Hasil Filter

16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (16004)

Halaman 170 / 321
INCB13739 DB05064
small molecule

INCB13739 is developed as a new treatment for type 2 diabetes. It is an orally available small molecule inhibitor of 11beta-HSD1 (11-beta hydroxysteroid dehydrogenase type 1). 11beta-HSD1 is an enzyme that appears to be critical to the development of type 2…

Kategori:
11-beta-Hydroxysteroid Dehydrogenase Type 1, antagonists & inhibitorsAmidesSulfones +1
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1
Waktu Paruh-
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Genetik -
INCB3284 DB05130
small molecule

INCB3284 is a CCR2 antagonist for Inflammation-driven Diseases.

Kategori:
Acids, CarbocyclicAmidesAmino Acids +3
Target Protein:
C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Inclacumab DB12246
biotech | CAS: 1256258-86-2

Inclacumab has been used in trials studying the treatment and prevention of Myocardial Infarction, Peripheral Arterial Disease (PAD), and Coronary Heart Disease, Graft Occlusion, Vascular.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Inclisiran Approved DB14901
biotech | CAS: 1639324-58-5

Inclisiran is a long-acting, synthetic small interfering RNA (siRNA) directed against proprotein convertase subtilisin-kexin type 9 (PCSK9), which is a serine protease that regulates plasma low-density lipoprotein cholesterol (LDL-C) levels. By binding to PCS…

Kategori:
Antisense Elements (Genetics)Compounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +16
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThere is limited in…
Genetik -
Incyclinide DB11647
small molecule | CAS: 15866-90-7

Incyclinide has been used in trials studying the treatment of HIV Infection, AIDS-related Kaposi Sarcoma, Brain and Central Nervous System Tumors, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Naphthacenes
Target Protein:
72 kDa type IV collagenase
Waktu Paruh-
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Indacaterol Approved DB05039
small molecule | CAS: 312753-06-3

Indacaterol is a novel, ultra-long-acting, rapid onset ?(2)-adrenoceptor agonist developed for Novartis for the once-daily management of asthma and chronic obstructive pulmonary disease. It was approved by the European Medicines Agency (EMA) on 30 November 20…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +17
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhIndacaterol serum c…
Vol. DistribusiAfter intravenous i…
KlirensRenal clearance of …
Genetik -
Indalpine DB08953
small molecule | CAS: 63758-79-2

Indalpine was one of the first selective serotonin reuptake inhibitors to reach the American market. It was initially marketed by Pharmuka. However, after the emergence of widespread concern regarding adverse effects caused by SSRIs, and reported hematologica…

Kategori:
Antidepressive AgentsCentral Nervous System AgentsCentral Nervous System Depressants +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Indanazoline DB13827
small molecule | CAS: 40507-78-6

Deskripsi belum tersedia.

Kategori:
Nasal PreparationsSympathomimetics, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 14Carbonic anhydrase 12 +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Indantadol DB12664
small molecule | CAS: 202844-10-8

Indantadol has been used in trials studying the treatment of Cough and Diabetic Peripheral Neuropathic Pain.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsIndenes +1
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh-
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Genetik -
Indapamide Approved DB00808
small molecule | CAS: 26807-65-8

The most significant modifiable risk factor for cardiovascular disease and the most prominent contributor to all-cause mortality is hypertension.[A204155] Characterized by an office blood pressure of ?140/90, hypertension is pervasive and impacts an estimated…

Kategori:
AmidesAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +26
Target Protein:
Solute carrier family 12 member 3Potassium voltage-gated channel subfamily KQT member 1
Waktu ParuhIndapamide is chara…
Vol. DistribusiSome sources report…
KlirensIndapamide's renal …
Genetik -
Indatraline DB17032
small molecule | CAS: 86939-10-8

Indatraline is a nonselective monoamine reuptake inhibitor.[A253022]

Kategori:
AminesIndenes
Target Protein:
Sodium-dependent dopamine transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1238517-16-2

Indatuximab ravtansine is under investigation in clinical trial NCT01001442 (Safety and Dose Determining Multi-dose Study of BT062 in Patients With Relapsed or Refractory Multiple Myeloma).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Indecainide Approved DB00192
small molecule | CAS: 74517-78-5

Indecainide is a rarely used antidysrhythmic. Indecainide has local anesthetic activity and belongs to the membrane stabilizing (Class 1) group of antiarrhythmic agents; it has electrophysiologic effects characteristic of the IC class of antiarrhythmics.

Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh-
Vol. Distribusi-
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Indeglitazar DB07724
small molecule | CAS: 835619-41-5

Deskripsi belum tersedia.

Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor delta +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Indenolol DB08952
small molecule | CAS: 60607-68-3

Indenolol is a drug of the beta-adrenergic blocker class.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +15
Waktu Paruh-
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Indian frankincense Approved DB14275
biotech

Indian frankincense is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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Indibulin DB06169
small molecule | CAS: 204205-90-3

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAmides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Indigo DB16862
small molecule | CAS: 482-89-3

Deskripsi belum tersedia.

Kategori:
Coloring AgentsCompounds used in a research, industrial, or household settingHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Aryl hydrocarbon receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Indigofera tinctoria leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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Indigotindisulfonic acid Approved DB11577
small molecule | CAS: 483-20-5

Indigotindisulfonic acid is a blue-colored dye with a variety of uses.[A32490,A32491,A32492,L2222] Its salt form, indigotindisulfonate sodium, is also known as indigo carmine, indigotine or FD&C Blue #2. This compound is an acid-base indicator and is used in …

Kategori:
Coloring AgentsCompounds used in a research, industrial, or household settingDiagnostic Agents +5
Target Protein:
Alpha adrenergic receptor
Waktu ParuhIn healthy adults g…
Vol. DistribusiThe volume of distr…
KlirensIn healthy adults g…
Genetik -
Indinavir Approved DB00224
small molecule | CAS: 150378-17-9

A potent and specific HIV protease inhibitor that appears to have good oral bioavailability. [PubChem]

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +33
Target Protein:
Gag-Pol polyproteinPol polyprotein
Waktu Paruh1.8 (± 0.4) …
Vol. Distribusi-
Klirens-
Genetik -
Indiplon DB12590
small molecule | CAS: 325715-02-4

Indiplon has been used in trials studying the treatment of Insomnia and Depression.

Kategori:
BenzazepinesCentral Nervous System AgentsCentral Nervous System Depressants +7
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Indirubin DB12379
small molecule | CAS: 479-41-4

Indirubin is under investigation in clinical trial NCT01735864 (Dosage Determination Trial for Indigo Naturalis Extract in Oil Ointment).

Kategori:
Antibiotics, AntineoplasticAntineoplastic AgentsColoring Agents +4
Target Protein:
Cytochrome P450 1A1Aryl hydrocarbon receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
AminesHeterocyclic Compounds, Fused-RingHydroxylamines
Target Protein:
Cyclin-dependent kinase 5 activator 1Cyclin-dependent kinase 2Aryl hydrocarbon receptor +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 244021-67-8

Deskripsi belum tersedia.

Target Protein:
Glycogen phosphorylase, muscle formCell division control protein 2 homolog
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Indisulam DB06370
small molecule | CAS: 165668-41-7

Deskripsi belum tersedia.

Kategori:
AmidesAntineoplastic AgentsCarbonic Anhydrase Inhibitors +15
Target Protein:
Carbonic anhydrase 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Indium DB11659
small molecule | CAS: 7440-74-6

Indium has been used in trials studying the basic science of Clear Cell Renal Cell Carcinoma.

Kategori:
AnionsElectrolytesElements +5
Waktu Paruh-
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Genetik -
small molecule | CAS: 131391-70-3

Deskripsi belum tersedia.

Waktu Paruh-
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Indium In-111 DB11916
small molecule | CAS: 15750-15-9

Indium In-111 is under investigation in clinical trial NCT00493454 (Ibritumomab Tiuxetan for Treatment of Non-Follicular CD20+ Indolent Lymphomas).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 156586-92-4

Deskripsi belum tersedia.

Waktu Paruh-
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Indium In-111 chloride Approved DB09490
small molecule | CAS: 50800-85-6

Indium In-111 Chloride is a diagnostic radiopharmaceutical agent intended for radiolabeling OncoScint (satumomab pendetide) or ProstaScint (capromab pendetide) used for _in vivo_ diagnostic imaging procedures and for radiolabeling Zevalin (ibritumomab tiuxeta…

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu Paruh2.8 days
Vol. DistribusiIndium In-111 Chlor…
KlirensIndium In-111 Chlor…
Genetik -
biotech | CAS: 138661-00-4

Indium In-111 imciromab pentetate is a mouse monoclonal antibody labelled with the radioisotope Indium-111 which was used for cardiac imaging under the trade name Myoscint, but was withdrawn in 1993.

Kategori:
Diagnostic Radiopharmaceuticals
Waktu Paruh-
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Indium In-111 oxyquinoline Approved DB09473
small molecule | CAS: 65389-08-4

Indium In 111 oxyquinoline (oxine) is a diagnostic radiopharmaceutical intended for radiolabeling of autologous leukocytes. It is composed of a 3:1 saturated complex of In-111 isotope and oxyquinoline. Indium-111 decays by isomeric transition and electron ca…

Kategori:
Radioactive Diagnostic AgentRadiopharmaceutical Activity
Waktu ParuhIndium In 111 decay…
Vol. Distribusi-
KlirensClearance from whol…
Genetik -
Indium In-111 pentetate Approved DB09425
small molecule | CAS: 135998-32-2

Indium In-111 pentetate disodium is a radioactive diagnostic indicated for use in radionuclide cisternography. Decay of In-111 by electron capture allows for detection with a gamma camera for visualization of the brain and spinal column.

