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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 163 / 236
Nitrendipine Approved DB01054
small molecule | CAS: 39562-70-4

Nitrendipine is a calcium channel blocker with marked vasodilator action. It is an effective antihypertensive agent and differs from other calcium channel blockers in that it does not reduce glomerular filtration rate and is mildly natriuretic, rather than so…

Kategori:
ACE Inhibitors and Calcium Channel BlockersAgents causing hyperkalemiaAntiarrhythmic agents +21
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitric acid DB15995
small molecule | CAS: 7697-37-2

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicCompounds used in a research, industrial, or household setting +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitrite Approved DB12529
small molecule | CAS: 14797-65-0

Nitrite is under investigation for the treatment of Heart Failure.

Kategori:
AnionsElectrolytesIons +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitroarginine DB04223
small molecule | CAS: 2149-70-4

An inhibitor of nitric oxide synthetase which has been shown to prevent glutamate toxicity. Nitroarginine has been experimentally tested for its ability to prevent ammonia toxicity and ammonia-induced alterations in brain energy and ammonia metabolites. (Neur…

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +3
Target Protein:
Nitric oxide synthase 1Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitroaspirin DB12445
small molecule | CAS: 175033-36-0

Nitroaspirin has been investigated for the treatment of Intermittent Claudication.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +19
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitrofural Approved DB00336
small molecule | CAS: 59-87-0

Nitrofural or nitrofurazone is a topical anti-infective agent effective against gram-negative and gram-positive bacteria. It is used for superficial wounds, burns, ulcers, and skin infections. Nitrofural has also been administered orally in the treatment of t…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Products, Insecticides and Repellents +15
Target Protein:
Glutathione reductase
Waktu Paruh5 hours
Vol. Distribusi-
Klirens-
Genetik -
Nitrofurantoin Approved DB00698
small molecule | CAS: 67-20-9

Nitrofurantoin is a nitrofuran antibiotic used to treat uncomplicated urinary tract infections.[L6856,L6859,L6862] Nitrofurantoin is converted by bacterial nitroreductases to electrophilic intermediates which inhibit the citric acid cycle as well as synthesis…

Kategori:
Agents causing hyperkalemiaAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
Probable pyruvate-flavodoxin oxidoreductaseOxygen-insensitive NADPH nitroreductase30S ribosomal protein S10
Waktu ParuhThe half life of ni…
Vol. DistribusiData regarding the …
KlirensThe clearance of ni…
Genetik -
Nitrogen Approved DB09152
small molecule | CAS: 7727-37-9

Nitrogen is a chemical element with symbol N and atomic number 7. At room temperature, it is a transparent, odorless diatomic gas. Liquid nitrogen is used principally in cryotherapy for removal of diseased skin. Liquid nitrogen helps in removal of skin lesi…

Kategori:
ElementsGasesMedical Gases +2
Waktu ParuhFor local use only.
Vol. DistribusiFor local use only.
KlirensFor local use only.
Genetik -
Nitroglycerin Approved DB00727
small molecule | CAS: 55-63-0

Nitroglycerin, also known as glyceryl trinitrate,[A180169] is an organic nitrate and a vasodilating agent [L38369] that was first discovered in 1847.[A249965] Originally used to dynamite, its antianginal effects were identified in the late 1860s after it prod…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAntianginal AgentsAntihypertensive Agents +14
Target Protein:
Epidermal growth factor receptorGuanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1 +1
Waktu ParuhFollowing intraveno…
Vol. DistribusiThe volume of distr…
KlirensThe estimated clear…
Genetik -
Nitroprusside Approved DB00325
small molecule | CAS: 15078-28-1

Nitroprusside serves as a source of nitric oxide, a potent peripheral vasodilator that affects both arterioles and venules (venules more than arterioles). Nitroprusside is often administered intravenously to patients who are experiencing a hypertensive emerge…

Kategori:
AnionsAntihypertensive AgentsArteriolar Smooth Muscle, Agents Acting On +20
Target Protein:
Guanylate cyclase soluble subunit alpha-1Guanylate cyclase soluble subunit beta-1Atrial natriuretic peptide receptor 1
Waktu ParuhApproximately 2 min…
Vol. Distribusi-
Klirens-
Genetik -
Nitrosoethane DB02646
small molecule | CAS: 925-91-7

Deskripsi belum tersedia.

