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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

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Hasil Pencarian (11778)

Halaman 169 / 236
small molecule

Deskripsi belum tersedia.

Target Protein:
Lactose operon repressor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Orticumab DB16653
biotech | CAS: 1314241-10-5

Orticumab is under investigation in clinical trial NCT04776629 (A Proof-of-activity Study With Orticumab in Subjects With Psoriasis and Cardiometabolic Risk Factors).

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Genetik -
biotech

Deskripsi belum tersedia.

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Orvepitant DB12427
small molecule | CAS: 579475-18-6

Orvepitant has been used in trials studying the treatment of Depressive Disorder, Depressive Disorder, Major, Post-Traumatic Stress Disorder, and Posttraumatic Stress Disorder (PTSD).

Kategori:
Antidepressive AgentsCentral Nervous System Depressants
Target Protein:
Substance-P receptor
Waktu Paruh-
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Genetik -
Oryctolagus cuniculus skin Approved DB10607
biotech

Oryctolagus cuniculus skin or pelt is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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OS2966 DB17207
biotech

OS2966 is a humanized integrin ?1 (CD29) blocking antibody currently evaluated for the treatment of acute myeloid leukemia, glioblastoma and ovarian cancer.[A254561, L47351]

Waktu Paruh-
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Osalmid DB16273
small molecule | CAS: 526-18-1

Osalmid is under investigation in clinical trial NCT03670173 (Safety and Efficacy Assessments of Osalmid in Multiple Myeloma).

Waktu Paruh-
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Osanetant DB04872
small molecule | CAS: 160492-56-8

Developed by Sanofi-Aventis (formerly Sanofi-Synthelabo), osanetant (SR-142801) is an NK3 receptor antagonist which was under development for the treatment of schizophrenia and other Central Nervous System (CNS) disorders. In a review of its R&D portfolio, th…

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +3
Target Protein:
Neuromedin-K receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osbond acid DB14088
small molecule | CAS: 25182-74-5

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Waktu Paruh-
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OSE-2101 DB17122
biotech

Deskripsi belum tersedia.

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Oseltamivir Approved DB00198
small molecule | CAS: 196618-13-0

Oseltamivir (marketed as the product Tamiflu?), is an antiviral neuraminidase inhibitor used for the treatment and prophylaxis of infection with influenza viruses A (including pandemic H1N1) and B. Oseltamivir exerts its antiviral activity by inhibiting the a…

Kategori:
AcetamidesAcetatesAmides +8
Target Protein:
NeuraminidaseSialidase-1Sialidase-2
Waktu ParuhPlasma concentratio…
Vol. DistribusiThe mean volume of …
KlirensRenal clearance (18…
Genetik -
small molecule | CAS: 187227-45-8

Deskripsi belum tersedia.

Kategori:
AcetamidesAcetatesAcids, Acyclic +8
Target Protein:
Neuraminidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSI-027 DB12387
small molecule | CAS: 936890-98-1

OSI-027 has been used in trials studying the treatment of Any Solid Tumor or Lymphoma.

Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
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OSI-7836 DB05837
small molecule

OSI-7836 is a member of the nucleoside class of cytotoxic drugs of which gemcitabine is the market leader. OSI Pharmaceuticals develops OSI-7836 as a next-generation gemcitabine. The anti-tumor activity of OSI-7836 appeares to be less schedule dependent than …

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosides
Waktu Paruh-
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OSI-7904L DB05457
small molecule

OSI-7904L is a liposome encapsulated thymidylate synthase inhibitor, which is indicated for use in advanced gastric and/or gastroesophageal adenocarcinoma (A-G/GEJA). Current treatments also inhibit thymidylate synthase but the innovative lipid coating of OSI…

Kategori:
Acids, AcyclicDicarboxylic AcidsHeterocyclic Compounds, Fused-Ring
Target Protein:
Thymidylate synthase
Waktu Paruh-
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OSI-930 DB05913
small molecule | CAS: 728033-96-3

OSI-930 is an orally active inhibitor of two clinically validated targets: c-Kit and the vascular endothelial growth factor receptor-2 (VEGFR-2). OSI-930 is designed to target both cancer cell proliferation and blood vessel growth (angiogenesis) in selected t…

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Vascular endothelial growth factor receptor 2Mast/stem cell growth factor receptor KitVascular endothelial growth factor receptor 1
Waktu Paruh-
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Osilodrostat Approved DB11837
small molecule | CAS: 928134-65-0

Osilodrostat is an inhibitor of 11?-hydroxylase (also referred to as CYP11B1), the enzyme that catalyzes the final step in the biosynthesis of endogenous cortisol.[L12123] It is used to lower circulating cortisol levels in the treatment of Cushing's disease, …

