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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Hasil Pencarian (17430)

Halaman 170 / 349
Grn163l DB05036
small molecule

GRN163L is a novel anti-cancer drug. It has been characterized preclinically and shown to inhibit telomerase in human tumor cells of many cancer types (including lung, breast, prostate, liver, and early stage of human breast cancer), in both cell culture syst…

Target Protein:
Telomerase-binding protein EST1AN-terminal kinase-like proteinProstaglandin E synthase 3 +1
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GRObeta DB18205
biotech

Deskripsi belum tersedia.

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small molecule | CAS: 141925-59-9

Growth hormone-releasing peptide 1 is under investigation in clinical trial NCT00381602 (A Phase II, Randomized, Cross-over, Vehicle-controlled, Double-blind, Multicenter Study of the Safety, Pharmacodynamics, and Preliminary Efficacy of GHRP-1/AG in Subjects…

Kategori:
Amino Acids, Peptides, and ProteinsGrowth Hormone-Releasing HormonePeptides
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GS 0573 DB08843
small molecule | CAS: 113852-41-8

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsHeterocyclic Compounds, Fused-RingImmunologic Factors +1
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GS-100 DB18337
biotech

GS-100 is an adeno-associated virus serotype 9 virus particle containing viral DNA that includes an expression cassette containing the human NGLY1 gene coding sequence

Kategori:
CyclohexanesCycloparaffinsLipids +3
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GS-441524 DB15686
small molecule | CAS: 1191237-69-0

GS-441524 is an adenosine nucleotide analog antiviral, similar to [remdesivir].[A203057,L13239] This molecule was patented in 2009.[L13775] _In vitro_ studies of GS-441524 have determined it has a higher EC<sub>50</sub> than remdesivir against a number of vir…

Kategori:
Adenine NucleotidesAnti-Infective AgentsAntiviral Agents +10
Target Protein:
Replicase polyprotein 1abRNA-directed RNA polymerase L
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GS-5745 DB12296
biotech | CAS: 1518996-49-0

GS-5745 has been used in trials studying the treatment of Tumors, Breast Cancer, Crohn's Disease, Colorectal Cancer, and Pancreatic Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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GS-6620 DB15222
small molecule | CAS: 1350735-70-4

GS-6620 is under investigation in clinical trial NCT01316237 (A Study Evaluating the Safety, Tolerability, Pharmacokinetics and Antiviral Activity of GS-6620 in Treatment Naïve Subjects With Chronic Hepatitis C Virus Infection).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Genome polyprotein
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GS-9191 DB15084
small molecule | CAS: 859209-84-0

GS-9191 is under investigation in clinical trial NCT00499967 (Safety and Effectiveness Study of an Experimental Topical Ointment (GS-9191) for the Treatment of Genital Warts).

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
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GS-9256 DB12876
small molecule | CAS: 1001094-46-7

GS-9256 has been used in trials studying the treatment of HCV Infection and Chronic Hepatitis C Infection.

Kategori:
AcidsAcids, NoncarboxylicAmino Acids, Peptides, and Proteins +4
Target Protein:
Gag-Pol polyprotein
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GS030-DP DB17847
biotech

GS030-DP is an optogenetic gene therapy being investigated for the treatment of retinitis pigmentosa. It targets retinal ganglion cells that encodes a light-sensitive channelrhodopsin, ChrimsonR-tdTomato (ChR-tdT), delivered by an AAV2.7m8 vector. It is a com…

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GSBR-1290 DB18551
small molecule

GSBR-1290 is a small molecule agonist of the GLP-1 receptor.

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GSI-136 DB12819
small molecule | CAS: 443989-01-3

GSI-136 has been used in trials studying the treatment of Alzheimer Disease.

Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
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GSK-1004723 DB12806
small molecule | CAS: 955359-72-5

Gsk1004723 has been investigated for the treatment of Allergic Rhinitis and Rhinitis, Allergic, Seasonal.

Kategori:
Histamine AntagonistsHistamine H1 AntagonistsPyridazines
Target Protein:
Histamine H3 receptorHistamine H1 receptor
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GSK-1059615 DB11962
small molecule | CAS: 958852-01-2

GSK1059615 has been used in trials studying the treatment of Lymphoma, Solid Tumours, Endometrial Cancer, Solid Tumor Cancer, and Metastatic Breast Cancer.

Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 3-kinase catalytic subunit type 3
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GSK-1292263 DB12627
small molecule | CAS: 1032823-75-8

GSK1292263 has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.

Target Protein:
Glucose-dependent insulinotropic receptor
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GSK-1521498 DB12886
small molecule | CAS: 1007573-18-3

GSK1521498 has been used in trials studying the treatment of Obesity and Alcoholism.