Target Protein:
Myoglobin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitrous acid Approved DB09112
small molecule | CAS: 7782-77-6

Nitrous acid (as sodium nitrite) is used as part of an intravenous mixture with sodium thiosulfate to treat cyanide poisoning. It is on the World Health Organization's List of Essential Medicines, a list of the most important medications needed in a basic hea…

Kategori:
AcidsAcids, NoncarboxylicAnions +16
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit betaMyoglobin
Waktu ParuhHalf life of 0.4-0.…
Vol. Distribusi-
Klirens-
Genetik -
Nitrous oxide Approved DB06690
small molecule | CAS: 10024-97-2

Nitrous oxide, commonly known as "laughing gas", is a chemical compound with the chemical formula N2O. At room temperature, it is a colorless non-flammable gas, with a pleasant, slightly sweet odor and taste. It is used in surgery and dentistry for its anesth…

Kategori:
Agents that produce hypertensionAnalgesicsAnalgesics, Non-Narcotic +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nitroxoline DB01422
small molecule | CAS: 4008-48-4

Nitroxoline is a urinary antibacterial agent active against susceptible gram-positive and gram-negative organisms commonly found in urinary tract infections. It is a hydroxyquinoline derivative unrelated to other classes of drugs.[A179251] Nitroxoline is acti…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +5
Target Protein:
Methionine aminopeptidase 2Magnesium cationManganese cation
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nivatrotamab DB16654
biotech | CAS: 2278244-14-5

Nivatrotamab is under investigation in clinical trial NCT03860207 (Study of the Safety and Efficacy of Humanized 3F8 Bispecific Antibody (Hu3f8-bsab) in Patients With Relapsed/refractory Neuroblastoma, Osteosarcoma and Other Solid Tumor Cancers).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nivocasan DB12720
small molecule | CAS: 908253-63-4

Nivocasan has been used in trials studying the treatment of HCV Infection and Nonalcoholic Steatohepatitis.

Target Protein:
Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nix-0699 DB17732
biotech

Deskripsi belum tersedia.

Kategori:
Anemia, Sickle Cell, drug therapyBiological ProductsComplex Mixtures +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nizatidine Approved DB00585
small molecule | CAS: 76963-41-2

A histamine H2 receptor antagonist with low toxicity that inhibits gastric acid secretion. The drug is used for the treatment of duodenal ulcers.

Kategori:
Acid ReducersAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +13
Target Protein:
Histamine H2 receptor
Waktu Paruh1-2 hours
Vol. Distribusi* 0.8 to 1.5 L/kg
Klirens* 40-60 L/h * 7 – …
Genetik -
biotech

These cells are prepared as universal off-the-shelf CAR-NK cells from cord blood with NKG2D-ACE2 proteins engineered as part of the CARs; the cell secretes IL-15 and GM-CSF. Chimeric antigen receptors (CARs) are artificial receptors consisting of an antibody-…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NKTT-120 DB17730
biotech

NKTT-120 is a recombinant humanized IgG1k monoclonal antibody to human invariant T cell receptor (iTCR).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NM-3 DB12818
small molecule | CAS: 181427-78-1

NM-3 has been used in trials studying the treatment of Neoplasms.

