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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 162 / 252
MK-0767 DB12055
small molecule | CAS: 934017-32-0

MK0767 has been used in trials studying the treatment of Dyslipidemia, Diabetes Mellitus, Type 2 Diabetes Mellitus, Diabetes Mellitus, Type 2, and Diabetes Mellitus, Type II, among others.

Kategori:
Sulfur Compounds
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MK-0773 DB16244
small molecule | CAS: 606101-58-0

MK-0773 is under investigation in clinical trial NCT00529659 (A Study of the Safety and Efficacy of MK-0773 in Women With Sarcopenia (Loss of Muscle Mass)(mk-0773-005)).

Kategori:
Fused-Ring CompoundsSteroids
Target Protein:
Androgen receptor
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MK-0777 DB12238
small molecule | CAS: 252977-51-8

MK-0777 has been used in trials studying the treatment of Schizophrenia, Anxiety Disorder, and Generalized Anxiety Disorder.

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MK-0873 DB13029
small molecule | CAS: 500355-52-2

MK-0873 has been used in trials studying the treatment of Rheumatoid Arthritis.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPhosphodiesterase 4 Inhibitors +1
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4D
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MK-1064 DB15028
small molecule | CAS: 1207253-08-4

MK-1064 is under investigation in clinical trial NCT02549014 (A Single Dose Study of the Safety, Pharmacokinetics and Pharmacodynamics of MK-1064 (MK-1064-001)).

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MK-1454 DB14721
small molecule

A synthetic cyclic dinucleotide (CDN) and agonist of stimulator of interferon genes protein (STING), with potential immunoactivating and antineoplastic activities. Upon intratumoral (IT) administration, STING agonist MK-1454 binds to STING and activates the S…

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MK-1496 DB12763
small molecule | CAS: 1037254-47-9

MK-1496 has been used in trials studying the treatment of Neoplasms and Malignant.

Target Protein:
Serine/threonine-protein kinase PLK1
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MK-2225 DB18240
biotech

Deskripsi belum tersedia.

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MK-2748 DB15371
small molecule | CAS: 1193902-95-2

MK-2748 is under investigation in clinical trial NCT01593735 (A Multiple Dose Study to Evaluate the Safety and Efficacy of MK-2748 in Hepatitis C-Infected Participants (MK-2748-002 AM1)).

Kategori:
Sulfur Compounds
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MK-3207 DB12424
small molecule | CAS: 957118-49-9

Mk3207 has been used in trials studying the treatment of Migraine and Migraine Disorders.

Kategori:
Receptors, Calcitonin Gene-Related Peptide, antagonists & inhibitors
Target Protein:
Calcitonin gene-related peptide type 1 receptor
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MK-3577 DB14957
small molecule | CAS: 1019112-29-8

MK-3577 is under investigation in clinical trial NCT00868790 (A Study of the Safety and Efficacy of MK-3577 in Participants With Type 2 Diabetes Mellitus (MK-3577-009)).

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MK-4541 DB17016
small molecule | CAS: 796885-38-6

MK-4541 is a 4-azasteroid and a selective androgen receptor modulator (SARM). MK-4541 acts as a dual selective SARM and is both a potent androgen receptor antagonist and a 5?-reductase inhibitor.[A252687]

Kategori:
Acids, AcyclicFused-Ring CompoundsSteroids
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MK-4721 DB05933
biotech

MK-4721 is a fully human monoclonal antibody directed to Agensys’ proprietary target Prostate Stem Cell Antigen (PSCA), an antigen expressed at significant levels on tumor cells from the majority of patients with all stages of prostate, pancreatic and bladder…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Prostate stem cell antigen
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MK-4830 DB17454
biotech

MK-4830 is a monoclonal antibody that targets the myeloid-specific immunoglobulin-like transcript (ILT) 4 receptor.

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MK-4965 DB08460
small molecule | CAS: 920035-77-4

MK-4965 is an HIV-1 reverse transcriptase inhibitor.

Kategori:
HIV Reverse Transcriptase, antagonists & inhibitors
Target Protein:
Gag-Pol polyprotein
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MK-5108 DB12556
small molecule | CAS: 1010085-13-8

MK-5108 has been used in trials studying the treatment of Cancer, Neoplasms, Tumors.

Kategori:
Acids, CarbocyclicCyclohexanesCycloparaffins +2
Target Protein:
Aurora kinase BAurora kinase A
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MK-6186 DB12999
small molecule | CAS: 1034474-19-5

MK6186 has been used in trials studying the treatment of HIV-1 Infection.