Kategori:
IndenesReceptors, Opioid, mu
Target Protein:
Mu-type opioid receptor
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GSK-2018682 DB11987
small molecule | CAS: 1034688-30-6

GSK2018682 has been investigated for the treatment of Multiple Sclerosis, Relapsing-Remitting.

Kategori:
Heterocyclic Compounds, Fused-RingOxazoles
Target Protein:
Sphingosine 1-phosphate receptor 1
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GSK-239512 DB15120
small molecule | CAS: 720691-69-0

GSK-239512 is under investigation in clinical trial NCT00474513 (An Imaging Study to Investigate the Distribution of GSK239512 in the Brain.).

Kategori:
Heterocyclic Compounds, Fused-RingHistamine Antagonists
Target Protein:
Histamine H3 receptor
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GSK-256066 DB12137
small molecule | CAS: 801312-28-7

Gsk256066 has been used in trials studying the treatment and diagnostic of SAR, Asthma, Mild Asthma, Allergic Rhinitis, and Seasonal Allergic Rhinitis, among others.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPhosphodiesterase 4 Inhibitors +3
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A
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GSK-2636771 DB11795
small molecule | CAS: 1372540-25-4

GSK2636771 has been used in trials studying the treatment of CANCER, LYMPHOMA, Solid Neoplasm, Recurrent Solid Neoplasm, and Advanced Malignant Neoplasm, among others.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsOxazines +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
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GSK-269962A DB17030
small molecule | CAS: 850664-21-0

GSK-269962A is a Rho kinase (ROCK) inhibitor with both ROCK1 and ROCK2 affinity.[A253012]

Kategori:
Oxazoles
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GSK-2879552 DB16895
small molecule | CAS: 1401966-69-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesCycloparaffins
Target Protein:
Lysine-specific histone demethylase 1A
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GSK-2881078 DB16888
small molecule | CAS: 1539314-06-1

Deskripsi belum tersedia.

Kategori:
Anabolic AgentsHeterocyclic Compounds, Fused-RingHormones +1
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GSK-2981278 DB16319
small molecule | CAS: 1474110-21-8

GSK-2981278 is under investigation in clinical trial NCT03004846 (A Study of GSK2981278 Ointment in Subjects With Plaque Psoriasis).

Kategori:
AmidesBenzene DerivativesSulfonamides +2
Target Protein:
Nuclear receptor ROR-gamma
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GSK-2982772 DB16875
small molecule | CAS: 1622848-92-3

Deskripsi belum tersedia.

Target Protein:
Receptor-interacting serine/threonine-protein kinase 1
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GSK-3117391 DB15440
small molecule | CAS: 1018673-42-1

GSK-3117391 is under investigation in clinical trial NCT02965599 (Efficacy, Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of GSK3117391 in Subjects With Rheumatoid Arthritis).

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GSK-356278 DB12542
small molecule | CAS: 720704-34-7

Gsk356278 has been used in trials studying the treatment and basic science of Anxiety Disorders, Huntington Disease, Depressive Disorder, Huntingtons Disease, and Depressive Disorder, Major, among others.

Kategori:
OxazolesSulfur Compounds
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4B
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GSK-364735 DB13119
small molecule | CAS: 863434-13-3

GSK-364735 (Naphthyridinone) has been used in trials studying the treatment of HIV-1 Infection and Infection, Human Immunodeficiency Virus.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Gag-Pol polyprotein
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GSK-376501 DB12654
small molecule | CAS: 1010412-80-2

GSK376501 has been used in trials studying the treatment and diagnostic of Type 2 Diabetes Mellitus.

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GSK-424887 DB12219
small molecule

Gsk424887 has been used in trials studying the basic science and treatment of Depressive Disorder and Anxiety Disorder.

Kategori:
AcetatesAcids, AcyclicAmides
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GSK-690693 DB12745
small molecule | CAS: 937174-76-0

GSK690693 has been used in trials studying the treatment of Tumor, CANCER, and Lymphoma.

Kategori:
Oxazoles
Target Protein:
RAC-gamma serine/threonine-protein kinase
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GSK-923295 DB06097
small molecule

GSK-923295 is a small-molecule inhibitor of the mitotic kinesin centromere-associated protein E (CENP-E), and the third novel drug candidate to arise from Cytokinetics' broad strategic alliance with GlaxoSmithKline (GSK). GSK-923295 demonstrated a broad spect…

Target Protein:
Centromere-associated protein E
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GSK-945237 DB15345
small molecule | CAS: 944406-54-6

GSK-945237 is under investigation in clinical trial NCT01039610 (A Single Center Four Part Study in Healthy Adult Subjects to Evaluate: the Safety, Tolerability and Pharmacokinetics of a Single Oral Dose and Repeat Escalating Oral Doses of GSK945237; the Effe…

Kategori:
Heterocyclic Compounds, Fused-Ring
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GSK159797 DB05043
small molecule

GSK159797 ('797) is an inhaled, longer-acting Beta2 agonist developed for the treatment of respiratory disease such as asthma and COPD.

