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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 167 / 282
Levofloxacin Approved DB01137
small molecule | CAS: 100986-85-4

Levofloxacin is a fluoroquinolone antibiotic and the optical S-(-) isomer of racemic [ofloxacin].[A190663] It reportedly carries 8 to 128-fold more activity against both gram-negative and gram-positive bacteria compared to R-(+)-ofloxacin[A190663] and remains…

Kategori:
4-QuinolonesAlimentary Tract and MetabolismAnti-Bacterial Agents +35
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu ParuhThe average termina…
Vol. DistribusiLevofloxacin is wid…
KlirensThe average apparen…
Genetik -
Levoglucose DB12970
small molecule | CAS: 921-60-8

Levoglucose has been used in trials studying the diagnostic of Bowel Cleansing Prior to Colonoscopy.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levoketoconazole Approved DB05667
small molecule | CAS: 142128-57-2

Cushing's syndrome (CS) is underpinned by chronic hypercortisolism leading to multisystem morbidity, including effects on the cardiovascular and endocrine systems, metabolic syndrome with accompanying changes in body composition, neuropsychiatric effects, cha…

Kategori:
Adrenal Cortex HormonesAntiadrenal PreparationsAnticorticosteroids +32
Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyaseCytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial +2
Waktu ParuhLevoketoconazole ha…
Vol. DistribusiLevoketoconazole ha…
Klirens-
Genetik -
Levoleucovorin Approved DB11596
small molecule | CAS: 68538-85-2

Levoleucovorin is the enantiomerically active form of Folinic Acid (also known as 5-formyl tetrahydrofolic acid or leucovorin). Commercially available leucovorin is composed of a 1:1 racemic mixture of the dextrorotary and levorotary isomers, while levoleucov…

Kategori:
AntidotesCoenzymesCompounds used in a research, industrial, or household setting +14
Target Protein:
Serine hydroxymethyltransferase
Waktu ParuhThe mean terminal h…
Vol. DistribusiData can't be found.
KlirensData can't be found.
Genetik -
Levomefolic acid Approved DB11256
small molecule | CAS: 31690-09-2

Levomefolic acid (INN) is the metabolite of folic acid (Vitamin B9) and it is a predominant active form of folate found in foods and in the blood circulation, accounting for 98% of folates in human plasma [A19276]. It is transported across the membranes inclu…

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +10
Waktu ParuhThe mean eliminatio…
Vol. DistribusiCirculates in its f…
Klirens-
Genetik -
Levomenol Approved DB13153
small molecule | CAS: 23089-26-1

Bisabolol, or more formally ?-(?)-bisabolol or also known as levomenol, (-)-alpha-Bisabolol is found in fats and oils. (-)-alpha-Bisabolol is isolated from essential oil of Matricaria chamomilla (German chamomile) (-)-alpha-Bisabolol belongs to the family of …

Kategori:
Biological ProductsComplex MixturesLipids +7
Waktu Paruh-
Vol. DistribusiTo demonstrate the …
Klirens-
Genetik -
Levomenthol Approved DB00825
small molecule | CAS: 2216-51-5

Menthol is a covalent organic compound made synthetically or obtained from peppermint or other mint oils. Forming clear or white waxy, crystalline substance, menthol is typically solid at room temperature. (-)-Menthol is the naturally-occurring and main form …

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntipruritics +16
Target Protein:
Transient receptor potential cation channel subfamily M member 8Transient receptor potential cation channel subfamily A member 1Transient receptor potential cation channel subfamily V member 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levomethadone DB13515
small molecule | CAS: 125-58-6

Deskripsi belum tersedia.

