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11778

Total database: 17430
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8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 172 / 236
Pam2csk4 DB16474
small molecule | CAS: 574741-81-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsDNA-Binding ProteinsExperimental Unapproved Treatments for COVID-19 +5
Target Protein:
Toll-like receptor 6Toll-like receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pamapimod DB19169
small molecule | CAS: 449811-01-2

Pamapimod is under investigation in clinical trial NCT05659459 (The KIN-FAST Trial (KIN001 for Accelerated Symptoms Termination) in Non Hospitalized Patients Infected With Sars-cov-2).

Kategori:
p38 Mitogen-Activated Protein Kinases, antagonists & inhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pamidronic acid Approved DB00282
small molecule | CAS: 40391-99-9

Pamidronic acid is a second generation, nitrogen containing bisphosphonate similar to [neridronic acid] and [alendronic acid].[A203111] Pamidronic acid was first described in the literature in 1977.[A203267] The second generation bisphosphonates are less comm…

Kategori:
Agents Causing Muscle ToxicityAntineoplastic AgentsBisphosphonates +7
Target Protein:
Farnesyl pyrophosphate synthaseHydroxylapatiteGeranylgeranyl pyrophosphate synthase +2
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
KlirensThe mean total clea…
Genetik -
Pamiparib DB14769
small molecule | CAS: 1446261-44-4

Pamiparib is under investigation in clinical trial NCT03933761 (Pamiparib in Fusion Positive, Reversion Negative High Grade Serous Ovarian Cancer or Carcinosarcoma With BRCA1/2 Gene Mutations If Progression on Substrate Poly ADP Ribose Polymerase Inhibitbor (…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 59763-91-6

Pancreatic Polypeptide has been investigated for the treatment of Diabetes Mellitus, Type 1.

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal AgentsHormones +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pancrelipase Approved DB00085
biotech | CAS: 53608-75-6

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase mixture was developed by Ortho-McNeil-Janssen Pharmace…

Kategori:
Alimentary Tract and MetabolismCarboxylic Ester HydrolasesComplex Mixtures +10
Target Protein:
Dietary fatDietary proteinDietary starch
Waktu ParuhPancrelipase acts l…
Vol. DistribusiPancrelipase acts l…
KlirensPancrelipase acts l…
Genetik -
Pancrelipase amylase Approved DB11065
biotech | CAS: 9000-90-2

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The amylases are enzymes that help in the chemical process of digestion…

Kategori:
AmylasesAmylases, antagonists & inhibitorsEnzymes +3
Target Protein:
Dietary starch
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Pancrelipase lipase Approved DB13147
biotech | CAS: 9001-62-1

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase lipase is an enzyme secreted by the pancreas that is r…

Kategori:
Carboxylic Ester HydrolasesEnzymesEnzymes and Coenzymes +4
Target Protein:
Dietary fat
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Pancrelipase protease Approved DB11066
biotech | CAS: 9001-94-9

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase protease is a mix of enzymes, formed by trypsin and ch…

Kategori:
EnzymesEnzymes and CoenzymesHydrolases +1
Target Protein:
Dietary protein
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Pancuronium Approved DB01337
small molecule | CAS: 16974-53-1

A bis-quaternary steroid that is a competitive nicotinic antagonist. As a neuromuscular blocking agent it is more potent than curare but has less effect on the circulatory system and on histamine release.