Kategori:
Antiadrenal PreparationsAnticorticosteroidsCortisol Synthesis Inhibitors +32
Target Protein:
Cytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial
Waktu ParuhThe elimination hal…
Vol. DistribusiThe median apparent…
KlirensData regarding the …
Genetik -
Osimertinib Approved DB09330
small molecule | CAS: 1421373-65-0

Osimertinib is an oral, third-generation epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI) drug developed by AstraZeneca Pharmaceuticals.[A7926,L43453] Its use is indicated for the treatment of metastatic non-small cell lung cancer (NSCL…

Kategori:
Acids, AcyclicAcrylatesAmides +29
Target Protein:
Epidermal growth factor receptor
Waktu ParuhThe population esti…
Vol. DistribusiThe mean volume of …
KlirensOral clearance is 1…
Genetik -
Osivelotor DB18071
small molecule | CAS: 2417955-18-9

Deskripsi belum tersedia.

Waktu Paruh-
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Osocimab DB14818
biotech | CAS: 2056878-75-0

Osocimab is under investigation in clinical trial NCT03276143 (Factor XIa inhibition for the prevention of venous Thromboembolism in Patients Undergoing Total Knee Arthroplasty).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Osoresnontrine DB16274
small molecule | CAS: 1189767-28-9

Osoresnontrine is under investigation in clinical trial NCT02281773 (A Study to Investigate the Efficacy, Safety and Tolerability of Four Different Doses of BI 409306 Compared to Placebo Given for 12 Weeks in Patients With Schizophrenia on Stable Antipsychoti…

Kategori:
Enzyme InhibitorsPhosphodiesterase Inhibitors
Target Protein:
High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A
Waktu Paruh-
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Ospemifene Approved DB04938
small molecule | CAS: 128607-22-7

Ospemifene is a new selective non-hormonal estrogen receptor modulator (SERM) that is used for the treatment of moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause. FDA approved on February 26, 2013.

Kategori:
Benzene DerivativesBenzylidene CompoundsCytochrome P-450 CYP2B6 Substrates +14
Target Protein:
Estrogen receptor
Waktu ParuhTerminal half-life …
Vol. Distribusi448 L
KlirensTotal body clearanc…
Genetik -
OSSM-007 DB18553
biotech

OSSM-007 consists of interferon-gamma primed allogeneic mesenchymal stem cells.

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Ostabolin-C DB05536
small molecule | CAS: 188899-65-2

Ostabolin C was under investigation in clinical trial NCT00787358 (A Proof-of-Concept Study Investigating the Safety and Efficacy of ZT-031 on Hip Fracture Healing in Men and Postmenopausal Women (SHIFT)).

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +3
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OSU-6162 DB19178
small molecule | CAS: 146798-66-5

OSU-6162 is under investigation in clinical trial NCT05641623 (OSU6162 as Add-on in Ssri/snri-resistant Depression).

Kategori:
Dopamine AgentsDopamine AntagonistsDopamine D2 Receptor Antagonists +2
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Osugacestat DB12006
small molecule | CAS: 1401066-79-2

Osugacestat (BMS-906024) has been used in trials studying the treatment of Cancer, Lymphoblastic Leukemia, Acute T-cell, and Precursor T-Cell Lymphoblastic Lymphoma.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
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OT-004 DB18276
biotech

Deskripsi belum tersedia.

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OT-15 DB17950
biotech

Deskripsi belum tersedia.

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OT-551 DB05650
small molecule | CAS: 627085-11-4

OT-551 is a novel small molecule that is topically dosed in an eye drop and has the unique ability to penetrate cell membranes and reach both the front and the back of the eye. It is intended to treat Age-related macular Degeneration (AMD), and preclinical re…

Target Protein:
Nuclear factor erythroid 2-related factor 2
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OT-730 DB16112
small molecule | CAS: 870809-51-1

OT-730 is under investigation in clinical trial NCT00753168 (Phase 1-2 Evaluation of OT-730 Eye Drops in Reducing the Intraocular Pressure in Patients With Ocular Hypertension or Open-angle Glaucoma).

Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
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Otamixaban DB06635
small molecule | CAS: 193153-04-7

Otamixaban is a novel direct Factor Xa (FXa) inhibitor. It is currently being developed by the French pharmaceutical company Sanofi-Aventis as a treatment for acute coronary syndrome.

Kategori:
AnticoagulantsAntithrombinsEnzyme Inhibitors +4
Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Otenabant DB11745
small molecule | CAS: 686344-29-6

Otenabant has been investigated for the treatment of Obesity.

