Hasil Filter

12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (12560)

Halaman 161 / 252
Mirabegron Approved DB08893
small molecule | CAS: 223673-61-8

Mirabegron is a sympathomimetic beta-3 adrenergic receptor agonist used to relax the smooth muscle of the bladder in the treatment of urinary frequency and incontinence. It is unique amongst overactive bladder treatment options in that, unlike other treatment…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-3 Receptor Agonists +32
Target Protein:
Beta-3 adrenergic receptorBeta-1 adrenergic receptor
Waktu ParuhThe mean terminal e…
Vol. DistribusiFollowing intraveno…
KlirensTotal plasma cleara…
Genetik -
Miramistin ion DB19386
small molecule | CAS: 91481-38-8

Miramistin ion is under investigation in clinical trial NCT05561816 (Efficacy and Safety of Dioxidin Versus Miramistin in Superficial Pyoderma).

Kategori:
AminesBenzylammonium CompoundsOnium Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miransertib DB14982
small molecule | CAS: 1313881-70-7

Miransertib is under investigation in clinical trial NCT01473095 (Phase 1 Dose Escalation Study of ARQ 092 in Adult Subjects With Advanced Solid Tumors and Recurrent Malignant Lymphoma).

Kategori:
AminesPyridines
Target Protein:
RAC-gamma serine/threonine-protein kinaseRAC-alpha serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miravirsen DB12851
biotech | CAS: 1072874-90-8

Miravirsen has been investigated for the treatment of Hepatitis C and Hepatitis C, Chronic.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirdametinib DB07101
small molecule | CAS: 391210-10-9

PD-0325901 has been used in trials studying the treatment and basic science of Melanoma, Solid Tumour, Solid Tumors, Advanced Cancer, and Breast Neoplasms, among others.

Kategori:
Acids, CarbocyclicAmidesAmines +3
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirfentanil DB09175
small molecule | CAS: 117523-47-4

Mirfentanil is a derivative of fentanyl that presents high selectivity for the mu opioid receptor. At lower doses, it antagonizes the analgesic effects of alfentanil and substitutes for naloxone in morphine-treated monkeys; however, it also reverses naloxone-…

Kategori:
Piperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miricorilant DB16234
small molecule | CAS: 1400902-13-7

Miricorilant is under investigation in clinical trial NCT03818256 (Study Evaluating the Safety, Efficacy, and Pharmacokinetics of Miricorilant (CORT118335) in Obese Adult Patients With Schizophrenia and Recent Weight Gain While Taking Antipsychotic Medication…

Kategori:
PyrimidinesPyrimidinones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirikizumab Approved DB14910
biotech | CAS: 1884201-71-1

Mirikizumab is a monoclonal antibody developed by Eli Lilly intended to treat ulcerative colitis. It inhibits the actions of interleukin-23 (IL-23), a pro-inflammatory cytokine that activates pathways contributing to the development of inflammatory diseases.[…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnti-Inflammatory Agents +16
Target Protein:
Interleukin-23 subunit alpha
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Mirococept DB06492
biotech | CAS: 507453-82-9

Mirococept (APT070) is a complement inhibitor currently under development for treatment of rheumatoid arthritis and I/RI. It is a truncated form of the human Complement Receptor 1 (CR1) linked to a unique Prodaptin™ construct that regulates the over-productio…

Target Protein:
Complement C3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirodenafil DB11792
small molecule | CAS: 862189-95-5

Mirodenafil has been used in trials studying the treatment and supportive care of Kidney Diseases, Urologic Diseases, Renal Insufficiency, Erectile Dysfunction, and Male Erectile Dysfunction.

Kategori:
AmidesEnzyme InhibitorsPhosphodiesterase 5 Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirogabalin DB11825
small molecule | CAS: 1138245-13-2

Mirogabalin has been used in trials studying the treatment of Post-herpetic Neuralgia, Pain Associated With Fibromyalgia, and Diabetic peripheral neuropathic pain.

