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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 163 / 252
Modimelanotide DB15314
small molecule | CAS: 926277-68-1

Modimelanotide is under investigation in clinical trial NCT01897519 (A Safety and Efficacy Trial of Multiple Dosing Regimens of ABT-719 for the Prevention of Acute Kidney Injury in Subjects Undergoing High Risk Surgery).

Kategori:
Pyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modipafant DB16237
small molecule | CAS: 122957-06-6

Modipafant is under investigation in clinical trial NCT02569827 (Celgosivir or Modipafant as Treatment for Adult Participants With Uncomplicated Dengue Fever in Singapore).

Kategori:
Pyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modithromycin DB16238
small molecule | CAS: 736992-12-4

Modithromycin is under investigation in clinical trial NCT00270517 (Comparative Study of EDP-420 Versus Another Antibiotic in the Treatment of Community Acquired Pneumonia).

Kategori:
LactonesPolyketides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modotuximab DB14827
biotech | CAS: 1310460-86-6

Modotuximab is under investigation in clinical trial NCT03549338 (Sym004 Versus Futuximab or Modotuximab in Patients With mCRC).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modufolin DB12676
small molecule | CAS: 31690-11-6

Modufolin is under investigation for the treatment of Osteosarcoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moexipril Approved DB00691
small molecule | CAS: 103775-10-6

Moexipril is a non-sulfhydryl containing precursor of the active angiotensin-converting enzyme (ACE) inhibitor moexiprilat. It is used to treat high blood pressure (hypertension). It works by relaxing blood vessels, causing them to widen. Lowering high blood …

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +14
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhMoexipril eliminati…
Vol. Distribusi* 183 L
Klirens* 441 mL/min
Genetik -
Moexiprilat DB14210
small molecule | CAS: 103775-14-0

The active metabolite of the prodrug [Moexipril].

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAngiotensin-Converting Enzyme Inhibitors +2
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mogamulizumab Approved DB12498
biotech | CAS: 1159266-37-1

Mogamulizumab is a humanized monoclonal antibody (mAb) directed against CC chemokine receptor 4 (CCR4) for the treatment of Mycosis Fungoides (MF) and Sézary Syndrome (SS), the most common subtypes of cutaneous T-cell lymphoma. Cutaneous T-cell lymphomas occu…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
C-C chemokine receptor type 4
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe central volume …
KlirensClearance is 12 mL/…
Genetik -
MOL-4239 DB16051
small molecule | CAS: 1204306-34-2

MOL-4239 is under investigation in clinical trial NCT01826201 (Paired Psoriasis Lesion, Comparative, Study to Evaluate MOL4239 in Psoriasis).

Target Protein:
Signal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Molgramostim DB12525
biotech | CAS: 99283-10-0

Molgramostim has been used in trials studying the treatment of Bronchiectasis, Cystic Fibrosis, Pulmonary Alveolar Proteinosis, Acute Respiratory Distress Syndrome, and Autoimmune Pulmonary Alveolar Proteinosis.

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic Agents +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Molibresib DB16239
small molecule | CAS: 1260907-17-2

Molibresib is under investigation in clinical trial NCT01943851 (A Dose Escalation Study to Investigate the Safety, Pharmacokinetics (PK), Pharmacodynamics (PD) and Clinical Activity of GSK525762 in Subjects With Relapsed, Refractory Hematologic Malignancies).

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Bromodomain-containing protein 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Molidustat DB15642
small molecule | CAS: 1154028-82-6

Molidustat is under investigation in clinical trial NCT03350321 (A Study of Molidustat for Correction of Renal Anemia in Non-dialysis Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Molnupiravir DB15661
small molecule | CAS: 2349386-89-4

Molnupiravir (EIDD-2801, MK-4482) is the isopropylester prodrug of [N4-hydroxycytidine].[A193014,A193026] With improved oral bioavailability in non-human primates, it is hydrolyzed _in vivo_, and distributes into tissues where it becomes the active 5’-triphos…

Kategori:
AminesAnti-Infective AgentsAntiinfectives for Systemic Use +13
Waktu ParuhThe half life of th…
Vol. Distribusi-
Klirens-
Genetik -
Molsidomine Approved DB09282
small molecule | CAS: 25717-80-0

Molsidomine is an orally active, long-acting vasodilator, which belongs to the class of medications known as syndnones. Interestingly, it is being studied as being a preventive measure in cerebral infarction [A31932].