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +19
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3
Waktu Paruh1.5 to 2.7 hours.
Vol. Distribusi* 241 to 280 mL/kg
Klirens* Plasma cl=1.1–1.9…
Genetik -
Panitumumab Approved DB01269
biotech | CAS: 339177-26-3

Panitumumab (ABX-EGF) is a recombinant human IgG2 monoclonal antibody that binds specifically to the human epidermal growth factor receptor (EGFR). This drug is an antineoplastic agent. Panitumumab was granted FDA approval on 27 September 2006.[L17663]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Epidermal growth factor receptor
Waktu Paruh7.5 days (range: 4-…
Vol. Distribusi-
Klirens* 4.9+/- 1.4 mL/kg/…
Genetik -
Panobacumab DB15342
biotech | CAS: 885053-97-4

Panobacumab is under investigation in clinical trial NCT00851435 (Safety and Pharmacokinetics of KBPA-101 in Hospital Acquired Pneumonia Caused by O11 Pseudomonas Aeruginosa).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Panobinostat Approved DB06603
small molecule | CAS: 404950-80-7

Panobinostat is an oral deacetylace (DAC) inhibitor approved on February 23, 2015 by the FDA for the treatment of multiple myeloma. The approval was accelerated based on progression-free survival, therefore confirmatory trials by the sponsor to demonstrate cl…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
Histone deacetylase 1Histone deacetylase
Waktu Paruh30 hours
Vol. Distribusi-
Klirens-
Genetik -
Pantethine Approved DB11190
small molecule | CAS: 16816-67-4

Pantethine is a naturally occurring compound synthesized in the body from pantothenic acid (vitamin B5) via addition of cysteamine. It consists of two molecules of pantetheine that form a dimer via disufide linkages, and acts as an intermediate in the product…

Kategori:
Alimentary Tract and MetabolismSulfhydryl CompoundsSulfur Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Panthenol Approved DB11204
small molecule | CAS: 16485-10-2

Panthenol is an alcohol derivative of pantothenic acid, a component of the B complex vitamins and an essential component of a normally functioning epithelium. Panthenol exists as a racemic mixture containing both the dextrorotatory form (dexpanthenol) and the…

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pantoprazole Approved DB00213
small molecule | CAS: 102625-70-7

Pantoprazole is a first-generation proton pump inhibitor (PPI) used for the management of gastroesophageal reflux disease (GERD), for gastric protection to prevent recurrence of stomach ulcers or gastric damage from chronic use of NSAIDs, and for the treatmen…

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesAcid ReducersAlimentary Tract and Metabolism +27
Target Protein:
Potassium-transporting ATPase alpha chain 1Potassium-transporting ATPase subunit betaN(G),N(G)-dimethylarginine dimethylaminohydrolase 1
Waktu ParuhAbout 1 hour[F3202]
Vol. DistribusiThe apparent volume…
Klirens**Adults**: With in…
Genetik -
Pantothenic acid Approved DB01783
small molecule | CAS: 79-83-4

Pantothenic acid, also called pantothenate or vitamin B5 (a B vitamin), is a water-soluble vitamin discovered by Roger J. Williams in 1919. For many animals, pantothenic acid is an essential nutrient as it is required to synthesize coenzyme-A (CoA), as well a…

Kategori:
AlanineAlimentary Tract and MetabolismAmino Acids +9
Target Protein:
Pantothenate kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Phosphopantothenoylcysteine decarboxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Papain Approved DB11193
biotech | CAS: 9001-73-4

Papain, also known as papaya proteinase I, is a cysteine protease (EC 3.4.22.2) enzyme that is found in species of papaya, _Carica papaya_ and _Vasconcellea cundinamarcensis_. The enzyme is found to be localized in the skin of papaya, and is collected from sl…

Kategori:
Cysteine EndopeptidasesCysteine ProteasesEndopeptidases +6
Target Protein:
Toll-like receptor 4
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Papaverine Approved DB01113
small molecule | CAS: 58-74-2

An alkaloid found in opium but not closely related to the other opium alkaloids in its structure or pharmacological actions. It is a direct-acting smooth muscle relaxant used in the treatment of impotence and as a vasodilator, especially for cerebral vasodila…

Kategori:
Alimentary Tract and MetabolismAlkaloidsBenzylisoquinolines +18
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4DcGMP-specific 3',5'-cyclic phosphodiesterase3',5'-cyclic-AMP phosphodiesterase 4B +2
Waktu Paruh0.5-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Paprika Approved DB10678
biotech

Paprika allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 873-75-6

Deskripsi belum tersedia.

