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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Hasil Pencarian (17430)

Halaman 162 / 349
Furaprevir DB12785
small molecule | CAS: 1435923-88-8

Furaprevir is under investigation in clinical trial NCT01523990 (A Study to Evaluate the Safety, Tolerability, and PK in Healthy Volunteers and HCV Genotype 1 Infected Patients).

Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaprofen DB06499
small molecule | CAS: 67700-30-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazabol DB01514
small molecule | CAS: 1239-29-8

Deskripsi belum tersedia.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazidin DB13475
small molecule | CAS: 1672-88-4

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazolidone DB00614
small molecule | CAS: 67-45-8

A nitrofuran derivative with antiprotozoal and antibacterial activity. Furazolidone binds bacterial DNA which leads to the gradual inhibition of monoamine oxidase. (From Martindale, The Extra Pharmacopoeia, 30th ed, p514)

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnti-Infective Agents +20
Target Protein:
DNA
Waktu Paruh10 minutes
Vol. Distribusi-
Klirens-
Genetik -
Furethidine DB01464
small molecule | CAS: 2385-81-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furfural DB16856
small molecule | CAS: 98-01-1

Deskripsi belum tersedia.

Kategori:
AldehydesFurans
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furosemide Approved DB00695
small molecule | CAS: 54-31-9

Furosemide is a potent loop diuretic that acts on the kidneys to ultimately increase water loss from the body. It is an anthranilic acid derivative.[L7958] Furosemide is used for edema secondary to various clinical conditions, such as congestive heart failure…

Kategori:
Acids, CarbocyclicAmidesAmines +30
Target Protein:
Solute carrier family 12 member 1Carbonic anhydrase 2G-protein coupled receptor 35
Waktu ParuhThe half-life from …
Vol. DistribusiThe volume of distr…
KlirensFollowing intraveno…
Genetik -
Furoyl-Leucine DB02215
small molecule

Deskripsi belum tersedia.

Target Protein:
Disintegrin and metalloproteinase domain-containing protein 28
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fursultiamine Approved DB08966
small molecule | CAS: 804-30-8

Compound used for therapy of thiamine deficiency. It has also been suggested for several non-deficiency disorders but has not yet proven useful. Fursultiamine is a vitamin B1 derivative.

Kategori:
MicronutrientsPyrimidinesSulfur Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furvina DB16547
small molecule | CAS: 189935-72-6

Furvina (G1) is an antimicrobial agent active against Gram-positive and Gram-negative bacteria, yeasts, and filamentous fungi. Furvina is marketed in Cuba as Dermofural®, an ointment containing G1 as the only active principle ingredient. It is used to treat d…

Kategori:
AlkenesAnti-Infective AgentsHydrocarbons, Acyclic
Target Protein:
30S ribosomal protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusafungine Approved DB08965
small molecule | CAS: 1393-87-9

Fusafungine is an antibiotic from Fusarium lateririum, and is used for the treatment of respiratory infections.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusarium compactum Approved DB10698
biotech

Fusarium compactum is a fungus which can provoke allergic reactions. Fusarium compactum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusarium graminearum Approved DB13907
biotech

Fusarium graminearum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusarium oxysporum Approved DB10806
biotech

Fusarium oxysporum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Fusarium oxysporum vasinfectum is a fungus which can provoke allergic reactions. Fusarium oxysporum vasinfectum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusicoccin DB01780
small molecule | CAS: 20108-30-9

Deskripsi belum tersedia.