Kategori:
Cardiac TherapyCardiovascular AgentsMorpholines +7
Target Protein:
Guanylate cyclase soluble subunit alpha-2
Waktu Paruh-
Vol. Distribusi98 L [L1369]
Klirensrenal excretion is …
Genetik -
Molybdate DB15878
small molecule | CAS: 14259-85-9

Deskripsi belum tersedia.

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Molybdate Mo-99 DB16587
small molecule | CAS: 72826-31-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1313-27-5

Deskripsi belum tersedia.

Kategori:
Air PollutantsAnionsElectrolytes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Momelotinib Approved DB11763
small molecule | CAS: 1056634-68-4

Momelotinib is a Janus Kinase 1 (JAK1) and 2 (JAK2) inhibitor. It is a competitive inhibitor of JAK ATP binding.[A261566] First approved by the FDA on September 15, 2023,[L48206] momelotinib is used to treat myelofibrosis.[L48186] Myelofibrosis (MF) is a grou…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +24
Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK3 +3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean (%CV) appa…
KlirensThe mean (%CV) clea…
Genetik -
Mometasone DB00764
small molecule | CAS: 105102-22-5

Mometasone is a corticosteroid not currently used in medical products. [Mometasone furoate] however, is still in use.

Kategori:
Adrenal Cortex HormonesAdrenalsAnti-Allergic Agents +29
Target Protein:
Glucocorticoid receptorProgesterone receptor
Waktu Paruh5.8 hours
Vol. Distribusi-
Klirens-
Genetik -
Mometasone furoate Approved DB14512
small molecule | CAS: 83919-23-7

Mometasone furoate is a corticosteroid drug that can be used for the treatment of asthma, rhinitis, and certain skin conditions[FDA Label][F4292,F4295]. It has a glucocorticoid receptor binding affinity 22 times stronger than [dexamethasone] and higher than m…

Kategori:
Adrenal Cortex HormonesAdrenalsAdrenergics, Inhalants +28
Target Protein:
Glucocorticoid receptorProgesterone receptor
Waktu ParuhThe terminal half l…
Vol. DistribusiSteady state volume…
KlirensThe clearance rate …
Genetik -
biotech

Momordica charantia fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monalizumab DB12824
biotech | CAS: 1228763-95-8

Monalizumab has been used in trials studying the treatment of Gynecologic Cancer, Chronic Lymphocytic Leukemia, and Squamous Cell Carcinoma of the Oral Cavity.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monarsen DB16946
biotech | CAS: 864021-55-6

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monastrol DB04331
small molecule | CAS: 254753-54-3

Deskripsi belum tersedia.

Kategori:
Antimitotic AgentsAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
Kinesin-like protein KIF11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monepantel DB18755
small molecule | CAS: 887148-69-8

Deskripsi belum tersedia.

Kategori:
AcetonitrilesNitriles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mongersen DB15019
biotech | CAS: 1443994-46-4

Mongersen is under investigation in clinical trial NCT02957474 (A Study to Evaluate the Effect of Food, Formulation Strength, and a Proton Pump Inhibitor on GED 0301 Pharmacokinetics in Healthy Adult Subjects).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nicotinate-nucleotide--dimethylbenzimidazole phosphoribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monoctanoin DB06801
small molecule | CAS: 502-54-5

Monoctanoin is used to dissolve cholesterol gallstones.

Kategori:
Acids, AcyclicFatty AcidsLipids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 15181-43-8

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAnions +10
Target Protein:
Glycogen phosphorylase, muscle form
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycoconjugatesGlycolipids +1
Target Protein:
Photosystem II protein D1 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Trypsin-2Subtilisin BPN'Serine protease 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monomethyl fumarate Approved DB14219
small molecule | CAS: 2756-87-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic AcidsImmunosuppressive Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 532-40-1

Deskripsi belum tersedia.

Kategori:
MicronutrientsPyrimidinesSulfur Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Montelukast Approved DB00471
small molecule | CAS: 158966-92-8

Montelukast was first approved for clinical use by the US FDA in 1998 as Merck's brand name Singulair.[L6301] The medication is a member of the leukotriene receptor antagonist (LTRA) category of drugs.[L6301,L6304,L6307,L6310,L6325,L6328,L6331] Although capab…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAgents to Treat Airway Disease +29
Target Protein:
Cysteinyl leukotriene receptor 1Polyunsaturated fatty acid 5-lipoxygenase
Waktu ParuhStudies have demons…
Vol. DistribusiThe steady-state vo…
KlirensThe plasma clearanc…
Genetik -
Monteplase DB12726
biotech | CAS: 156616-23-8

Monteplase has been used in trials studying the treatment of Pulmonary Embolism.