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GSK2245035 DB16076
small molecule | CAS: 1207629-49-9

GSK2245035 is under investigation in clinical trial NCT02833974 (Effect of the GSK2245035 on the Allergen-induced Asthmatic Response).

Kategori:
Heterocyclic Compounds, Fused-RingPurines
Target Protein:
Toll-like receptor 7
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GSK2256098 DB16106
small molecule | CAS: 1224887-10-8

GSK2256098 is under investigation in clinical trial NCT02523014 (Vismodegib and FAK Inhibitor GSK2256098 in Treating Patients With Progressive Meningiomas).

Kategori:
AminesHydroxy AcidsHydroxylamines +1
Target Protein:
Focal adhesion kinase 1
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GSK232802 DB16110
small molecule | CAS: 843661-24-5

GSK232802 is under investigation in clinical trial NCT00604825 (Treatment of Hot Flashes/flushes in Postmenopausal Women (WARM Study)).

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GSK2798745 DB16033
small molecule | CAS: 1419609-94-1

GSK2798745 is under investigation in clinical trial NCT03372603 (A Study to Assess the Effectiveness and Side Effects of GSK2798745 in Participants With Chronic Cough).

Kategori:
Heterocyclic Compounds, Fused-Ring
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GsMtx-4 DB17861
biotech

GsMtx-4 is a peptide found in tarantula venom that inhibits mechanosensitive ion channel (MSC) activity.

Kategori:
Amino Acids, Peptides, and ProteinsArthropod VenomsBiological Factors +5
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GT 389-255 DB05894
small molecule

Peptimmune’s lead product GT 389-255, is a novel lipase inhibitor and fat binding hydrogel polymer conjugate for the treatment of obesity which has completed single and multiple ascending dose (SAD and MAD) Phase I trials. It is expected to block fat absorpti…

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GT-AS DB17883
biotech

GT-AS recombinant adeno-associated virus serotype 9 vector containing the transgene UBE3A encoding for ubiquitin protein ligase E3A/E6-AP.

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GTA002 DB17187
biotech

Deskripsi belum tersedia.

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GTB-3550 DB18494
biotech

GTB-3550 is a single-chain, tri-specific scFv recombinant fusion protein conjugate composed of the variable regions of the heavy and light chains of anti-CD16 and anti-CD33 antibodies and a modified form of Interleukin 15 (IL-15).

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GTI 2040 DB05801
small molecule

GTI-2040 is a substance that is being studied as a treatment for cancer. It belongs to the family of drugs called antisense oligonucleotides.

Target Protein:
Ribonucleoside-diphosphate reductase subunit M2
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GTI-2040 DB15030
biotech | CAS: 236391-66-5

GTI-2040 is under investigation in clinical trial NCT00084643 (GTI-2040, Oxaliplatin, and Capecitabine in Treating Patients With Locally Advanced or Metastatic Colorectal Cancer or Other Solid Tumors).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
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GTI-2501 DB05406
small molecule

GTI-2501 is a novel antisense drug which has shown a favorable safety profile in preclinical studies, and in a phase I clinical trial. The drug is in a phase II clinical trial in combination with docetaxel for the treatment of hormone refractory prostate canc…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
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GTP-506 DB17682
biotech

GTP-506 is a gene therapy formed by two vectors, a nuclease vector targeting gene editing in the well-characterized PCSK9 gene locus and a therapeutic donor vector that inserts the OTC gene to provide the desired genetic correction.

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GTS-21 DB05708
small molecule | CAS: 148372-04-7

GTS-21 (also known as DMBX-A), is a novel, small-molecule, orally active and selective alpha-7 nicotinic acetylcholine (nACh) receptor agonist that has demonstrated memory and cognition enhancement activity in human clinical trials. Athenagen licensed the exc…

Kategori:
Benzene DerivativesCholinergic AgentsCholinergic Agonists +5
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
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GTX-102 DB16981
biotech

GTX-102 is an antisense oligonucleotide designed to target and inhibit the expression of UBE3A-AS. It is being investigated for the treatment of Angelman Syndrome.[L46772]

Kategori:
Antisense Oligonucleotide Specific to the Antisense Transcript of UBE3A
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