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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 170 / 315
ION283 DB18162
biotech

Deskripsi belum tersedia.

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ION356 DB19389
biotech

Deskripsi belum tersedia.

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ION582 DB18158
biotech

Deskripsi belum tersedia.

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IONIS-FGFR4Rx DB16198
biotech | CAS: 1416376-17-4

IONIS-FGFR4Rx is under investigation in clinical trial NCT02476019 (A Safety, Tolerability, PK, and PD Study of Once Weekly ISIS-FGFR4RX SC in Obese Patients).

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IONIS-HBVRx DB16202
biotech | CAS: 1403787-62-1

IONIS-HBVRx is under investigation in clinical trial NCT04544956 (A Mechanistic Study of GSK3228836 With Fine Needle Aspiration (FNA) in Participants With Chronic Hepatitis B).

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Iopamidol Approved DB08947
small molecule | CAS: 60166-93-0

Iopamidol is a contrast agent developed by Bracco with nonionic, low-osmolar properties.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +11
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Iopentol DB13861
small molecule | CAS: 89797-00-2

Iopentol is used as a contrast medium.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +6
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Iophendylate Approved DB01187
small molecule | CAS: 99-79-6

Iophendylate is a mixture of isomers used as contrast medium, mainly for brain and spinal cord visualization. Iophendylate is a myelographic oil-ester (U.S. Patent 2,348,231). Iophendylate, which was never shown to be safe, was initially introduced for use in…

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingContrast Media +6
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Iopodic acid Approved DB09333
small molecule | CAS: 5587-89-3

Iopodic acid, also known by the name of ipodate, is classified as a cholecystographic agent formed by a weak organic acid that contains a tri-iodinated benzene ring with iodine at positions 2, 4 and 6.[A32080] Due to its particular structure, it presents a hi…

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingContrast Media +6
Target Protein:
Thyroxine 5-deiodinase
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small molecule | CAS: 873438-87-0

Deskripsi belum tersedia.

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small molecule | CAS: 873438-88-1

Iopofosine I-131 (NM-404 I-131) is under investigation in clinical trial NCT01495663 (Dose Escalation Study of I-131-CLR1404 in Subjects With Cancer That Does Not Respond to Treatment or Has Returned).

Kategori:
AlcoholsBenzene DerivativesEthers +12
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Iopromide Approved DB09156
small molecule | CAS: 73334-07-3

Iopromide is a low osmolar, non-ionic X-ray contrast agent for intravascular administration. It functions as a contrast agent by opacifying blood vessels in the flow path of the contrast agent, permitting radiographic visualization of the internal structures …

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingContrast Media +8
Waktu ParuhAfter intravenous a…
Vol. DistribusiThe total volume of…
KlirensThe mean total and …
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Iopydol DB13389
small molecule | CAS: 5579-92-0

Deskripsi belum tersedia.

Kategori:
Contrast MediaNon-Watersoluble X-Ray Contrast MediaX-Ray Contrast Media, Iodinated
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small molecule | CAS: 9062-07-1

iota-Carrageenan is under investigation in clinical trial NCT01944631 (Iota-Carrageenan Nasal Spray in Common Cold).

Kategori:
CarbohydratesPolysaccharides
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Iothalamic acid Approved DB09133
small molecule | CAS: 2276-90-6

Iothalamic acid is an iodine containing organic anion used as a diagnostic contrast agent.

Kategori:
Acids, CarbocyclicAlcoholsAmino Sugars +16
Waktu ParuhIn patients with no…
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Iotroxic acid DB08945
small molecule | CAS: 51022-74-3

Iotroxic acid is a contrast medium molecule.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +7
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Ioversol Approved DB09134
small molecule | CAS: 87771-40-2

Ioversol is a non-ionic compound with a tri-iodinated benzene ring used as a contrast dye in diagnostic procedures to visualize different types of organs and tissues.[L41780] Iodine has a high atomic density, which gives it the ability to attenuate X-rays.[L4…

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +11
Waktu ParuhThe elimination hal…
Vol. DistribusiIn adults, the volu…
KlirensIn healthy voluntee…
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IOWH-032 DB12959
small molecule | CAS: 1191252-49-9

Iowh032 has been investigated for the treatment of Cholera, Diarrhea, and Secretory Diarrhea.

