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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (14063)

Halaman 161 / 282
K-777 DB17760
small molecule | CAS: 502960-90-9

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +5
Target Protein:
Cruzipain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
K201 free base DB02929
small molecule | CAS: 145903-06-6

Deskripsi belum tersedia.

Target Protein:
Annexin A5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KAb201 DB17210
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Kaempferia galanga root Approved DB14288
biotech

Kaempferia galanga root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Kaempherol DB01852
small molecule | CAS: 520-18-3

Deskripsi belum tersedia.

Target Protein:
Polyunsaturated fatty acid 5-lipoxygenasePolyunsaturated fatty acid lipoxygenase ALOX15Aldo-keto reductase family 1 member B1 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KAHR-102 DB17427
biotech

KAHR-102 is a dual signaling protein fusing cytotoxic T-lymphocyte-associated protein 4 (CTLA-4) to the Fas-ligand (FasL).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
KAI-1678 DB16211
biotech | CAS: 1041004-14-1

KAI-1678 is under investigation in clinical trial NCT01106716 (Safety and Efficacy Study of KAI-1678 to Treat Pain in Subjects With Postherpetic Neuralgia).

Kategori:
Amino Acids, Peptides, and ProteinsProtein Kinase C-epsilon, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kanamycin Approved DB01172
small molecule | CAS: 59-01-8

Kanamycin (also known as kanamycin A) is an aminoglycoside bacteriocidal antibiotic, available in oral, intravenous, and intramuscular forms, and used to treat a wide variety of infections. Kanamycin is isolated from the bacterium Streptomyces kanamyceticus a…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAminoglycoside Antibacterials +16
Target Protein:
30S ribosomal protein S1216S ribosomal RNA
Waktu Paruh2.5 hours
Vol. Distribusi-
Klirens-
Genetik -
KAND567 DB16511
small molecule | CAS: 911715-90-7

KAND567, a small molecule, blocks the fractaline (CX3CL1) receptor, which mediates the immune system response to inflammation[L32908]. Because COVID-19 involves cytotoxic cells associated with this pathway, KAND567 is currently being tested as a treatment for…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
CX3C chemokine receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kaolin Approved DB01575
small molecule | CAS: 1332-58-7

Kaolin is a layered silicate mineral. Kaolin is used in ceramics, medicine, coated paper, as a food additive, in toothpaste, as a light diffusing material in white incandescent light bulbs, and in cosmetics. Until the early 1990s it was the active substance o…

Kategori:
Alimentary Tract and MetabolismAluminium CompoundsAluminum Silicates +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kappadione Approved DB09332
small molecule | CAS: 131-13-5

Kappadione is a Vitamin K derivative (chemically, it is menadiol sodium diphosphate), previously approved by FDA prior to 1982 and marketed by Lilly Marketing for this drug has been discontinued and is not available in North America [L1543]. It has been found…

Target Protein:
ProthrombinCoagulation factor VIICoagulation factor IX +4
Waktu ParuhMean elimination ha…
Vol. DistribusiIn a study of rabbi…
KlirensThe plasma clearanc…
Genetik -
Kava Approved DB01322
small molecule | CAS: 9000-38-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
KB-141 DB03176
small molecule | CAS: 219691-94-8

An anticholesteremic agent.

Kategori:
Acids, CarbocyclicBenzene DerivativesEthers +2
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KB001 DB05222
biotech

KB001 is a Humaneered™ PEGylated monoclonal antibody fragment for the treatment of life-threatening Pseudomonas aeruginosa infections, a common problem of cystic fibrosis and mechanically ventilated patients.

Target Protein:
Low calcium response locus protein V
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KB002 DB05194
small molecule

KB002 is an engineered human IgG1k antibody engineered human. It is developed for the treatment of autoimmune diseases, initially rheumatoid arthritis.

