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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 165 / 282
Lasofoxifene Approved DB06202
small molecule | CAS: 180916-16-9

Lasofoxifene is a non-steroidal 3rd generation selective estrogen receptor modulator (SERM) that selectively binds to both ER? and ER? with high affinity. It is a naphthalene derivative marketed for prevention and treatment of osteoporosis and for the treatme…

Kategori:
Genito Urinary System and Sex HormonesNaphthalenesSelective Estrogen Receptor Modulators +1
Target Protein:
Fusion glycoprotein F0Estrogen receptorEstrogen receptor beta +1
Waktu ParuhElimination half-li…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Latamoxef Approved DB04570
small molecule | CAS: 64952-97-2

Latamoxef is a broad- spectrum beta-lactam antibiotic similar in structure to the cephalosporins except for the substitution of an oxaazabicyclo moiety for the thiaazabicyclo moiety of certain cephalosporins. It has been proposed especially for the meningitid…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 3Penicillin-binding protein 1A +2
Waktu Paruh1.6 hours
Vol. Distribusi8.51 L
Klirens-
Genetik -
Latanoprost Approved DB00654
small molecule | CAS: 130209-82-4

Latanoprost is a prodrug analog of prostaglandin F2 alpha that is used to treat elevated intraocular pressure (IOP). It was initially approved by the FDA in 1998. Latanoprost is the first topical prostaglandin F2 alpha analog used for glaucoma treatment.[A184…

Kategori:
Antiglaucoma Preparations and MioticsAntihypertensive AgentsAutacoids +18
Target Protein:
Prostaglandin F2-alpha receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
Latanoprost acid Approved DB19360
small molecule | CAS: 41639-83-2

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Latanoprostene bunod Approved DB11660
small molecule | CAS: 860005-21-6

Latanoprostene Bunod has been used in trials studying the treatment of Glaucoma, Ocular Hypertension, Open-Angle Glaucoma, Open Angle Glaucoma, and Intraocular Pressure. As of November 2, 2017 the FDA approved Bausch + Lomb's Vyzulta (latanoprostene bunod …

Kategori:
Antiglaucoma Preparations and MioticsAutacoidsBiological Factors +12
Target Protein:
Prostaglandin F2-alpha receptor
Waktu ParuhThe half-life after…
Vol. DistribusiUnfortunately there…
KlirensSince latanoprost a…
Genetik -
Latiglutenase DB06326
biotech | CAS: 1360452-96-5

Deskripsi belum tersedia.

Kategori:
Celiac Disease, drug therapyEnzymesEnzymes and Coenzymes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Latozinemab DB16978
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Latrepirdine DB11725
small molecule | CAS: 3613-73-8

Latrepirdine has been investigated for the treatment of Alzheimer's Disease and Huntington's Disease.

Kategori:
Alzheimer DiseaseHeterocyclic Compounds, Fused-Ring
Target Protein:
5-hydroxytryptamine receptor 6Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Latrunculin A DB02621
small molecule | CAS: 76343-93-6

Latrunculin A is an actin binding macrolide purified from the red sea sponge Latrunculia magnifica. It is under investigation for the treatment of cancer. It disrupts actin polymerization, prevents mitotic spindle formation and thus cell replication.

Kategori:
PoriferaSulfur CompoundsThiazoles
Target Protein:
Actin, alpha skeletal muscleGelsolinIota toxin component Ia
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Latrunculin B DB08080
small molecule | CAS: 76343-94-7

Latrunculin B is a 14-membered macrolide attached to 2-thiazolidinone moiety, isolated from Red Sea sponge _Latrunculia magnifica_.

Kategori:
PoriferaSulfur CompoundsThiazoles
Target Protein:
Actin, alpha skeletal muscleMyocardin-related transcription factor AProtein spire homolog 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lauric acid Approved DB03017
small molecule | CAS: 143-07-7

Lauric acid is an inexpensive, non-toxic and safe to handle compound often used in laboratory investigations of melting-point depression. Lauric acid is a solid at room temperature but melts easily in boiling water, so liquid lauric acid can be treated with v…

Kategori:
Fatty AcidsLipids
Target Protein:
Toll-like receptor 4LactotransferrinPhospholipase A2, membrane associated +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Laurocapram Approved DB17308
small molecule | CAS: 59227-89-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 112-16-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 16610-63-2

Deskripsi belum tersedia.

