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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 168 / 236
ONT-093 DB14069
small molecule | CAS: 216227-54-2

ONT-093 is an orally bioavailable inhibitor of P-glycoprotein (P-gp). In pre-clinical studies, ONT-093 could inhibit P-gp and reverse multidrug resistance at nM concentrations with no effect on paclitaxel pharmacokinetics.

Kategori:
Drug Resistance, MultipleP-glycoprotein inhibitors
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
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Ontamalimab DB15298
biotech | CAS: 2098790-40-8

Ontamalimab is under investigation in clinical trial NCT03627091 (Efficacy and Safety Study of SHP647 as Maintenance Treatment in Participants With Moderate to Severe Crohn's Disease (CARMEN CD 307)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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Onternabez DB18076
small molecule | CAS: 256934-39-1

Deskripsi belum tersedia.

Kategori:
Cannabinoid Receptor AgonistsCannabinoids and similarsHormones +3
Waktu Paruh-
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Ontorpacept DB17116
biotech | CAS: 2131089-46-6

Deskripsi belum tersedia.

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Ontuxizumab DB16270
biotech | CAS: 946415-62-9

Ontuxizumab is a humanized monoclonal antibody that targets endosialin or tumour endothelial marker 1 (TEM-1). It is under investigation in clinical trial NCT01574716 (Sarcoma Study of Morab-004 Utilization: Research and Clinical Evaluation).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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biotech | CAS: 1620643-19-7

Onvitrelin ucalontide is under investigation in clinical trial NCT01485848 (EP-100 Plus Paclitaxel Versus Paclitaxel Alone in Patients With Ovarian Cancer).

Waktu Paruh-
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OP-145 DB05672
biotech | CAS: 732984-79-1

OP-145 is a synthetic antimicrobial peptide developed from human cathelicidin LL-37.

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Opaganib DB12764
small molecule | CAS: 915385-81-8

Opaganib, also known as ABC294640, is a selective [sphingosine kinase-2 (SK2)](https://go.drugbank.com/polypeptides/Q9NRA0) inhibitor that is orally administered.[L27436] This drug has potential anticancer, anti-inflammatory, and antiviral activities, with po…

Kategori:
Bridged-Ring CompoundsCycloparaffins
Target Protein:
Sphingosine kinase 2
Waktu Paruh-
Vol. Distribusi-
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Opaviraline DB07884
small molecule | CAS: 178040-94-3

Deskripsi belum tersedia.

Kategori:
Antiviral AgentsHeterocyclic Compounds, Fused-RingNon-Nucleoside Reverse Transcriptase Inhibitors
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
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OPB-111077 DB16630
small molecule

OPB-111077 is a novel inhibitor of STAT3 and mitochondrial oxidative phosphorylation. It has demonstrated promising anticancer activity in preclinical models.

Target Protein:
Signal transducer and activator of transcription 3
Waktu Paruh-
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OPC1 DB17944
biotech

OPC1 is an oligodendrocyte progenitor cell therapy being investigated for the treatment of acute spinal cord injury.[L47082]

Waktu Paruh-
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Opebacan DB06161
biotech | CAS: 206254-79-7

Deskripsi belum tersedia.

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Opelconazole DB18251
small molecule | CAS: 1931946-73-4

Deskripsi belum tersedia.

Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
Deoxyribose-phosphate aldolaseDeoxyribose-phosphate aldolase
Waktu Paruh-
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Opicapone Approved DB11632
small molecule | CAS: 923287-50-7

Opicapone is a potent, reversible, and peripherally-acting third-generation inhibitor of catechol-o-methyltransferase (COMT), an enzyme involved in the breakdown of various catecholamines including dopamine.[A36938, A203048] Many patients with Parkinson’s dis…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsBCRP/ABCG2 Substrates +25
Target Protein:
Catechol O-methyltransferase
Waktu ParuhThe mean eliminatio…
Vol. DistribusiFollowing oral admi…
KlirensFollowing oral admi…
Genetik -
Opicinumab DB14959
biotech | CAS: 1422268-07-2

Opicinumab is under investigation in clinical trial NCT02641041 (Safety, Tolerability, and Pharmacokinetics of Single and Multiple Doses of BIIB033 in Healthy Japanese Participants).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Opipramol DB12930
small molecule | CAS: 315-72-0

Opipramol has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders.

Kategori:
Adrenergic AgentsAgents that produce hypertensionAgents that reduce seizure threshold +16
Waktu Paruh-
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Opiranserin DB16271
small molecule | CAS: 1441000-45-8

Opiranserin is under investigation in clinical trial NCT03997838 (Evaluate the Efficacy and Safety of VVZ-149 Injections for the Treatment of Post-operative Pain Following Abdominoplasty).

