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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
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13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 162 / 272
Lintitript DB04867
small molecule | CAS: 136381-85-6

Lintitript is a new, highly specific and potent CCK-A receptor antagonist.

Kategori:
Heterocyclic Compounds, Fused-RingHormone AntagonistsHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Cholecystokinin receptor type A
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Lintuzumab DB14877
biotech | CAS: 166089-32-3

Lintuzumab is under investigation in clinical trial NCT00016159 (Chemotherapy Plus Monoclonal Antibody in Treating Patients With Acute Promyelocytic Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
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biotech | CAS: 2209911-94-2

Lintuzumab actinium Ac-225 is under investigation in clinical trial NCT00672165 (Targeted Atomic Nano-Generators (Actinium-225-Labeled Humanized Anti-CD33 Monoclonal Antibody HuM195) in Patients With Advanced Myeloid Malignancies).

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Linvoseltamab DB17447
biotech

Linvoseltamab is an investigational bispecific antibody. It promotes the interaction of B-cell maturation antigen (BCMA) on multiple myeloma cells with CD3-expressing T cells.

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Linzagolix Approved DB17083
small molecule | CAS: 935283-04-8

Linzagolix is a non-peptide, selective antagonist of the gonadotropin-releasing hormone (GnRH) receptor. It has been studied for the treatment of estrogen-dependent conditions such as uterine fibroids and endometriosis.[A253642,A253647] It is similar to other…

Kategori:
Anti-Gonadotropin-Releasing HormonesBCRP/ABCG2 SubstratesCytochrome P-450 CYP2C8 Inhibitors +18
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe half-life of li…
Vol. DistribusiAfter seven days of…
KlirensThe geometric mean …
Genetik -
LioCyx-M004 DB17368
biotech

LioCyx-M004 are autologous T cells transduced with a retroviral vector encoding a hepatitis B virus antigen-specific T cell receptor.

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Liothyronine Approved DB00279
small molecule | CAS: 6893-02-3

Liothyronine is a thyroidal hormone T3 which is normally produced by the thyroid gland in a ratio 4:1 when compared with T4: T3. Liothyronine is the active form of thyroxine which is composed in a basic chemical structure by a tyrosine with bound iodine.[T457…

Kategori:
Agents used to treat hypothyroidismDrugs that are Mainly Renally ExcretedHormones +12
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor betaProliferating cell nuclear antigen
Waktu ParuhThe half-life of li…
Vol. DistribusiThe reported volume…
KlirensThere are no report…
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small molecule | CAS: 20196-64-9

Liothyronine I-131 has been used in trials studying the treatment of Tricuspid Atresia and Heart Defects, Congenital.

Kategori:
Thyroxine-binding globulin substrates
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Liotrix Approved DB01583
small molecule | CAS: 8065-29-0

Liotrix is a synthetically derived thyroid hormone replacement preparation. It consists of levothyroxine sodium (thyroxine, T4) and liothyronine sodium (triiodothyronine, T3) in a 4 to 1 ratio by weight. Liotrix was developed when it was believed that serum l…

Kategori:
Agents used to treat hypothyroidismAmino AcidsAmino Acids, Aromatic +19
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
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Lipegfilgrastim Approved DB13200
biotech | CAS: 1117844-87-7

Lipegfilgrastim, previously known as XM22, is a pegylated, recombinant granulocyte colony-stimulating factor (G-CSF) that was synthetized using a highly site-specific glycoPEGylation technology [A32665]. It is used as an alternate to [DB00019] for prophylacti…

Kategori:
Adjuvants, ImmunologicAlcoholsAmino Acids, Peptides, and Proteins +17
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe average termina…
Vol. DistribusiLipegfilgrastim has…
KlirensIn a phase 1, multi…
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LipidRescue DB18163
biotech

Deskripsi belum tersedia.

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Lipoic acid Approved DB00166
small molecule | CAS: 1200-22-2

A vitamin-like antioxidant.

Kategori:
Alimentary Tract and MetabolismAntioxidantsBiological Factors +15
Target Protein:
Lipoyl amidotransferase LIPT1, mitochondrialSodium-dependent multivitamin transporterLipoyl synthase, mitochondrial
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small molecule

Liposome-encapsulated form of prostaglandin E1 (Liprostin) is known to be a potent vasodilator and platelet inhibitor as well as an anti-inflammatory and anti-thrombotic agent. The liposomal formulation of PGE-1 changes the drug’s dynamics and improve its the…

Target Protein:
Platelet glycoprotein Ib alpha chain
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Lipotecan DB17385
small molecule | CAS: 1432468-79-5

Deskripsi belum tersedia.

