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12560

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9109 (72.5%)
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12560 (100.0%)

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Halaman 164 / 252
Mosunetuzumab Approved DB15434
biotech | CAS: 1905409-39-3

Mosunetuzumab is a humanized anti-CD20/CD3 bispecific antibody.[L42230] It can recognize and bind two different targets simultaneously, CD20 on cancer B-cells and CD3 on T-cells, allowing it to redirect T-cell cytotoxic activity to cancer cells.[A249320] The …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +13
Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3 epsilon chain
Waktu ParuhMosunetuzumab has a…
Vol. DistribusiThe estimated centr…
KlirensThe mean steady-sta…
Genetik -
Motesanib DB05575
small molecule | CAS: 453562-69-1

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingNicotinic Acids +3
Target Protein:
Vascular endothelial growth factor receptor 2Mast/stem cell growth factor receptor Kit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 246252-06-2

Motexafin gadolinium is studied in the treatment of cancer by Pharmacyclics. It may make tumor cells more sensitive to radiation therapy, improve tumor images using magnetic resonance imaging (MRI), and kill cancer cells. It belongs to the family of drugs cal…

Kategori:
Antineoplastic AgentsBiological FactorsCompounds used in a research, industrial, or household setting +9
Target Protein:
Peroxiredoxin-5, mitochondrialThioredoxin reductase 1, cytoplasmicThioredoxin reductase 2, mitochondrial +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 246252-04-0

Motexafin lutetium (MLu) is a second-generation photosensitizer for photodynamic therapy (PDT) of cancer. It belongs to the family of drugs called metallotexaphyrins. Also called lutetium texaphyrin. Motexafin lutetium is a pentadentate aromatic metallotexaph…

Kategori:
Biological FactorsCoordination ComplexesDermatologicals +5
Target Protein:
Prostate-specific antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Motixafortide Approved DB14939
biotech | CAS: 664334-36-5

Motixafortide is a cyclic peptide hematopoietic stem cell mobilizer used to improve stem cell collection prior to autologous transplantation.[L48116] Hematopoietic stem cell transplantation (HSCT) is commonly employed in the context of hematologic cancers - h…

Kategori:
Amino Acids, Peptides, and ProteinsHematopoietic Stem Cell MobilizerPeptides
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhThe effective half-…
Vol. DistribusiIn a typical patien…
KlirensIn a typical patien…
Genetik -
Motretinide DB13368
small molecule | CAS: 56281-36-8

Deskripsi belum tersedia.

Kategori:
AlkenesAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moxaverine DB12251
small molecule | CAS: 10539-19-2

Moxaverine has been investigated for the treatment of Retina, Ocular Physiology, and Regional Blood Flow.

Kategori:
Alimentary Tract and MetabolismAlkaloidsAutonomic Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moxestrol DB13418
small molecule | CAS: 34816-55-2

Deskripsi belum tersedia.

Kategori:
Estradiol CongenersEstrogen AntagonistsEstrogenic Steroids, Alkylated +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moxetumomab pasudotox Approved DB12688
biotech | CAS: 1020748-57-5

CD22 is a lineage-restricted B-cell antigen that is expressed solely in on B-chronic lymphocytic leukemia, hairy cell leukemia, acute lymphocytic leukemiathe and Burkitt's lymphoma. The predecessor of Moxetumab pasudotox (MxP), named BL22, was first created b…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
B-cell receptor CD22Elongation factor 2
Waktu ParuhMxP presents a shor…
Vol. DistribusiThe mean volume of …
KlirensThe mean systemic c…
Genetik -
Moxidectin Approved DB11431
small molecule | CAS: 113507-06-5

Moxidectin is a potent, broad-spectrum endectocide (antiparasitic that is active against endo- and ecto-parasites) with activity against nematodes, insects, and acari. It was first used in cattle followed by an approved use in general animals. It is a semi-sy…

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +9
Target Protein:
Glutamate-gated chloride channelGABA-A gated chloride channelABC transporters
Waktu ParuhMoxidectin reporter…
Vol. DistribusiMoxidectin presents…
KlirensThe apparent cleara…
Genetik -
Moxifloxacin Approved DB00218
small molecule | CAS: 151096-09-2

