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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 171 / 236
P-57AS3 DB06569
small molecule | CAS: 384329-61-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
P-Anisic Acid DB02795
small molecule | CAS: 100-09-4

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +5
Target Protein:
Phospholipase A2Group IIE secretory phospholipase A2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
P-BCMA-101 DB17371
biotech

P-BCMA-101 is an autologous CAR-T therapy developed using Poseida’s piggyBac platform technology.

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small molecule | CAS: 104504-45-2

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +3
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1Tyrosine--tRNA ligase, cytoplasmic
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 76410-58-7

p-Boronophenylalanine is under investigation in clinical trial NCT00039572 (Boron Neutron Capture Therapy in Treating Patients With Glioblastoma Multiforme or Melanoma Metastatic to the Brain).

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 74-11-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates
Target Protein:
4-chlorobenzoyl CoA ligase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 90736-23-5

p-Fluorofentanyl is an opioid analgesic being an analogue of fentanyl developed by Janssen Pharmaceutica in the 1960s. p-Fluorofentanyl was sold briefly on the US black market in the early 1980s, before the introduction of the Federal Analog Act which for the…

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p-Heptylphenol DB03941
small molecule | CAS: 1987-50-4

Deskripsi belum tersedia.

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Genetik -
small molecule | CAS: 1126-48-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Target Protein:
Carbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
P-Nitrophenol DB04417
small molecule | CAS: 100-02-7

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesNitro CompoundsPhenols
Target Protein:
Sulfotransferase 1A1Alpha-amylase 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 104-03-0

Deskripsi belum tersedia.

Kategori:
Acids, Carbocyclic
Target Protein:
Penicillin G acylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
p-Quaterphenyl DB12794
small molecule | CAS: 135-70-6

p-Quaterphenyl has been used in trials studying the treatment of Malaria.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 70-55-3

Deskripsi belum tersedia.

Kategori:
AmidesBenzene DerivativesSulfonamides +2
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 12Carbonic anhydrase 6 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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PA3-17 DB18569
biotech

PA3-17 is CD7-directed chimeric antigen receptor (CAR) T-cell therapy.

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Pabinafusp alfa DB15633
biotech | CAS: 2140211-48-7

Pabinafusp alfa is under investigation in clinical trial NCT03568175 (A Study of JR-141 in Patients With Mucopolysaccharidosis II).

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PAC-113 DB05756
small molecule

PAC-113 an anti-fungal, for the treatment of oral candidiasis infections. It is a 12 amino-acid antimicrobial peptide derived from a naturally occurring histatin protein found in saliva. In vitro studies demonstrate that it has potent anti-fungal activity aga…

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Pacanalotamab DB17254
biotech | CAS: 2251756-52-0

Deskripsi belum tersedia.

Waktu Paruh-
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PACAP38 DB17073
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCardiovascular Agents +9
Waktu Paruh-
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Paclitaxel Approved DB01229
small molecule | CAS: 33069-62-4

Paclitaxel is a chemotherapeutic agent marketed under the brand name Taxol among others. Used as a treatment for various cancers, paclitaxel is a mitotic inhibitor that was first isolated in 1971 from the bark of the Pacific yew tree which contains endophytic…

Kategori:
Agents Causing Muscle ToxicityAlbuminsAmino Acids, Peptides, and Proteins +42
Target Protein:
Tubulin beta-1 chainApoptosis regulator Bcl-2Nuclear receptor subfamily 1 group I member 2
Waktu ParuhWhen a 24 hour infu…
Vol. Distribusi* 227 to 688 L/m^2 …
Klirens* 21.7 L/h/m2 [Dose…
Genetik -
small molecule | CAS: 186040-50-6

Deskripsi belum tersedia.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
Waktu Paruh-
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small molecule | CAS: 199796-52-6

A combination of [docosahexaenoic Acid] (a natural fatty acid) and [paclitaxel] (an anticancer drug) being studied in the treatment of cancer. It is a type of mitotic inhibitor.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
Target Protein:
Apoptosis regulator Bcl-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1075214-55-9

Three paclitaxel molecules linked by a cleavable succinyl ester linkage to a brain peptide vector, Angiopep-2, conjugate named ANG1005.

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsCardiotoxic antineoplastic agents +5
Waktu Paruh-
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Pacmilimab DB18873
biotech | CAS: 2145091-51-4

Pacmilimab is under investigation in clinical trial NCT04596150 (Study to Evaluate the Safety and Antitumor Activity of CX-2009 Monotherapy and in Combination With CX-072 in Advanced Breast Cancer).