Kategori:
AnalgesicsBridged-Ring CompoundsGabapentinoids +1
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirostipen DB06453
small molecule | CAS: 244130-01-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirtazapine Approved DB00370
small molecule | CAS: 85650-52-8

Mirtazapine is a tetracyclic _piperazino-azepine_ antidepressant agent that was initially approved for the treatment of major depressive disorder (MDD) in the Netherlands in 1994.[A177946] This drug was first manufactured by Organon Inc., and received FDA app…

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +38
Target Protein:
5-hydroxytryptamine receptor 2A5HT3 serotonin receptorAlpha-2A adrenergic receptor +4
Waktu Paruh20-40 hours [FDA la…
Vol. DistribusiThe volume of distr…
KlirensTotal body clearanc…
Genetik -
Mirvetuximab DB16235
biotech | CAS: 1453084-36-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirvetuximab soravtansine Approved DB12489
biotech | CAS: 1453084-37-1

Mirvetuximab soravtansine-gynx (IMGN853) is an antibody-drug conjugate (ADC) formed by a monoclonal antibody (M9346A) that targets folate receptor alpha (FR?), covalently joined by a cleavable disulfide linker to the genotoxic compound DM4 (also known as sora…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Folate receptor alpha
Waktu ParuhAfter the first dos…
Vol. DistribusiMirvetuximab soravt…
KlirensThe total plasma cl…
Genetik -
Misetionamide DB18098
small molecule | CAS: 856785-75-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Misonidazole DB11716
small molecule | CAS: 13551-87-6

Misonidazole is under investigation in clinical trial NCT00038038 (Assessment of Head and Neck Tumor Hypoxia Using 18F-Fluoromisonidazole).

Kategori:
Anti-Infective AgentsAntineoplastic AgentsAntiparasitic Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Misoprostol Approved DB00929
small molecule | CAS: 59122-46-2

Misoprostol is a prostaglandin analog used to reduce the risk of NSAID related ulcers, manage miscarriages, prevent post partum hemorrhage, and also for first trimester abortions.[L7616,L7619,A181589,A181583,A181697] The stimulation of prostaglandin receptors…

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAlimentary Tract and Metabolism +24
Target Protein:
Prostacyclin receptorProstaglandin E2 receptor EP3 subtypeProstaglandin E2 receptor EP2 subtype +2
Waktu ParuhThe half life of an…
Vol. DistribusiData regarding the …
KlirensBecause of the rapi…
Genetik -
Mitapivat Approved DB16236
small molecule | CAS: 1260075-17-9

Mitapivat is a novel, first-in-class pyruvate kinase activator. It works to increase the activity of erythrocyte pyruvate kinase, a key enzyme involved in the survival of red blood cells. Defects in the pyruvate kinase enzyme in various red blood cells disord…

Kategori:
Anemia, Hemolytic, Congenital, drug therapyBlood and Blood Forming OrgansCytochrome P-450 CYP1A2 Substrates +27
Target Protein:
Pyruvate kinase PKLRAromatase
Waktu ParuhIn patients with py…
Vol. DistribusiThe mean volume of …
KlirensPopulation pharmaco…
Genetik -
Mitazalimab DB15225
biotech | CAS: 2055640-86-1

Mitazalimab is under investigation in clinical trial NCT02379741 (ADC-1013 First-in-Human Study).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitemcinal DB06587
small molecule | CAS: 154738-42-8

Mitemcinal (GM-611) is a novel erythromycin-derived prokinetic agent that acts as an agonist at the motilin receptor.

Kategori:
Anti-Bacterial AgentsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +5
Target Protein:
Motilin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitiglinide DB01252
small molecule | CAS: 145375-43-5

Mitiglinide is a drug for the treatment of type 2 diabetes. It may stimulate insulin secretion in beta-cells by closing off ATP dependant potassium ion channels.