Kategori:
AlcoholsBenzene DerivativesBenzyl Compounds
Target Protein:
Alcohol dehydrogenase 1C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paraldehyde Approved DB09117
small molecule | CAS: 123-63-7

Paraldehyde was initially introduced into medical practice in the United Kingdom in 1882 by the Italian physician Vincenzo Cervello. It is classified as a central nervous system (CNS) depressant and has also been found to be an effective anticonvulsant, hypno…

Kategori:
AcetaldehydeAnticonvulsantsCentral Nervous System Agents +4
Waktu ParuhThe mean half life …
Vol. Distribusi-
Klirens-
Genetik -
Paramethadione Approved DB00617
small molecule | CAS: 115-67-3

Paramethadione is an anticonvulsant in the oxazolidinedione class. It is associated with fetal trimethadione syndrome, which is also known as paramethadione syndrome.

Kategori:
AnticonvulsantsCentral Nervous System DepressantsCytochrome P-450 CYP2C8 Substrates +7
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1GVoltage-dependent T-type calcium channel subunit alpha-1I
Waktu Paruh12 to 24 hours (how…
Vol. Distribusi-
Klirens-
Genetik -
Paramethasone DB01384
small molecule | CAS: 53-33-8

A glucocorticoid with the general properties of corticosteroids. It has been used by mouth in the treatment of all conditions in which corticosteroid therapy is indicated except adrenal-deficiency states for which its lack of sodium-retaining properties makes…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +27
Target Protein:
Corticosteroid-binding globulinGlucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paramethasone acetate Approved DB14657
small molecule | CAS: 1597-82-6

Deskripsi belum tersedia.

Kategori:
Fused-Ring CompoundsPregnadienesPregnadienetriols +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parathiazine DB15978
small molecule | CAS: 84-08-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 172867-62-8

Parathyroid Hormone-Related Protein 1-36 is under investigation in clinical trial NCT00853723 (Comparison Study of Pthrp and PTH to Treat Osteoporosis).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsHormones +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pardoprunox DB12061
small molecule | CAS: 269718-84-5

Pardoprunox has been used in trials studying the treatment of Early Stage Parkinson's Disease and Advanced Stage Parkinson's Disease. Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parecoxib Approved DB08439
small molecule | CAS: 198470-84-7

Parecoxib is a water-soluble and injectable prodrug of valdecoxib. It is marketed as Dynastat in the European Union. Parecoxib is a COX2 selective inhibitor in the same category as celecoxib (Celebrex) and rofecoxib (Vioxx). As it is injectable, it can be use…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +18
Target Protein:
Prostaglandin G/H synthase 2Lactotransferrin
Waktu Paruh22 minutes (parecox…
Vol. Distribusi-
Klirens-
Genetik -
Pargeverine DB15783
small molecule | CAS: 13479-13-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pargyline Approved DB01626
small molecule | CAS: 555-57-7

Pargyline is a monoamine oxidase inhibitor with antihypertensive properties.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAmines +12
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2259927-72-3

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paritaprevir Approved DB09297
small molecule | CAS: 1216941-48-8

Paritaprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into ni…

Kategori:
AmidesAmino AcidsAmino Acids, Cyclic +27
Target Protein:
Genome polyproteinGag-Pol polyprotein
Waktu Paruh5.5 hr [FDA Label]
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
Paromomycin Approved DB01421
small molecule | CAS: 7542-37-2

An oligosaccharide antibiotic produced by various streptomyces. [PubChem]

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmebicides +10
Target Protein:
30S ribosomal protein S1016S ribosomal RNASmall ribosomal subunit protein uS2 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paroxetine Approved DB00715
small molecule | CAS: 61869-08-7