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Pacritinib Approved DB11697
small molecule | CAS: 937272-79-2

Myelofibrosis (MF) is a rare disorder characterized by hematopoietic abnormalities and fibrosis within the bone marrow.[L40793] The underlying cause of primary MF is unknown, but secondary MF can arise in patients with a history of polycythemia vera or essent…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +29
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK2Receptor-type tyrosine-protein kinase FLT3
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Pactimibe DB12971
small molecule | CAS: 189198-30-9

Pactimibe has been used in trials studying the treatment of Atherosclerosis and Coronary Heart Disease.

Kategori:
Heterocyclic Compounds, Fused-RingIndolesSterol O-Acyltransferase, antagonists & inhibitors
Target Protein:
Liver carboxylesterase 1
Waktu Paruh-
Vol. Distribusi-
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Padeliporfin Approved DB15575
small molecule | CAS: 759457-82-4

Padeliporfin is a water-soluble chlorophyll derivative and cytotoxic photosensitizer used for vascular-targeted photodynamic therapy for malignancies.[A244559] Vascular-targeted photodynamic therapy (VTP), or vascular targeted photochemotherapy, is a focal tr…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Waktu ParuhThe estimated half-…
Vol. DistribusiIn healthy men rece…
KlirensFollowing administr…
Genetik -
Padimate O Approved DB11570
small molecule | CAS: 21245-02-3

Padimate O is an active sunscreen agent in cosmetics and over-the-counter sunscreen drug products in concentrations up to 8%, as regulated by the FDA [L2153]. It is a structurally-related compound to [DB02362] that absorbs UV-B rays to prevent photodamage. It…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +7
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Padnarsertib DB19243
small molecule | CAS: 1643913-93-2

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAcrylatesAmides +2
Target Protein:
Serine/threonine-protein kinase PAK 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Padsevonil DB14977
small molecule | CAS: 1294000-61-5

Padsevonil is under investigation in clinical trial NCT03695094 (A Study in Participants With Epilepsy, to Evaluate the Pharmacokinetics, Safety and Tolerability of Oxcarbazepine on Padsevonil).

Kategori:
AnticonvulsantsCentral Nervous System AgentsCentral Nervous System Depressants +3
Target Protein:
Synaptic vesicle glycoprotein 2A
Waktu Paruh-
Vol. Distribusi-
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Pafolacianine Approved DB15413
small molecule | CAS: 1628423-76-6

Pafolacianine, or OTL38, is a folate analogue conjugated with a fluorescent dye that absorbs light in the near-infrared (NIR) spectrum [A242572] within a range of 760 nm to 785 nm, with a peak absorption of 776 nm. It emits fluorescence within a range of 790 …

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic AgentsDiagnostic Uses of Chemicals +10
Target Protein:
Folate receptor alpha
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean plasma cle…
Genetik -
Pagibaximab DB17786
biotech | CAS: 595566-61-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pagoclone DB04903
small molecule | CAS: 133737-32-3

Pagoclone is an anxiolytic drug from the cyclopyrrolone family, which is related to other more well known drugs such as the sleeping medication zopiclone. It is one of a relatively recently developed class of medicines known as the nonbenzodiazepines, which h…

Kategori:
Central Nervous System DepressantsGABA AgentsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3
Waktu Paruh-
Vol. Distribusi-
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Palazestrant DB18971
small molecule | CAS: 2092925-89-6

Palazestrant is under investigation in clinical trial NCT06016738 (OP-1250 (Palazestrant) vs. Standard of Care for the Treatment of ER+/HER2- Advanced Breast Cancer).

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Palbociclib Approved DB09073
small molecule | CAS: 571190-30-2

Palbociclib is a piperazine pyridopyrimidine[A176792] that acts in the cell cycle machinery. It is a second generation cyclin-dependent kinase inhibitor[A176798] selected from a group of pyridopyrimidine compounds due to its favorable physical and pharmaceuti…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +21
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe mean apparent d…
KlirensThe mean apparent o…
Genetik -
Palifermin Approved DB00039
biotech | CAS: 162394-19-6

Palifermin is a recombinant human keratinocyte growth factor (KGF). It is 140 residues long, and is produced using E. coli. Palifermin was granted FDA approval on 15 December 2004.[L17933]

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsDetoxifying Agents for Antineoplastic Treatment +6
Target Protein:
Fibroblast growth factor receptor 2Fibroblast growth factor receptor 1Basement membrane-specific heparan sulfate proteoglycan core protein
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
Paliperidone Approved DB01267
small molecule | CAS: 144598-75-4

