Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 170 / 236
Oxametacin DB13308
small molecule | CAS: 27035-30-9

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAntiinflammatory and Antirheumatic ProductsAntiinflammatory and Antirheumatic Products, Non-Steroids +1
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxamic Acid DB03940
small molecule | CAS: 471-47-6

Amino-substituted glyoxylic acid derivative. [PubChem]

Kategori:
Acids, AldehydicAmino AcidsAmino Acids, Peptides, and Proteins +1
Target Protein:
4-aminobutyrate aminotransferase, mitochondrialL-lactate dehydrogenaseL-lactate dehydrogenase +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxamniquine Approved DB01096
small molecule | CAS: 21738-42-1

An anthelmintic with schistosomicidal activity against Schistosoma mansoni, but not against other Schistosoma spp. Oxamniquine causes worms to shift from the mesenteric veins to the liver where the male worms are retained; the female worms return to the mesen…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +15
Target Protein:
DNA
Waktu Paruh1-2.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Oxantel DB13670
small molecule | CAS: 36531-26-7

Deskripsi belum tersedia.

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxaprotiline DB09307
small molecule | CAS: 56433-44-4

Oxaprotiline is a norepinephrine reuptake inhibitor of the tetracyclic antidepressant family that is related to maprotiline. This drug was never marketed. Oxaprotiline is a racemic mixture of the isomers levoprotiline and dextroprotiline. Levoprotiline is the…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnthracenes +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxatomide Approved DB12877
small molecule | CAS: 60607-34-3

Oxatomide has been used in trials studying the treatment of Muscular Dystrophy, Duchenne.

Kategori:
Anti-Allergic AgentsAnti-Asthmatic AgentsAntihistamines for Systemic Use +8
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxazepam Approved DB00842
small molecule | CAS: 604-75-1

Oxazepam is an intermediate-acting, 3-hydroxybenzodiazepine used in the treatment of alcohol withdrawal and anxiety disorders. Oxazepam, like related 3-hydroxybenzodiazepine [lorazepam], is considered less susceptible to pharmacokinetic variability based on p…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepine hypnotics and sedatives +16
Target Protein:
GABA(A) ReceptorTranslocator proteinGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1824-74-4

Deskripsi belum tersedia.

Kategori:
BenzazepinesBenzodiazepines and benzodiazepine derivativesBenzodiazepinones +2
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxazolam DB15491
small molecule | CAS: 24143-17-7

Deskripsi belum tersedia.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OXB-301 DB19269
biotech

OXB-301 is under investigation in clinical trial NCT00397345 (Trovax Renal Immunotherapy Survival Trial).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxcarbazepine Approved DB00776
small molecule | CAS: 28721-07-5

Oxcarbazepine is an anti-epileptic medication used in the treatment of partial onset seizures that was first approved for use in the United States in 2000.[L8627,L8630,L8633] It is a structural derivative of [carbamazepine][A186101] and exerts a majority of i…

Kategori:
Anti-epileptic AgentAnticonvulsantsCarboxamide Derivatives +29
Target Protein:
Sodium channel protein type 11 subunit alphaSodium channel protein
Gen Terkait:
HLA-B
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensPlasma clearance of…
Genetik 1 Varian
Oxeladin Approved DB04822
small molecule | CAS: 468-61-1

Withdrawn from the Canadian, US, and UK markets in 1976 due to carcinogenicity.

Kategori:
Acids, CarbocyclicAntitussive AgentsCentral Nervous System Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxetacaine Approved DB12532
small molecule | CAS: 126-27-2

Oxetacaine, also called oxethazaince, is a potent surface analgesic with the molecular formula N, N-bis-(N-methyl-N-phenyl-t-butyl-acetamide)-beta-hydroxyethylamine that conserves its unionized form at low pH levels. Its actions have shown to relieve dysphagi…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAnestheticsAnesthetics, Local +5
Target Protein:
Gastrin
Waktu ParuhOxetacaine presents…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Oxfendazole DB11446
small molecule | CAS: 53716-50-0

Oxfendazole is a sulfoxide metabolite of fenbendazole. This benzimidazole antihelminthic protects livestock from roundworm. strongyles, and pinworn.

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OXI-4503 DB05143
small molecule | CAS: 288847-35-8

OXI-4503 is investigated in clinical trials for treating cancer/tumors. OXI-4503 is a solid. OXI-4503 blocks and destroys tumor vasculature, resulting in extensive tumor cell death and necrosis. OXI-4503 (combretastatin A1 di-phosphate / CA1P) is a unique and…

Kategori:
AcidsAcids, NoncarboxylicAnions +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
ActVA 6 protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 9032-53-5

Deskripsi belum tersedia.

Kategori:
BiopolymersBlood and Blood Forming OrgansCarbohydrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxidronic acid Approved DB14159
small molecule | CAS: 15468-10-7

Deskripsi belum tersedia.

Kategori:
OrganophosphonatesOrganophosphorus Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxitropium DB12086
small molecule | CAS: 99571-64-9

Oxitropium has been investigated for the treatment of Pulmonary Disease, Chronic Obstructive.