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsDrugs Used in Diabetes +4
Target Protein:
ATP-binding cassette sub-family C member 8ATP-sensitive inward rectifier potassium channel 10Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitiperstat DB18963
small molecule | CAS: 1933460-19-5

Mitiperstat is under investigation in clinical trial NCT05492877 (An Efficacy and Safety Study of Mitiperstat (AZD4831) (MPO Inhibitor) vs Placebo in the Treatment of Moderate to Severe COPD.).

Target Protein:
Myeloperoxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mito-4509 DB05846
small molecule

Mito-4509 is a non-feminizing estrogen analog that could affect mitochondrial metabolic pathways. It is used to treat Parkinson's Disease, Alzheimer's Disease, Retinal Disorders and other neurologic Disorders.

Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitobronitol DB13543
small molecule | CAS: 488-41-5

Deskripsi belum tersedia.

Kategori:
AlcoholsAlkylating DrugsAntineoplastic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitoguazone DB12967
small molecule | CAS: 459-86-9

Mitoguazone has been used in trials studying the treatment of Lymphoma, HIV Infections, and Lymphoma, Non-Hodgkin.

Kategori:
AmidinesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +2
Target Protein:
S-adenosylmethionine decarboxylase proenzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitometh DB12117
small molecule | CAS: 107465-03-2

Mitometh is under investigation for the treatment of Adenocarcinoma, Oropharyngeal Neoplasms, Nasopharyngeal Carcinoma, Non-small Cell Lung Cancer, and Stage IV Non-small Cell Lung Cancer, among others. Mitometh has been investigated for the treatment of Lung…

Kategori:
Hydrocarbons, ChlorinatedHydrocarbons, Halogenated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitomycin Approved DB00305
small molecule | CAS: 50-07-7

Mitomycin is an antineoplastic antibiotic first isolated by Japanese microbiologists in the 1950s from cultures of _Streptomyces caespitosus_.[L12867,A193419] It is an alkylating agent that inhibits DNA synthesis (and, at higher concentrations, RNA and protei…

Kategori:
Alkylating ActivityAlkylating DrugsAntibiotics, Antineoplastic +19
Target Protein:
DNA
Waktu Paruh8-48 min
Vol. Distribusi-
Klirens-
Genetik -
Mitomycin A DB19369
small molecule | CAS: 4055-39-4

Deskripsi belum tersedia.

Kategori:
AzirinesHeterocyclic Compounds, Fused-RingIndolequinones +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitoquinone DB05063
small molecule | CAS: 444890-41-9

Mitoquinone is based on a novel technology, targeted lipophilic cations, that transport and concentrate antioxidants into the mitochondria -- organelles inside cells that provide energy for life processes -- where they accumulate up to a thousand fold. In 200…

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitotane Approved DB00648
small molecule | CAS: 53-19-0

Mitotane is an adrenolytic isomer of the insecticide dichlorodiphenyldichloroethane (DDD) - itself a metabolite of dichlorodiphenyltrichloroethane (DDT) - that inhibits cells of the adrenal cortex and their production of hormones. It has been in use since 195…

Kategori:
Adrenal Cytotoxic AgentsAntineoplastic AgentsAntineoplastic Agents, Hormonal +15
Target Protein:
Cytochrome P450 11B1, mitochondrialEstrogen receptorProgesterone receptor +2
Waktu ParuhThe plasma terminal…
Vol. DistribusiMitotane is extensi…
Klirens-
Genetik -
Mitoxantrone Approved DB01204
small molecule | CAS: 65271-80-9

An anthracenedione-derived antineoplastic agent.

Kategori:
AnalgesicsAnthracenesAnthracyclines and Related Substances +30
Target Protein:
DNA topoisomerase 2-betaDNADNA topoisomerase 2-alpha
Waktu Paruh75 hours
Vol. Distribusi* 1000 L/m2
Klirens* 21.3 L/hr/m2 [Eld…
Genetik -
Mitsugumin-53 DB16969
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitumomab DB06462
biotech | CAS: 216503-58-1

Mitumomab, an anti-BEC-2 monoclonal antibody derived from mice, was previously studied to treat small cell lung carcinoma in combination with BCG vaccination.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MIV-701 DB05736
small molecule

MIV-701 is a selective, potent inhibitor of the protease Cathepsin K. It is developed for the treatment of osteoporosis.

