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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 169 / 321
Imgatuzumab DB14884
biotech | CAS: 959963-46-3

Imgatuzumab is under investigation in clinical trial NCT01326000 (A Study of RO5083945 in Combination With FOLFIRI Versus FOLFIRI Plus Cetuximab or FOLFIRI Alone as Second Line Treatment in Patients With Metastatic Colorectal Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
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IMGN632 DB17337
biotech

Deskripsi belum tersedia.

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Imidacloprid DB11421
small molecule | CAS: 105827-78-9

Imidacloprid is a neonicotinoid, which is a class of neuro-active insecticides modeled after nicotine. Imidacloprid is a patented chemical, Imidacloprid is manufactured by Bayer Cropscience (part of Bayer AG) and sold under trade names Kohinor, Admire, Advant…

Kategori:
AgrochemicalsCholinergic AgentsCompounds used in a research, industrial, or household setting +4
Target Protein:
CHRNA7-FAM7A fusion protein
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Imidafenacin DB09262
small molecule | CAS: 170105-16-5

Imidafenacin is an antispasmodic agent with anticholinergic effects. It antagonizes muscarinic receptors in the bladder to reduce the frequency of urination in the treatment of overactive bladder. It is marketed in Japan under the tradenames Staybla by Ono Ph…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCytochrome P-450 CYP3A Substrates +8
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3
Waktu ParuhThe half life of el…
Vol. DistribusiThe estimated volum…
KlirensThe estimated clear…
Genetik -
Imidapril DB11783
small molecule | CAS: 89371-37-9

Imidapril has been investigated for the treatment of Kidney, Polycystic, Autosomal Dominant.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +7
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Imidazole DB03366
small molecule | CAS: 288-32-4

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsThromboxane-A Synthase, antagonists & inhibitors
Target Protein:
Monomeric sarcosine oxidaseNicotinate-nucleotide--dimethylbenzimidazole phosphoribosyltransferaseMyoglobin +23
Waktu Paruh-
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Genetik -
small molecule | CAS: 36364-49-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +16
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small molecule | CAS: 1072-84-0

Imidazole-4-carboxylic acid is under investigation in clinical trial NCT00583895 (Safety and Efficacy Study of Imcooh Cream in Patients Suffering From Moderate Atopic Dermatitis).

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small molecule

Deskripsi belum tersedia.

Target Protein:
Endoglucanase 5A
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Methionine aminopeptidase
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Imidocarb DB11521
small molecule | CAS: 27885-92-3

Imidocarb is a urea derivative used in veterinary medicine as an antiprotozoal agent for the treatment of infection with Babesia and other parasites.

Kategori:
AmidesAminesAnilides +7
Target Protein:
Acetylcholinesterase
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Imidurea Approved DB14075
small molecule | CAS: 39236-46-9

Imidurea is an antimicrobial preservative used in cosmetics. It acts as a formaldehyde releaser.

Kategori:
AmidesCell-mediated ImmunityIncreased Histamine Release +2
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Imifoplatin DB17120
small molecule | CAS: 1339960-28-9

Deskripsi belum tersedia.

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Imiglitazar DB12511
small molecule | CAS: 250601-04-8

Imiglitazar has been used in trials studying the treatment of Diabetes Mellitus.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
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Imiglucerase Approved DB00053
biotech | CAS: 154248-97-2

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 0.09 to 0.15 L/kg
Klirens* 14.5 +/- 4.0 mL/m…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
D-amino-acid oxidase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
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Imipenem Approved DB01598
small molecule | CAS: 64221-86-9

Imipenem is a semisynthetic thienamycin that has a wide spectrum of antibacterial activity against gram-negative and gram-positive aerobic and anaerobic bacteria, including many multiresistant strains.[label] It is stable to many beta-lactamases. Similar comp…

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +12
Target Protein:
Penicillin-binding protein 2Penicillin-binding protein 1BPenicillin-binding protein 1A +3
Waktu ParuhWhen given via IV i…
Vol. DistribusiThe reported volume…
KlirensThe total clearance…
Genetik -
Imipramine Approved DB00458
small molecule | CAS: 50-49-7

Imipramine, the prototypical tricyclic antidepressant (TCA), is a dibenzazepine-derivative TCA. TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individ…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +70
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +21
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhImipramine has a me…
Vol. DistribusiImipramine has a hi…
KlirensImipramine has a me…
Genetik 9 Varian
small molecule | CAS: 6829-98-7

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Imiquimod Approved DB00724
small molecule | CAS: 99011-02-6