Moxifloxacin is a synthetic fluoroquinolone antibiotic agent. Bayer AG developed the drug (initially called BAY 12-8039) and it is marketed worldwide (as the hydrochloride) under the brand name Avelox (in some countries also Avalox) for oral treatment.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +18
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +3
Waktu Paruh11.5-15.6 hours (si…
Vol. Distribusi* 1.7 to 2.7 L/kg
Klirens* 12 +/- 2 L/hr
Genetik -
Moxisylyte Approved DB09205
small molecule | CAS: 54-32-0

Moxisylyte, denominated as thymoxamine in the UK, is a specific and orally active ?1-adrenergic antagonist.[T45] According to the WHO, moxisylyte is approved since 1987[T91] and in the same year, it acquired the denomination of orphan product by the FDA.[L117…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +17
Target Protein:
Alpha-1D adrenergic receptorAlpha adrenergic receptor
Waktu ParuhThe half-life of mo…
Vol. DistribusiIn preclinical tria…
KlirensIn preclinical tria…
Genetik -
Moxonidine Approved DB09242
small molecule | CAS: 75438-57-2

Moxonidine is a new-generation centrally acting antihypertensive drug approved for the treatment of mild to moderate essential hypertension. It is suggested to be effective in cases where other agents such as thiazides, beta-blockers, ACE inhibitors, and calc…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +8
Target Protein:
Alpha-2C adrenergic receptorAlpha-2B adrenergic receptorAlpha-2A adrenergic receptor +1
Waktu ParuhPlasma elimination …
Vol. Distribusi1.8±0.4L/kg. [FDA l…
KlirensAdministered twice …
Genetik -
Mozenavir DB02102
small molecule | CAS: 174391-92-5

Deskripsi belum tersedia.

Kategori:
Amides
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MP-0250 DB17218
biotech | CAS: 1816305-70-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MP4 DB05313
small molecule

MP4 is a hemoglobin-based oxygen carrier designed to serve as an alternative for blood transfusions. It is free of harmful vasoactivity and provides targeted oxygen delivery to tissues at risk of oxygen deprivation.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPB-1523 DB18334
small molecule

MPB-1523 is a contrast agent comprising PEGylated iron oxide nanoparticles.[L48161]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPI-674 DB05749
small molecule

MPI-674 is an aromatase inhibitor (AI) with a well-established, multi-year chronic safety and tolerability profile. AIs are a class of drugs that reduce the amount of estrogen circulating in the body by binding to and inhibiting the enzyme aromatase, which i…

Target Protein:
Aromatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPT-0L055 DB17136
small molecule | CAS: 2069950-14-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPT0B640 DB16512
small molecule

MPT0B640 was under investigation in clinical trials NCT04526717 for COVID-19 infection and NCT04294875 for locally advanced or metastatic solid malignancies.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRK-003 DB17015
small molecule | CAS: 623165-93-5

MRK-003 is a potent and selective ?-secretase inhibitor developed by Merck. It is the preclinical analog of [MK-0752], a drug in clinical development.[A252682]

Kategori:
Amyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme InhibitorsGamma Secretase Inhibitors and Modulators +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRK-409 DB13993
small molecule | CAS: 233275-76-8

MRK-409 is a GABA-A receptor agonist [A31972].

Kategori:
Anti-Anxiety AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-1345 DB18739
biotech

mRNA-1345 is an investigational RSV vaccine.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3351 DB17718
biotech

mRNA-3351 is a modified mRNA encoding the UGT1A1 gene. Developed by Moderna, it is currently being investigated as the treatment for Crigler-Najjar syndrome

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3705 DB17668
biotech

mRNA-3705 is an investigational mRNA encoding methylmalonic CoA mutase (MUT) enzyme. Developed by Moderna TX Inc., it is being investigated for the treatment of methylmalonic academia.[A258843]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3745 DB18554
biotech

mRNA-3745 is a lipid nanoparticle (LNP) encapsulated with nucleoside-modified, codon-optimized mRNAs encoding human glucose 6-phosphatase (G6Pase).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3927 DB17669
biotech

mRNA-3927 is an investigational mRNA therapy that consists of two mRNAs that encode for the alpha and beta subunits of the mitochondrial enzyme propionyl-CoA carboxylase (PCC) encapsulated within a lipid nanoparticle (LNP). Developed by Moderna Inc., it is be…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRT-2359 DB18015
small molecule | CAS: 2803881-11-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRT5005 DB18260
biotech