Kategori:
Oxazoles
Target Protein:
Cystic fibrosis transmembrane conductance regulator
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Ioxaglic acid Approved DB09313
small molecule | CAS: 59017-64-0

Ioxaglic acid is marketed as Hexabrix. This drug is an ionic tri-iodinated benzoate used as a low-osmolality contrast agent during diagnostic imaging procedures. Like other organic iodine compounds, ioxaglic acid blocks x-rays and is opaque in its appearance …

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu ParuhHexabrix 320 is rap…
Vol. DistribusiIoxaglate salts cro…
Klirens245 ml/kg [L1886]
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Ioxilan Approved DB09135
small molecule | CAS: 107793-72-6

Ioxilan is a tri-iodinated diagnostic contrast agent. Intravascular injection results in opacification of vessels in the path of flow of the contrast medium, permitting radiographic visualization of the internal structures of the human body until significant …

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Acids, CarbocyclicBenzene DerivativesBenzoates +11
Waktu ParuhAn initial fast dis…
Vol. DistribusiIoxilan is distribu…
KlirensThe total clearance…
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Ioxitalamic acid Approved DB13444
small molecule | CAS: 28179-44-4

Ioxitalamate is an ionic iodinated contrast medium.[A27209] It is a first-generation contrast media formed by an ionic monomer with a high osmolarity of 1500-1800 mOsm/kg.[A33006] Ioxitalamic acid in the salt forms of sodium and meglumine was developed by Lie…

Kategori:
Acids, CarbocyclicAlcoholsAmino Sugars +12
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe total clearance…
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IP-2018 DB19049
small molecule | CAS: 881387-68-4

IP-2018 is under investigation in clinical trial NCT04686916 (Clinical Trial Studying the Efficacy and Safety of IP2018 in Depressed, Erectile Dysfunction (ED) Patients).

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IP501 DB06450
small molecule

IP-501 is an investigational antifibrotic compound being tested for the treatment of alcohol-induced liver disease and chronic hepatitis-C-induced cirrhosis. The compound was developed by Indevus Pharmaceuticals.

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Ipafricept DB15045
biotech | CAS: 1391727-24-4

Ipafricept is under investigation in clinical trial NCT01608867 (A Dose Escalation Study of OMP-54F28 in Subjects With Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +10
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Ipamorelin DB12370
small molecule | CAS: 170851-70-4

Ipamorelin has been investigated for the treatment of Ileus.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Growth hormone secretagogue receptor type 1
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Ipatasertib DB11743
small molecule | CAS: 1001264-89-6

Ipatasertib has been used in trials studying the treatment of Cancer, Neoplasms, Solid Cancers, Breast Cancer, and Gastric Cancer, among others.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors +1
Target Protein:
RAC-alpha serine/threonine-protein kinase
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Ipecac Approved DB13293
small molecule | CAS: 8012-96-2

Ipecac is obtained from the plant _Cephaelis ipecacuanha_ and contains a number of emetic alkaloids including emetine and cephaeline.[L2753] Ipecac was approved by Health Canada as an OTC but all those products are now discontinued.[L1113] The FDA does not ha…

Kategori:
Agents Causing Muscle ToxicityAntidotesAutonomic Agents +15
Waktu ParuhThe effect of ipeca…
Vol. DistribusiThe volume of distr…
KlirensThe urinary excreti…
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IPH 1101 DB05754
small molecule

IPH 1101 is a chemically-synthesized structural analog of non-conventional bacterial phosphoantigens which specifically activate the V?9V?2 T cell subset. IPH 1101 is the most advanced drug candidate of the ?? T cell platform

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IPH 2101 DB06049
biotech | CAS: 1000676-42-5

IPH-2101 (NN-1975), a fully human monoclonal antibody developed for patients with acute myeloid leukemia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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IPI-493 DB13023
small molecule | CAS: 64202-81-9

IPI-493 has been used in trials studying the treatment of Advanced Malignancies.

Kategori:
AmidesHSP90 Heat-Shock Proteins, antagonists & inhibitorsLactams +2
Target Protein:
Heat shock protein HSP 90-alpha
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IPI-549 DB16296
small molecule | CAS: 1693758-51-8

IPI-549 is under investigation in clinical trial NCT03795610 (Window of Opportunity Study of IPI-549 in Patients With Locally Advanced HPV+ and HPV- Head and Neck Squamous Cell Carcinoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
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Ipidacrine DB13668
small molecule | CAS: 62732-44-9

Deskripsi belum tersedia.

Kategori:
Anti-Dementia DrugsCholinesterase InhibitorsHeterocyclic Compounds, Fused-Ring +3
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Ipilimumab Approved DB06186
biotech | CAS: 477202-00-9

Ipilimumab is a fully humanized IgG1 monoclonal antibody that blocks cytotoxic T lymphocyte antigen-4 (CTLA-4).[L12126] Blocking CTLA-4 removes an inhibitory signal from reducing the activity of T lymphocytes.[A35065,A35080,L12126] Ipilimumab was developed by…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntibodies +21
Target Protein:
Cytotoxic T-lymphocyte protein 4
Waktu ParuhIpilimumab has a ha…
Vol. DistribusiThe volume of distr…
KlirensIpilimumab has a cl…
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IPL-344 DB16958
small molecule | CAS: 877120-59-7

Deskripsi belum tersedia.