Kategori:
Drugs Used in Addictive DisordersDrugs Used in Opioid DependenceNervous System
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levomilnacipran Approved DB08918
small molecule | CAS: 96847-54-0

Levomilnacipran is a selective serotonin and norepinephrine reuptake inhibitor (SNRI), although it is a more potent inhibitor of norepinephrine reuptake than serotonin reuptake.[A261181, A38560] Levomilnacipran is the more active 1S,2R-enantiomer in the racem…

Kategori:
Adrenergic Uptake InhibitorsAgents producing tachycardiaAntidepressive Agents +27
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporter
Waktu ParuhThe apparent termin…
Vol. DistribusiLevomilnacipran is …
KlirensFollowing oral admi…
Genetik -
small molecule | CAS: 154357-42-3

Levonadifloxacin is under investigation in clinical trial NCT03405064 (Comparative Study of Levonadifloxacin (IV and Oral) With Linezolid (IV and Oral) in Acute Bacterial Skin and Skin Structure Infections (ABSSSI)).

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levonordefrin Approved DB06707
small molecule | CAS: 829-74-3

Levonordefrin acts as a topical nasal decongestant and vasoconstrictor, most often used in dentistry.

Kategori:
Adrenergic AgonistsAgents producing tachycardiaAgents that produce hypertension +9
Target Protein:
Alpha-1D adrenergic receptorAlpha-1B adrenergic receptorAlpha-1A adrenergic receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levonorgestrel Approved DB00367
small molecule | CAS: 797-63-7

Levonorgestrel (LNG) is a synthetic progestogen similar to [Progesterone] used in contraception and hormone therapy.[A181988,T659] Also known as Plan B, it is used as a single agent in emergency contraception, and as a hormonal contraceptive released from an …

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +23
Target Protein:
Progesterone receptor3-oxo-5-alpha-steroid 4-dehydrogenase 1Estrogen receptor +3
Waktu ParuhThe elimination hal…
Vol. DistribusiOne pharmacokinetic…
KlirensClearance was found…
Genetik -
small molecule | CAS: 230313-75-4

Levophencynonate is under investigation in clinical trial NCT02299804 (A Clinical Trial to Evaluate Efficacy and Safety of Levophencynonate Hydrochloride in Patient With Vertigo).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2338-37-6

Levopropoxyphene is a stereoisomer of propoxyphene in the form of 2S, 3R enantiomer. It was sold as an antitussive, but it was removed from the market in the 70s.[T133] Levopropoxyphene was developed by Lilly and FDA approved on March 21st, 1962. This drug pr…

Kategori:
Acids, AcyclicAgents that reduce seizure thresholdAntitussive Agents +3
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levosalbutamol Approved DB13139
small molecule | CAS: 34391-04-3

Levosalbutamol, or levalbuterol, is a short-acting ?2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructive pulmonary disease (COPD). [Salbutamol] has been marketed as a racemic mixture, although beta2-agonist activity resides …

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +15
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh3.3 - 4 hours
Vol. Distribusi-
Klirens-
Genetik -
Levosimendan Approved DB00922
small molecule | CAS: 141505-33-1

Levosimendan increases calcium sensitivity to myocytes by binding to troponin C in a calcium dependent manner. This increases contractility without raising calcium levels. It also relaxes vascular smooth muscle by opening adenosine triphosphate sensitive pota…

Kategori:
Antiarrhythmic agentsCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy +14
Target Protein:
Troponin C, slow skeletal and cardiac musclesATP-sensitive inward rectifier potassium channel 11ATP-sensitive inward rectifier potassium channel 8 +1
Waktu ParuhEliminination half-…
Vol. Distribusi-
Klirens-
Genetik -
Levosulpiride DB16021
small molecule | CAS: 23672-07-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntipsychotic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levothyroxine Approved DB00451
small molecule | CAS: 51-48-9

Levothyroxine is a synthetically produced form of thyroxine, a major endogenous hormone secreted by the thyroid gland.[F4633] Also known as L-thyroxine or the brand name product Synthroid, levothyroxine is used primarily to treat hypothyroidism, a condition w…

Kategori:
Agents used to treat hypothyroidismAmino AcidsAmino Acids, Aromatic +16
Target Protein:
Integrin alpha-VIntegrin beta-3Thyroid hormone receptor alpha +1
Waktu ParuhT<sub>4</sub> half-…
Vol. Distribusi-
Klirens-
Genetik -
Levotofisopam DB19073
small molecule | CAS: 82059-51-6

Levotofisopam is under investigation in clinical trial NCT01519687 (Study of Levotofisopam 50 Mg Three Times a Day (TID) Administered for 7 Days on Hyperuricemia and Gout).

