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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 172 / 282
LY2140023 DB05096
small molecule

LY2140023 is an investigational drug from Lilly, which is being developed as a new treatment option for schizophrenia. LY2140023 is an oral "prodrug," meaning it is devoid of intrinsic biological activity and, once administered, is metabolized to provide the …

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
Metabotropic glutamate receptor 2Metabotropic glutamate receptor 3
Waktu Paruh-
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LY2181308 DB05141
small molecule

LY2181308 is investigated in clinical trials for treating solid tumors. LY2181308 is a solid. LY2181308 is directed against a molecular target called survivin. LY2181308 is known to target baculoviral IAP repeat-containing protein 5. LY2181308 is an anti-sens…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Baculoviral IAP repeat-containing protein 5
Waktu Paruh-
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LY2275796 DB05165
small molecule

LY2275796 is a second-generation antisense anti-cancer drug candidate for clinical development. LY2275796 targets eukaryotic initiation factor- 4E (eIF-4E), a protein involved in the translation of key growth and survival factors that drive tumor progression,…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Eukaryotic translation initiation factor 4E
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
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LY249543 DB04322
small molecule

Deskripsi belum tersedia.

Target Protein:
C-1-tetrahydrofolate synthase, cytoplasmic
Waktu Paruh-
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LY2828360 DB16074
small molecule | CAS: 1231220-79-3

LY2828360 is under investigation in clinical trial NCT01319929 (A Study of LY2828360 in Patients With Osteoarthritic Knee Pain).

Kategori:
Cannabinoid Receptor AgonistsCannabinoids and similarsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
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LY374571 DB02358
small molecule

Deskripsi belum tersedia.

Target Protein:
C-1-tetrahydrofolate synthase, cytoplasmic
Waktu Paruh-
Vol. Distribusi-
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Lycopene Approved DB11231
small molecule | CAS: 502-65-8

Lycopene is a naturally occurring red carotenoid pigment that is responsible for red to pink colors seen in tomatoes, pink grapefruit, and other foods [A27242]. Having a chemical formula of C40H56, lycopene is a tetraterpene assembled from eight isoprene unit…

Kategori:
AlkenesAnti-Inflammatory AgentsAnticarcinogenic Agents +13
Waktu Paruh-
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Klirens-
Genetik -
biotech

Vaccine against Lyme disease that contains lipoprotein OspA, an outer surface protein of Borrelia burgdorferi sensu stricto ZS7, as expressed by Escherichia coli. Lipoprotein OspA is a single polypeptide chain of 257 amino acids with lipids covalently bonded …

Target Protein:
Toll-like receptor 2
Waktu Paruh1.2 hours (mammalia…
Vol. Distribusi-
Klirens-
Genetik -
Lymecycline Approved DB00256
small molecule | CAS: 992-21-2

Lymecycline is a broad-spectrum second-generation tetracycline antibiotic used for the treatment of acne and other susceptible bacterial infections.[L13880,L13883] It has been proven a cost-effective alternative to treatment with [minocycline] with comparable…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
30S ribosomal protein S4
Waktu ParuhThe half-life of ly…
Vol. DistribusiLymecycline is lipo…
KlirensLymecycline is part…
Genetik -
Lynestrenol Approved DB12474
small molecule | CAS: 52-76-6

Lynestrenol is a progestin and prodrug of [norethisterone].

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +25
Waktu Paruh-
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Lypressin Approved DB14642
small molecule | CAS: 50-57-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntidiuretic AgentsCardiovascular Agents +20
Target Protein:
Vasopressin V1a receptorVasopressin V2 receptorVasopressin V1b receptor
Waktu Paruh-
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Genetik -
small molecule

Lysergic acid 2,4-dimethylazetidide is under investigation in clinical trial NCT02765802 (A Study to Evaluate Pegylated Interferon Lambda Monotherapy in Patients With Chronic Hepatitis Delta Virus Infection).

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small molecule | CAS: 50-37-3

Debate continues over the nature and causes of chronic flashbacks. Explanations in terms of LSD physically remaining in the body for months or years after consumption have been discounted by experimental evidence. Some say HPPD is a manifestation of post-trau…

Kategori:
Agents that produce hypertensionAlkaloidsAntidepressive Agents +18
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2B +1
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Lysine Approved DB00123
small molecule | CAS: 56-87-1

Lysine (abbreviated as Lys or K) is an ?-amino acid with the chemical formula HO2CCH(NH2)(CH2)4NH2. This amino acid is an essential amino acid, which means that humans cannot synthesize it. Its codons are AAA and AAG. Lysine is a base, as are arginine and his…

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +10
Target Protein:
High affinity cationic amino acid transporter 1Cationic amino acid transporter 4Cationic amino acid transporter 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lysozyme DB13260
biotech | CAS: 12650-88-3

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseDermatologicals +6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
LYT-200 DB18179
biotech

LYT-200 is a fully human IgG4 monoclonal antibody directed against galectin-9.