Target Protein:
Cathepsin K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MIV-711 DB15599
small molecule

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsAntineoplastic AgentsAntirheumatic Agents
Target Protein:
Cathepsin K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mivelsiran DB19003
biotech | CAS: 2572991-83-2

Mivelsiran is under investigation in clinical trial NCT06393712 (A Phase 2 Trial of ALN-APP in Patients With Cerebral Amyloid Angiopathy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mizagliflozin DB19036
small molecule | CAS: 666843-10-3

Mizagliflozin is under investigation in clinical trial NCT05721729 (Effect of Mizagliflozin Repeat Dosing on Adverse Events and Postprandial Glucose Excursions).

Kategori:
CarbohydratesGlycosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mizolastine Approved DB12523
small molecule | CAS: 108612-45-9

Mizolastine is under investigation in clinical trial NCT01928316 (A Bioequivalence Study of Domestic (Made in China) and Imported Mizolastine Tablets in Healthy Volunteers).

Kategori:
Antihistamines for Systemic UseCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +9
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mizoribine DB12617
small molecule | CAS: 50924-49-7

Mizoribine has been investigated for the treatment of Rheumatoid Arthritis.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Infective Agents +15
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0249 DB11910
small molecule | CAS: 1167574-41-5

MK0249 has been used in trials studying the treatment of Hypopnea Syndrome, Alzheimer's Disease, Paranoid Schizophrenia, Sleep Apnea, Obstructive, and Excessive Daytime Sleepiness, among others.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Target Protein:
Histamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0354 DB05939
small molecule | CAS: 851776-28-8

MK-0354, is an orally administered drug candidate under development by Merck for the treatment of atherosclerosis and related disorders. It targets G protein-coupled receptor, or GPCR, that have the potential to regulate plasma lipid profiles, including HDL, …

Target Protein:
Hydroxycarboxylic acid receptor 2G-protein coupled estrogen receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0482 DB17453
biotech

MK-0482 is a novel humanized IgG4 monoclonal antibody targeting the immunoglobulin-like transcript (ILT) 3.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0533 DB15242
small molecule | CAS: 668455-28-5

MK-0533 is under investigation in clinical trial NCT00543959 (Efficacy and Tolerability of MK0533 in Patients With Type 2 Diabetes (0533-005)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0557 DB12168
small molecule | CAS: 328232-95-7

MK0557 has been investigated for the treatment of Schizophrenia and Paranoid Schizophrenia.

Kategori:
Cycloparaffins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0668 DB15791
small molecule | CAS: 865110-07-2

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +3
Target Protein:
Integrin beta-1Integrin alpha-4VLA-4 (very late antigen-4)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0686 DB12563
small molecule | CAS: 578727-68-1

MK0686 has been used in trials studying the treatment of Osteoarthritis, Pain, Postoperative, and Neuralgia, Postherpetic.

Kategori:
AcetatesAcids, AcyclicAcids, Carbocyclic +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0731 DB08037
small molecule | CAS: 845256-65-7

MK-0731 is a kinesin spindle protein inhibitor and antineoplastic agent.

Target Protein:
Kinesin-like protein KIF11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0736 DB15209
small molecule | CAS: 719272-79-4

MK-0736 is under investigation in clinical trial NCT00679055 (A Study of How MK-0736 Affects Arterial Plaque (0736-006)(TERMINATED)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0752 DB12852
small molecule | CAS: 471905-41-6

Mk 0752 is under investigation in clinical trial NCT00572182 (MK0752 in Treating Young Patients With Recurrent or Refractory CNS Cancer).

Kategori:
Acids, AcyclicAmyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme Inhibitors +5
Target Protein:
Gamma-secretase subunit PEN-2NicastrinGamma-secretase subunit APH-1B +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 8001–8050 dari 12560
Sebelumnya Halaman 161 / 252 Berikutnya