Target Protein:
Vascular endothelial growth factor A, long formVascular endothelial growth factor BVascular endothelial growth factor C +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NM-702 DB05505
small molecule

Nissan Chemical and Taisho have been jointly developing NM-702, a drug for the treatment of arteriosclerosis obliterans. M-702 is an orally active inhibitor of phosphodiesterase and thromboxane synthetase. In Japan, Phase 2 studies are being conducted for …

Target Protein:
Thromboxane-A synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NM3086 DB17719
biotech

NM3086 is a recombinant, humanized, aglycosylated, IgG1-kappa anti-properdin monoclonal antibody being developed by Novelmed Therapeutics Inc.[L46193]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NMD-670 DB18466
small molecule | CAS: 2354321-33-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 357400-14-7

NNC-55-0396 is a T-type Ca(2+) channel inhibitor.[A253047]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NNI-351 DB18048
small molecule | CAS: 929607-23-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NNZ-2591 DB15601
small molecule | CAS: 847952-38-9

NNZ-2591 (cyclo-L-glycyl-L-2-allylproline)[A189390] is an investigational synthetic analog of cyclic glycine-proline (cGP), a breakdown product of human insulin-like growth factor 1 (IGF-1), that has been chemically modified to increase its half-life, stabili…

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPiperazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nofazinlimab DB18852
biotech | CAS: 2377845-98-0

Nofazinlimab is under investigation in clinical trial NCT04194775 (A Study of Nofazinlimab (CS1003) in Subjects With Advanced Hepatocellular Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nogapendekin alfa Approved DB18740
biotech | CAS: 1622189-43-8

Nogapendekin alfa is a human IL-15N72D variant. It is one of the active ingredients in Anktiva, a combination product also containing [inbakicept], where a single inbakicept is complexed with two nogapendekin alfa components.[L50592] This combination product …

Kategori:
Amino Acids, Peptides, and ProteinsInterleukin-15Proteins +2
Target Protein:
Interleukin-2 receptor subunit betaCytokine receptor common subunit gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Glycogen phosphorylase, muscle formLactase-like proteinLactase/phlorizin hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nolasiban DB16259
small molecule | CAS: 1477482-19-1

Nolasiban is under investigation in clinical trial NCT03081208 (Phase 3 Placebo Controlled Study of Nolasiban to Improve Pregnancy Rates in Women Undergoing IVF/ICSI).

Kategori:
AminesHydroxylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nolatrexed DB12912
small molecule | CAS: 147149-76-6

Nolatrexed is under investigation in clinical trial NCT00012324 (Nolatrexed Dihydrochloride Compared With Doxorubicin in Treating Patients With Recurrent or Unresectable Liver Cancer).

Kategori:
AntimetabolitesAntineoplastic AgentsEnzyme Inhibitors +5
Target Protein:
Thymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 153050-21-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomacopan DB14991
biotech | CAS: 875125-19-2

Nomacopan is under investigation in clinical trial NCT03427060 (Coversin in PNH in Patients With Resistance to Eculizumab Due to Complement C5 Polymorphisms).

Kategori:
Recombinant Protein Inhibitor of Complement Factor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomegestrol acetate Approved DB13981
small molecule | CAS: 58652-20-3

Nomegestrol acetate, also known as NOMAC, is a progestin used in oral contraceptives, menopausal hormone therapy, and for the treatment of gynecological disorders.

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +14
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomifensine Approved DB04821
small molecule | CAS: 24526-64-5

Nomifensine, formerly marketed as Merital capsules, was associated with an increased incidence of hemolytic anemia. The approved application holder removed Merital capsules from the market on January 23, 1986. FDA published a notice of its determination that …

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsDopamine Agents +8
Target Protein:
D(2) dopamine receptorSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nomlabofusp DB17903
biotech | CAS: 2548202-05-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nona-arginine DB12648
small molecule | CAS: 143413-47-2

Nona-arginine is under investigation in clinical trial NCT00264706 (PolyArginine Treated vEiN grafTs (PATENT)).

