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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 168 / 321
Ieramilimab DB16419
biotech | CAS: 2137049-37-5

Ieramilimab is under investigation in clinical trial NCT02460224 (Safety and Efficacy of LAG525 Single Agent and in Combination With PDR001 in Patients With Advanced Malignancies.).

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Ifebemtinib DB17570
small molecule | CAS: 1227948-82-4

Deskripsi belum tersedia.

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Ifenprodil DB08954
small molecule | CAS: 23210-56-2

N-methyl-D-aspartate (NMDA) receptors (NMDARs) are members of the ionotropic glutamate receptor family, with key roles in brain development and neurological function.[A220118, A220128] NMDARs are heterotetramers that typically involve a dimer of dimers of bot…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +12
Target Protein:
Glutamate receptor ionotropic, NMDA 2BChymotrypsin-like elastase family member 1Glutamate receptor ionotropic, NMDA 1 +3
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Iferanserin DB11686
small molecule | CAS: 58754-46-4

Iferanserin has been investigated for the treatment of Hemorrhoids.

Kategori:
Acids, CarbocyclicAntidepressive AgentsCentral Nervous System Depressants +2
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Ifetroban DB12321
small molecule | CAS: 143443-90-7

Ifetroban has been used in trials studying the treatment of Skin Diseases, Autoimmune Diseases, Pathologic Processes, Scleroderma, Limited, and Scleroderma, Diffuse, among others.

Kategori:
Antiplatelet agentsHematologic Agents
Target Protein:
Thromboxane A2 receptor
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biotech | CAS: 2407582-19-6

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Ifidancitinib DB16191
small molecule | CAS: 1236667-40-5

Ifidancitinib is under investigation in clinical trial NCT03585296 (A Study of ATI-502 Topical Solution for the Treatment of Atopic Dermatitis).

Kategori:
Adrenal Cortex HormonesFused-Ring CompoundsNorpregnanes +4
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK1
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biotech | CAS: 2484870-92-8

Deskripsi belum tersedia.

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Ifosfamide Approved DB01181
small molecule | CAS: 3778-73-2

Ifosfamide is a chemotherapeutic agent chemically related to the nitrogen mustards and a synthetic analog of cyclophosphamide. It is active as an alkylating agent and an immunosuppressive agent.

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +46
Target Protein:
DNANuclear receptor subfamily 1 group I member 2
Waktu Paruh7-15 hours. The eli…
Vol. DistribusiIfosfamide volume o…
Klirens* 2.4±0.33 L/h/m^2 …
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IFx-Hu2.0 DB18396
biotech

IFx-Hu2.0 is an investigational cancer vaccine. It is composed of plasmid DNA encoding the streptococcal membrane protein, Emm55, contained within a cationic polymer.

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IGN101 DB06500
biotech

IGN101 is an antibody-based cancer vaccine directed against epithelial cancers. It consists of 500 ug 17-1A antibody adsorbed on aluminum hydroxide.

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IGN301 DB05117
biotech

IGN301 is a cancer vaccine based on an anti-idiotypic antibody which provokes an immune response to Lewis Y. Lewis Y is a carbohydrate molecule expressed on the surface of tumor cells of epithelial origin (e.g. lung, intestinal, breast, prostate or ovarian ca…

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IGN311 DB04988
biotech

IGN311 is a humanized monoclonal antibody (mab) against the Lewis Y carbohydrate antigen, a blood-group-related oligosaccharide.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2
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Iguratimod DB12233
small molecule | CAS: 123663-49-0

Iguratimod is under investigation in Rheumatoid Arthritis.

Kategori:
AmidesBenzopyransHeterocyclic Compounds, Fused-Ring +3
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IK-930 DB18149
small molecule

IK-930 is an oral, paralog-selective TEAD inhibitor.

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IKT-001Pro DB17307
small molecule

Deskripsi belum tersedia.

Kategori:
Kinase Inhibitor
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IL-2 pDNA DB05935
small molecule

Vical incorporated has initiated a human Phase 1 study of an investigational method of delivering interleukin-2 (IL-2), a potent immune system stimulant, for patients with recurrent metastatic melanoma.