Kategori:
CarbohydratesMycotoxins
Target Protein:
14-3-3 protein epsilon
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusidic acid Approved DB02703
small molecule | CAS: 6990-06-3

An antibiotic isolated from the fermentation broth of Fusidium coccineum. (From Merck Index, 11th ed) It acts by inhibiting translocation during protein synthesis. It is often used topically in creams and eyedrops but is available in systemic formulations inc…

Kategori:
Agents Causing Muscle ToxicityAnti-Bacterial AgentsAnti-Infective Agents +35
Target Protein:
Elongation factor GChloramphenicol acetyltransferaseChloramphenicol acetyltransferase 3
Waktu ParuhApproximately 5 to …
Vol. Distribusi-
Klirens-
Genetik -
Futibatinib Approved DB15149
small molecule | CAS: 1448169-71-8

Futibatinib is an inhibitor of Fibroblast Growth Factor receptor (FGFR), which comprises a group of receptor tyrosine kinases that play a key role in cell proliferation, differentiation, migration, and survival. FGFR was investigated in oncology as a therapeu…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +10
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +1
Waktu ParuhThe mean (CV%) elim…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Futuximab DB15262
biotech | CAS: 1310460-85-5

Futuximab is under investigation in clinical trial NCT01955473 (Japanese Phase 1 Trial of Sym004 in Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fx-1006A DB05352
small molecule

Fx-1006A is a small molecule compound with the potential to treat genetic disorders, such as familial amyloid cardiomyopathy (FAC) and familial amyloid polyneuropathy (FAP).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FX06 DB05685
biotech

FX06 is a naturally occurring peptide derived from the neo-N-terminus of fibrin (Bbeta(15-42)). It prevents leukocyte migration through the gap junctions of endothelial cells. FX06 has proven safe in acute and subchronic toxicological studies and recently ent…

Target Protein:
Cadherin-5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G100 DB17244
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G17DT Immunogen DB04914
biotech

G17DT Immunogen is a vaccine that neutralizes gastrin-17, a hormone required for the growth of a number of cancers of the gastrointestinal tract. It is in phase III trials for advanced pancreatic cancer as a monotherapy and in combination with gemcitabine. It…

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsComplex Mixtures +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G207 DB05827
biotech

G207 is cancer-killing viruses, so-called oncolytic viruses, for the treatment of various forms of cancer developed by MediGene AG. These viruses are specific herpes simplex viruses, or HSVs, generally known as the cause of cold sores. MediGene uses these vir…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G305 DB17292
biotech

G305 is a [recombinant NY-ESO-1 protein] plus glucopyranosyl lipid A (GLA) in a stable emulsion (SE). G305 is an active component of CMB305 along with [LV305].[L47346]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G4460 DB06359
biotech

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Target Protein:
Transcriptional activator Myb
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G4544 DB05244
small molecule

G4544 is an oral gallium compound that enables oral absorption of the active ingredient contained in Ganite™ (gallium nitrate injection). It targets bone tissue and is actively incorporated into bone mineral at sites where bone is metabolically active.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gabaculine DB02054
small molecule | CAS: 87980-11-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicCyclohexanesCycloparaffins +2
Target Protein:
Ornithine aminotransferase, mitochondrialGlutamate-1-semialdehyde 2,1-aminomutase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gabapentin Approved DB00996
small molecule | CAS: 60142-96-3

Gabapentin is a structural analogue of the inhibitory neurotransmitter gamma-aminobutyric acid ([GABA]) that was first approved for use in the United States in 1993.[L8717] It was originally developed as a novel anti-epileptic for the treatment of certain typ…

Kategori:
Acids, AcyclicAcids, CarbocyclicAmines +24
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1Gamma-aminobutyric acid type B receptor subunit 2Gamma-aminobutyric acid type B receptor subunit 1 +5
Waktu ParuhThe elimination t<s…
Vol. DistribusiThe apparent volume…
KlirensBoth the plasma cle…
Genetik -
Gabapentin enacarbil Approved DB08872
small molecule | CAS: 478296-72-9

Gabapentin enacarbil is marketed under the name Horizant. It is a prodrug of gabapentin, and indicated in adults for the treatment of Restless Legs Syndrome (RLS) and postherpetic neuralgia (PHN).

