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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 168 / 282
Ligufalimab DB17542
biotech | CAS: 2428381-55-7

Ligufalimab is a humanized immunoglobulin G4 (IgG4) monoclonal antibody targeting leukocyte surface antigen CD47. It is under investigation in clinical trial NCT04900350 (A Trial of AK117 (Anti-cd47) in Patients With Myelodysplastic Syndrome).

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Ligustrazine DB19074
small molecule | CAS: 1124-11-4

Ligustrazine is under investigation in clinical trial NCT05942352 (Clinical Study of Ligustrazine in Treating Alcohol Addiction).

Kategori:
Antiplatelet agentsCardiovascular AgentsVasodilating Agents
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Lilotomab DB19076
biotech | CAS: 1453362-55-4

Lilotomab is under investigation in clinical trial NCT01796171 (A Phase 1/2 Study of Betalutin for Treatment of Relapsed Non-hodgkin Lymphoma).

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Limaprost DB09211
small molecule | CAS: 74397-12-9

Limaprost (as Limaprost alfadex; CAS number 88852-12-4) is an oral prostaglandin E1 analog. Prostaglandins act on a variety of cells such as vascular smooth muscle cells causing constriction or dilation, on platelets causing aggregation or disaggregation and …

Kategori:
AnticoagulantsAutacoidsBiological Factors +11
Target Protein:
Prostaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtypeProstaglandin E2 receptor EP3 subtype +1
Waktu ParuhThe mean half life …
Vol. Distribusi-
KlirensMean total clearanc…
Genetik -
small molecule | CAS: 138-86-3

Limonene, (+/-)- is under investigation in clinical trial NCT05525260 (Limonene for Pulmonary Nodule Chemoprevention).

Kategori:
Cyclohexane MonoterpenesCyclohexanesCyclohexenes +3
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Linaclotide Approved DB08890
small molecule | CAS: 851199-59-2

Linaclotide is a synthetic 14-amino acid cyclic peptide [A260271] and first-in-class guanylate cyclase-C (G-CC) agonist.[A260271, L47211] Linaclotide is structurally related to human guanylin and uroguanylin, paracrine peptide hormones that are endogenous act…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +7
Target Protein:
Guanylyl cyclase C
Waktu ParuhThere is no availab…
Vol. DistribusiGiven that linaclot…
KlirensNo information is a…
Genetik -
Linafexor DB18031
small molecule | CAS: 2499656-04-9

Deskripsi belum tersedia.

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Linagliptin Approved DB08882
small molecule | CAS: 668270-12-0

Linagliptin is a DPP-4 inhibitor developed by Boehringer Ingelheim for the treatment of type II diabetes [L9557]. Linagliptin differs from other DPP-4 inhibitors in that it has a non-linear pharmacokinetic profile, is not primarily eliminated by the renal sys…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +24
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhThe terminal half l…
Vol. DistribusiA single intravenou…
KlirensTotal clearance of …
Genetik -
Lincomycin Approved DB01627
small molecule | CAS: 154-21-2

Lincomycin is a lincosamide antibiotic first isolated from the soil bacterium _Streptomyces lincolnensis_ in Lincoln, Nebraska.[A190621] Clinical use of lincomycin has largely been superseded by its semisynthetic derivative [clindamycin] due to its higher eff…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
23S ribosomal RNA
Waktu ParuhLincomycin has a bi…
Vol. DistribusiLincomycin administ…
KlirensLincomycin administ…
Genetik -
Lindane Approved DB00431
small molecule | CAS: 58-89-9

An organochlorine insecticide that has been used as a pediculicide and a scabicide. Lindane has been banned in California, United Kingdom, Australia, and many western countries due to concerns about neurotoxicity and adverse effects on the environment. In Can…

Kategori:
Agents that reduce seizure thresholdAgrochemicalsAntiparasitic Products, Insecticides and Repellents +9
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-1Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2 +7
Waktu Paruh18 hours
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Linerixibat DB11729
small molecule | CAS: 1345982-69-5

GSK2330672 has been investigated for the treatment of Diabetes Mellitus, Type 2.

