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Halaman 17 / 46
Estradiol acetate Approved DB13952
small molecule | CAS: 4245-41-4

Estradiol acetate is a pro-drug ester of [DB00783], a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex hormone. As a pro-dru…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +24
Target Protein:
Estrogen receptorEstrogen receptor betaNuclear receptor subfamily 1 group I member 2 +7
Waktu Paruh-
Vol. DistribusiThe distribution of…
Klirens-
Genetik -
Estradiol benzoate Approved DB13953
small molecule | CAS: 50-50-0

Estradiol Benzoate is a pro-drug ester of [DB00783], a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex hormone. As a pro-dr…

Kategori:
Adrenal Cortex HormonesBCRP/ABCG2 InhibitorsContraceptive Agents, Hormonal +35
Target Protein:
Estrogen receptorEstrogen receptor betaNuclear receptor subfamily 1 group I member 2 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Estradiol cypionate Approved DB13954
small molecule | CAS: 313-06-4

Estradiol Cypionate is a pro-drug ester of [DB00783], a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex hormone. As a pro-d…

Kategori:
Adrenal Cortex HormonesBCRP/ABCG2 InhibitorsContraceptive Agents, Female +38
Target Protein:
Estrogen receptorEstrogen receptor betaNuclear receptor subfamily 1 group I member 2 +7
Waktu Paruh-
Vol. DistribusiThe distribution of…
Klirens-
Genetik -
Estradiol dienanthate Approved DB13955
small molecule | CAS: 7732-97-0

Estradiol Dienanthate is a pro-drug ester of [DB00783], a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex hormone. As a pro…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +31
Target Protein:
Estrogen receptorEstrogen receptor betaNuclear receptor subfamily 1 group I member 2 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Estradiol valerate Approved DB13956
small molecule | CAS: 979-32-8

Estradiol Valerate (also known as E2V) is a pro-drug ester of [DB00783], a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex …

Kategori:
Adrenal Cortex HormonesBCRP/ABCG2 InhibitorsContraceptive Agents, Female +38
Target Protein:
Estrogen receptorEstrogen receptor betaNuclear receptor subfamily 1 group I member 2 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eszopiclone Approved DB00402
small molecule | CAS: 138729-47-2

Eszopiclone, marketed by Sepracor under the brand-name Lunesta, is a nonbenzodiazepine hypnotic drug used to treat insomnia. It is the active stereoisomer of zopiclone, belonging to the class of drugs known as _cyclopyrrolones_.[A179638,L6850] Cyclopyrrolone …

Kategori:
Benzodiazepine hypnotics and sedativesCentral Nervous System AgentsCentral Nervous System Depressants +18
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Translocator proteinGABA(A) Receptor +3
Waktu ParuhThe half-life is 6.…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Etafedrine Approved DB11587
small molecule | CAS: 48141-64-6

Etafedrine (INN) or ethylephedrine is a long-acting bronchodilator and has been an ingredient combined with other drugs in the brand names Nethaprin [A32757] and Dalmacol [L2568]. It was previously available as both the free base and as the hydrochloride salt…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +10
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhIt has a plasma hal…
Vol. DistribusiSimilar to ephedrin…
Klirens-
Genetik -
Etanercept Approved DB00005
biotech | CAS: 185243-69-0

Dimeric fusion protein consisting of the extracellular ligand-binding portion of the human 75 kilodalton (p75) tumor necrosis factor receptor (TNFR) linked to the Fc portion of human IgG1.[L14862,A216522] The Fc component of etanercept contains the CH2 domain…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAnti-Inflammatory Agents +18
Target Protein:
Tumor necrosis factorLymphotoxin-alphaHigh affinity immunoglobulin gamma Fc receptor I +6
Waktu ParuhEtanercept has a me…
Vol. DistribusiPopulation pharmaco…
KlirensEtanercept has a me…
Genetik -
Etesevimab DB15897
biotech | CAS: 2423948-94-9

Etesevimab (LY-CoV016, also known as JS016) is a fully human and recombinant monoclonal antibody that targets the SARS-CoV-2 surface spike protein receptor binding domain.[L16651,L16661] Under the EUA granted in February 2021, etesevimab is used in combinatio…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etevritamab DB17211
biotech | CAS: 2329692-74-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethinamate Approved DB01031
small molecule | CAS: 126-52-3

Ethinamate is a short-acting sedative-hypnotic medication used to treat insomnia. Like many such similar medications, the regular use of ethinamate can result in the development of drug tolerance in a patient. Nevertheless, the medication itself is generally …