Target Protein:
Farnesyl pyrophosphate synthaseGeranylgeranyl pyrophosphate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 27836-64-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LAVA-051 DB18395
biotech

LAVA-051 is a humanized V?9V?2-T cell-engaging bispecific antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavender oil Approved DB14566
biotech | CAS: 8000-28-0

Deskripsi belum tersedia.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavendustin A DB16768
small molecule | CAS: 125697-92-9

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesEnzyme InhibitorsTyrosine Kinase Inhibitors
Target Protein:
Epidermal growth factor receptorTyrosine-protein kinase Lck
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavendustin b DB16760
small molecule | CAS: 125697-91-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavoltidine DB12884
small molecule | CAS: 76956-02-0

Lavoltidine has been used in trials studying the diagnostic of Reflux, Gastroesophageal and Gastroesophageal Reflux Disease.

Kategori:
Gastric Acid Lowering AgentsHistamine AgentsHistamine Antagonists +2
Target Protein:
Histamine H2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lawsone DB04744
small molecule | CAS: 83-72-7

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsColoring Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LAX-101 DB05301
small molecule | CAS: 909712-41-0

LAX-101 treats hungtington’s disease, not just the symptoms but the disease itself. The active molecule in LAX-101 is Eicosapentaenoic Acid (EPA). All molecules of EPA are identical. The molecules of EPA found in LAX-101 are identical to the molecules of EPA …

Target Protein:
Phospholipase D1Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lazertinib Approved DB16216
small molecule | CAS: 1903008-80-9

Lazertinib is an oral, third-generation, epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI).[A264299, A264304] Lazertinib was first approved in South Korea on January 18, 2021, for the treatment of _EGFR_ T790M mutation-positive non-small…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +14
Target Protein:
Epidermal growth factor receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Lazuvapagon DB19046
small molecule | CAS: 2379889-71-9

Lazuvapagon is under investigation in clinical trial NCT03116191 (Trial of SK-1404 for Nocturia Due to Nocturnal Polyuria in Japanese Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LB-100 DB15412
small molecule | CAS: 1632032-53-1

LB-100 is under investigation in clinical trial NCT03886662 (A Study of LB-100 in Patients With Low or Intermediate-1 Risk Myelodysplastic Syndromes (MDS)).

Kategori:
Antineoplastic AgentsEnzyme Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LB-102 DB19214
small molecule | CAS: 2227154-23-4

LB-102 is under investigation in clinical trial NCT06179108 (Randomized, Double-blinded, Placebo-controlled, Evaluating the Treatment With LB-102 in Patients With Acute Schizophrenia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LCL-161 DB12085
small molecule | CAS: 1005342-46-0

LCL161 has been used in trials studying the treatment of Leukemia, Neoplasms, Solid Tumors, Breast Cancer, and Ovarian Cancer, among others.

Kategori:
Antineoplastic AgentsProto-Oncogene Proteins c-bcl-2, antagonists & inhibitorsSulfur Compounds
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2Baculoviral IAP repeat-containing protein 3 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LDN-193189 DB18051
small molecule | CAS: 1062368-24-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lebrikizumab Approved DB11914
biotech | CAS: 953400-68-5

Lebrikizumab is a monoclonal antibody that binds to IL-13 with high affinity and slow off-rate.[L51374] It binds to a different epitope compared [tralokinumab].[A262874,A262879] On November 17, 2023, lebrikizumab was approved by the EMA under the brand nam…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAntibodies +10
Target Protein:
Interleukin-13
Waktu ParuhThe mean eliminatio…
Vol. DistribusiBased on a populati…
KlirensIn the population P…
Genetik -
Lecanemab Approved DB14580
biotech | CAS: 1260393-98-3