Kategori:
Central Nervous SystemDiagnostic RadiopharmaceuticalsRadioactive Diagnostic Agent +1
Waktu ParuhIndium 111 decays b…
Vol. Distribusi-
Klirens-
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Indium In-111 pentetreotide Approved DB11835
small molecule | CAS: 139096-04-1

Indium In 111 pentetreotide (Octreoscan) has been used in trials studying the diagnostic of SARCOIDOSIS, Solid Tumors, and cushing syndrome.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic RadiopharmaceuticalsHormones +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 138955-27-8

Tumor associated glycoprotein (TAG) 72 (B72.3) monoclonal antibody conjugated with Indium 111 for radioimaging colon tumors. Satumomab Pendetide (trade name: OncoScint®) is no longer commercially available.

Kategori:
AcetatesAcids, AcyclicAmines +14
Target Protein:
Tumor-associated glycoprotein 72 (TAG-72)
Waktu Paruh0.8 hours (mammalia…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 139096-04-1

Deskripsi belum tersedia.

Kategori:
Radioactive Diagnostic Agent
Waktu Paruh-
Vol. Distribusi-
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Indobufen DB12545
small molecule | CAS: 63610-08-2

Indobufen has been used in trials studying the supportive care and prevention of Atrial Fibrillation.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Indocyanine green Approved DB16024
small molecule | CAS: 3599-32-4

Deskripsi belum tersedia.

Kategori:
Cardiac FunctionColoring AgentsCompounds used in a research, industrial, or household setting +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Indocyanine green acid form Approved DB09374
small molecule | CAS: 28782-33-4

Indocyanine Green is a water soluble, tricarbocyanine dye with a peak spectral absorption at 800 nm. The chemical name for Indocyanine Green is 1 H-Benz[e]indolium, 2-[7-[1,3-dihydro-1,1-dimethyl-3-(4-sulfobutyl)-2H-benz[e] indol-2-ylidene]-1,3,5-heptatrienyl…

Kategori:
BSEP/ABCB11 SubstratesCardiac FunctionColoring Agents +6
Waktu ParuhICG has a half-life…
Vol. DistribusiICG distribution in…
KlirensClearance of dyes w…
Genetik -
Indole DB04532
small molecule | CAS: 120-72-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
EndolysinNicotinate-nucleotide--dimethylbenzimidazole phosphoribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 700-06-1

Indole 3 Carbinol is under investigation in clinical trial NCT00033345 (Indole-3-Carbinol in Preventing Breast Cancer in Nonsmoking Women Who Are at High Risk For Breast Cancer).

Kategori:
Anticarcinogenic AgentsAntineoplastic AgentsCompounds used in a research, industrial, or household setting +2
Target Protein:
NF-kappa-B inhibitor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydratesCompounds used in a research, industrial, or household setting +8
Target Protein:
Tryptophan synthase alpha chainTryptophan synthase beta chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Tryptophan synthase alpha chainTryptophan synthase beta chainTryptophan synthase alpha chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Indoleacetamide DB08652
small molecule | CAS: 879-37-8

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Target Protein:
Aralkylamine dehydrogenase light chainAralkylamine dehydrogenase heavy chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 87-51-4

Deskripsi belum tersedia.

Kategori:
Growth SubstancesHeterocyclic Compounds, Fused-RingIndoles +1
Target Protein:
Group IIE secretory phospholipase A2S-phase kinase-associated protein 1Kynurenine--oxoglutarate transaminase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 830-96-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
Group IIE secretory phospholipase A2Aspartate aminotransferaseAromatic-amino-acid aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Indomethacin Approved DB00328
small molecule | CAS: 53-86-1

Indometacin, or indomethacin, is a non-steroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic, and antipyretic properties. NSAIDs consist of agents that are structurally unrelated; the NSAID chemical classification of indometacin is an ind…

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +49
Target Protein:
Prostaglandin G/H synthase 2Phospholipase A2, membrane associatedHuman Cyclooxygenases +8
Waktu ParuhIndometacin disposi…
Vol. DistribusiThe volume of distr…
KlirensIn a clinical pharm…
Genetik -
Indopan DB01446
small molecule | CAS: 299-26-3

Indopan (alpha-methyltryptamine) is a stimulant and psychoactive drug which produces effects similar to 3,4-methylenedioxy-N-methylamphetamine (MDMA), despite being structurally dissimilar. It was developed in the 1960's by Upjohn with the intention for use a…

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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