Kategori:
AminesAzepinesSulfur Compounds +1
Target Protein:
Ileal sodium/bile acid cotransporter
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Linezolid Approved DB00601
small molecule | CAS: 165800-03-3

Linezolid is a synthetic antibiotic which is used for the treatment of infections caused by aerobic Gram-positive bacteria. Its effects are bacteriostatic against both enterococci and staphylococci and bactericidal against most isolates of streptococci.[L3296…

Kategori:
AcetamidesAcetatesAcids, Acyclic +22
Target Protein:
23S ribosomal RNA
Waktu ParuhThe elimination hal…
Vol. DistribusiAt steady-state, th…
KlirensTotal clearance of …
Genetik -
Linifanib DB06080
small molecule | CAS: 796967-16-3

Linifanib (ABT-869) is a small molecule vascular endothelial growth factor (VEGF) receptor-based kinase inhibitor that is designed to suppress tumor growth by preventing the formation of new blood vessels that supply the tumor with oxygen and nutrients and by…

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Vascular endothelial growth factor receptor 3Receptor-type tyrosine-protein kinase FLT3Vascular endothelial growth factor receptor 1 +3
Waktu Paruh-
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Linoleic acid Approved DB14104
small molecule | CAS: 60-33-3

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, EssentialFatty Acids, Omega-6 +3
Target Protein:
Fatty acid-binding protein, adipocyte
Waktu Paruh-
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Linopirdine DB13806
small molecule | CAS: 105431-72-9

Deskripsi belum tersedia.

Kategori:
Cardiovascular AgentsCentral Nervous System AgentsCompounds used in a research, industrial, or household setting +8
Target Protein:
Potassium voltage-gated channel subfamily KQT member 3
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Linopristin DB19296
small molecule | CAS: 325965-23-9

Linopristin is an antibiotic of the streptogramin B class. It is one part of the combination product NXL 103, along with [Virginiamycin M1]. The combination product was under investigation in clinical trials NCT00653172 and NCT00949130 for treatment of variou…

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Linperlisib DB17235
small molecule | CAS: 1702816-75-8

Deskripsi belum tersedia.

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Linrodostat DB14986
small molecule | CAS: 1923833-60-6

Linrodostat is under investigation in clinical trial NCT03247283 (Pharmacokinetics and Metabolism Study in Healthy Male Participants).

Kategori:
AcetatesAcids, AcyclicAmides +2
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Linseed oil DB11357
biotech | CAS: 66071-03-2

Linseed oil is a rich source of ?-Linolenic acid extracted from the dried, ripened seeds of the flax plant *Linum usitatissimum*. Other fatty acids contained in linseed oil include palmitic acid, stearic acid, oleic acid and linolenic acid. Linseed oil is par…

Kategori:
Biological ProductsComplex MixturesFats +5
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Linsitinib DB06075
small molecule | CAS: 867160-71-2

An orally bioavailable small molecule inhibitor of the insulin-like growth factor 1 receptor (IGF-1R) with potential antineoplastic activity. IGF-1R inhibitor OSI-906 selectively inhibits IGF-1R, which may result in the inhibition of tumor cell proliferation …

Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
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Lintuzumab DB14877
biotech | CAS: 166089-32-3

Lintuzumab is under investigation in clinical trial NCT00016159 (Chemotherapy Plus Monoclonal Antibody in Treating Patients With Acute Promyelocytic Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
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biotech | CAS: 2209911-94-2

Lintuzumab actinium Ac-225 is under investigation in clinical trial NCT00672165 (Targeted Atomic Nano-Generators (Actinium-225-Labeled Humanized Anti-CD33 Monoclonal Antibody HuM195) in Patients With Advanced Myeloid Malignancies).

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Linzagolix Approved DB17083
small molecule | CAS: 935283-04-8

Linzagolix is a non-peptide, selective antagonist of the gonadotropin-releasing hormone (GnRH) receptor. It has been studied for the treatment of estrogen-dependent conditions such as uterine fibroids and endometriosis.[A253642,A253647] It is similar to other…

Kategori:
Anti-Gonadotropin-Releasing HormonesBCRP/ABCG2 SubstratesCytochrome P-450 CYP2C8 Inhibitors +18
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe half-life of li…
Vol. DistribusiAfter seven days of…
KlirensThe geometric mean …
Genetik -
Liothyronine Approved DB00279
small molecule | CAS: 6893-02-3

Liothyronine is a thyroidal hormone T3 which is normally produced by the thyroid gland in a ratio 4:1 when compared with T4: T3. Liothyronine is the active form of thyroxine which is composed in a basic chemical structure by a tyrosine with bound iodine.[T457…

Kategori:
Agents used to treat hypothyroidismDrugs that are Mainly Renally ExcretedHormones +12
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor betaProliferating cell nuclear antigen
Waktu ParuhThe half-life of li…
Vol. DistribusiThe reported volume…
KlirensThere are no report…
Genetik -
small molecule | CAS: 20196-64-9

Liothyronine I-131 has been used in trials studying the treatment of Tricuspid Atresia and Heart Defects, Congenital.