MRT5005 is a human cystic fibrosis transmembrane conductance regulator (hCFTR) messenger RNA (mRNA) complexed with branched polyethyleneimine (bPEI).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRT5201 DB17656
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
MRx-4DP0004 DB15751
biotech

MRx-4DP0004 is a lyophilised formulation of the Bifidobacterium breve strain of commensal bacteria. It is a live biotherapeutic derived from the microbiota of a healthy human infant.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRx0518 DB17523
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MS-1819 DB15004
biotech

MS-1819 is under investigation in clinical trial NCT03481803 (A Phase IIa Study With Escalating Dose of MS1819-SD).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MSX-122 DB12715
small molecule | CAS: 897657-95-3

MSX-122 has been used in trials studying the treatment of Solid Tumors.

Kategori:
Receptors, CXCR4, antagonists & inhibitors
Target Protein:
C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MTL-CEBPA DB18143
biotech

MTL-CEBPA is a SMARTICLES liposomal formulation of MTL-501, a small activating RNA (saRNA) oligonucleotide.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
OxidoreductaseNitrous-oxide reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mubodina DB17616
biotech

Mubodina is an investigational drug developed by Adienne Pharma & Biotech. It is a recombinant human minibody directed against complement component C5. It was investigated in various conditions including primary membranoproliferative glomerulonephritis and ty…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Dendritic Cell (DC) Therapy is a newly emerging and potent form of immune therapy that amplifies the actions of the body's own immune system to help fight cancer, AIDS and other serious conditions. The Dendritic Cell is an immune cell whose role is the recogn…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Mucor circinelloides f. circinelloides allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Mucor circinelloides f. lusitanicus allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mufemilast DB18075
small molecule | CAS: 1255909-03-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MUL001 DB18534
biotech

MUL001 is live attenuated strain of _Salmonella typhimurium_ being investigated for the treatment of schwannomas.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MultiStem DB15742
biotech

MultiStem is an intravenously-administered, off-the-shelf proprietary product developed which comprises Multipotent Adult Progenitor Cells (MAPCs). Like mesenchymal stem cells, MAPCs are derived from bone-marrow stroma and are non-hematopoietically adherent. …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Muparfostat DB05808
small molecule | CAS: 1020105-89-8

Muparfostat (PI-88) is a mixture of highly sulfated, monophosphorylated mannose oligosaccharides, derived from the extracellular phosphomannan of the yeast Pichia (Hansenula) holstii, with potential antiangiogenic activity.

Kategori:
CarbohydratesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mupirocin Approved DB00410
small molecule | CAS: 12650-69-0

Mupirocin, formerly termed pseudomonic acid A,[A178531] is a novel antibacterial agent with a unique chemical structure and mode of action apart from other antibiotic agents. Produced by fermentation using the organism _Pseudomonas fluorescens_, mupirocin is …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics for Topical Use +12
Target Protein:
Isoleucine--tRNA ligase
Waktu ParuhIn healthy male vol…
Vol. DistribusiNo information avai…
KlirensNo information avai…
Genetik -
Muplestim DB12431
biotech | CAS: 148641-02-5

Muplestim is under investigation in clinical trial NCT00002258 (A Phase I, Open Label Trial to Evaluate the Safety, Tolerance and Biological Effects of SDZ ILE-964 (Recombinant Human Interleukin-3, RhIL-3) in HIV Infected Patients With Cytopenia).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Muraglitazar DB06510
small molecule | CAS: 331741-94-7

Muraglitazar (Bristol-Myers Squibb/Merck) is a new agent under investigation for the treatment of patients with type 2 diabetes. It belongs to a novel class of drugs that target the peroxisome proliferator-activated receptors, both alpha and gamma subtypes. I…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsCytochrome P-450 CYP1A2 Substrates +6
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mureletecan DB15020
small molecule | CAS: 246527-99-1

Mureletecan is under investigation in clinical trial NCT00004076 (PNU 166148 in Treating Patients With Metastatic Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Murepavadin DB14777
small molecule | CAS: 944252-63-5

Murepavadin is under investigation in clinical trial NCT02110459 (Pharmacokinetics and Safety of POL7080 in Patients With Renal Impairment).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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