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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 164 / 236
Norethynodrel Approved DB09371
small molecule | CAS: 68-23-5

A synthetic progestational hormone with actions and uses similar to those of PROGESTERONE. It has been used in the treatment of functional uterine bleeding and endometriosis. As a contraceptive, it has usually been administered in combination with MESTRANOL.

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +18
Target Protein:
Estrogen receptorAndrogen receptorSex hormone-binding globulin
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Norfenefrine DB13378
small molecule | CAS: 536-21-0

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +14
Waktu Paruh-
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Norfloxacin Approved DB01059
small molecule | CAS: 70458-96-7

A synthetic fluoroquinolone (fluoroquinolones) with broad-spectrum antibacterial activity against most gram-negative and gram-positive bacteria. Norfloxacin inhibits bacterial DNA gyrase.

Kategori:
4-QuinolonesAgents Causing Muscle ToxicityAnti-Bacterial Agents +24
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA topoisomerase 4 subunit A +4
Waktu Paruh3-4 hours
Vol. Distribusi-
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Genetik -
Norflurane Approved DB13116
small molecule | CAS: 811-97-2

Norflurane is under investigation in clinical trial NCT01673061 (Vapocoolant Spray for Numbing Small Boils Before Incision and Drainage).

Kategori:
Aerosol PropellantsAerosolsAlkanes +8
Waktu Paruh-
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Norgestimate Approved DB00957
small molecule | CAS: 35189-28-7

Norgestimate was first described in the literature in 1977.[A191068] It was developed by Ortho Pharmaceutical Corporation as part of an effort to develop new hormonal contraceptives with reduced adverse effects.[A191068] It is commonly formulated with [ethiny…

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +27
Target Protein:
Progesterone receptorEstrogen receptorAndrogen receptor
Waktu ParuhNorgestimate is rap…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Norgestomet DB11440
small molecule | CAS: 25092-41-5

Norgestomet, also known as 11?-methyl-17-hydroxy-19-norprogesterone acetate, is a steroidal progestin used in veterinary medicine to control estrus and ovulation in cattle.

Kategori:
Fused-Ring CompoundsPregnanesPregnenes +2
Waktu Paruh-
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Norgestrel Approved DB09389
small molecule | CAS: 6533-00-2

Norgestrel is synthetic steroidal progestin that is used in combination with ethinyl estradiol for oral contraception. Norgestrel is composed of a racemic mixture of two stereoisomers, dextronorgestrel and levonorgestrel. However, only the levorotary enantio…

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +20
Target Protein:
Progesterone receptor3-oxo-5-alpha-steroid 4-dehydrogenase 1Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norleucine DB15458
small molecule | CAS: 327-57-1

Norleucine is under investigation in clinical trial NCT00081952 (Amino Acid Therapy for Hot Flashes in Postmenopausal Women).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAminocaproates
Target Protein:
Hepatocyte nuclear factor 1-alpha
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Normethadone Approved DB11609
small molecule | CAS: 467-85-6

Normethadone is used as an opioid antitussive in combination with [DB11610]. It is marketed in Canada by Valeant under the tradename Cophylac.

Kategori:
AnalgesicsAntitussive AgentsCentral Nervous System Agents +10
Waktu Paruh-
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Genetik -
small molecule | CAS: 156126-12-4

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Waktu Paruh-
Vol. Distribusi-
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Nortriptyline Approved DB00540
small molecule | CAS: 72-69-5

Nortriptyline hydrochloride, the active metabolite of [amitriptyline], is a tricyclic antidepressant (TCA).[L11878] It is used in the treatment of major depression and is also used off-label for chronic pain and other conditions.[L11881]

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +59
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +12
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +4
Waktu ParuhThe average plasma …
Vol. DistribusiThe apparent volume…
KlirensThe average plasma …
Genetik 7 Varian
small molecule | CAS: 99697-24-2

norUrsodeoxycholic acid is under investigation in clinical trial NCT03872921 (Norursodeoxycholic Acid vs Placebo in PSC).

Kategori:
Bile Acids and SaltsCholanesCholic Acids +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Noscapine Approved DB06174
small molecule | CAS: 128-62-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntitussive AgentsCentral Nervous System Agents +12
Target Protein:
Sigma non-opioid intracellular receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Novobiocin Approved DB01051
small molecule | CAS: 303-81-1

Novobiocin is an antibiotic compound derived from _Streptomyces niveus_. It has a chemical structure similar to coumarin. Novobiocin binds to DNA gyrase and blocks adenosine triphosphatase (ATPase) activity. (From Reynolds, Martindale The Extra Pharmacopoeia,…

Kategori:
AminocoumarinsAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA gyrase subunit B +1
Waktu Paruh6 hours
Vol. Distribusi-
Klirens-
Genetik -
Novolimus DB19085
small molecule | CAS: 151519-50-5

Novolimus is under investigation in clinical trial NCT04483791 (Dynamx Bioadaptor Hong Kong Registry).