Kategori:
Amino Acids, Peptides, and ProteinsFurin, antagonists & inhibitorsPeptides
Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nonacog beta pegol Approved DB13933
biotech | CAS: 1175512-71-6

Nonacog beta pegol is a recombinant coagulation factor IX derivative. It is produced without animal-derived materials and with an attached 40kDa polyethylene glycol (PEG) molecule for peptide activation by a site-directed glycoPEGylation. Once activated, the …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +10
Target Protein:
Coagulation factor VIICoagulation factor VIIICoagulation factor X
Waktu ParuhThe mean half-life …
Vol. DistribusiThe volume of distr…
KlirensMean clearance in c…
Genetik -
Nonan-1-Ol DB03143
small molecule | CAS: 28473-21-4

Deskripsi belum tersedia.

Target Protein:
ATP synthase subunit c, sodium ion specific
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nonivamide DB11324
small molecule | CAS: 2444-46-4

Nonivamide is found in herbs and spices. It is an alkaloid from the Capsicum species. The structures of [DB06774] and nonivamide differ only slightly with respect to the fatty acid moiety of the side chain (8-methyl nonenoic acid versus nonanoic acid) [F31]. …

Kategori:
Acids, CarbocyclicAlkaloidsAlkenes +20
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu ParuhAbout 7 minutes [F3…
Vol. Distribusi-
Klirens-
Genetik -
Nonoxynol-9 Approved DB06804
small molecule | CAS: 26027-38-3

Nonoxynol-9 (N-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives. When present in the vagina during intercourse, they immobilize/inactivate/damage and/or kill sperms without eliciting systemic …

Kategori:
Adrenal Cortex HormonesAlcoholsAntispermatogenic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NOP-1A DB15208
small molecule | CAS: 1283095-70-4

NOP-1A is under investigation in clinical trial NCT01198197 (PET Brain and Whole Body Distribution Studies for Nociceptin/Orphanin FQ Peptide (NOP) Receptor Using [11C]NOP-1A).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
nor-NOHA DB02381
small molecule | CAS: 189302-40-7

N-Hydroxy-nor-L-arginine (nor-NOHA) is under investigation in clinical trial NCT02009527 (Arginase Inhibition in Ischemia-reperfusion Injury).

Target Protein:
Arginase-2, mitochondrialArginase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norclobazam DB17092
small molecule | CAS: 22316-55-8

Deskripsi belum tersedia.

Kategori:
AnticonvulsantsBenzazepinesCentral Nervous System Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norclozapine DB05766
small molecule | CAS: 6104-71-8

ACP-104, or N-desmethylclozapine, is the major metabolite of clozapine, and is being developed by ACADIA as a novel, stand-alone therapy for schizophrenia. It combines an atypical antipsychotic efficacy profile with the added potential benefit of enhanced cog…

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +4
Target Protein:
Muscarinic acetylcholine receptor M1D(2) dopamine receptorD(3) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norelgestromin Approved DB06713
small molecule | CAS: 53016-31-2

Norelgestromin is a drug used in contraception. Norelgestromin is the active progestin responsible for the progestational activity that occurs in women after application of ORTHO EVRA patch.

Kategori:
Adrenal Cortex HormonesAminesCombination Contraceptives (with Estrogen and derivatives) +17
Target Protein:
Progesterone receptorAlbuminAndrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norethandrolone DB12787
small molecule | CAS: 52-78-8

Norethandrolone is under investigation in clinical trial NCT00700544 (Treatment Outcome in Elderly Patients).

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3836-23-5

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Norethisterone Approved DB00717
small molecule | CAS: 68-22-4

Norethisterone, also known as norethindrone, is a synthetic progestational hormone belonging to the 19-nortestosterone-derived class of progestins.[A10367] It is further classified as a second-generation progestin, along with [levonorgestrel] and its derivati…

Kategori:
Adrenal Cortex HormonesAnti-Gonadotropin-Releasing HormonesCombination Contraceptives (with Estrogen and derivatives) +34
Target Protein:
Progesterone receptorAndrogen receptorGlucocorticoid receptor
Waktu ParuhThe half-life of no…
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
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