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IL15-NK Cell DB15725
biotech

Natural killer (NK) cells can be incubated with ‘feeder cells’ expressing certain cytokines prior to maturation to enhance their activity. In particular, incubation with IL-15 allows NK cells to lyse a broad range of fresh and cultured tumor targets that the …

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Ilacirnon DB16066
small molecule | CAS: 1100318-47-5

Ilacirnon (CCX-140) is under investigation in clinical trial NCT01440257 (A Study to Evaluate the Effect of CCX140-B on Urinary Albumin Excretion in Subjects With Type 2 Diabetes and Albuminuria).

Target Protein:
C-C chemokine receptor type 2
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Ilaprazole DB11964
small molecule | CAS: 172152-36-2

Ilaprazole has been investigated in Helicobacter Infections.

Kategori:
Anti-Ulcer AgentsBenzimidazolesGastric Acid Lowering Agents +5
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Ilepatril DB06604
small molecule | CAS: 473289-62-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingProdrugs
Target Protein:
NeprilysinAngiotensin-converting enzyme
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Ilepcimide DB16942
small molecule | CAS: 82857-82-7

Deskripsi belum tersedia.

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biotech

Ilex paraguariensis leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Ilginatinib DB12784
small molecule | CAS: 1239358-86-1

NS-018 has been used in trials studying the treatment of Primary Myelofibrosis, Post-Polycythemia Vera Myelofibrosis, and Post-Essential Thrombocythemia Myelofibrosis.

Target Protein:
Tyrosine-protein kinase JAK2
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Ilodecakin DB06449
small molecule | CAS: 149824-15-7

Deskripsi belum tersedia.

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Ilomastat DB02255
small molecule | CAS: 142880-36-2

Ilomastat is a broad-spectrum matrix metalloproteinase inhibitor.

Kategori:
AminesAmino Acids, Peptides, and ProteinsEnzyme Inhibitors +7
Target Protein:
Interstitial collagenaseMatrix metalloproteinase-14Neutrophil collagenase +8
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Iloperidone Approved DB04946
small molecule | CAS: 133454-47-4

Iloperidone is a benzisoxazole [A263557] and an atypical antipsychotic agent that was first approved by the FDA on May 6, 2009.[A3024] It is considered to be a second-generation antipsychotic drug [A263552] with multiple receptor binding profile, although it …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +31
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +14
Waktu ParuhThe observed mean e…
Vol. DistribusiThe apparent volume…
KlirensIloperidone has an …
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Iloprost Approved DB01088
small molecule | CAS: 78919-13-8

Iloprost is an analog of prostacyclin (PGI2; epoprostenol), an endogenous prostanoid mainly produced in the vascular endothelium. It is more stable than prostacyclin, which is short-lived.[A263326] Iloprost consists of a mixture of the 4R and 4S diastereoisom…

Kategori:
Agents Causing Muscle ToxicityAntiplatelet agentsAutacoids +16
Target Protein:
Prostacyclin receptorProstaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtype +6
Waktu ParuhThe half-life of il…
Vol. DistribusiFollowing intraveno…
KlirensClearance in normal…
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Ilorasertib DB11694
small molecule | CAS: 1227939-82-3

Ilorasertib has been used in trials studying the treatment of Myelodysplasia, Solid Neoplasm, Advanced Cancers, Advanced Solid Tumors, and Acute Myelogenous Leukemia, among others.

Kategori:
AmidesAminesAntineoplastic Agents +4
Target Protein:
Aurora kinase AAurora kinase BAurora kinase C
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ILS-920 DB15422
small molecule | CAS: 892494-07-4

ILS-920 is under investigation in clinical trial NCT00827190 (Study Evaluating Single Ascending Doses Of ILS-920).

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Iltamiocel DB19059
biotech

Deskripsi belum tersedia.

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Iluzanebart DB18275
biotech | CAS: 2733621-19-5

Deskripsi belum tersedia.

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ILY101 DB05059
small molecule

ILY101 is a metal-free, non-absorbed polymeric drug designed for the selective binding and removal of phosphate anions from the gastrointestinal tract. ILY101 is being developed for the treatment of hyperphosphatemia in CKD patients on dialysis and works by …

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small molecule | CAS: 1422365-93-2

Deskripsi belum tersedia.

Kategori:
Amidines
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IMA901 DB06628
biotech

IMA901 is a vaccine consists of tumor-associated peptides (TUMAPs).

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Imagabalin DB12105
small molecule | CAS: 610300-07-7

Imagabalin has been investigated in Generalized Anxiety Disorder.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Anxiety AgentsCentral Nervous System Depressants
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
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Imalumab DB15558
biotech | CAS: 1430205-07-4

Imalumab is under investigation in clinical trial NCT02540356 (Phase 1/2a Two-arm Dose-escalation Study of BAX69 in Subjects With Malignant Ascites of Ovarian Cancer).