Kategori:
Antidepressive AgentsBenzazepinesCentral Nervous System Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levovirin DB06523
small molecule | CAS: 206269-27-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lexanersen DB17933
biotech | CAS: 2073015-40-2

Lexanersen is an antisense oligonucleotide under investigation for use as a disease-modifying therapy in Huntington's disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1390631-57-8

Lexaptepid pegol has been used in trials studying the treatment of Anemia, Inflammation, Chronic Diseases, End Stage Renal Disease, and Anemia of Chronic Disease.

Kategori:
Anti-Inflammatory AgentsNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lexatumumab DB06599
biotech | CAS: 845816-02-6

Lexatumumab is a fully humanized, high-affinity immunoglobulin G(1 lambda) monoclonal antibody (mAb).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +7
Target Protein:
Tumor necrosis factor receptor superfamily member 10B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LFA703 DB03932
small molecule

Deskripsi belum tersedia.

Target Protein:
Integrin alpha-L
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LG-100268 DB01941
small molecule | CAS: 153559-76-3

LG-100268 is a retinoid X receptor (RXR) selective compound.

Kategori:
LigandsNaphthalenesPyridines
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor RXR-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD-1550 DB05785
small molecule | CAS: 178600-20-9

LGD-1550 is an orally-active synthetic aromatic retinoic acid agent with potential antineoplastic and chemopreventive activities.

Kategori:
AlkenesBiological FactorsCarotenoids +8
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor betaRetinoic acid receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD-2226 DB08089
small molecule | CAS: 328947-93-9

An androgen receptor modulator.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD-3303 DB13937
small molecule | CAS: 917891-35-1

An androgen receptor modulator.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD-6972 DB14779
small molecule | CAS: 1207989-09-0

LGD-6972 is under investigation in clinical trial NCT01919684 (Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of LGD-6972 in Healthy Subjects and Subjects With Type 2 Diabetes Mellitus).

Kategori:
Acids, CarbocyclicAlkanesAlkanesulfonic Acids +7
Target Protein:
Glucagon receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD2941 DB05234
small molecule

LGD2941 is a non-steroidal, selective androgen receptor modulator (SARM) developed jointly by Ligand and TAP.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGH-447 DB14943
small molecule | CAS: 1210608-43-7

LGH-447 is under investigation in clinical trial NCT02160951 (Dose Escalation Study of LGH447 in Japanese Patients With Relapsed and/or Refractory Hematologic Malignancies).

Target Protein:
Serine/threonine-protein kinase pim-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LH-708 DB17636
small molecule | CAS: 1616758-14-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Liafensine DB14878
small molecule | CAS: 1198790-53-2

Liafensine is under investigation in clinical trial NCT00892840 (Multiple-Ascending Dose Study).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Libivirumab DB17748
biotech | CAS: 569658-79-3

Libivirumab is an investigational monoclonal antibody. It is one of the active ingredients in HepeX-B, a drug product containing two human monoclonal antibodies to the hepatitis B virus (HBV) surface antigen.[A259202]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licaminlimab DB18936
biotech | CAS: 1688648-13-6

Licaminlimab is under investigation in clinical trial NCT05896670 (Safety and Efficacy of Licaminlimab Ophthalmic Suspension for the Treatment of Dry Eye Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licochalcone A DB19281
small molecule | CAS: 58749-22-7

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFabaceae +5
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licofelone DB04725
small molecule | CAS: 156897-06-2

Developed by the German pharmaceutical company, Merckle GmbH, together with EuroAlliance partners Alfa Wassermann and Lacer, licofelone (ML3000) is a dual COX/LOX inhibitor and the first member of this new class of analgesic and anti-inflammatory drugs. It is…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +15
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenaseProstaglandin G/H synthase 2Group IIE secretory phospholipase A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licogliflozin DB15048
small molecule | CAS: 1291094-73-9

Licogliflozin is under investigation in clinical trial NCT03320941 (A Dose-finding Study to Evaluate the Change in Weight After Treatment With LIK066 in Japanese Patients With Obesity).