Kategori:
Alkaloids
Target Protein:
DNA topoisomerase 1
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biotech

Deskripsi belum tersedia.

Kategori:
Carboxylic Ester HydrolasesEnzymesEnzymes and Coenzymes +3
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biotech | CAS: 118731-97-8

Deskripsi belum tersedia.

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biotech | CAS: 8046-19-3

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +2
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Lirafugratinib DB18300
small molecule | CAS: 2549174-42-5

Deskripsi belum tersedia.

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Liraglutide Approved DB06655
biotech | CAS: 204656-20-2

Victoza contains liraglutide, a synthetic analog of human glucagon-like peptide-1(GLP-1) and acts as a GLP-1 receptor agonist.[Label,A6932] Liraglutide is 97% similar to native human GLP-1, differing primarily by substituting arginine for lysine at position 3…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +17
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhTerminal half life …
Vol. Distribusi13L[Label].
Klirens1.2L/h[Label].
Genetik -
Lirentelimab DB16728
biotech | CAS: 2283348-97-8

Lirentelimab is under investigation in clinical trial NCT04856891 (A Study of Lirentelimab (AK002) in Patients With Active Eosinophilic Duodenitis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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LIS-1 DB18388
biotech

LIS-1 is an immunoglobulin G (IgG) polyclonal antibody that binds to human T cells.

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Lisaftoclax DB18054
small molecule | CAS: 2180923-05-9

Lisaftoclax is a novel, orally active, selective and potent BCL-2 inhibitor

Kategori:
Benzene DerivativesNitro Compounds
Target Protein:
Apoptosis regulator Bcl-2
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Lisavanbulin DB15224
small molecule | CAS: 1263384-43-5

Lisavanbulin is under investigation in clinical trial NCT02895360 (Phase 1/2a Study of BAL101553 as 48-hour Infusions in Patients With Advanced Solid Tumors or Recurrent Glioblastoma).

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalHeterocyclic Compounds, Fused-Ring +2
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Lisdexamfetamine Approved DB01255
small molecule | CAS: 608137-32-2

Lisdexamfetamine is a prodrug of [dextroamphetamine], a central nervous system stimulant known as d-amphetamine,[A40246] covalently attached to the naturally occurring amino acid L-lysine.[A2230] Lisdexamfetamine is the first chemically formulated prodrug sti…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +17
Target Protein:
Trace amine-associated receptor 1
Waktu ParuhPlasma concentratio…
Vol. DistribusiDextroamphetamine, …
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Lisinopril Approved DB00722
small molecule | CAS: 76547-98-3

Lisinopril is an angiotensin converting enzyme inhibitor (ACEI) used to treat hypertension, heart failure, and myocardial infarction.[L8384,L8387,L8390] Lisinopril and [captopril] are the only ACEIs that are not prodrugs.[A184853] It functions by inhibition o…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +20
Target Protein:
Angiotensin-converting enzymeRenin
Waktu ParuhLisinopril has an e…
Vol. DistribusiThe apparent volume…
KlirensA 30kg child has a …
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Lisocabtagene maraleucel Approved DB16582
biotech

Lisocabtagene maraleucel is a chimeric antigen receptor (CAR) T-cell therapy, similar to [brexucabtagene autoleucel] and [axicabtagene ciloleucel].[A228493,L31588] Lisocabtagene maraleucel is a genetically modified autologous T-cell therapy that targets CD19,…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy +3
Target Protein:
B-lymphocyte antigen CD19
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Lisofylline DB12406
small molecule | CAS: 100324-81-0

Lisofylline has been investigated for the treatment of Type 1 Diabetes Mellitus.

Kategori:
Adjuvants, ImmunologicAnalgesicsAnalgesics, Non-Narcotic +12
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biotech

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Lisuride Approved DB00589
small molecule | CAS: 18016-80-3

An ergot derivative that acts as an agonist at dopamine D2 receptors (dopamine agonists). It may also act as an antagonist at dopamine D1 receptors, and as an agonist at some serotonin receptors (serotonin agonists).

Kategori:
Agents that produce hypertensionAlkaloidsAnalgesics +27
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor +12
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Lithium carbonate Approved DB14509
small molecule | CAS: 554-13-2

Lithium has been used to treat manic episodes since the 19th century[A176642]. Though it is widely used, its mechanism of action is still unknown[FDA Label][A14585,A176642,A176651,L5843]. Lithium carbonate has a narrow therapeutic range and so careful monitor…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +26
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu ParuhThe half life of li…
Vol. DistribusiApparent volume of …
KlirensClearance is genera…
Genetik -
Lithium cation DB01356
small molecule | CAS: 7439-93-2

Lithium was used during the 19th century to treat gout. Lithium salts such as lithium carbonate (Li2CO3), lithium citrate, and lithium orotate are mood stabilizers. They are used in the treatment of bipolar disorder, since unlike most other mood altering drug…

Kategori:
Antidepressive AgentsAntimanic AgentsAntipsychotic Agents +11
Target Protein:
Glycogen synthase kinase-3 betaInositol monophosphatase 1Inositol monophosphatase 2 +1
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Lithium hydroxide Approved DB14506
small molecule | CAS: 1310-65-2

Used for tryptophan determinations in proteins & foods.