Kategori:
Agents producing tachycardiaAlkaloidsAnticholinergic Agents +9
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxogluric acid DB08845
small molecule | CAS: 328-50-7

Oxogluric acid (?-Ketoglutarate) is not approved for any indication in the world but is an investigational drug in the United States. In the United States a phase I clinical trial is investigating whether oxogluric acid precursors found in nutritional supplem…

Kategori:
Acids, AcyclicDicarboxylic AcidsGlutarates +2
Target Protein:
Aspartate aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxolinic acid DB13627
small molecule | CAS: 14698-29-4

Deskripsi belum tersedia.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxomemazine DB13820
small molecule | CAS: 3689-50-7

Deskripsi belum tersedia.

Kategori:
Antihistamines for Systemic UseHeterocyclic Compounds, Fused-RingPhenothiazine Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 19771-63-2

Procysteine has been used in trials studying the treatment of HIV Infections.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Cyclic +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxprenolol Approved DB01580
small molecule | CAS: 6452-71-7

A beta-adrenergic antagonist used in the treatment of hypertension, angina pectoris, arrhythmias, and anxiety.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +32
Target Protein:
Beta-1 adrenergic receptorBeta-3 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Oxybenzone Approved DB01428
small molecule | CAS: 131-57-7

Oxybenzone is an organic compound used in sunscreens. It is a derivative of benzophenone. It forms colorless crystals that are readily soluble in most organic solvents. It is used as an ingredient in sunscreen and other cosmetics because it absorbs UV-A ultra…

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingCosmetics +6
Target Protein:
Hormone-sensitive lipaseProgesterone receptorAndrogen receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxybutynin Approved DB01062
small molecule | CAS: 5633-20-5

Overactive bladder (OAB) is a common condition negatively impacting the lives of millions of patients worldwide. Due to its urinary symptoms that include nocturia, urgency, and frequency, this condition causes social embarrassment and a poor quality of life.…

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAnticholinergic Agents +23
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1
Waktu ParuhThe plasma eliminat…
Vol. DistribusiOxybutynin has a wi…
Klirens-
Genetik -
Oxycodone Approved DB00497
small molecule | CAS: 76-42-6

Oxycodone is a semisynthetic opioid analgesic derived from thebaine in Germany in 1917.[A178696] It is currently indicated as an immediate release product for moderate to severe pain and as an extended release product for chronic moderate to severe pain requi…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +21
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Waktu ParuhThe apparent elimin…
Vol. Distribusi2.6L/kg.[Label]
KlirensTotal plasma cleara…
Genetik -
Oxyfedrine DB13398
small molecule | CAS: 15687-41-9

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-Agonists +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxygen Approved DB09140
small molecule | CAS: 7782-44-7

Oxygen is an element displayed by the symbol O, and atomic number 8. It is an essential element for human survival. Decreased oxygen levels may be treated with medical oxygen therapy. Treatment with oxygen serves to increase blood oxygen levels and also exer…

Kategori:
ChalcogensElementsGases +3
Target Protein:
Cytochrome c oxidase subunit 1NADPH oxidase 1
Waktu ParuhApproximately 122.2…
Vol. Distribusi-
Klirens-
Genetik -
Oxymatrine DB16276
small molecule | CAS: 16837-52-8

Oxymatrine is under investigation in clinical trial NCT02202473 (Oxymatrine Plus Lamivudine Combination Therapy Versus Lamivudine Monotherapy for Chronic Hepatitis B Infected Subjects).

Kategori:
AlkaloidsAnti-Infective AgentsAntiarrhythmic agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxymetazoline Approved DB00935
small molecule | CAS: 1491-59-4

Oxymetazoline is an imidazole derivative and a potent, direct-acting alpha (?)-adrenergic agonist with affinity to both ?<sub>1</sub>- and ?<sub>2</sub>-adrenoceptors.[A215542] Oxymetazoline is available in various formulations with a wide variety of clinical…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +25
Target Protein:
Alpha-1A adrenergic receptorAlpha-2A adrenergic receptorAlpha-2B adrenergic receptor +7
Waktu ParuhFollowing ocular ad…
Vol. DistribusiThere is limited in…
KlirensThere is limited in…
Genetik -
Oxymetholone Approved DB06412
small molecule | CAS: 434-07-1

Oxymetholone is a synthetic anabolic steroid marketed under the brand name Anapolon by Hoffmann La Roche Limitedand used in the treatment of osteoporosis, anaemia, and as an agent to stimulate muscle growth in malnourished or underdeveloped patients. Anabolic…

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +20
Target Protein:
Androgen receptorNatriuretic peptides B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxymorphone Approved DB01192
small molecule | CAS: 76-41-5

An opioid analgesic with actions and uses similar to those of morphine, apart from an absence of cough suppressant activity. It is used in the treatment of moderate to severe pain, including pain in obstetrics. It may also be used as an adjunct to anesthesia …

Kategori:
AdjuvantsAdjuvants, AnesthesiaAlkaloids +22
Target Protein:
Mu-type opioid receptorDelta-type opioid receptor
Waktu Paruh1.3 (+/-0.7) hours
Vol. Distribusi-
Klirens-
Genetik -
Oxypertine DB13403
small molecule | CAS: 153-87-7