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +6
Target Protein:
Sodium-dependent multivitamin transporterVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent calcium channel subunit alpha-2/delta-2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensRenal clearance of …
Genetik -
Gabexate DB12831
small molecule | CAS: 39492-01-8

Gabexate is a synthetic serine protease inhibitor which has been used as an anticoagulant. It also known to decrease production of inflammatory cytokines. Gabexate has been investigated for use in cancer, ischemia-reperfusion injury, and pancreatitis.[A19218,…

Kategori:
AmidinesAnticoagulantsEnzyme Inhibitors +4
Target Protein:
Plasma kallikreinProthrombinPlasminogen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gaboxadol DB06554
small molecule | CAS: 64603-91-4

Gaboxadol also known as 4,5,6,7-tetrahydroisoxazolo(5,4-c)pyridin-3-ol (THIP) is an experimental sleep aid drug developed by Lundbeck and Merck, who reported increased deep sleep without the reinforcing effects of benzodiazepines. Development of Gaboxadol was…

Kategori:
AnalgesicsAnestheticsAnticonvulsants +8
Target Protein:
Gamma-aminobutyric acid receptor subunit delta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gacyclidine DB13096
small molecule | CAS: 68134-81-6

Gacyclidine has been used in trials studying the treatment of Tinnitus.

Kategori:
Central Nervous System AgentsCompounds used in a research, industrial, or household settingCyclohexanes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gadobenic acid Approved DB00743
small molecule | CAS: 113662-23-0

Gadobenic acid, usually available in the salt form gadobenate dimeglumine, is a linear MRI gadolinium-based contrast agent (GBCA) used primarily for MR imaging of the liver.[A263086] It differs from other GBCAs due to the benzene ring that confers weak protei…

Kategori:
AlcoholsAmino SugarsCarbohydrates +14
Target Protein:
Albumin
Waktu ParuhGadobenate ion has …
Vol. DistribusiThe volume of distr…
KlirensThe total plasma cl…
Genetik -
Gadobutrol Approved DB06703
small molecule | CAS: 770691-21-9

Gadobutrol is a second-generation extracellular non-ionic macrocyclic GBCA (gadolinium-based contrast agent) used in magnetic resonance imaging (MRI) in adults and children older than 2 years of age. Due to its physicochemical properties, gadobutrol is formu…

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +5
Waktu ParuhFor adult patients,…
Vol. DistribusiIn children aged 2 …
KlirensIn healthy subjects…
Genetik -
Gadodiamide Approved DB00225
small molecule | CAS: 131410-48-5

Gadodiamide is a linear, non-ionic gadolinium-based contrast agent (GBCA) that is used in magnetic resonance imaging (MRI) procedures to assist in the visualization of blood vessels.[A263086,A263091] GBCAs constitute the largest group of MR agents, and they a…

Kategori:
AcetatesAcids, AcyclicAmines +13
Waktu ParuhThe mean distributi…
Vol. DistribusiThe volume of distr…
KlirensThe renal and plasm…
Genetik -
Gadofosveset trisodium Approved DB06705
small molecule | CAS: 193901-90-5

Gadofosveset trisodium is an intravenous contrast agent used with magnetic resonance angiography(MRA), which is a non-invasive way of imaging blood vessels. The agent allows for the vascular system to be imaged more clearly by the MRA. In this way, gadofosves…

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +11
Target Protein:
Albumin
Waktu Paruh18.5 hours
Vol. Distribusi48 ± 16 mL/kg
Klirens6.57 ± 0.97 mL/h/kg…
Genetik -
Gadolinium Approved DB12091
small molecule | CAS: 7440-54-2

Gadolinium is under investigation in Hypertension, ACUTE KIDNEY INJURY, and Chronic Kidney Disease. Gadolinium has been investigated for the basic science of CAD, Multiple Sclerosis, and Coronary Artery Disease.

Kategori:
Anti-Inflammatory AgentsCompounds used in a research, industrial, or household settingContrast Media +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22541-19-1

Deskripsi belum tersedia.