Waktu Paruh-
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Genetik -
small molecule | CAS: 156021-12-4

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acetylcholinesterase
Waktu Paruh-
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M-032 DB17258
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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M-2698 DB15431
small molecule | CAS: 1379545-95-5

M-2698 is under investigation in clinical trial NCT01971515 (First-in-Human Dose Escalation Trial in Subjects With Advanced Malignancies).

Target Protein:
RAC-alpha serine/threonine-protein kinaseRAC-gamma serine/threonine-protein kinaseRibosomal protein S6 kinase beta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 6640-24-0

m-Chlorophenylpiperazine has been used in trials studying the treatment of Alcoholism.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNeurotransmitter Agents +7
Target Protein:
5-hydroxytryptamine receptor 1E5-hydroxytryptamine receptor 75-hydroxytryptamine receptor 6 +4
Waktu Paruh-
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Genetik -
small molecule | CAS: 1637-75-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzamides and benzamide derivatives +3
Target Protein:
Kynureninase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
M0002 DB05091
small molecule

M0002 is an orally-active selective vasopressin antagonist that inhibits water re-absorption from the kidneys. It is a vasopressin 2 antagonist and represents a new class of compounds – aquaretics – that produce profound diuresis without loss of electrolytes.…

Target Protein:
Vasopressin V2 receptor
Waktu Paruh-
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Genetik -
M002 DB18318
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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M012 DB18243
biotech

Deskripsi belum tersedia.

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Macelignan DB14129
small molecule | CAS: 107534-93-0

Macelignan is an NSAID with antioxidant, free radical scavenging, and neuroprotective activities.

Kategori:
Benzene DerivativesBenzyl Compounds
Waktu Paruh-
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Macimorelin Approved DB13074
small molecule | CAS: 381231-18-1

Macimorelin, a novel and orally active ghrelin mimetic that stimulates GH secretion, is used in the diagnosis of adult GH deficiency (AGHD). More specifically, macimorelin is a peptidomimetic growth hormone secretagogue (GHS) that acts as an agonist of GH sec…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +11
Target Protein:
Growth hormone secretagogue receptor type 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Macitentan Approved DB08932
small molecule | CAS: 441798-33-0

Macitentan is a dual endothelin receptor antagonist used in the treatment of pulmonary arterial hypertension (PAH).[L35890] It was first approved by the FDA in 2013. Macitentan differs from its predecessor [bosentan] in part due to its lower risk of hepatotox…

Kategori:
AmidesAntihypertensive AgentsAntihypertensives for Pulmonary Arterial Hypertension +13
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu ParuhThe half-life of el…
Vol. DistribusiMacitentan has an a…
KlirensClearance data was …
Genetik -
biotech

Maclura tricuspidata whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Macozinone DB14821
small molecule | CAS: 1377239-83-2

Macozinone is under investigation in clinical trial NCT03036163 (Phase 1 Study of PBTZ169).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsDrugs for Treatment of Tuberculosis +1
Waktu Paruh-
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Madecassic acid DB14037
small molecule | CAS: 18449-41-7

Deskripsi belum tersedia.

Kategori:
Terpenes
Waktu Paruh-
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Madecassoside DB15532
small molecule | CAS: 34540-22-2

Deskripsi belum tersedia.

Kategori:
Terpenes
Waktu Paruh-
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Maduramicin DB11525
small molecule | CAS: 84878-61-5

Maduramicin is an antiprotozoal agent used in veterinary medicine as prophylaxis against coccidiosis. It is a naturally occurring compound which was first isolated from the actinomycete, Actinomadura rubra.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsIonophores
Waktu Paruh-
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Mafenide Approved DB06795
small molecule | CAS: 138-39-6

Mafenide is a sulfonamide-type antimicrobial agent used to treat severe burns. It acts by reducing the bacterial population present in the burn tissue and promotes healing of deep burns.[L36773] In 1998, mafenide acetate was approved under the FDA’s accelerat…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 12Carbonic anhydrase 14 +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mafosfamide DB12083
small molecule | CAS: 88859-04-5

Mafosfamide has been used in trials studying the treatment of Lymphoma, Leukemia, Meningeal Neoplasm, and Brain and Central Nervous System Tumors.

Kategori:
Adjuvants, ImmunologicAntineoplastic AgentsHydrocarbons, Halogenated +6
Waktu Paruh-
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Genetik -
Maftivimab Approved DB15899
biotech | CAS: 2135632-36-7

Ebola virus (EBOV) remains an important human pathogen within the _Ebolavirus_ genus, having been responsible for at least 17 known outbreaks with an average case fatality rate of 43.92%.[A221825] Immune therapy using monoclonal antibodies (mAbs) is becoming …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Envelope glycoprotein
Waktu ParuhMaftivimab administ…
Vol. DistribusiMaftivimab administ…
KlirensMaftivimab administ…
Genetik -
Magnesium Approved DB14513
small molecule | CAS: 7439-95-4