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsIndole Derivatives +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxyphenisatin acetate Approved DB14627
small molecule | CAS: 115-33-3

Oxyphenisatin acetate is the pro-drug of [oxyphenisatin] (3,3-bis(4-hydroxyphenyl)-1H-indol-2-one). The FDA withdrew its approval for the use of oxyphenisatin acetate due to safety reasons.[L43942]

Kategori:
Gastrointestinal AgentsHeterocyclic Compounds, Fused-RingIndoles +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxyphenonium Approved DB00219
small molecule | CAS: 14214-84-7

A quaternary ammonium anticholinergic agent with peripheral side effects similar to those of atropine. It is used as an adjunct in the treatment of gastric and duodenal ulcer, and to relieve visceral spasms. The drug has also been used in the form of eye drop…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAmines +12
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxypurinol DB05262
small molecule | CAS: 2465-59-0

Oxypurinol, an inhibitor of xanthine oxidase, is a metabolite of allopurinol.

Kategori:
Enzyme InhibitorsPyrazolesPyrimidines +1
Target Protein:
Xanthine dehydrogenase/oxidase
Waktu Paruh23.3 +/- 6.0 hours
Vol. Distribusi-
Klirens-
Genetik -
Oxytetracycline Approved DB00595
small molecule | CAS: 79-57-2

A tetracycline analog isolated from the actinomycete streptomyces rimosus and used in a wide variety of clinical conditions.

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAnti-Bacterial Agents +16
Target Protein:
30S ribosomal protein S930S ribosomal protein S416S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxytocin Approved DB00107
biotech | CAS: 50-56-6

Sir Henry H. Dale first identified oxytocin and its uterine contractile properties in 1906.[A229008,A228593,A229108] Like all other neurohypophysial hormones, oxytocin is composed of nine amino acids with a disulfide bridge between the Cys 1 and 6 residues.[A…

Kategori:
Amino Acids, Peptides, and ProteinsGenito Urinary System and Sex HormonesHormones +15
Target Protein:
Oxytocin receptorVasopressin V1b receptorVasopressin V2 receptor +1
Waktu ParuhThe plasma half-lif…
Vol. Distribusi-
KlirensIn a study that obs…
Genetik -
Ozagrel DB12017
small molecule | CAS: 82571-53-7

Ozagrel has been used in trials studying the treatment of Dry Eye Syndromes.

Kategori:
Acids, AcyclicAcrylatesCardiovascular Agents +6
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ozanimod Approved DB12612
small molecule | CAS: 1306760-87-1

Ozanimod is a once-daily sphingosine 1-phosphate receptor modulator for the treatment of relapsing Multiple Sclerosis (MS) and inflammatory bowel disease. It was developed by Celgene (now acquired by Bristol-Myers Squibb) [L11025] and was approved by the FDA …

Kategori:
Antineoplastic and Immunomodulating AgentsBCRP/ABCG2 SubstratesCytochrome P-450 CYP2C8 Substrates +13
Target Protein:
Sphingosine 1-phosphate receptor 1Sphingosine 1-phosphate receptor 5
Waktu ParuhThe half-life of oz…
Vol. DistribusiThe average volume …
KlirensThe mean apparent o…
Genetik -
Ozarelix DB12581
small molecule | CAS: 295350-45-7

Ozarelix has been used in trials studying the treatment of Prostate Cancer, Benign Prostatic Hypertrophy, and Benign Prostatic Hyperplasia (BPH).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ozekibart DB18675
biotech | CAS: 2539847-03-3

Ozekibart is a tetravalent recombinant humanized IgG1 agonist antibody targeting the human TRAIL death receptor 5 (DR5). It is being investigated for the treatment of chondrosarcoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ozenoxacin Approved DB12924
small molecule | CAS: 245765-41-7

To date, ozenoxacin has been used in trials studying the treatment of impetigo. As of December 11, 2017 the FDA approved Ferrer Internacional S.A.'s Xepi (ozenoxacin 1%) as a topically applied cream indicated for the treatment of impetigo caused by *Staphy…

Kategori:
AminesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
DNA gyrase subunit ADNA topoisomerase 4 subunit ADNA gyrase subunit B +1
Waktu Paruh-
Vol. DistribusiOzenoxacin undergoe…
KlirensOzenoxacin undergoe…
Genetik -
Ozoralizumab DB12014
biotech | CAS: 1167985-17-2

Ozoralizumab has been used in trials studying the treatment of Rheumatoid Arthritis and Active Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2460400-11-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Target Protein:
Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
P-113D DB04987
biotech | CAS: 190673-60-0

P-113D is a novel 12 amino-acid antimicrobial peptide drug derived from histatins, which are compounds found naturally in human saliva. It is being pursued as a potential treatment for cystic fibrosis by Demegen, Inc.

Kategori:
Amino Acids, Peptides, and ProteinsAntimicrobial Cationic PeptidesAntimicrobial Peptides +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
P-2045 Re-188 DB17204
biotech | CAS: 934712-65-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 8451–8500 dari 11778
Sebelumnya Halaman 170 / 236 Berikutnya