Kategori:
Cannabinoid Receptor AntagonistsCannabinoids and similarsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
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Genetik -
Oteracil Approved DB03209
small molecule | CAS: 937-13-3

Oteracil is an adjunct to antineoplastic therapy, used to reduce the toxic side effects associated with chemotherapy. Approved by the European Medicines Agency (EMA) in March 2011, Oteracil is available in combination with [DB09257] and [DB09256] within the c…

Kategori:
Triazines
Waktu ParuhFollowing a single …
Vol. DistribusiAlthough no intrave…
Klirens-
Genetik -
Oteseconazole Approved DB13055
small molecule | CAS: 1340593-59-0

Oteseconazole is an azole metalloenzyme inhibitor that targets fungal CYP51.[L41635] CYP51, also known as 14? demethylase, participates in the formation of ergosterol, a compound that plays a vital role in the integrity of cell membranes.[L41635,A247020] By b…

Kategori:
14-alpha Demethylase InhibitorsAntifungal AgentsAntiinfectives for Systemic Use +5
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhThe median terminal…
Vol. DistribusiOn average, the vol…
KlirensClinical phase I st…
Genetik -
OTL-103 DB17593
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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OTL-201 DB17652
biotech

OTL-201 is an investigational hematopoietic stem cell (HSC) gene therapy being developed by Orchard Therapeutics for the treatment of mucopolysaccharidosis type IIIA (MPS-IIIA). It consists of a lentiviral vector to insert a functional copy of the human N-Sul…

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Otlertuzumab DB16275
biotech | CAS: 1372645-37-8

Otlertuzumab is under investigation in clinical trial NCT01188681 (Safety and Efficacy Study of TRU-016 Plus Bendamustine vs. Bendamustine in Relapsed Chronic Lymphocytic Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Leukocyte antigen CD37
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OTX-2002 DB17246
biotech

OTX-2002 is a bicistronic messenger ribonucleic acid (mRNA) encoding for ZF-DNMT and ZF-KRAB proteins, encapsulated in a lipid nanoparticle (LNP).

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Ovatodiolide DB19264
small molecule | CAS: 3484-37-5

Ovatodiolide is under investigation in clinical trial NCT04220411 (A Study for AR100DP1 in Mild to Moderate Atopic Dermatitis (AD)).

Kategori:
Terpenes
Waktu Paruh-
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Ovemotide DB19156
biotech | CAS: 181477-91-8

Ovemotide is under investigation in clinical trial NCT00357461 (Ipilimumab With or Without Vaccine Therapy in Treating Patients With Previously Treated Stage IV Melanoma).

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Oxabact DB17676
biotech

Deskripsi belum tersedia.

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Oxabolone DB01500
small molecule | CAS: 4721-69-1

Deskripsi belum tersedia.

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small molecule | CAS: 1254-35-9

Oxabolone cipionate is the C17? cypionate ester and a prodrug of [DB01500]. A synthetic anabolic-androgenic (AAS) steroid, it is a derivative of 19-nortestosterone (nandrolone). It is considered as a performance enhancing drug thus is prohibited from use in s…

Kategori:
Alimentary Tract and MetabolismAnabolic Agents for Systemic UseAnabolic Steroids +11
Waktu Paruh-
Vol. Distribusi-
KlirensThe elimination on …
Genetik -
Oxaceprol DB13363
small molecule | CAS: 33996-33-7

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +6
Waktu Paruh-
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Oxacillin Approved DB00713
small molecule | CAS: 66-79-5

An antibiotic similar to [flucloxacillin] used in resistant staphylococci infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1A +7
Waktu Paruh20 to 30 minutes
Vol. Distribusi-
Klirens-
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Oxaflozane DB13457
small molecule | CAS: 26629-87-8

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNervous System +2
Waktu Paruh-
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Oxalic Acid DB03902
small molecule | CAS: 144-62-7

A strong dicarboxylic acid occurring in many plants and vegetables. It is produced in the body by metabolism of glyoxylic acid or ascorbic acid. It is not metabolized but excreted in the urine. It is used as an analytical reagent and general reducing agent. […

Kategori:
Acids, AcyclicCompounds used in a research, industrial, or household settingDicarboxylic Acids +6
Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
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Oxaliplatin Approved DB00526
small molecule | CAS: 61825-94-3

Oxaliplatin is a platinum-based chemotherapy drug in the same family as cisplatin and carboplatin. Compared to cisplatin the two amine groups are replaced by diamino cyclohexane (DACH) group to provide a greater antitumor effect.[A797] However, this leads to …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +9
Target Protein:
DNA
Waktu ParuhThe decline of ultr…
Vol. DistribusiAfter a single 2-ho…
KlirensPlatinum was cleare…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Citrate synthase, mitochondrialMalate dehydrogenaseSepiapterin reductase +2
Waktu Paruh-
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Genetik -
small molecule | CAS: 328-42-7

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic AcidsKeto Acids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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