Waktu Paruh-
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Opium Approved DB11130
small molecule | CAS: 8008-60-4

Opium is the first substance of the diverse group of the opiates. It has been known for a long time, and the first evidence of a poppy culture dates from 5 thousand years by the Sumerians. During the years, opium was used as a sedative and hypnotic, but it wa…

Kategori:
Alimentary Tract and MetabolismAnalgesicsAntidiarrheals +25
Target Protein:
Delta-type opioid receptorKappa-type opioid receptorMu-type opioid receptor
Waktu ParuhThe half-life of op…
Vol. DistribusiOpium presents a la…
Klirens-
Genetik -
Oprelvekin Approved DB00038
biotech | CAS: 145941-26-0

Oprelvekin, the active ingredient in Neumega®, is recombinant Interleukin-11 (IL-11), which is produced in Escherichia coli (E. coli) by recombinant DNA technology. With a molecular mass of approximately 19,000 daltons, the non-glycosylated protein is 177 ami…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Interleukin-11 receptor subunit alpha
Waktu Paruh6.9 +/- 1.7 hrs
Vol. Distribusi-
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OptPA DB18325
biotech

Optimized tPA (OptPA; W253R/R275S-tPA) is an engineered variant of tPA designed to exhibit reduced neurotoxicity.[A261486]

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Orantinib DB12072
small molecule | CAS: 252916-29-3

Orantinib has been used in trials studying the treatment of Lung Cancer, Breast Cancer, Kidney Cancer, Gastric Cancer, and Prostate Cancer, among others.

Kategori:
Acids, AcyclicAlkaloidsEnzyme Inhibitors +9
Target Protein:
Vascular endothelial growth factor receptor 2Aurora kinase AFibroblast growth factor receptor 1 +2
Waktu Paruh-
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Orbifloxacin DB11443
small molecule | CAS: 113617-63-3

Orbifloxacin is a fluoroquinolone antibiotic. It is marketed by Schering-Plough Animal Health and approved for certain infections in dogs.

Kategori:
4-QuinolonesAnti-Bacterial AgentsCytochrome P-450 CYP1A2 Inhibitors +8
Waktu Paruh-
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ORC-13661 DB18903
small molecule | CAS: 1979935-33-5

ORC-13661 is under investigation in clinical trial NCT05730283 (Prevention of Ototoxicity in NTM Patients Treated With IV Amikacin).

Kategori:
AmidesSulfur Compounds
Waktu Paruh-
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Ordesekimab DB16649
biotech | CAS: 2394931-19-0

Ordesekimab is under investigation in clinical trial NCT02633020 (Study to Evaluate the Efficacy and Safety of AMG 714 in Adult Patients With Type II Refractory Celiac Disease).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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ORE-1001 DB12271
small molecule | CAS: 305335-31-3

ORE1001 has been used in trials studying the treatment of Mild to Moderate Ulcerative Colitis. It is an ACE2 inhibitor.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins
Target Protein:
Angiotensin-converting enzyme 2Carboxypeptidase N catalytic chainCarboxypeptidase N subunit 2
Waktu Paruh-
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Oregano Approved DB10677
biotech

Oregano allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Genetik -
small molecule

Deskripsi belum tersedia.

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Oregovomab DB04964
biotech | CAS: 213327-37-8

Oregovomab is a murine monoclonal antibody that attaches to the tumor-associated antigen CA125.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Mucin-16
Waktu Paruh-
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Orelabrutinib DB16272
small molecule | CAS: 1655504-04-3

Orelabrutinib is under investigation in clinical trial NCT04305197 (A Study of ICP-022 in Patients With Systemic Lupus Erythematosus (SLE)).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +1
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
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Orellanine DB19263
small molecule | CAS: 37338-80-0

Orellanine is under investigation in clinical trial NCT05287945 (Study of Orellanine in Metastatic Clear-cell or Papillary Renal Cell Carcinoma).

Kategori:
AgaricalesPyridines
Waktu Paruh-
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Orforglipron DB18964
small molecule | CAS: 2212020-52-3

Orforglipron is under investigation in clinical trial NCT06010004 (A Long-term Safety Study of Orforglipron (LY3502970) in Participants With Type 2 Diabetes).

Kategori:
Oxazoles
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
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ORG-25435 DB12312
small molecule | CAS: 256456-73-2

Org 25435 has been used in trials studying the treatment of Anaesthesia.

Kategori:
Benzene Derivatives
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
Waktu Paruh-
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ORG-25935 DB12220
small molecule | CAS: 1147011-84-4

Org 25935 has been used in trials studying the treatment of Alcoholism, Schizophrenia, and Panic Disorder.

Kategori:
Naphthalenes
Target Protein:
Sodium- and chloride-dependent glycine transporter 1
Waktu Paruh-
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ORG-31710 DB15585
small molecule | CAS: 118968-41-5

ORG-31710 is a progestational hormone antagonist.