Kategori:
Acids, Acyclic
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 1
Waktu Paruh2.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Ethylenediamine Approved DB14189
small molecule | CAS: 107-15-3

Ethylenediamine is an organic compound that is used as a building block for the production of many other chemical products. It is also used as an excipient in many pharmacological preparations such as creams. Notably, ethylenediamine is a contact sensitizer c…

Kategori:
AllergensAminesAntigens +6
Target Protein:
Dihydropteroate synthase
Waktu ParuhEthylenediamine has…
Vol. DistribusiVd = 0.133 l/kg [A3…
Klirens-
Genetik -
Etigilimab DB18854
biotech | CAS: 2044984-83-8

Etigilimab is under investigation in clinical trial NCT04761198 (A Study of Etigilimab and Nivolumab in Subjects With Locally Advanced or Metastatic Tumors.).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etranacogene dezaparvovec Approved DB16791
biotech | CAS: 2156583-26-3

Hemophilia B - also called factor IX deficiency or Christmas disease - is an X-linked genetic disorder resulting in an absence or deficiency of clotting factor IX.[L44176] Clotting factors, including factor IX, are necessary components of the signaling cascad…

Kategori:
Adeno-associated Viral Vector TherapiesBlood and Blood Forming OrgansBlood Coagulation Factors +2
Target Protein:
Coagulation factor IX
Waktu Paruh-
Vol. DistribusiIn a study to evalu…
KlirensIn a clinical study…
Genetik -
Etravirine Approved DB06414
small molecule | CAS: 269055-15-4

Etravirine is an antiretroviral agent more specifically classified as a Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI). Etraverine is used clinically for the treatment of human immunodeficiency virus type 1 (HIV-1) infection. On January 18, 2007, the …

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiinfectives for Systemic Use +24
Target Protein:
Gag-Pol polyproteinGag-Pol polyproteinReverse transcriptase/RNaseH
Waktu ParuhHalf life of 9.05-4…
Vol. DistribusiDistribution of etr…
KlirensRenal clearance of …
Genetik -
Etrolizumab DB12189
biotech | CAS: 1044758-60-2

Inflammatory bowel disease (IBD), including ulcerative colitis and Crohn's disease, is typified by a chronic gastrointestinal inflammatory microenvironment, driven in part by the excessive infiltration and retention of intestinal-homing lymphocytes.[A244564, …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Integrin beta-7
Waktu ParuhEtrolizumab adminis…
Vol. DistribusiModelling of etroli…
KlirensEtrolizumab has a m…
Genetik -
Eucalyptol DB03852
small molecule | CAS: 470-82-6

Eucalyptol is naturally produced cyclic ether and monoterpenoid. Eucalyptol is an ingredient in many brands of mouthwash and cough suppressant. It controls airway mucus hypersecretion and asthma via anti-inflammatory cytokine inhibition. Eucalyptol is an effe…

Kategori:
AgrochemicalsAlcoholsAnti-Infective Agents +29
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eucalyptus globulus leaf Approved DB14320
biotech

Eucalyptus globulus leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eucalyptus oil Approved DB11114
biotech | CAS: 8000-48-4

Eucalyptus oil is a distilled oil derived from the leaves of the tree Eucalyptus. It is shown to be effective in reducing pain, swelling, and inflammation via its modulatory effect on the immune response. It is also shown to exhibit antibacterial activity aga…

Kategori:
Biological ProductsComplex MixturesDrugs that are Mainly Renally Excreted +6
Waktu ParuhStudies have determ…
Vol. DistribusiStudies have determ…
KlirensStudies have determ…
Genetik -
Evalstotug DB19410
biotech | CAS: 2460399-39-5

Evalstotug is under investigation in clinical trial NCT05271604 (A Phase 2 Open Label Study of BA3021 in Patients With Recurrent or Metastatic Squamous Cell Carcinoma of the Head and Neck).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 308064-97-3

Evening primrose oil comes from the extraction from _Oenothera biennis_ seeds and it is commonly used as an alternative source for omega-6 essential fatty acids. In its composition it presents some fatty acids such as [DB00132] and [DB13854].[A33131] Evening …

Kategori:
Agents that reduce seizure thresholdAngiospermsAnti-Inflammatory Agents +26
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Evinacumab Approved DB15354
biotech | CAS: 1446419-85-7

Evinacumab is a recombinant human IgG4 monoclonal antibody targeted against angiopoietin-like protein 3 (ANGPTL3) and the first drug of its kind. The ANGPTL family of proteins serve a number of physiologic functions - including involvement in the regulation o…