Lecanemab is a recombinant humanized immunoglobulin gamma 1 (IgG1) monoclonal antibody directed against aggregated soluble and insoluble forms of amyloid beta (A?), which are implicated in the pathophysiology of Alzheimer’s disease.[L44537] Lecanemab works to…

Kategori:
Alzheimer DiseaseAlzheimer Disease, drug therapyAmino Acids, Peptides, and Proteins +12
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe mean value (95%…
KlirensThe clearance of le…
Genetik -
Lecithin DB15834
small molecule | CAS: 8002-43-5

A complex mixture of phospholipids, glycolipids, triglycerides, phosphatidylcholines, phosphatidylethanolamines, and phosphatidylinositols.

Kategori:
Biological ProductsComplex MixturesCompounds used in a research, industrial, or household setting +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 8030-76-0

A complex mixture of phospholipids; glycolipids; and triglycerides; with substantial amounts of phosphatidylcholines; phosphatidylethanolamines; and phosphatidylinositols, which are sometimes loosely termed as 1,2-diacyl-3-phosphocholines. Lecithin is a compo…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lecozotan DB12540
small molecule | CAS: 434283-16-6

Lecozotan has been used in trials studying the treatment of Alzheimer Disease.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT1 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 15-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ledipasvir Approved DB09027
small molecule | CAS: 1256388-51-8

Ledipasvir is a direct acting antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized int…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +10
Target Protein:
Genome polyproteinNonstructural protein 5A
Waktu ParuhThe median terminal…
Vol. Distribusi-
Klirens-
Genetik -
Lefamulin Approved DB12825
small molecule | CAS: 1061337-51-6

Lefamulin is a pleuromutilin antibiotic used for the treatment of bacterial community-acquired pneumonia. A pleuromotilin is a more recently developed type of antibiotic that is derived from the fungus, Pleurotus mutilus.[A183206] Lefamulin is available in in…

Kategori:
AcetatesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
50S ribosomal protein L22
Waktu ParuhThe average elimina…
Vol. DistribusiThe average volume …
KlirensThe total body clea…
Genetik -
Leflunomide Approved DB01097
small molecule | CAS: 75706-12-6

Leflunomide is a pyrimidine synthesis inhibitor belonging to the DMARD (disease-modifying antirheumatic drug) class of drugs, which are chemically and pharmacologically very heterogeneous. Leflunomide was approved by FDA and in many other countries (e.g., Can…

Kategori:
AdjuvantsAgents Causing Muscle ToxicityAntineoplastic and Immunomodulating Agents +16
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialDihydroorotate dehydrogenase (quinone), mitochondrialAryl hydrocarbon receptor +1
Gen Terkait:
CYP1A2
Waktu Paruh2 weeks
Vol. Distribusi* 0.13 L/kg
Klirens-
Genetik 1 Varian
Leflutrozole DB19047
small molecule | CAS: 143030-47-1

Leflutrozole is under investigation in clinical trial NCT02908074 (A 6 Month Safety Extension Study of MBGS205).

Kategori:
Aromatase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lemborexant Approved DB11951
small molecule | CAS: 1369764-02-2

Lemborexant is a novel dual orexin receptor antagonist used in the treatment of insomnia characterized by difficulties with sleep onset and/or sleep maintenance.[L10863] Recent research in the field of sleep disorders has revealed that insomnia is likely driv…

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP2B6 Inducers +17
Target Protein:
Orexin/Hypocretin receptor type 1Orexin receptor type 2
Waktu ParuhThe half-life for l…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Lemuteporfin DB04980
small molecule | CAS: 215808-49-4

Lemuteporfin, under development by QLT Incorporated, is a benzoporphyrin-derived chlorin-like photosensitizer. It is intended for the treatment of beign prostatic hyperplasia.