Magnesium is classified as an alkaline earth metal and has 2 hydration shells.[A19349] The element can be found in abundance in the hydrosphere and in mineral salts such as dolomite and magnesium carbonate.[A19349] Common dietary sources of magnesium incl…

Kategori:
ElementsLaxativesMagnesium Compounds +6
Waktu ParuhMagnesiums biologic…
Vol. DistribusiAccording to a phar…
Klirens-
Genetik -
Magnesium acetate Approved DB13996
small molecule | CAS: 142-72-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAgents that produce neuromuscular block (indirect)Fatty Acids +3
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh-
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Genetik -
small molecule | CAS: 16674-78-5

Magnesium acetate tetrahydrate is a hydrated form of anhydrous magnesium acetate salt with the chemical formula of Mg(CH3COO)2 • 4H2O. As a salt form of magnesium, magnesium acetate is one of the bioavailable forms of magnesium and forms a very water soluble …

Kategori:
Agents that produce neuromuscular block (indirect)Laxatives
Target Protein:
Glutamate (NMDA) receptor
Waktu ParuhElimination half-li…
Vol. DistribusiMagnesium ions disp…
Klirens-
Genetik -
Magnesium Aluminum Silicate Approved DB11230
small molecule | CAS: 1327-43-1

Magnesium aluminum silicate is a naturally occurring mineral obtained from silicate ores of the montmorillonite group [A32782]. It is refined to a powder for use in cosmetic and pharmaceutical applications as an absorbent, anticaking agent, opacifying agent, …

Kategori:
Agents that produce neuromuscular block (indirect)MineralsPharmaceutic Aids +1
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small molecule | CAS: 28184-71-6

Deskripsi belum tersedia.

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Magnesium cation Approved DB01378
small molecule | CAS: 22537-22-0

Magnesium hydroxide is used primarily in "Milk of Magnesia", a white aqueous, mildly alkaline suspension of magnesium hydroxide formulated at about 8%w/v. Milk of magnesia is primarily used to alleviate constipation, but can also be used to relieve indigestio…

Kategori:
Agents that produce neuromuscular block (indirect)Calculi Dissolution AgentIncreased Large Intestinal Motility +9
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh-
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Magnesium citrate Approved DB11110
small molecule | CAS: 3344-18-1

Magnesium citrate is a low volume and osmotic cathartic agent. The cathartic action works primarily through the high osmolarity of the solution which draws large amounts of fluid into space where is used.[T215] Magnesium citrate is considered by the FDA as an…

Kategori:
Acids, AcyclicAgents that produce neuromuscular block (indirect)Alimentary Tract and Metabolism +15
Waktu ParuhThe study of the ha…
Vol. Distribusi-
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Magnesium gluconate Approved DB13749
small molecule | CAS: 59625-89-7

Magnesium gluconate is a magnesium salt of gluconate. It demonstrates the highest oral bioavailability of magnesium salts [L2608] and is used as a mineral supplement. Magnesium is ubiquitous in the human body, and is naturally present in many foods, added to …

Kategori:
Acids, AcyclicAgents that produce neuromuscular block (indirect)Alimentary Tract and Metabolism +7
Waktu Paruh-
Vol. DistribusiAbout 60% of the ma…
KlirensThe kidney plays a …
Genetik -
Magnesium hydroxide Approved DB09104
small molecule | CAS: 1309-42-8

Magnesium hydroxide is an inorganic compound. It is naturally found as the mineral brucite. Magnesium hydroxide can be used as an antacid or a laxative in either an oral liquid suspension or chewable tablet form. Additionally, magnesium hydroxide has smoke …

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAlkalies +22
Waktu ParuhN/A
Vol. DistribusiThe peak action and…
KlirensMagnesium hydroxide…
Genetik -
small molecule | CAS: 14452-57-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAluminum and magnesium containing antacidsAnions +15
Waktu Paruh-
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small molecule | CAS: 7757-87-1

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAgents that produce neuromuscular block (indirect) +10
Waktu Paruh-
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Magnesium silicate Approved DB13249
small molecule | CAS: 1343-88-0

Magnesium silicate is a compound of magnesium oxide and silicon. It is the magnesium salt of silicic acid containing an unspecified amount of water. The molecular formula can be expressed more clearly as MgSiO3.xH2O.[T186] It is known as talc and it presents …

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAluminum and magnesium containing antacids +9
Waktu ParuhThe very low absorp…
Vol. DistribusiThe very low absorp…
KlirensThe very low absorp…
Genetik -
Magnesium sulfate Approved DB00653
small molecule | CAS: 7487-88-9

A small colorless crystal used as an anticonvulsant, a cathartic, and an electrolyte replenisher in the treatment of pre-eclampsia and eclampsia. It causes direct inhibition of action potentials in myometrial muscle cells. Excitation and contraction are uncou…

Kategori:
Agents causing hyperkalemiaAgents that produce neuromuscular block (indirect)Alimentary Tract and Metabolism +38
Target Protein:
Voltage-dependent L-type calcium channel
Waktu Paruh43.2 hours (for new…
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 8551–8600 dari 14063
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