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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 170 / 282
Losmapimod DB12270
small molecule | CAS: 585543-15-3

Losmapimod has been investigated for the prevention of Chronic Obstructive Pulmonary Disease.

Kategori:
Cycloparaffinsp38 Mitogen-Activated Protein KinasesProtein Kinase Inhibitors
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Loteprednol Approved DB00873
small molecule | CAS: 129260-79-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAndrostadienesAndrostanes +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Loteprednol etabonate Approved DB14596
small molecule | CAS: 82034-46-6

Loteprednol Etabonate (LE) is a topical corticoid anti-inflammatory. It is used in ophthalmic solution for the treatment of steroid responsive inflammatory conditions of the eye such as allergic conjunctivitis, uveitis, acne rosacea, superficial punctate kera…

Kategori:
Adrenal Cortex HormonesAndrostadienesAndrostanes +9
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe only data avail…
KlirensLoteprednol etabona…
Genetik -
Lotilaner Approved DB17992
small molecule | CAS: 1369852-71-0

Lotilaner is an ectoparasiticide that is a member of the isoxazoline family of compounds.[L47546] Lotilaner has largely been used for veterinary uses as an antiparasitic agent to treat flea and tick infestations in animals.[A260746, L47556] Lotilaner consists…

Kategori:
Antiparasitic AgentsEctoparasiticideEctoparasiticides, Incl. Scabicides +2
Target Protein:
Gaba-gated chloride channel, putative
Waktu ParuhThe effective half-…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Lovastatin Approved DB00227
small molecule | CAS: 75330-75-5

Lovastatin, also known as the brand name product Mevacor, is a lipid-lowering drug and fungal metabolite derived synthetically from a fermentation product of _Aspergillus terreus_.[A174550] Originally named Mevinolin, lovastatin belongs to the statin class of…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBSEP/ABCB11 Substrates +21
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-LHistone deacetylase 2
Waktu ParuhLovastatin half-lif…
Vol. DistribusiLovastatin is able …
Klirens-
Genetik -
Lovotibeglogene autotemcel Approved DB18680
biotech

Lovotibeglogene autotemcel consists of autologous hematopoietic stem and progenitor cells transduced with the BB305 lentiviral vector encoding a modified ?-globin gene. Specifically, lovotibeglogene autotemcel provides a functional copy of a modified beta-glo…

Kategori:
Autologous Cultured CellAutologous Hematopoietic Stem Cell-Based Gene TherapyGenetic Therapy
Target Protein:
Hemoglobin subunit beta
Waktu ParuhLovotibeglogene aut…
Vol. DistribusiLovotibeglogene aut…
KlirensLovotibeglogene aut…
Genetik -
biotech

Ingredient used in over-the-counter medications.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Loxapine Approved DB00408
small molecule | CAS: 1977-10-2

An antipsychotic agent used in schizophrenia. [PubChem]

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +24
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 2C +30
Waktu ParuhOral-4 hours
Vol. Distribusi-
Klirens-
Genetik -
Loxicodegol DB14146
small molecule | CAS: 1211231-76-3

Loxicodegol was developed by Nektar Therapeutics as an opioid analgesic with low abuse potential for the treatment of chronic pain [L3263]. The lack of abuse potential is believed to be due to the drug's slow rate of entry into brain, a unique characteristic …

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingOpiate Alkaloids +1
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhLoxicodegol has a h…
Vol. DistribusiLoxicodegol has a s…
KlirensLoxicodegol has a c…
Genetik -
Loxoprofen Approved DB09212
small molecule | CAS: 68767-14-6

Loxoprofen is a propionic acid derivative non-steroidal anti-inflammatory drug. It is marketed under the trade name Loxonin in Brazil, Mexico and Japan by Sankyo, as Loxomac in India, and as Oxeno in Argentina. A transdermal preparation was approved for use i…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +13
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe elimination hal…
Vol. DistribusiLoxoprofen has a vo…
KlirensMost of the drug as…
Genetik -
Loxoribine DB17589
small molecule | CAS: 121288-39-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LP-184 DB18215
small molecule | CAS: 924835-67-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LP-2307 DB17470
biotech

LP-2307 is an investigational allogeneic large multivalent immunogen (LMI) vaccine developed by Avanir. It was investigated for melanoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LP-284 DB18006
small molecule | CAS: 2412580-47-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LPT-99 DB17142
small molecule | CAS: 1263477-83-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LSALT Peptide DB16472
biotech

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LSP-GR3 DB16934
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LSTA1 DB17346
biotech | CAS: 1392278-76-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LSZ-102 DB15362
small molecule | CAS: 2135600-76-7