Kategori:
Gadolinium-based Contrast AgentMagnetic Resonance Contrast Activity
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gadopentetic acid Approved DB00789
small molecule | CAS: 80529-93-7

A complex of gadolinium with a chelating agent, diethylenetriamine penta-acetic acid (DTPA see pentetic acid), that is given to enhance the image in cranial and spinal MRIs. (From Martindale, The Extra Pharmacopoeia, 30th ed, p706)

Kategori:
AcetatesAcids, AcyclicAmines +12
Target Protein:
6-phosphogluconate dehydrogenase, decarboxylating
Waktu ParuhDistribution half l…
Vol. Distribusi* 266 ± 43 mL/kg
Klirens* 1.94 +/- 0.28 mL/…
Genetik -
Gadopiclenol Approved DB17084
small molecule | CAS: 933983-75-6

Gadopiclenol is a gadolinium-based contrast agent (GBCA) based on a pyclen macrocyclic structure. It is indicated for use with magnetic resonance imaging (MRI) to detect and visualize lesions with abnormal vascularity in the central nervous system and the bod…

Kategori:
Contrast MediaDiagnostic Uses of ChemicalsGadolinium-based Contrast Agent +5
Waktu ParuhGadopiclenol has a …
Vol. DistribusiAt steady state, th…
KlirensGadopiclenol has a …
Genetik -
Gadoteric acid Approved DB09132
small molecule | CAS: 72573-82-1

Gadoteric acid, commonly used in the salt form gadoterate meglumine, is a macrocyclic, ionic gadolinium-based contrast agent (GBCA).[A263131] It is composed of the organic acid DOTA (1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid) used for its chel…

Kategori:
AlcoholsAmino SugarsCarbohydrates +12
Waktu ParuhFollowing an intrav…
Vol. DistribusiThe volume of distr…
KlirensIn healthy subjects…
Genetik -
Gadoteridol Approved DB00597
small molecule | CAS: 120066-54-8

Gadoteridol is a macrocyclic nonionic gadolinium that provides contrast enhancement of the brain, spine, and surrounding tissues, resulting in improved visualization (compared with unenhanced MRI) of lesions with abnormal vascularity or those thought to disru…

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +10
Waktu ParuhThe elimination hal…
Vol. DistribusiThe plasma distribu…
KlirensThe renal and plasm…
Genetik -
Gadoversetamide Approved DB00538
small molecule | CAS: 131069-91-5

Gadoversetamide, marketed under the trade name OptiMARK, is a gadolinium compound used as a contrast agent in magnetic resonance imaging (MRI), particularly imaging of the brain, spine and liver.

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +6
Waktu ParuhDistribution 13.3 &…
Vol. Distribusi* 162 ± 25 mL/kg [n…
Klirens* 72 +/- 16.3 mL/hr…
Genetik -
Gadoxetic acid Approved DB08884
small molecule | CAS: 135326-11-3

Gadoxetic acid (gadoxetate) is a paramagnetic gadolinium-containing ionic linear contrast agent in which its salt form, gadoxetate disodium, is used for intravenous injection. Ethoxybenzyl diethylenetriaminepentaacetic acid is the moiety that chelates with a …

Kategori:
AcetatesAcids, AcyclicAmines +13
Waktu ParuhThe mean terminal e…
Vol. DistribusiThe total volume of…
KlirensA total serum clear…
Genetik -
Galactose Approved DB11735
small molecule | CAS: 59-23-4

Galactose has been used in trials studying the treatment and diagnosis of Hepatitis C, Hepatic Cancer, Wilsons Disease, Diabetic Macular Oedema, and Focal Segmental Glomerulosclerosis, among others. There are even proposals for its use in accelerating senesce…

Kategori:
CarbohydratesContrast MediaDiagnostic Agents +4
Waktu ParuhReadily accessible …
Vol. DistribusiIt has been documen…
KlirensIn subjects with no…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Histo-blood group ABO system transferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 8051–8100 dari 17430
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