Imiquimod is an immune response modifier that acts as a toll-like receptor 7 agonist. Imiquimod is commonly used topically to treat warts on the skin of the genital and anal areas. Imiquimod does not cure warts, and new warts may appear during treatment. Imiq…

Kategori:
Adjuvants, ImmunologicAminoquinolinesAntineoplastic Agents +17
Target Protein:
Toll-like receptor 7Toll-like receptor 8
Waktu Paruh20 hours (topical d…
Vol. Distribusi-
Klirens-
Genetik -
Imlifidase Approved DB15258
biotech | CAS: 1947415-68-0

Chronic kidney disease (CKD) is a progressive and irreversible disease that represents a significant burden for both the individual and healthcare system at large.[A225916] Currently available treatments for end-stage renal disease are limited to dialysis and…

Kategori:
Antineoplastic and Immunomodulating AgentsEndopeptidasesImmunosuppressive Agents +2
Target Protein:
IgG heavy chain
Waktu ParuhThe mean distributi…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Imlunestrant DB19043
small molecule | CAS: 2408840-26-4

Imlunestrant is under investigation in clinical trial NCT05514054 (A Study of Imlunestrant Versus Standard Endocrine Therapy in Participants With Early Breast Cancer).

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Estrogen receptor
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IMM-0306 DB19309
biotech

IMM-0306 (bispecific antibody-trap selectively targeting cd47 and cd20) is under investigation in clinical trial NCT05805943 (Study of IMM0306 in Patients With Relapsed or Refractory Cd20-positive B-cell Non-hodgkin's Lymphoma).

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IMM-101 DB15850
biotech

IMM-101 is a heat-inactivated immune-activating mycobacterial product. It has shown to be safe and well tolerated to complement conventional cancer therapy for patients with melanoma and pancreatic ductal adenocarcinoma[A220013,A220018,A220023]. Studies with …

Kategori:
Biological ProductsComplex MixturesMelanoma, therapy +1
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IMM101 DB15851
biotech

IMM-101 is a heat-inactivated immune-activating mycobacterial product. It has shown to be safe and well tolerated to complement conventional cancer therapy for patients with melanoma and pancreatic ductal adenocarcinoma [PMID: 21930686; PMID: 30107850; PMID: …

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IMMU-114 DB18458
biotech

IMMU-114 is antibody-drug conjugate consisting of humanized anti-HLA-DR IgG4 monoclonal antibody specific for alpha-chain linked to SN-38 via a CL2A linker.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Immucillin-G DB02230
small molecule

Deskripsi belum tersedia.

Kategori:
Purine-Nucleoside Phosphorylase, antagonists & inhibitorsPyrimidines
Target Protein:
Purine nucleoside phosphorylase
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Immucin DB17403
biotech

Deskripsi belum tersedia.

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biotech | CAS: 1807503-77-0

Deskripsi belum tersedia.

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Imolamine DB09284
small molecule | CAS: 318-23-0

Imolamine is a compound with a molecular weight of 260.33 g/mol with the formula diethyl[2-{5-imino-3-phenyl-4,5-dihydro-1,2,3-oxadiazol,-4-yl)ethyl]amine. It is developed under the brand name Coremax by Novartis consumer health SA.

Kategori:
Cardiac TherapyCardiovascular AgentsOxazoles +2
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Implitapide DB04852
small molecule | CAS: 177469-96-4

Implitapide is a microsomal triglyceride transfer protein (MTP)-inhibitor.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu Paruh-
Vol. Distribusi-
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Imrecoxib DB12354
small molecule | CAS: 395683-14-4

Imrecoxib has been used in trials studying the treatment of Knee Osteoarthritis.

Kategori:
AnionsElectrolytesHydrogen Sulfide +2
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
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Imsidolimab DB16658
biotech | CAS: 2102543-86-0

Imsidolimab is under investigation in clinical trial NCT03633396 (A Study to Evaluate the Efficacy and Safety of ANB019 in Subjects With Palmoplantar Pustulosis).