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Ipragliflozin DB11698
small molecule | CAS: 761423-87-4

Ipragliflozin is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsCarbohydrates +6
Target Protein:
Sodium/glucose cotransporter 2
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Ipratropium Approved DB00332
small molecule | CAS: 60205-81-4

Ipratropium is a quaternary ammonium derivative of [atropine][A176957] that acts as an anticholinergic agent.[A176939] It is commonly administered through inhalation which allows producing a local effect without presenting a significant systemic absorption.[A…

Kategori:
Adrenergics, InhalantsAgents producing tachycardiaAgents to Treat Airway Disease +19
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2
Waktu ParuhIpratropium present…
Vol. DistribusiIpratropium has a v…
KlirensThe average clearan…
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Iprazochrome DB13541
small molecule | CAS: 7248-21-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAntidepressive AgentsAntimigraine Preparations +10
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Ipriflavone DB13618
small molecule | CAS: 35212-22-7

Deskripsi belum tersedia.

Kategori:
BenzopyransBone RemodelingChromones +6
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Iprindole DB13496
small molecule | CAS: 5560-72-5

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +14
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Iproniazid DB04818
small molecule | CAS: 54-92-2

Withdrawn from the Canadian market in July 1964 due to interactions with food products containing tyrosine.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +18
Target Protein:
Amine oxidase [flavin-containing] AAmine oxidase [flavin-containing] B
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Iptacopan Approved DB16200
small molecule | CAS: 1644670-37-0

Iptacopan is a small-molecule factor B inhibitor previously investigated as a potential treatment for the rare blood disease paroxysmal nocturnal hemoglobinuria (PNH) by inhibiting the complement factor B.[A262566] Factor B is a positive regulator of the alte…

Kategori:
Acids, CarbocyclicAntineoplastic and Immunomodulating AgentsBenzene Derivatives +8
Target Protein:
Complement factor B
Waktu ParuhThe half-life (t<su…
Vol. DistribusiAfter administratio…
KlirensThe clearance of ip…
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IQP-0528 DB14888
small molecule | CAS: 301297-45-0

IQP-0528 is under investigation in clinical trial NCT03082690 (ImQuest (IQP) DuoGel Phase 1 Pharmacokinetic Study).

Kategori:
Anti-HIV AgentsPyrimidines
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IR-901 DB17932
biotech | CAS: 146446-23-3

Deskripsi belum tersedia.

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IR208 DB05106
biotech

IR208 is a synthetic T-Cell receptor peptide vaccine developed by Immune Response Corporation. It contains three peptides (BV5S2, BV6S5 and BV13S1) expressed by T-Cells in over 90% of MS patients. IR208 is currently undergoing Phase II studies in a 200-p…

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IR501 DB06464
biotech

IR501 (Ravax) is a potential first-in-class vaccine for the treatment of Rheumatoid Arthritis. It specifically targets autoreactive T-cells, reducing their activity. It was last known to be in phase III clinical trials.

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Iratumumab DB05550
biotech | CAS: 640735-09-7

Immunoglobulin G1, anti-(human CD30 (antigen)) (human monoclonal MDX-060 heavy chain), disulfide with human monoclonal MDX-060 light chain, dimer. Molecular weight is approximately 170,000 daltons. In phase I/II clinical trials for treatment of CD30+ lymphoma…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Tumor necrosis factor receptor superfamily member 8
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Irbesartan Approved DB01029
small molecule | CAS: 138402-11-6

Irbesartan is an angiotensin receptor blocker (ARB) indicated to treat hypertension or diabetic nephropathy.[L7456,L7459] It can also be used as part of a combination product with [hydrochlorothiazide] for patients not well controlled or not expected to be we…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin 2 Receptor Blocker +24
Target Protein:
Type-1 angiotensin II receptorTranscription factor Jun
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensTotal plasma cleara…
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Irdabisant DB12900
small molecule | CAS: 1005402-19-6

Irdabisant has been used in trials studying Cognitive Impairment.

Kategori:
Receptors, Histamine H3
Target Protein:
Histamine H3 receptor
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Irinotecan Approved DB00762
small molecule | CAS: 97682-44-5

Irinotecan is a topoisomerase inhibitor used for chemotherapy. It is a water-soluble analogue of [camptothecin], which is extracted from the Chinese tree _Camptotheca acuminate_.[A263376] The bis-piperidine side chain in the structure of irinotecan bestows en…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +29
Target Protein:
DNA topoisomerase I, mitochondrialDNA topoisomerase 1
Gen Terkait:
SLCO1B1 UGT1A1 UGT1A7 +2
Waktu ParuhAfter intravenous i…
Vol. DistribusiFollowing intraveno…
KlirensThe mean (± standar…
Genetik 5 Varian
IRL-1620 DB06138
small molecule | CAS: 142569-99-1

SPI-1620 is an endothelin B receptor agonist. In animal models SPI-1620 selectively and transiently increases tumor blood flow allowing increased delivery of anticancer agents to the tumor. It is being developed as an adjunct to chemotherapy.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
Target Protein:
Endothelin receptor type B
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