Paroxetine is a selective serotonin reuptake inhibitor (SSRI) drug commonly known as Paxil. It has a variety of uses, including the treatment of anxiety disorders, major depression, posttraumatic stress disorder, and symptoms of menopause, among others.[T653]…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAntidepressive Agents +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporter5-hydroxytryptamine receptor 2A +9
Gen Terkait:
ABCB1 CYP2D6 CYP2D6 +4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiParoxetine has a la…
KlirensThe apparent oral c…
Genetik 7 Varian
PARPI F-18 DB18657
small molecule | CAS: 1883580-48-0

PARPI F-18 is a diagnostic agent under investigation for use in the management of glioblastoma multiforme.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parsaclisib DB14867
small molecule | CAS: 1426698-88-5

Parsaclisib is under investigation in clinical trial NCT03126019 (An Open-Label Study of Parsaclisib in Relapsed or Refractory Follicular Lymphoma (CITADEL-203)).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsPhosphatidylinositol-3-kinase (Pi3K) inhibitors +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parsatuzumab DB14897
biotech | CAS: 1312797-14-0

Parsatuzumab is under investigation in clinical trial NCT01366131 (Study Evaluating the Safety and Efficacy of MEGF0444A in Combination With Carboplatin, Paclitaxel and Bevacizumab in Patients With Advanced or Recurrent Non-Squamous Non-Small Cell Lung Cancer…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Parsley Approved DB10647
biotech

Parsley allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PASBN DB03078
small molecule

Deskripsi belum tersedia.

Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pascopyrum smithii pollen Approved DB10719
biotech

Pascopyrum smithii pollen is the pollen of the Pascopyrum smithii plant. Pascopyrum smithii pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pasireotide Approved DB06663
small molecule | CAS: 396091-73-9

Pasireotide is a synthetic long-acting cyclic hexapeptide with somatostatin-like activity. It is marketed as a diaspartate salt called Signifor, which is used in the treatment of Cushing's disease.

Kategori:
Amino Acids, Peptides, and ProteinsBradycardia-Causing AgentsCytochrome P-450 CYP3A Inhibitors +22
Target Protein:
Somatostatin receptor type 3Somatostatin receptor type 1Somatostatin receptor type 2 +1
Waktu ParuhThe half-life is 12…
Vol. DistribusiPasireotide is wide…
KlirensThe clearance in he…
Genetik -
Passalora fulva Approved DB10817
biotech

Passalora fulva is a fungus which can provoke allergic reactions. Passalora fulva extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Passiflora incarnata flower Approved DB13974
biotech

Deskripsi belum tersedia.

Kategori:
Central Nervous System DepressantsHerbs and Natural ProductsHypnotics and Sedatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PAT-1251 DB16735
small molecule | CAS: 2098884-52-5

PAT-1251 is under investigation in clinical trial NCT04054245 (PAT-1251 in Treating Patients With Primary Myelofibrosis, Post-polycythemia Vera Myelofibrosis, or Post-essential Thrombocytosis Myelofibrosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PAT-SM6 DB17406
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pateclizumab DB14997
biotech | CAS: 1202526-59-7

Pateclizumab is under investigation in clinical trial NCT01225393 (A Study to Evaluate the Efficacy and Safety of MLTA3698A in Combination With a Disease-Modifying Anti-Rheumatic Drug (DMARD) Compared With Adalimumab in Combination With a DMARD in Patients Wi…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Patent Blue Approved DB13967
small molecule | CAS: 25305-77-5

Patent blue is aniline dye and it is one of the most common dyes used.[A32573] It is a sodium or calcium salt of diethylammonium hydroxide inner salt.[A32574] It has the chemical designation of (4-(alpha-(p-(diethylamino)phenyl)-2,4-disulfobenzylidene)-2,5-cy…

Kategori:
AminesAniline CompoundsColoring Agents +4
Target Protein:
Albumin
Waktu ParuhThe elimination hal…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Patidegib DB12655
small molecule | CAS: 1037210-93-7

Patidegib has been investigated for the treatment of Conventional Chondrosarcoma.

Kategori:
Alkaloids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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