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IMT-288 DB19068
small molecule | CAS: 637771-94-9

IMT-288 is under investigation in clinical trial NCT01730638 (Immunotep for Patients With Medullary Thyroid Carcinoma.).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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IMT504 DB17792
biotech

IMT504, a non-CpG 24-mer oligodeoxynucleotide, is an immunomodulatory oligonucleotide currently being investigated as a rabies vaccine.[A259467]

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
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IN01 DB16434
biotech

The IN01 Vaccine, sponsored by the Instituto Oncologico Dr Rosell, IN3BIO, and PANGAEA, is a compound containing recombinant bacteria[L30543]. These cultures contain EGF-4-EGF with the cholera toxin B-subunit domain G33D sequence[L30543]. Administration of th…

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Genetik -
biotech

Developed by Sinopharm's Wuhan Institute of Biological Products co., this vaccine consists of the WIV04 strain of SARS-CoV-2. This strain was isolated from a patient in Wuhan, cultivated in a Vero cell line, and then subsequently inactivated using B-propiolac…

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biotech

The SARS-CoV-2 Inactivated Vaccine is a purified vaccine that contains multiple antigens from the virus and is inactivated in Vero Cells[A219758]. This vaccine specifically was developed in collaboration with the Chinese Academy of Medical Sciences, West Chin…

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Inalimarev DB17332
biotech | CAS: 685563-13-7

Deskripsi belum tersedia.

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Inarigivir DB15062
small molecule | CAS: 475650-36-3

Inarigivir is under investigation in clinical trial NCT03434353 (Study to Evaluate the Antiviral Activity of Inarigivir (GS-9992) Plus Tenofovir Alafenamide (TAF) for 12 Weeks in Adults With Chronic Hepatitis B (CHB)).

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small molecule | CAS: 942123-43-5

Inarigivir soproxil is under investigation in clinical trial NCT03434353 (Study to Evaluate the Antiviral Activity of Inarigivir (GS-9992) Plus Tenofovir Alafenamide (TAF) for 12 Weeks in Adults With Chronic Hepatitis B (CHB)).

Target Protein:
Nucleotide-binding oligomerization domain-containing protein 2
Waktu Paruh-
Vol. Distribusi-
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Inavolisib Approved DB15275
small molecule | CAS: 2060571-02-8

_PIK3CA_ is one of the most frequently mutated oncogenes, with the resulting mutated p110? protein it encodes playing a central role in tumor cell proliferation.[A264563] Chemotherapeutic agents targeting the PI3K p110? catalytic subunit have shown antitumor …

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +4
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe total clearance…
Genetik -
Inbakicept DB16479
biotech | CAS: 2135939-52-3

Inbakicept is a dimeric human IL-15 receptor ? (IL-15R?) sushi domain/human IgG1 Fc fusion protein. It is one of the active ingredients in Anktiva, a combination product also containing [nogapendekin alfa], where a single inbakicept is complexed with two noga…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsExperimental Unapproved Treatments for COVID-19 +4
Target Protein:
Interleukin-2 receptor subunit betaCytokine receptor common subunit gamma
Waktu Paruh-
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INBRX-101 DB18384
biotech

INBRX-101 is a recombinant human alpha-1 antitrypsin (AAT)-Fc fusion protein.

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Incadronic acid DB06255
small molecule | CAS: 124351-85-5

Incadronate, or YM-175,[A202769] is a nitrogen containing bisphosphonate. Along with being investigated to treat hypercalcemia of malignancy,[A202862] it has also been investigated in the treatment of myeloma, leukemia, and other cancers.[A14426,A14431,A14427…

Kategori:
Antineoplastic AgentsBisphosphonatesBone Density Conservation Agents +2
Target Protein:
Farnesyl pyrophosphate synthaseCaspase-3Caspase-4 +1
Waktu ParuhIncadronate has a b…
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INCB-054329 DB16894
small molecule | CAS: 1628607-64-6

Deskripsi belum tersedia.

Kategori:
Antineoplastic Agents
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INCB-057643 DB16054
small molecule | CAS: 1820889-23-3

INCB-057643 is under investigation in clinical trial NCT02959437 (Azacitidine Combined With Pembrolizumab and Epacadostat in Subjects With Advanced Solid Tumors (ECHO-206)).

Kategori:
AcidsAcids, NoncarboxylicAntineoplastic Agents +1
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INCB-086550 DB18901
small molecule | CAS: 2230911-59-6

INCB-086550 is under investigation in clinical trial NCT04629339 (Study of INCB086550 in Select Solid Tumors).

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INCB-9471 DB12960
small molecule | CAS: 869769-98-2

INCB-9471 is a novel, orally available CCR5 antagonist that is part of a new class of drugs to treat HIV/AIDS. It is a potent, selective inhibitor of the HIV-1 virus.

Kategori:
Receptors, CCR4, antagonists & inhibitors
Target Protein:
C-C chemokine receptor type 5
Waktu Paruh-
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