Kategori:
Amino Acids, Peptides, and ProteinsAngiopoietin-like 3 InhibitorAngiopoietin-like 3 Inhibitors +8
Target Protein:
Angiopoietin-related protein 3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Evolocumab Approved DB09303
biotech | CAS: 1256937-27-5

Evolocumab is a monoclonal antibody designed for the treatment of hyperlipidemia by Amgen. It is a subcutaneous injection approved by the FDA for individuals on maximum statin therapy who still require additional LDL-cholesterol lowering. It is approved for b…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu Paruh-
Vol. Distribusi-
KlirensEvolocumab showed n…
Genetik -
Evorpacept DB17573
biotech | CAS: 2484949-51-9

evorpacept is under investigation in clinical trial NCT04755244 (A Study of Evorpacept (ALX148) With Venetoclax and Azacitidine for Acute Myeloid Leukemia (ASPEN-05)).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Holoclar (_ex vivo_ expanded autologous human corneal epithelial cells containing stem cells) is a stem cell therapy used to treat limbal stem cell deficiencies.[L48375]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exagamglogene autotemcel Approved DB15572
biotech

Sickle cell disease (SCD) is a genetic disorder characterized by the production of abnormal sickle-shaped red blood cells (called hemoglobin S, HbS) that initiate a pathophysiology resulting in severe pain, progressive multi-organ damage, and premature death.…

Kategori:
Autologous Cultured CellBlood and Blood Forming Organs
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exbivirumab DB17747
biotech | CAS: 569658-80-6

Exbivirumab is an investigational monoclonal antibody. It is one of the active ingredients in HepeX-B, a drug product containing two human monoclonal antibodies to the hepatitis B virus (HBV) surface antigen.[A259202]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exemestane Approved DB00990
small molecule | CAS: 107868-30-4

Exemestane is an oral steroidal aromatase inhibitor used in the adjuvant treatment of hormonally-responsive (also called hormone-receptor-positive, estrogen-responsive) breast cancer in postmenopausal women. It irreversibly binds to the active site of the enz…

Kategori:
AndrostanesAndrostenesAntineoplastic Agents +14
Target Protein:
Aromatase
Waktu Paruh24 hours
Vol. Distribusi-
Klirens-
Genetik -
Exidavnemab DB19452
biotech | CAS: 2438229-02-6

Exidavnemab is under investigation in clinical trial NCT06671938 (Safety, Tolerability, and Pharmacokinetics of Exidavnemab in Patients With Parkinson's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exlinkibart DB17474
biotech | CAS: 2642171-64-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EXOB-001 DB18257
biotech

EXOB-001 consists of extracellular vesicles derived from cultured human umbilical cord mesenchymal stromal cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ezabenlimab DB17483
biotech | CAS: 2249882-54-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ezatiostat DB05460
small molecule | CAS: 168682-53-9

Ezatiostat is investigated in clinical trials for treating myelodysplastic syndrome. This compound belongs to the peptides. These are compounds containing an amide derived from two or more amino carboxylic acid molecules (the same or different) by formation o…

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Glutathione S-transferase P
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ezetimibe Approved DB00973
small molecule | CAS: 163222-33-1

Ezetimibe is a lipid-lowering compound that inhibits intestinal cholesterol and phytosterol absorption. The discovery and research of this drug began in the early 1990s, after the intravenous administration of radiolabelled ezetimibe in rats revealed that it …

Kategori:
Anticholesteremic AgentsAzetinesBCRP/ABCG2 Substrates +20
Target Protein:
NPC1-like intracellular cholesterol transporter 1Sterol O-acyltransferase 1Aminopeptidase N
Waktu ParuhBoth ezetimibe and …
Vol. DistribusiThe relative volume…
KlirensThere are no pharma…
Genetik -
Factor IX Complex (Human) Approved DB11330
biotech | CAS: 37224-63-8

Factor IX Complex is a sterile, lyophilized concentrate composed of a number of Vitamin K-dependent clotting factors found in functioning human plasma. Also known as prothrombin complex concentrate, products containing this complex often include Factor IX (an…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Factor XIII (human) Approved DB12909
biotech | CAS: 9013-56-3

Factor XIII (human) is a heat-treated, lyophilized concentrate of coagulation factor XIII, an endogenous enzyme responsible for the crosslinking of fibrin and an essential component of the coagulation cascade [FDA Label]. For people with congenital deficiency…

Kategori:
AcyltransferasesAmino Acids, Peptides, and ProteinsAminoacyltransferases +14
Waktu Paruh6.6 ±2.29 days [FDA…
Vol. DistribusiVss = 51.1 mL/kg (v…
Klirens0.25 ±0.09 mL/hr/kg…
Genetik -
Fallypride DB15167
small molecule | CAS: 166173-78-0