Kategori:
LactonesPolyketides
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
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NOX-100 DB05799
small molecule

NOX-100 is the new nitric oxide (NO) neutralizing agent being developed by San Diego-based Medinox -- demonstrated its effectiveness and potential as a therapeutic to treat hemorrhagic shock. NOX-100 is the first in a series of proprietary NO neutralizing com…

Waktu Paruh-
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NOX-700 DB05464
small molecule

NOX-700, an new orally active dithiocarbamate-based nitric oxide (NO) blocking agent that is in development for the treatment of diabetes mellitus (type 2 diabetes). In animal studies, NOX-700 lowered serum glucose, improved glucose tolerance, and reduced the…

Kategori:
Acids, AcyclicCarbamatesSulfur Compounds
Target Protein:
Nuclear factor NF-kappa-B p100 subunitNuclear factor NF-kappa-B p105 subunit
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NP-10679 DB18040
small molecule | CAS: 2914889-88-4

Deskripsi belum tersedia.

Waktu Paruh-
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NP-6A4 DB17599
biotech

NP-6A4 is a peptide designed to specifically bind and activate angiotensin II receptor type 2 (AT2R). It has an Orphan Drug designation from the FDA for pediatric cardiomyopathy.[A258523]

Waktu Paruh-
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NP-G2-044 DB14995
small molecule | CAS: 1807454-59-6

NP-G2-044 is under investigation in clinical trial NCT03199586 (Phase 1 Clinical Trial of Metastasis Inhibitor NP-G2-044 in Patients With Advanced or Metastatic Solid Tumors (Including Lymphoma)).

Kategori:
Heterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Fascin
Waktu Paruh-
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Genetik -
NPT520-34 DB17920
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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NRC-AN-019 DB17110
small molecule | CAS: 879507-25-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +2
Waktu Paruh-
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NRX-1074 DB11784
small molecule | CAS: 1421866-48-9

NRX-1074 has been used in trials studying the treatment of Schizophrenia.

Waktu Paruh-
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NS-2359 DB05805
small molecule | CAS: 195875-68-4

NS2359 is a triple monoamine re-uptake inhibitor with a new, unique drug profile expected to yield important benefits compared to existing treatments of depression. Enhancing the function of the three neurotransmitters serotonin, noradrenalin and dopamine, NS…

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds +1
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NS-3728 DB05835
small molecule | CAS: 265646-85-3

NS3728 is an orally active chloride channel blocker for the treatment of cancer.

Kategori:
AmidesAminesAnilides +3
Waktu Paruh-
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NS-8593 DB16897
small molecule | CAS: 875755-39-8

Deskripsi belum tersedia.

Kategori:
AminesNaphthalenes
Waktu Paruh-
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NSC-663284 DB17038
small molecule | CAS: 383907-43-5

NSC-663284 is a potent quinolinedione Cdc25 phosphatase inhibitor.[A253052]

Kategori:
cdc25 Phosphatases, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
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NSI-189 DB16230
small molecule | CAS: 1270138-40-3

NSI-189 is under investigation in clinical trial NCT02695472 (Study of NSI-189 for Major Depressive Disorder).

Kategori:
AminesPyridines
Waktu Paruh-
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NSI-566 DB17954
biotech

NSI-566 is a stem cell therapy consisting of human spinal cord-derived neural stem cells. Developed by Seneca Biopharma, it is being investigated for the treatment of amyotrophic lateral sclerosis (ALS), stroke, and chronic spinal cord injury (cSCI).[L47097]

Waktu Paruh-
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NT 13 DB16953
small molecule | CAS: 117928-93-5

Deskripsi belum tersedia.

Waktu Paruh-
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NT-102 DB18112
small molecule | CAS: 1607447-79-9

Deskripsi belum tersedia.

Waktu Paruh-
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NT-219 DB17490
small molecule | CAS: 1198078-60-2

Deskripsi belum tersedia.