Paliperidone is the primary active metabolite of risperidone. The mechanism of action is unknown but it is likely to act via a similar pathway to risperidone. It has been proposed that the drug's therapeutic activity in schizophrenia is mediated through a com…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +37
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptorD(4) dopamine receptor +12
Waktu ParuhThe terminal elimin…
Vol. Distribusi* 487 L
Klirens-
Genetik -
Paliroden DB05454
small molecule | CAS: 188396-77-2

Paliroden is an orally active neurotrophic, non-peptidic compound that activates synthesis of endogenous neurotrophines. Studies show that use of paliroden increased the rate of formation of both neural progenitors and mature neurons. It is indicated for use …

Target Protein:
Glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
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Palivizumab Approved DB00110
biotech | CAS: 188039-54-5

Humanized monoclonal antibody (IgG1k) produced by recombinant DNA technology, directed to an epitope in the A antigenic site of the F protein of respiratory syncytial virus (RSV). Synagis is a composite of human (95%) and murine (5%) antibody sequences. The h…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +15
Target Protein:
Fusion glycoprotein F0Low affinity immunoglobulin gamma Fc region receptor III-BComplement C1r subcomponent +6
Waktu Paruh18-20 days (in adul…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14967-68-1

Palladium Pd-103 is under investigation in clinical trial NCT00247312 (Pd-103 Dose De-Escalation for Early Stage Prostate Cancer: A Prospective Randomized Trial).

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Palm oil DB14377
biotech | CAS: 8002-75-3

Palm oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesDietary Fats +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palmitic Acid Approved DB03796
small molecule | CAS: 57-10-3

A common saturated fatty acid found in fats and waxes including olive oil, palm oil, and body lipids.

Kategori:
Enzyme InhibitorsFatty AcidsLipids +1
Target Protein:
Fatty acid-binding protein, adipocyteFatty acid-binding protein 5Alpha-lactalbumin +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 373-49-9

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, UnsaturatedLipids
Target Protein:
UDP-3-O-[3-hydroxymyristoyl] N-acetylglucosamine deacetylaseFatty-acid peroxygenaseBifunctional cytochrome P450/NADPH--P450 reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 147732-56-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 221227-05-0

Deskripsi belum tersedia.

Waktu Paruh-
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Palonosetron Approved DB00377
small molecule | CAS: 135729-56-5

Palonosetron (INN, trade name Aloxi) is an antagonist of 5-HT3 receptors that is indicated for the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV). It is the most effective of the 5-HT3 antagonists in controlling delayed CINV nause…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +22
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu ParuhApproximately 40 ho…
Vol. Distribusi* 8.3 ± 2.5 L/kg
Klirens* 160 +/- 35 mL/h/kg
Genetik -
Palopegteriparatide Approved DB18676
biotech | CAS: 2222514-07-8

Palopegteriparatide is a parathyroid hormone (PTH) analog. Palopegteriparatide is a prodrug consisting of PTH(1-34) conjugated to a methoxy polyethylene glycol carrier (mPEG) via a proprietary TransCon Linker.[L51134] PTH(1-34) contains the N-terminal part of…

Kategori:
Calcium HomeostasisParathyroid Hormones and AnaloguesSystemic Hormonal Preparations, Excl. Sex Hormones and Insulins +1
Target Protein:
Parathyroid hormone/parathyroid hormone-related peptide receptor
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe estimated appar…
KlirensThe estimated clear…
Genetik -
Palovarotene Approved DB05467
small molecule | CAS: 410528-02-8

Fibrodysplasia Ossificans Progressiva (FOP), with an estimated worldwide prevalence of one in 2 million individuals, is an exceptionally rare genetic disorder.[A244920] FOP is caused by a gain-of-function mutation in the ACVR1/ALK2 gene which results in progr…

Kategori:
BCRP/ABCG2 InhibitorsBenzene DerivativesBenzylidene Compounds +17
Target Protein:
Retinoic acid receptor gamma
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean (SD) appar…
KlirensThe apparent total …
Genetik -
Paltusotine DB16277
small molecule | CAS: 2172870-89-0

Paltusotine is under investigation in clinical trial NCT04261712 (A Study to Evaluate the Long-term Safety and Efficacy of Paltusotine for the Treatment of Acromegaly (ACROBAT Advance)).

Target Protein:
Somatostatin receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palucorcel DB17955
biotech

Palucorcel is an investigational stem cell therapy consisting of human umbilical tissue-derived cells. Developed by Janssen Biotech, it is being investigated for the treatment of various conditions such as amyotrophic lateral sclerosis (ALS) and macular degen…

Waktu Paruh-
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