Fallypride is under investigation in clinical trial NCT02310360 (Striatal and Extra-striatal Dopamine Release in Response to Food in Healthy Humans).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Faricimab Approved DB15303
biotech | CAS: 1607793-29-2

Retinal vascular diseases (RVDs) such as diabetic macular edema (DME), age-related macular degeneration (AMD), and retinal vein occlusion (RVO) are typically caused by retinal ischemia and subsequent neovascularization (NV).[A225985, A225990, A225995] Vascula…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Target Protein:
Vascular endothelial growth factor A, long formAngiopoietin-2
Waktu ParuhFaricimab has an es…
Vol. Distribusi-
Klirens-
Genetik -
Farletuzumab DB05595
biotech | CAS: 896723-44-7

Farletuzumab (MORAb-003) is a fully humanized monoclonal antibody against the folate receptor alpha, for the potential treatment of epithelial ovarian cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Target Protein:
Folate receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fasinumab DB12157
biotech | CAS: 1190239-42-9

Fasinumab is a human IgG1k monoclonal antibody targeted against nerve growth factor (NGF). It is currently under investigation for the treatment osteoarthritic pain[A241045] and has demonstrated significantly greater pain relief and functional improvement as …

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +11
Target Protein:
Beta-nerve growth factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fazpilodemab DB18924
biotech | CAS: 2517935-02-1

Fazpilodemab is under investigation in clinical trial NCT04171765 (A Study to Evaluate the Efficacy, Safety, and Pharmacokinetics of BFKB8488A Compared With Placebo in Participants With Non-alcoholic Steatohepatitis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FB-825 DB17598
biotech

FB-825 is an investigational humanized monoclonal antibody that targets the C?mX domain of the membrane-bound IgE (mIgE), causing a depletion of mIgE positive B-cells. It is currently being investigated for immune disorders, such as atopic dermatitis and hype…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FBX-101 DB18340
biotech

FBX-101 is an adeno-associated virus serotype rhesus 10 vector expressing the human galactocerebrosidase (GALC) gene

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FCX-013 DB18218
biotech

FCX-013 consists of human dermal fibroblasts genetically modified with a lentiviral vector expressing metalloproteinase-1 (MMP-1).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Febuxostat Approved DB04854
small molecule | CAS: 144060-53-7

Febuxostat is a non-purine xanthine oxidase (XO) inhibitor.[A39743] In early 2008, febuxostat was granted marketing authorization by the European Commission for the treatment of chronic hyperuricemia and gout.[A230548] In the following year, the FDA for appro…

Kategori:
Antigout PreparationsAntirheumatic AgentsBCRP/ABCG2 Inhibitors +15
Target Protein:
Xanthine dehydrogenase/oxidase
Waktu ParuhThe apparent mean t…
Vol. DistribusiThe apparent steady…
KlirensFollowing oral admi…
Genetik -
Fecal microbiota Approved DB17743
biotech

Fecal microbiota, given either as a rectal transplant or in an oral formulation of live spores, is an FDA-approved option to prevent the recurrence of _Clostridioides difficile_ infection (CDI) in patients given an antibacterial treatment for recurrent CDI.[A…

Kategori:
Miscellaneous Therapeutic Agents
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Fenfluramine Approved DB00574
small molecule | CAS: 458-24-2

Dravet syndrome is a pediatric encephalopathy that typically manifests within the first year of life following exposure to elevated temperatures. It is characterized by recurrent pharmacoresistant seizures, which increase in frequency and severity with diseas…

Kategori:
Alimentary Tract and MetabolismAminesAnticonvulsants +27
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 2C +4
Waktu ParuhFenfluramine has an…
Vol. DistribusiFenfluramine has an…
KlirensFenfluramine has a …
Genetik -
Fenobam DB12931
small molecule | CAS: 57653-26-6

Fenobam is under investigation in clinical trial NCT00637221 (Open Label Study Investigating Safety and Efficacy of Fenobam anhydrous 50 mg - 150 mg on Prepulse Inhibition Tests and Continuous Performance Tasks, Adults With Fragile X Syndrome).

Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenproporex DB01550
small molecule | CAS: 16397-28-7

Fenproporex is an orally active stimulant drug, which was developed in the 1960s. It is used as an appetite suppressant and a treatment for obesity. It is listed as an illicit substance in many countries due to addiction issues and listed as a prohibited subs…

Kategori:
AminesDrugs that are Mainly Renally ExcretedEthylamines +2
Waktu Paruh-
Vol. Distribusi-
KlirensThe amphetamine met…
Genetik -
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