Target Protein:
Insulin receptor substrate 2Insulin receptor substrate 1Signal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NTLA-2002 DB17597
biotech

NTLA-2002 is a lipid nanoparticle encapsulating single guide RNA (G012267) targeting the human KLKB1 gene and messenger RNA (mRNA000042) encoding Cas9. It is an investigational therapy designed to knock out the target gene kallikrein B1 (KLKB1) to reduce plas…

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NU1025 DB02690
small molecule | CAS: 90417-38-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Poly [ADP-ribose] polymerase 1
Waktu Paruh-
Vol. Distribusi-
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NUC-7738 DB19148
small molecule | CAS: 2348493-39-8

NUC-7738 is under investigation in clinical trial NCT03829254 (A Safety, Pharmacokinetic and Clinical Activity Study of NUC-7738 in Patients With Advanced Solid Tumours and Lymphoma).

Kategori:
Benzene DerivativesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Nurulimab DB18946
biotech | CAS: 2168561-20-2

Nurulimab is under investigation in clinical trial NCT05732805 (A Clinical Study of BCD-217 (Nurulimab + Prolgolimab) Followed by Anti-pd-1 Compared to Anti-pd-1 Monotherapy as First-line Treatment in Subjects With Unresectable/metastatic Melanoma).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates
Waktu Paruh-
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Nutlin-3 DB17039
small molecule | CAS: 548472-68-0

Nutlin-3 is a small molecule inhibitor that targets p53-Mdm2 interaction.[A253057]

Kategori:
Stereoisomerism
Target Protein:
Cellular tumor antigen p53
Waktu Paruh-
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Nutmeg Approved DB10676
biotech

Nutmeg allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +2
Waktu Paruh-
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Nuvaxovid Approved DB15810
biotech

SARS-CoV-2, the causative agent of COVID-19, relies on the interaction between its trimeric spike (S) glycoprotein and angiotensin-converting enzyme 2 (hACE2) expressed on host cells in order to establish a productive infection in humans.[A243789] Antibodies …

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
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biotech | CAS: 8046-97-7

Deskripsi belum tersedia.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NV-07a DB05845
small molecule

NV-07a is topical skin repair compound protecting skin from sun-induced immunosuppression and UV-induced damage.

Waktu Paruh-
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NV-5138 DB19180
small molecule | CAS: 2095886-80-7

NV-5138 is under investigation in clinical trial NCT06235905 (Open-label of SPN-820 in Adults With Major Depressive Disorder).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +1
Waktu Paruh-
Vol. Distribusi-
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NV-52 DB05673
small molecule

NV-52 is an investigational synthetic flavonoid thromboxane synthase (TXS) inhibitor developed for the maintenance of remission in inflammatory bowel disease.

Target Protein:
Thromboxane-A synthase
Waktu Paruh-
Vol. Distribusi-
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NVP-LEQ-506 DB12857
small molecule | CAS: 1204975-42-7

LEQ506 has been used in trials studying the treatment of Advanced Solid Tumors, Recurrent or Refractory Medulloblastoma, and Locally Advanced or Metastatic Basal Cell Carcinoma.

Target Protein:
Protein smoothened
Waktu Paruh-
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NX-1207 DB05493
small molecule

NX-1207 is an investigational new drug for BPH, whose chemical entity and mechanism of action remain undisclosed. Nymox Pharmaceutical Corporation recently completed studies of NX-1207 for treatment of benign prostatic hyperplasia (BPH).

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
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Genetik -
biotech

NY-ESO-1 peptide vaccine is an investigational cancer immunotherapy. It contains a peptide derived from the cancer-testis antigen (NY-ESO-1).

Waktu Paruh-
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Nylidrin Approved DB06152
small molecule | CAS: 447-41-6

Nylidrin, also known as _buphenine_ belongs to the category of drugs called _vasodilators_, which relax blood vessels and increase blood flow. Nylidrin is a peripheral vasodilator. Some studies show the evidence of improving cognitive impairment in selected i…

Kategori:
2-Amino-1-Phenylethanol DerivativesAdrenergic AgentsAdrenergic Agonists +29
Target Protein:
Interferon alpha/beta receptor 2Voltage-dependent T-type calcium channel subunit alpha-1I
Waktu ParuhDuration of action …
Vol. Distribusi-
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Nystatin Approved DB00646
small molecule | CAS: 1400-61-9

Nystatin is a polyene antifungal drug that has broad-spectrum fungicidal and fungistatic activity against a number of yeasts and fungi, most notably _Candida_ species.[L10686] It is one of the most effective antifungal agents synthesized by bacteria, in this …

Kategori:
Alimentary Tract and MetabolismAnti-Infective AgentsAntidiarrheals, Intestinal Antiinflammatory/antiinfective Agents +17
Target Protein:
Ergosterol
Waktu Paruh-
Vol. DistribusiNystatin is not abs…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
4-hydroxy-tetrahydrodipicolinate synthase
Waktu Paruh-
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Genetik -
NZ-1002 DB17688
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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