LSZ-102 is under investigation in clinical trial NCT02734615 (Phase I/Ib Trial of LSZ102 Single Agent or LSZ102 + LEE011 or LSZ102 + BYL719 in ER+ Breast Cancers).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LT2003 DB18359
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LTX-109 DB12711
small molecule | CAS: 1166254-80-3

LTX-109 has been investigated for the treatment of Atopic Dermatitis, Mild Eczema/Dermatoses, and Gram-positive, Skin Infections.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptidomimetics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LTX-315 DB12748
small molecule | CAS: 1345407-05-7

LTX-315 has been used in trials studying the treatment of Cancer, Lymphoma, Melanoma, Carcinoma, and Breast Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LU-31130 DB05828
small molecule

LU-31130 is a rapid acting therapy developed by H. Lundbeck A/S to treat Psychosis, Schizophrenia and Schizoaffective Disorders. It acts at the Dopamine D4 receptors in the cortex and has low affinity for D2 receptors, adrenoceptors, muscarinic and histaminer…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lubazodone DB09196
small molecule | CAS: 161178-07-0

Lubazodone (YM-992, YM-35,995) is an arylpiperazine antidepressant which was being developed as a treatment for depression and obsessive compulsive disorder, and reached phase II clinical trials, but was discontinued. It acts as a serotonin reuptake inhibitor…

Kategori:
Oxazines
Target Protein:
5-hydroxytryptamine receptor 2ASodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lubiprostone Approved DB01046
small molecule | CAS: 136790-76-6

Lubiprostone is a medication used in the management of idiopathic chronic constipation. A prostaglandin E1 derivative, lubiprostone is a bicyclic fatty acid that activates ClC-2 chloride channels located on the apical side of the gastrointestinal epithelial c…

Kategori:
Alimentary Tract and MetabolismChloride Channel AgonistsDrugs for Constipation +9
Target Protein:
Chloride channel protein 2
Waktu Paruh0.9 to 1.4 hours
Vol. Distribusi-
Klirens-
Genetik -
Lucanthone DB04967
small molecule | CAS: 479-50-5

One of the schistosomicides, it has been replaced largely by hycanthone and more recently praziquantel. (From Martindale The Extrapharmacopoeia, 30th ed., p46). It is currently being tested as a radiation sensitizer.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +7
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA repair nuclease/redox regulator APEX1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lucatumumab DB06360
biotech | CAS: 903512-50-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Tumor necrosis factor receptor superfamily member 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lucerastat DB14872
small molecule | CAS: 141206-42-0

Lucerastat is under investigation in clinical trial NCT03425539 (Efficacy and Safety of Lucerastat Oral Monotherapy in Adult Subjects With Fabry Disease).

Kategori:
AlkaloidsCarbohydratesImines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lucinactant Approved DB04897
biotech | CAS: 825600-90-6

Lucinactant is a new synthetic peptide-containing surfactant for intratracheal use. It contains sinapultide, a novel, hydrophobic, 21-amino acid peptide (leucine and lysine repeating units, KL4 peptide) designed to mimic human surfactant protein-B (SB-P). Mor…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lucitanib DB11845
small molecule | CAS: 1058137-23-7

Lucitanib has been used in trials studying the treatment of ER+, MBC, SCLC, HER2+, and NSCLC, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Vascular endothelial growth factor receptor 2 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lufenuron DB11424
small molecule | CAS: 103055-07-8

Lufenuron is used in veterinary for the control of flea.

Kategori:
Acids, CarbocyclicAgrochemicalsAmides +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luliconazole Approved DB08933
small molecule | CAS: 187164-19-8

Luliconazole is a topical antifungal agent that acts by unknown mechanisms but is postulated to involve altering the synthesis of fungi cell membranes. It was approved by the FDA (USA) in November 2013 and is marketed under the brand name Luzu. Luliconazole i…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +10
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhThe half life of lu…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of lu…
Genetik -
Lulizumab pegol DB15441
biotech | CAS: 1421830-13-8

Lulizumab pegol is under investigation in clinical trial NCT02843659 (Proof of Concept Study to Evaluate the Efficacy and Safety of BMS-931699 (Lulizumab) or BMS-986142 in Primary Sjögren's Syndrome).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsAntibodies, Monoclonal +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumacaftor Approved DB09280
small molecule | CAS: 936727-05-8

Lumacaftor is a drug used in combination with [DB08820] as the fixed dose combination product Orkambi for the management of Cystic Fibrosis (CF) in patients aged 6 years and older. Cystic Fibrosis is an autosomal recessive disorder caused by one of several di…