Kategori:
Lithium CompoundsNarrow Therapeutic Index Drugs
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Litifilimab DB18864
biotech | CAS: 2407378-48-5

Litifilimab is under investigation in clinical trial NCT05531565 (A Study to Assess the Efficacy and Safety of BIIB059 (Litifilimab) in Participants With Active Subacute Cutaneous Lupus Erythematosus (SCLE) And/or Chronic Cutaneous Lupus Erythematosus (CCLE) …

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Litoxetine DB15038
small molecule | CAS: 86811-09-8

Litoxetine is under investigation in clinical trial NCT03397771 (DBPC Trial to Evaluate the Safety, Tolerability and Efficacy of Oral Litoxetine in Subjects With Urinary Incontinence).

Target Protein:
Sodium-dependent serotonin transporter
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Litronesib DB11861
small molecule | CAS: 910634-41-2

Litronesib has been used in trials studying the treatment of Solid Tumors, Ovarian Cancer, Gastric Cancer, Prostate Cancer, and Acute Leukaemia, among others.

Kategori:
AmidesSulfonesSulfur Compounds +1
Target Protein:
Kinesin-like protein KIF11
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Lividomycin A DB04728
small molecule | CAS: 36441-41-5

Deskripsi belum tersedia.

Target Protein:
Telomerase reverse transcriptase
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Livmoniplimab DB18939
biotech | CAS: 2412004-88-5

Livmoniplimab is under investigation in clinical trial NCT06109272 (A Study to Assess the Dose, Adverse Events, and Change in Disease Activity of Livmoniplimab as an Intravenous (IV) Solution in Combination With Budigalimab as an IV Solution in Adult Particip…

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Livoletide DB15188
small molecule | CAS: 1088543-62-7

Livoletide is under investigation in clinical trial NCT03790865 (Effects of Livoletide (AZP-531) on Food-related Behaviors in Patients With Prader-Willi Syndrome).

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsHormones +3
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Lixisenatide Approved DB09265
biotech | CAS: 320367-13-3

Lixisenatide is a glucagon-like peptide-1 (GLP-1) receptor agonist used in the treatment of type II diabetes mellitus (T2DM). It is sold by Sanofi-Aventis under the brand name Adlyxin in the US[L763] and Lyxumia in the EU.[L764] Adlyxin recieved FDA approval …

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +11
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhFollowing the admin…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Lixivaptan DB06666
small molecule | CAS: 168079-32-1

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzazepines +3
Target Protein:
Histidine decarboxylaseVasopressin V2 receptor
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biotech | CAS: 2461531-19-9

Lixmabegagene relduparvovec, formerly known as LYS-GM101, is a recombinant adeno-associated virus vector serotype rh.10 (AAVrh.10) carrying the human ?-galactosidase gene (GBL1). It is under development for the treatment of GM1 gangliosidosis.[L45929]

Kategori:
Adeno-associated Viral Vector Therapies
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Lixudebart DB19244
biotech | CAS: 2749515-10-2

Lixudebart, an investigational first-in-class monoclonal antibody, aims to reverse fibrosis.[L50833]

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Lixumistat DB18748
small molecule | CAS: 1422365-93-2

Deskripsi belum tersedia.

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LJ-2698 DB18018
small molecule | CAS: 945457-84-1

Deskripsi belum tersedia.

Kategori:
Adenosine A3 Receptor AntagonistsNeurotransmitter AgentsNucleic Acids, Nucleotides, and Nucleosides +5
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LJP-538 DB17810
biotech

Deskripsi belum tersedia.

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LJP-539 DB17811
biotech

Deskripsi belum tersedia.

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LL-37 DB16532
biotech

LL-37 is a human cathelicidin that inhibits viral replication and while also playing a role in host defense against infection.

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LLL-3348 DB05771
biotech

The botanical drug product LLL-3348 is a once-daily oral formulation for treatment of chronic stable plaque type psoriasis.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +1
Target Protein:
Interleukin-10
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LM-030 DB18283
small molecule | CAS: 1122484-55-2

Deskripsi belum tersedia.

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