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBlood Proteins +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Montmorillonite DB13654
small molecule | CAS: 1318-93-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAluminium CompoundsAluminum Silicates +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moperone DB13554
small molecule | CAS: 1050-79-9

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsButyrophenone DerivativesCentral Nervous System Depressants +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morclofone DB13558
small molecule | CAS: 31848-01-8

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesCough and Cold PreparationsKetones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morella cerifera pollen Approved DB10457
biotech

Morella cerifera pollen is the pollen of the Morella cerifera plant. Morella cerifera pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moricizine Approved DB00680
small molecule | CAS: 31883-05-3

An antiarrhythmia agent used primarily for ventricular rhythm disturbances.

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ic +15
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh2 hours (range 1.5-…
Vol. Distribusi* 300 L
Klirens-
Genetik -
Morin DB16770
small molecule | CAS: 480-16-0

Deskripsi belum tersedia.

Kategori:
AntioxidantsBenzopyransBiological Factors +8
Target Protein:
Estrogen receptor betaSolute carrier family 22 member 12Fatty acid synthase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morinamide DB13417
small molecule | CAS: 952-54-5

Deskripsi belum tersedia.

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsDrugs for Treatment of Tuberculosis
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morinidazole DB15098
small molecule | CAS: 92478-27-8

Morinidazole is under investigation in clinical trial NCT03380793 (A Trial to Assess the Efficacy and Safety of Morinidazole in Patients With Appendicitis).

Kategori:
ImidazolesNitro Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morniflumate DB09285
small molecule | CAS: 65847-85-0

Morniflumate is a non-steroidal anti-inflammatory drug with antipyretic properties. It is the morpholinoethyl ester of niflumic acid [L1496]. In one study, post morniflumate ingestion, physical examination and clinical symptoms of those with bronchitis show…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +14
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Polyunsaturated fatty acid 5-lipoxygenase +2
Waktu Paruh2h [L1498]
Vol. Distribusi-
Klirens45 ml/min [L1498]
Genetik -
Moroctocog alfa Approved DB13999
biotech | CAS: 284036-24-4

Moroctocog alfa, also known as BDDrFVIII (B domain deleted recombinant factor VIII), is a recombinant DNA-based drug with functional characteristics comparable to those of endogenous coagulation Factor VIII, the essential human blood clotting protein that is …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu ParuhMean terminal elimi…
Vol. DistribusiMean steady-state v…
KlirensMean clearance = 4.…
Genetik -
Moroxydine DB13597
small molecule | CAS: 3731-59-7

Deskripsi belum tersedia.

Kategori:
AmidinesAnti-Infective AgentsAntiinfectives for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morphine Approved DB00295
small molecule | CAS: 57-27-2

Morphine, the main alkaloid of opium, was first obtained from poppy seeds in 1805.[A176035] It is a potent analgesic, though its use is limited due to tolerance, withdrawal, and the risk of abuse.[A176050] Morphine is still routinely used today, though there …

Kategori:
AlkaloidsAnalgesicsAnesthetics +25
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Gen Terkait:
ABCB1 OPRM1
Waktu ParuhMorphine has a half…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik 2 Varian
Mosapride DB11675
small molecule | CAS: 112885-41-3

Mosapride is under investigation for the treatment and prevention of Postoperative Ileus and Gastric Peroral Endoscopic Pyloromyotomy (G-POEM). Mosapride has been investigated for the treatment and diagnostic of Constipation, Type 2 Diabetes, Functional Dyspe…

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmides +13
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosedipimod DB12592
small molecule | CAS: 221139-79-3

Mosedipimod has been used in trials studying the supportive care and treatment of Chemotherapy-induced Neutropenia.

Kategori:
Experimental Unapproved Treatments for COVID-19Lipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosliciguat DB19425
small molecule | CAS: 2231749-54-3

Mosliciguat is under investigation in clinical trial NCT06635850 (A Phase 2 Study of Mosliciguat in PH-ILD).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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