Target Protein:
Gag-Pol polyprotein
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MK-6325 DB15249
small molecule | CAS: 1263814-52-3

MK-6325 is under investigation in clinical trial NCT01329913 (Safety, Pharmacokinetics, and Pharmacodynamics of MK-6325 in Hepatitis C Virus (HCV) Infections (MK-6325-003)).

Target Protein:
Genome polyprotein
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MK-7145 DB11968
small molecule | CAS: 1255204-84-2

MK-7145 has been used in trials studying the treatment of Hypertension and Renal Insufficiency.

Kategori:
Heterocyclic Compounds, Fused-Ring
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MK-7288 DB17094
small molecule | CAS: 936626-07-2

Deskripsi belum tersedia.

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MK-8189 DB19153
small molecule | CAS: 1424371-93-6

MK-8189 is under investigation in clinical trial NCT04624243 (Efficacy and Safety of MK-8189 in Participants With an Acute Episode of Schizophrenia (MK-8189-008)).

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MK-8245 DB13024
small molecule | CAS: 1030612-90-8

MK-8245 has been used in trials studying the treatment of Type 2 Diabetes Mellitus.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
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MK-8666 DB14937
small molecule | CAS: 1544739-75-4

MK-8666 is under investigation in clinical trial NCT01971554 (Safety, Tolerability, Pharmacodynamics, and Pharmacokinetics of MK-8666 in Participants With Type 2 Diabetes Mellitus (MK-8666-003)).

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MK-8777 DB18904
small molecule | CAS: 1026791-61-6

MK-8777 is under investigation in clinical trial NCT00610649 (Trial to Determine the Maximum Tolerated Dose (MTD) Based on Safety and Tolerability, of Org 26576 in Participants With Major Depressive Disorder (174001/P05704/MK-8777-001)).

Kategori:
Isoxazoles
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MKC-1 DB05608
small molecule | CAS: 125313-92-0

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 2Cyclin-dependent kinase 1
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MKC1106-PP DB06030
small molecule

MKC1106-PP is a 3-component investigational vaccine made up of a DNA plasmid (pPRA-PSM) and 2 peptides E-PRA and E-PSM. The plasmid portion is a recombinant plasmid expressing segments of the 2 target antigens, PRAME and PSMA. MKC1106-PP was under investigati…

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MLN-977 DB05431
small molecule | CAS: 175212-04-1

MLN-977 is a small molecule compound that inhibits the production of leukotrienes, especially 5-lipoxygenase. It is developed by PharmaEngine to treat asthma and chronic obstructive pulmonary disease.

Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
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MLN0415 DB05183
small molecule

MLN0415 is a novel, small molecule IKK2 inhibitor, discovered by Millennium scientists. In preclinical studies, MLN0415 was shown to decrease NF-kB activation and down-regulate the expression of a number of inflammatory proteins. Because inflammatory proteins…

Target Protein:
Inhibitor of nuclear factor kappa-B kinase subunit beta
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MLN2222 DB06503
biotech

MLN2222 is a novel, proprietary recombinant protein that blocks both the C3 and C5 convertases, which are essential components of the complement activation pathway.

Target Protein:
Complement factor B
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MLN2704 DB06513
biotech

A Phase 1/2 trial (NCT00070837) evaluated the safety, dosage, and pharmacokinetics of MLN2704 in patients with metastatic androgen-independent prostate cancer.

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MLN3897 DB06505
small molecule | CAS: 849105-26-6

MLN3897, a novel CCR1 inhibitor, disrupts osteoclast formation and blocks the interaction between multiple myeloma cells and osteoclasts.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
C-C chemokine receptor type 1
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MLN576 DB06517
small molecule | CAS: 346689-77-8

XR11576 (MLN576) is a novel monophenazine with a mechanism of action that includes interaction with both topoisomerase (Topo) I and II.[A234609]

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +3
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MLN8054 DB13061
small molecule | CAS: 869363-13-3

MLN8054 has been used in trials studying the treatment of Colon Neoplasm, Breast Neoplasm, Bladder Neoplasm, Pancreatic Neoplasm, and Advanced Malignancies.

