated with the C5 inhibiting monoclonal antibody [eculizumab].[A2350…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsComplement Inactivating Agents +6
Target Protein:
Complement C3
Waktu ParuhThe median half lif…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
biotech | CAS: 1448590-54-2

Pegcrisantaspase is under investigation in clinical trial NCT02257684 (A Dose Confirmation and Pharmacokinetic Study of Pegcrisantaspase Administered as Intravenous (IV) Infusion in Children and Young Adults With Acute Lymphoblastic Leukemia (ALL) /Lymphoblas…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegenzileukin DB17495
biotech | CAS: 2573074-47-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegfilgrastim Approved DB00019
biotech | CAS: 208265-92-3

Pegfilgrastim is a PEGylated form of the recombinant human granulocyte colony-stimulating factor (G-CSF) analogue, [filgrastim].[A187601] The drug is approved for use to decrease the incidence of infection, as manifested by febrile neutropenia, in susceptible…

Kategori:
Adjuvants, ImmunologicAlcoholsAmino Acids, Peptides, and Proteins +21
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe serum half-life…
Vol. DistribusiPegfilgrastim appea…
KlirensPegfilgrastim has a…
Genetik -
Peginesatide Approved DB08894
biotech | CAS: 913976-27-9

Peginesatide is a synthetic peptide attached to polyethylene glycol for the treatment of anemia. The polyethylene glycol moiety helps make the drug less immunogenic and prolongs its plasma half-life. Chemically, peginesatide is designed to mimic the pharmacol…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsAntianemic Preparations +10
Target Protein:
Erythropoietin receptor
Waktu ParuhIV dose, healthy su…
Vol. DistribusiIV dose, dialysis p…
KlirensSystemic clearance,…
Genetik -
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