Kategori:
AlcoholsBlood Glucose Lowering AgentsCarbohydrates +2
Target Protein:
Sodium/glucose cotransporter 1Sodium/glucose cotransporter 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lidocaine Approved DB00281
small molecule | CAS: 137-58-6

Ever since its discovery and availability for sale and use in the late 1940s, lidocaine has become an exceptionally commonly used medication [T583]. In particular, lidocaine's principal mode of action in acting as a local anesthetic that numbs the sensations …

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAgents that reduce seizure thresholdAmides +49
Target Protein:
Sodium channel protein type 11 subunit alphaSodium channel protein type 10 subunit alphaSodium channel protein type 9 subunit alpha +5
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe mean systemic c…
Genetik -
Lidoflazine Approved DB13766
small molecule | CAS: 3416-26-0

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +13
Target Protein:
Sodium channel protein type 3 subunit alphaEquilibrative nucleoside transporter 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lidorestat DB07063
small molecule | CAS: 245116-90-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingIndoles +1
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1401812-88-1

Lifastuzumab vedotin is under investigation in clinical trial NCT01363947 (Safety and Pharmacokinetics of Escalating Doses of DNIB0600A in Participants With Non-Small Cell Lung Cancer (NSCLC) and Platinum Resistant Ovarian Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lifibrol DB12448
small molecule | CAS: 96609-16-4

Lifibrol has been used in trials studying the basic science of Hyperlipoproteinemia and Hypercholesterolemia.

Kategori:
Acids, CarbocyclicAlcoholsBenzene Derivatives +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lifileucel Approved DB17107
biotech | CAS: 2306267-74-1

Lifileucel is a tumour-derived autologous T cell immunotherapy composed of a suspension of tumour-derived T cells from the patient [L50171] which undergo isolation, ex vivo expansion, and activation[A263341] Lifileucel was granted accelerated approval by the …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lifirafenib DB14773
small molecule | CAS: 1446090-79-4

Lifirafenib is under investigation in clinical trial NCT03641586 (The Study of BGB-283 in Chinese Subjects With Local Advanced or Metastatic Malignant Solid Tumor).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase B-raf
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lifitegrast Approved DB11611
small molecule | CAS: 1025967-78-5

Lifitegrast is a FDA approved drug for the treatment of keratoconjunctivitis sicca (dry eye syndrome). It is a tetrahydroisoquinoline derivative and lymphocyte function-associated antigen-1 ( LFA-1) antagonist that was discovered through the rational design p…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +18
Target Protein:
Intercellular adhesion molecule 1Integrin alpha-L
Waktu ParuhNot possible to cal…
Vol. Distribusi-
KlirensNot possible to cal…
Genetik -
Ligandrol DB13934
small molecule | CAS: 1165910-22-4

Ligandrol is an investigational selective androgen receptor modulator (SARM) for treatment of conditions such as muscle wasting and osteoporosis.

Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ligelizumab DB11856
biotech | CAS: 1322627-61-1

Ligelizumab is a humanized IgG1k monoclonal antibody targeted against immunoglobulin E (IgE). Similar in mechanism to [omalizumab], another IgE-directed monoclonal antibody, ligelizumab has a distinct binding epitope as compared to its peer (with a small degr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Immunoglobulin heavy constant epsilon
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Light green SF yellowish Approved DB11183
small molecule | CAS: 5141-20-8

Light green SF yellowish is a green triarylmethane dye that is used in the preparation of the staining solution which is widely used as a counterstain. It is used in histological applications and other labratory settings, and usually exists as a disodium salt…

Kategori:
AminesArylsulfonatesArylsulfonic Acids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Light mineral oil Approved DB11579
small molecule | CAS: 92062-35-6

Deskripsi belum tersedia.

Kategori:
Basic Ointments and Protectants
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 8301–8350 dari 14063
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