Kategori:
Thyroxine-binding globulin substrates
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Liotrix Approved DB01583
small molecule | CAS: 8065-29-0

Liotrix is a synthetically derived thyroid hormone replacement preparation. It consists of levothyroxine sodium (thyroxine, T4) and liothyronine sodium (triiodothyronine, T3) in a 4 to 1 ratio by weight. Liotrix was developed when it was believed that serum l…

Kategori:
Agents used to treat hypothyroidismAmino AcidsAmino Acids, Aromatic +19
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu Paruh-
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Lipegfilgrastim Approved DB13200
biotech | CAS: 1117844-87-7

Lipegfilgrastim, previously known as XM22, is a pegylated, recombinant granulocyte colony-stimulating factor (G-CSF) that was synthetized using a highly site-specific glycoPEGylation technology [A32665]. It is used as an alternate to [DB00019] for prophylacti…

Kategori:
Adjuvants, ImmunologicAlcoholsAmino Acids, Peptides, and Proteins +17
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe average termina…
Vol. DistribusiLipegfilgrastim has…
KlirensIn a phase 1, multi…
Genetik -
Lipoic acid Approved DB00166
small molecule | CAS: 1200-22-2

A vitamin-like antioxidant.

Kategori:
Alimentary Tract and MetabolismAntioxidantsBiological Factors +15
Target Protein:
Lipoyl amidotransferase LIPT1, mitochondrialSodium-dependent multivitamin transporterLipoyl synthase, mitochondrial
Waktu Paruh-
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Lipotecan DB17385
small molecule | CAS: 1432468-79-5

Deskripsi belum tersedia.

Kategori:
Alkaloids
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
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biotech | CAS: 8046-19-3

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +2
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Lirafugratinib DB18300
small molecule | CAS: 2549174-42-5

Deskripsi belum tersedia.

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Liraglutide Approved DB06655
biotech | CAS: 204656-20-2

Victoza contains liraglutide, a synthetic analog of human glucagon-like peptide-1(GLP-1) and acts as a GLP-1 receptor agonist.[Label,A6932] Liraglutide is 97% similar to native human GLP-1, differing primarily by substituting arginine for lysine at position 3…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +17
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhTerminal half life …
Vol. Distribusi13L[Label].
Klirens1.2L/h[Label].
Genetik -
Lirentelimab DB16728
biotech | CAS: 2283348-97-8

Lirentelimab is under investigation in clinical trial NCT04856891 (A Study of Lirentelimab (AK002) in Patients With Active Eosinophilic Duodenitis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Lisaftoclax DB18054
small molecule | CAS: 2180923-05-9

Lisaftoclax is a novel, orally active, selective and potent BCL-2 inhibitor

Kategori:
Benzene DerivativesNitro Compounds
Target Protein:
Apoptosis regulator Bcl-2
Waktu Paruh-
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Lisavanbulin DB15224
small molecule | CAS: 1263384-43-5

Lisavanbulin is under investigation in clinical trial NCT02895360 (Phase 1/2a Study of BAL101553 as 48-hour Infusions in Patients With Advanced Solid Tumors or Recurrent Glioblastoma).

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalHeterocyclic Compounds, Fused-Ring +2
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Lisdexamfetamine Approved DB01255
small molecule | CAS: 608137-32-2

Lisdexamfetamine is a prodrug of [dextroamphetamine], a central nervous system stimulant known as d-amphetamine,[A40246] covalently attached to the naturally occurring amino acid L-lysine.[A2230] Lisdexamfetamine is the first chemically formulated prodrug sti…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +17
Target Protein:
Trace amine-associated receptor 1
Waktu ParuhPlasma concentratio…
Vol. DistribusiDextroamphetamine, …
Klirens-
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Lisinopril Approved DB00722
small molecule | CAS: 76547-98-3