Kategori:
EstranesFused-Ring CompoundsSteroids
Target Protein:
Progesterone receptor
Waktu Paruh-
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ORG-34517 DB05423
small molecule | CAS: 189035-07-2

ORG-34517 is currently under investigation by Organon for the treatment of depression. It has potential to treat a number of diseases such as Cushing’s disease, hypertension, diabetes, glaucoma etc, in which the activity of metabolites corticosterone and cor…

Kategori:
DioxolesFused-Ring CompoundsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Glucocorticoid receptor
Waktu Paruh-
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OriCar-017 DB17280
biotech

Deskripsi belum tersedia.

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Oridonin DB19086
small molecule | CAS: 28957-04-2

Oridonin is under investigation in clinical trial NCT05130892 (Effect of Inflammasome Inhibitor on Hscrp in Patients After PCI).

Kategori:
DiterpenesTerpenes
Waktu Paruh-
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Orilanolimab DB15312
biotech | CAS: 2066544-85-0

Orilanolimab is under investigation in clinical trial NCT03075878 (A Safety Study of SYNT001 in Subjects With Chronic, Stable Warm Autoimmune Hemolytic Anemia (WAIHA)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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Orismilast DB19042
small molecule | CAS: 1353546-86-7

Orismilast is under investigation in clinical trial NCT05190419 (Study to Assess the Efficacy and Safety of Orismilast in Psoriasis).

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Oritavancin Approved DB04911
small molecule | CAS: 171099-57-3

Oritavancin is a glycopeptide antibiotic used for the treatment of skin infections. It was developed by The Medicines Company (acquired by Novartis).[L12858] Oritavancin was initially approved by the FDA in 2014 and formulated to combat susceptible gram-posit…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +24
Target Protein:
Dihydropteroate synthasePeptidoglycan precursorsBacterial cell wall peptide bridging segments +1
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of or…
Genetik -
ORM-12741 DB12057
small molecule | CAS: 610782-82-6

ORM-12741 has been used in trials studying the basic science and treatment of Alzheimer's Disease.

Kategori:
Adrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +2
Target Protein:
Alpha-2C adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORM-13070 C-11 DB15324
small molecule | CAS: 1227170-74-2

ORM-13070 C-11 is under investigation in clinical trial NCT00735774 (Suitability of 11C-ORM-13070 as a PET Tracer).

Kategori:
Carbon Radioisotopes
Waktu Paruh-
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Ormeloxifene DB13310
small molecule | CAS: 31477-60-8

Ormeloxifene is a third-generation selective estrogen receptor (ER) modulator. In India, ormeloxifene has been marketed since the 1990s as a non-hormonal, non-steroidal oral contraceptive taken once a week,[A251450] and it was later introduced for the treatme…

Kategori:
Adrenal Cortex HormonesBenzopyransChromans +13
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu ParuhIn healthy, non-lac…
Vol. DistribusiIn healthy women, t…
KlirensIn healthy, non-lac…
Genetik -
Ornidazole DB13026
small molecule | CAS: 16773-42-5

Ornidazole has been used in trials studying the prevention of Elective Colorectal Surgery.

Kategori:
AmebicidesAnti-Infective AgentsAntibacterials for Systemic Use +13
Waktu Paruh-
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Ornipressin DB13464
biotech | CAS: 3397-23-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsCoagulants +18
Waktu Paruh-
Vol. Distribusi-
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Ornithine Approved DB00129
small molecule | CAS: 70-26-8

Produced during the urea cycle, ornithine is an amino acid produced from the splitting off of urea from arginine. L-Ornithine allows for the disposal of excess nitrogen and acts as a precursor of citrulline and arginine.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Basic +9
Target Protein:
Ornithine aminotransferase, mitochondrialOrnithine transcarbamylase, mitochondrialArginase-1 +7
Waktu Paruh-
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Orotidylic acid DB02957
small molecule | CAS: 2149-82-8

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPyrimidine Nucleotides +3
Waktu Paruh-
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ORP-101 DB16072
small molecule | CAS: 1820753-68-1

ORP-101 is under investigation in clinical trial NCT04129619 (A Comparison of the Effects of ORP-101 Versus Placebo in Adult Patients With Irritable Bowel Syndrome With Diarrhea (IBS-D)).

Target Protein:
Mu-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
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Orphenadrine Approved DB01173
small molecule | CAS: 83-98-7

A muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.

Kategori:
Agents producing tachycardiaAminesAnti-Dyskinesia Agents +41
Target Protein:
Glutamate receptor ionotropic, NMDA 2DGlutamate receptor ionotropic, NMDA 1Glutamate receptor ionotropic, NMDA 3B +4
Waktu Paruh13-20 hours
Vol. Distribusi-
Klirens-
Genetik -
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