Kategori:
AlcoholsBiological FactorsGlycols +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lemzoparlimab DB17572
biotech | CAS: 2377483-71-9

Lemzoparlimab is under investigation in clinical trial NCT04912063 (Study to Evaluate Adverse Events and Movement of Lemzoparlimab in Body When Used Intravenously (IV) With Azacitidine Subcutaneously or IV and Venetoclax Orally in Participants With Acute Myel…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenabasum DB12193
small molecule | CAS: 137945-48-3

Ajulemic acid has been used in trials studying the treatment of Cystic Fibrosis, Dermatomyositis, and Diffuse Cutaneous Systemic Sclerosis.

Kategori:
Agents producing tachycardiaCannabinoid Receptor AgonistsCannabinoids and similars +5
Target Protein:
Tumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenacapavir Approved DB15673
small molecule | CAS: 2189684-44-2

HIV/AIDS remains an area of concern despite the introduction of numerous successful therapies, mainly due to the emergence of multidrug resistance and patient difficulty in adhering to treatment regimens.[A244170, A244175] Lenacapavir is a first-in-class caps…

Kategori:
AcetatesAcids, AcyclicAmides +17
Target Protein:
Gag-Pol polyprotein
Waktu ParuhThe median half-lif…
Vol. DistribusiThe steady state vo…
KlirensLenacapavir clearan…
Genetik -
Lenalidomide Approved DB00480
small molecule | CAS: 191732-72-6

Lenalidomide (previously referred to as CC-5013) is an immunomodulatory drug with potent antineoplastic, anti-angiogenic, and anti-inflammatory properties.[A228553] It is a 4-amino-glutamyl analogue of [thalidomide] [A228543] and like thalidomide, lenalidomid…

Kategori:
Acids, CarbocyclicAngiogenesis InhibitorsAngiogenesis Modulating Agents +18
Target Protein:
Tumor necrosis factorProtein cereblonTumor necrosis factor ligand superfamily member 11 +2
Waktu ParuhIn healthy subjects…
Vol. DistribusiIn healthy male sub…
KlirensThe renal clearance…
Genetik -
Leniolisib Approved DB16217
small molecule | CAS: 1354690-24-6

Leniolisib is a potent and selective inhibitor of phosphoinositide 3-kinase ? (PI3K?). The FDA approved leniolisib on March 24, 2023, making it the first treatment for activated phosphoinositide 3-kinase delta syndrome (APDS).[L45758] APDS is a primary immuno…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +14
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu ParuhThe effective half-…
Vol. DistribusiThe systemic decay …
KlirensIn one study, healt…
Genetik -
Lenomorelin DB11895
biotech | CAS: 258279-04-8

Lenomorelin has been investigated for the treatment and basic science of Cancer, Alcoholism, Metabolism, Hypopituitarism, and Frailty Syndrome, among others.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenvatinib Approved DB09078
small molecule | CAS: 417716-92-8

Lenvatinib is a receptor tyrosine kinase (RTK) inhibitor that inhibits the kinase activities of vascular endothelial growth factor (VEGF) receptors VEGFR1 (FLT1), VEGFR2 (KDR), and VEGFR3 (FLT4). Lenvatinib also inhibits other RTKs that have been implicated i…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +41
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +7
Waktu ParuhThe terminal elimin…
Vol. Distribusi-
Klirens-
Genetik -
Lenvervimab DB17814
biotech | CAS: 2055006-79-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenzilumab DB15148
biotech | CAS: 1229575-09-0

Lenzilumab is under investigation in clinical trial NCT02546284 (Study of Lenzilumab in Previously Treated Patients With Chronic Myelomonocytic Leukemia (CMML)).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lepirudin Approved DB00001
biotech | CAS: 138068-37-8

Lepirudin is a recombinant hirudin formed by 65 amino acids that acts as a highly specific and direct thrombin inhibitor.[L41539,L41569] Natural hirudin is an endogenous anticoagulant found in _Hirudo medicinalis_ leeches.[L41539] Lepirudin is produced in yea…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombin Proteins +12
Target Protein:
Prothrombin
Waktu ParuhLepirudin has an in…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of le…
Genetik -
Leptazoline B DB15552
small molecule

Leptazoline B is a polar oxazoline from the Cyanobacterium Leptolyngbya sp. Also see [Leptazoline A], [Leptazoline C], and [Leptazoline D].

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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