Lisinopril is an angiotensin converting enzyme inhibitor (ACEI) used to treat hypertension, heart failure, and myocardial infarction.[L8384,L8387,L8390] Lisinopril and [captopril] are the only ACEIs that are not prodrugs.[A184853] It functions by inhibition o…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +20
Target Protein:
Angiotensin-converting enzymeRenin
Waktu ParuhLisinopril has an e…
Vol. DistribusiThe apparent volume…
KlirensA 30kg child has a …
Genetik -
Lisocabtagene maraleucel Approved DB16582
biotech

Lisocabtagene maraleucel is a chimeric antigen receptor (CAR) T-cell therapy, similar to [brexucabtagene autoleucel] and [axicabtagene ciloleucel].[A228493,L31588] Lisocabtagene maraleucel is a genetically modified autologous T-cell therapy that targets CD19,…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy +3
Target Protein:
B-lymphocyte antigen CD19
Waktu Paruh-
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Lisofylline DB12406
small molecule | CAS: 100324-81-0

Lisofylline has been investigated for the treatment of Type 1 Diabetes Mellitus.

Kategori:
Adjuvants, ImmunologicAnalgesicsAnalgesics, Non-Narcotic +12
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biotech

Deskripsi belum tersedia.

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Lisuride Approved DB00589
small molecule | CAS: 18016-80-3

An ergot derivative that acts as an agonist at dopamine D2 receptors (dopamine agonists). It may also act as an antagonist at dopamine D1 receptors, and as an agonist at some serotonin receptors (serotonin agonists).

Kategori:
Agents that produce hypertensionAlkaloidsAnalgesics +27
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor +12
Waktu Paruh-
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Lithium carbonate Approved DB14509
small molecule | CAS: 554-13-2

Lithium has been used to treat manic episodes since the 19th century[A176642]. Though it is widely used, its mechanism of action is still unknown[FDA Label][A14585,A176642,A176651,L5843]. Lithium carbonate has a narrow therapeutic range and so careful monitor…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +26
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu ParuhThe half life of li…
Vol. DistribusiApparent volume of …
KlirensClearance is genera…
Genetik -
Lithium cation DB01356
small molecule | CAS: 7439-93-2

Lithium was used during the 19th century to treat gout. Lithium salts such as lithium carbonate (Li2CO3), lithium citrate, and lithium orotate are mood stabilizers. They are used in the treatment of bipolar disorder, since unlike most other mood altering drug…

Kategori:
Antidepressive AgentsAntimanic AgentsAntipsychotic Agents +11
Target Protein:
Glycogen synthase kinase-3 betaInositol monophosphatase 1Inositol monophosphatase 2 +1
Waktu Paruh-
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Lithium hydroxide Approved DB14506
small molecule | CAS: 1310-65-2

Used for tryptophan determinations in proteins & foods.

Kategori:
Lithium CompoundsNarrow Therapeutic Index Drugs
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small molecule | CAS: 29126-50-9

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDermatologicalsDicarboxylic Acids +2
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu Paruh-
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Litifilimab DB18864
biotech | CAS: 2407378-48-5

Litifilimab is under investigation in clinical trial NCT05531565 (A Study to Assess the Efficacy and Safety of BIIB059 (Litifilimab) in Participants With Active Subacute Cutaneous Lupus Erythematosus (SCLE) And/or Chronic Cutaneous Lupus Erythematosus (CCLE) …

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Litronesib DB11861
small molecule | CAS: 910634-41-2

Litronesib has been used in trials studying the treatment of Solid Tumors, Ovarian Cancer, Gastric Cancer, Prostate Cancer, and Acute Leukaemia, among others.

Kategori:
AmidesSulfonesSulfur Compounds +1
Target Protein:
Kinesin-like protein KIF11
Waktu Paruh-
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Lividomycin A DB04728
small molecule | CAS: 36441-41-5

Deskripsi belum tersedia.

Target Protein:
Telomerase reverse transcriptase
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Livmoniplimab DB18939
biotech | CAS: 2412004-88-5

Livmoniplimab is under investigation in clinical trial NCT06109272 (A Study to Assess the Dose, Adverse Events, and Change in Disease Activity of Livmoniplimab as an Intravenous (IV) Solution in Combination With Budigalimab as an IV Solution in Adult Particip…

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Livoletide DB15188
small molecule | CAS: 1088543-62-7

Livoletide is under investigation in clinical trial NCT03790865 (Effects of Livoletide (AZP-531) on Food-related Behaviors in Patients With Prader-Willi Syndrome).

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsHormones +3
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