Kategori:
Heterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Aurora kinase A
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MM-093 DB05512
biotech

MM-093 is a recombinant version of human alpha-fetoprotein (hAFP), an immunomodulatory serum protein normally produced at very high levels by the fetus and present in low levels in the blood of adults and children. Research on AFP suggests that it may play a …

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MM-111 DB17983
biotech | CAS: 1361108-53-3

MM-111 is a novel bispecific antibody fusion protein that co-targets the the epidermal growth factor family receptor tyrosine kinases, ERBB2 and ERBB3.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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MMDA DB01442
small molecule | CAS: 13674-05-0

MMDA, or 3-methoxy-4,5-methylenedioxyamphetamine, is a member of the amphetamine drug class with stimulant and psychedelic properties. It also acts as an entheogen and an entactogen. MMDA bears resemblance to the psychopharmacologically active essential oils …

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +11
Target Protein:
5-hydroxytryptamine receptor 2ASodium-dependent dopamine transporterSodium-dependent serotonin transporter +5
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MMI-175 DB02378
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-secretase 1
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MN-246 DB05981
small molecule

MN-246 is a novel ß3-adrenergic receptor agonist developed for the treatment of urinary incontinence by MediciNova Inc.

Target Protein:
Beta-3 adrenergic receptor
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MN-305 DB05339
small molecule

MN-305 is a novel, potent and highly selective serotonin 5-HT1A receptor agonist under development by MediciNova for the treatment of anxiety disorders beginning with Generalized Anxiety Disorder (GAD).

Target Protein:
5-hydroxytryptamine receptor 1A
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Mobocertinib Approved DB16390
small molecule | CAS: 1847461-43-1

Mobocertinib is a kinase inhibitor targeted against human epidermal growth factor receptor (EGFR). It is used specifically in the treatment of non-small cell lung cancer (NSCLC) caused by exon 20 insertion mutations in the _EGFR_ gene,[L38368] which are typic…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +15
Target Protein:
Epidermal growth factor receptor
Waktu ParuhAt steady-state, th…
Vol. DistribusiThe mean apparent v…
KlirensAt steady-state, th…
Genetik -
Mocemestrocel DB19154
biotech

Deskripsi belum tersedia.

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Mocravimod DB18151
small molecule | CAS: 509092-16-4

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
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MOD-5014 DB17715
biotech

MOD-5014 is a long-acting carboxy-terminal peptide (CTP)-modified Factor IIa.[A259088] It is being investigated for the treatment of hemophilia.[L46173]

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Modafinil Approved DB00745
small molecule | CAS: 68693-11-8

Modafinil is a stimulant drug marketed as a 'wakefulness promoting agent' and is one of the stimulants used in the treatment of narcolepsy. Narcolepsy is caused by dysfunction of a family of wakefulness-promoting and sleep-suppressing peptides, the orexins, w…

Kategori:
Benzene DerivativesBenzhydryl CompoundsCentral Nervous System Agents +35
Target Protein:
Sodium-dependent dopamine transporterAlpha-1B adrenergic receptor
Gen Terkait:
COMT COMT
Waktu Paruh23-215 hours
Vol. Distribusi* 0.9 L/kg
Klirens-
Genetik 2 Varian
Modakafusp alfa DB16399
biotech

Modakafusp alfa is under investigation in clinical trial NCT03215030 (A Study to Investigate the Safety, Tolerability, Efficacy, Pharmacokinetics, and Immunogenicity of TAK-573 in Participants With Refractory Multiple Myeloma (MM)).

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Moderna COVID-19 Vaccine Approved DB15654
biotech

The Moderna COVID-19 Vaccine (mRNA-1273) is a novel mRNA-based vaccine encapsulated in a lipid nanoparticle that encodes for a full-length pre-fusion stabilized spike (S) protein of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2). Coronavirus dis…

Kategori:
Biological ProductsCOVID-19 VaccinesExperimental Unapproved Treatments for COVID-19 +5
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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Modified vaccinia ankara Approved DB15483
biotech

Modified Vaccinia Ankara (MVA) refers to an attenuated strain of the Vaccinia virus. Vaccines using MVA are live and non-replicating, and are produced using Modified Vaccinia Ankara-Bavarian Nordic (MVA-BN).[L42660,L42670]

Kategori:
Anti-Infective AgentsAntiviral AgentsBiological Products +5
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biotech | CAS: 2171576-44-4

Modified vaccinia virus Ankara-85A antigen is under investigation in clinical trial NCT00953927 (A Study of MVA85A in Healthy Infants).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBacterial Vaccines +8
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