Kategori:
AminesCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +21
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe half-life of lu…
Vol. DistribusiFollowing oral admi…
KlirensThe typical apparen…
Genetik -
Lumasiran Approved DB15935
biotech | CAS: 1834610-13-7

Lumasiran is a small interfering RNA used in the treatment of primary hyperoxaluria type 1 (PH1).[L23554] This condition, caused by a deficiency in the enzyme alanine-glyoxylate aminotransferase, leads to an accumulation of oxalate, causing calcium crystal fo…

Kategori:
Alimentary Tract and MetabolismAntisense Elements (Genetics)Cytochrome P-450 CYP2C8 Inhibitors +12
Target Protein:
2-Hydroxyacid oxidase 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent centra…
KlirensThe apparent plasma…
Genetik -
Lumateperone Approved DB06077
small molecule | CAS: 313368-91-1

Schizophrenia is a complex mental illness and impacts approximately 1% of the population.[L10902] Although there are several antipsychotics including [aripiprazole], [paliperidone] and [clozapine] available for clinical use, they are generally accompanied by …

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +21
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 2AD(2) dopamine receptor +1
Waktu ParuhLumateperone's half…
Vol. DistribusiThe volume of distr…
KlirensLumateperone's clea…
Genetik -
Lumefantrine Approved DB06708
small molecule | CAS: 82186-77-4

Lumefantrine is an antimalarial agent used to treat acute uncomplicated malaria. It is administered in combination with artemether for improved efficacy. This combination therapy exerts its effects against the erythrocytic stages of <i>Plasmodium spp.</i> and…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +11
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh~ 4.5 days
Vol. Distribusi-
Klirens-
Genetik -
Lumefantrine co-artemether Approved DB13085
small molecule | CAS: 141204-94-6

Lumefantrine Co-Artemether (Riamet) has been investigated for the treatment of Malaria, Malaria, Falciparum, Malaria in Pregnancy, Uncomplicated Malaria, and Uncomplicated Knowlesi Malaria. Lumefantrine Co-Artemether is a tablet formulation of artemether and …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumichrome DB04345
small molecule | CAS: 1086-80-2

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +3
Target Protein:
Flavin reductase (NADPH)Riboflavin biosynthesis protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumicitabine DB14808
small molecule | CAS: 1445385-02-3

Lumicitabine is under investigation in clinical trial NCT03010059 (A Study to Assess the Relative Bioavailability of JNJ64041575 Administered as 2 Different New Concept Formulations (Oral Suspension and Tablet) Compared to Their Respective Current Formulation…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumiflavin DB04726
small molecule | CAS: 1088-56-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumiliximab DB06162
biotech | CAS: 357613-86-6

Lumiliximab is a chimeric monoclonal antibody which is used as an immunosuppressive drug. It is a primatized anti-CD23 macaque/human chimeric antibody that inhibits the production of the IgE antibody, for the potential treatment of allergic conditions. Lumili…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Low affinity immunoglobulin epsilon Fc receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luminol DB18536
small molecule | CAS: 521-31-3

Deskripsi belum tersedia.

Kategori:
Compounds used in a research, industrial, or household settingIndicators and ReagentsLaboratory Chemicals +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumiracoxib Approved DB01283
small molecule | CAS: 220991-20-8

Lumiracoxib is a COX-2 selective non-steroidal anti-inflammatory drug (NSAID). On August 11, 2007, Australia's Therapeutic Goods Administration (TGA, the Australian equivalent of the FDA) cancelled the registration of lumiracoxib in Australia due to concerns …

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +21
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhTerminal half-life …
Vol. Distribusi-
Klirens-
Genetik -
Lumretuzumab DB12683
biotech | CAS: 1448327-63-6

Lumretuzumab has been used in trials studying the treatment of Neoplasms, Breast Cancer, Squamous Non-Small Cell Lung Cancer, and Non-Squamous Non-Small Cell Lung Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lunasine DB16223
small molecule | CAS: 6901-22-0

Lunasine is under investigation in clinical trial NCT02709330 (ALS Reversals - Lunasin Regimen).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lunresertib DB19241
small molecule | CAS: 2719793-90-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lunsekimig DB19009
biotech | CAS: 2770858-49-4

Lunsekimig is under investigation in clinical trial NCT06102005 (Dose Ranging Study of Lunsekimig Compared With Placebo-control in Adult Participants With Moderate-to-severe Asthma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lupeol DB12622
small molecule | CAS: 545-47-1

Lupeol has been investigated for the treatment of Acne.

Kategori:
Anti-Inflammatory AgentsPentacyclic TriterpenesTerpenes +1
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaNeutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luprostiol DB11425
small molecule | CAS: 67110-79-6

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +6
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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