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Imaradenant DB16192
small molecule | CAS: 1321514-06-0

Imaradenant is under investigation in clinical trial NCT03381274 (Oleclumab (MEDI9447) Egfrm NSCLC Novel Combination Study).

Target Protein:
Adenosine receptor A2a
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Imatinib Approved DB00619
small molecule | CAS: 152459-95-5

Imatinib is a small molecule kinase inhibitor that revolutionized the treatment of cancer, particularly chronic myeloid leukemia, in 2001.[A249305] It was deemed a "miracle drug" due to its clinical success, as oncologist Dr. Brian noted that "complete hemato…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +51
Target Protein:
Breakpoint cluster region proteinInduced myeloid leukemia cell differentiation protein Mcl-1Mast/stem cell growth factor receptor Kit +8
Waktu ParuhFollowing oral admi…
Vol. DistribusiPopulation pharmaco…
KlirensTypically, clearanc…
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Imazaquin DB04582
small molecule

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingHerbicides +3
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IMC-1C11 DB06101
biotech

IMC-1C11 is an anti-angiogenesis agent. It is a chimeric anti-kinase insert domain-containing receptor (KDR) antibody that blocks VEGFR-KDR interaction and inhibits VEGFR-induced endothelial cell proliferation. IMC-1C11 is used for treatment of patients with …

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3
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biotech | CAS: 138660-99-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
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IMCY-0141 DB17019
biotech

IMCY-0141 is a synthetic peptide based on MOG (Myelin Oligodendrocyte Glycoprotein), a dominant autoantigen, designed to stop the progression of multiple sclerosis (MS) and the destruction of the myelin sheath protecting the nerves.[L43287]

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Imdevimab Approved DB15940
biotech | CAS: 2415933-40-1

Imdevimab is a monoclonal antibody combined with [casirivimab] in Regeneron's antibody cocktail known as REGEN-COV2 for the treatment of COVID-19.[L23539] This drug is a combination of antibodies derived from humanized VelocImmune® mice in addition to blood …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Spike glycoprotein
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Imdusiran DB19014
biotech | CAS: 2839476-19-4

Imdusiran is under investigation in clinical trial NCT06245291 (Study of Imdusiran (AB-729) in Combination With Intermittent Dosing of Durvalumab in Subjects With Chronic HBV Infection).

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Imeglimin DB12509
small molecule | CAS: 775351-65-0

Imeglimin has been used in trials studying the treatment of Type 2 Diabetes Mellitus.

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsDrugs Used in Diabetes
Target Protein:
5'-AMP-activated protein kinase catalytic subunit alpha-15'-AMP-activated protein kinase subunit beta-15'-AMP-activated protein kinase subunit gamma-1
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Imelasomeran Approved DB17090
biotech | CAS: 2763208-92-8

Imelasomeran was first approved in Canada on September 1, 2022, as one-half of Moderna's Spikevax Bivalent COVID-19 mRNA vaccine.[L45320] It encodes for the viral spike protein of the Omicron BA.1 variant of SARS-CoV-2, a particularly infectious variant of co…

Kategori:
COVID-19 VaccinesmRNA VaccinesVaccines +1
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Imetelstat Approved DB14909
small molecule | CAS: 868169-64-6

Imetelstat is a first-in-class 18-amino acid oligonucleotide that directly and competitively inhibits human telomerase.[A263973] It is used to treat anemia in patients with myelodysplastic syndromes (MDS), a group of hematologic disorders characterized by ine…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +6
Target Protein:
Telomerase reverse transcriptaseHuman telomerase RNA component
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
Klirens-
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Imexon DB05003
small molecule | CAS: 59643-91-3

Imexon is currently being studied for the treatment of pancreatic, lung, breast, prostate, melanoma, and multiple myeloma cancers. It belongs to the family of drugs called cyanoaziridine derivatives. Also called Amplimexon. Imexon is a cyanoaziridine derivati…

Kategori:
Ketones
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2Ribonucleoside-diphosphate reductase large subunit
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IMG-7289 DB15126
small molecule | CAS: 1990504-34-1

IMG-7289 is under investigation in clinical trial NCT03136185 (IMG-7289 in Patients With Myelofibrosis).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysine-specific histone demethylase 1A
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