Target Protein:
Granulocyte-macrophage colony-stimulating factor receptor subunit alphaGranulocyte-macrophage colony-stimulating factorGM-CSF receptor alpha subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KB105 DB18224
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KB3305 DB06349
small molecule | CAS: 639520-46-0

KB3305 is an investigational liver selective antagonist for the glucocorticoid receptor, developed by Karo Bio for the treatment of Type 2 Diabetes.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesBile Acids and Salts +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KB407 DB18223
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KBP-COVID-19 DB15858
biotech

The KBP-201 COVID-19 Vaccine was developed by British American Tobacco’s (BAT) U.S. biotech subsidiary, Kentucky BioProcessing (KBP). KBP cloned COVID-19’s genetic sequence, identified a potential antigen, and then inserted it into tobacco plants for reproduc…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
KD7040 DB05214
small molecule

KD7040 is a topically-delivered inducible nitric oxide synthase (iNOS) inhibitor for the treatment of neuropathic pain. The KD7040 IND was filed in 4Q06, and a Phase Ib clinical trial began 2Q07. It is being developed by Kalypsys.

Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kelatorphan DB08040
small molecule | CAS: 92175-57-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsCentral Nervous System Agents +4
Target Protein:
Aminopeptidase NGlutamyl aminopeptidaseLeukotriene A-4 hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KER-047 DB19111
small molecule | CAS: 2248154-85-8

KER-047 is under investigation in clinical trial NCT05927012 (A Study to Evaluate the Safety and Preliminary Efficacy of a Response-guided Dose Titration of KER-047 in the Treatment of Functional IDA (Iron Deficiency Anemia).).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ketamine Approved DB01221
small molecule | CAS: 6740-88-1

Ketamine is an NMDA receptor antagonist with a potent anesthetic effect.[A31869] It was developed in 1963 as a replacement for phencyclidine (PCP) by Calvin Stevens at Parke Davis Laboratories. It started being used for veterinary purposes in Belgium and in 1…

Kategori:
Agents producing tachycardiaAmino AcidsAmino Acids, Acidic +35
Target Protein:
Glutamate receptor ionotropic, NMDA 3A5-hydroxytryptamine receptor 3ANeuronal acetylcholine receptor subunit alpha-7 +11
Waktu ParuhThe reported half-l…
Vol. DistribusiThe apparent volume…
KlirensThe clearance rate …
Genetik -
Ketanserin DB12465
small molecule | CAS: 74050-98-9

Ketanserin has been investigated for the treatment of Septic Shock, Severe Sepsis, and Diabetic Foot Ulcer.

Kategori:
Antidepressive AgentsAntihypertensive AgentsAntiplatelet agents +11
Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ketazolam Approved DB01587
small molecule | CAS: 27223-35-4

Ketazolam is a benzodiazepine derivative with anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant activity. Ketazolam is not approved in Canada or America.

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +16
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh26-200 hours
Vol. Distribusi-
Klirens-
Genetik -
Ketobemidone DB06738
small molecule | CAS: 469-79-4

Ketobemidone is a powerful opioid analgesic. It also has some NMDA-antagonist properties. This makes it useful for some types of pain that don't respond well to other opioids. The most commonly cited equalisation ratio for analgesic doses is 25 mg of ketobemi…

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +20
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Waktu ParuhPlasma half-life: 2…
Vol. Distribusi-
Klirens-
Genetik -
Ketocaine DB16020
small molecule | CAS: 1092-46-2

Deskripsi belum tersedia.

Kategori:
Ketones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ketoconazole Approved DB01026
small molecule | CAS: 65277-42-1

Ketoconazole is an imidazole antifungal agent used in the prevention and treatment of a variety of fungal infections.[FDA Label] It functions by preventing the synthesis of ergosterol, the fungal equivalent of cholesterol, thereby increasing membrane fluidity…

Kategori:
14-alpha Demethylase InhibitorsAgents causing hyperkalemiaAnti-Infective Agents +55
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol 14-alpha demethylaseSteroid 17-alpha-hydroxylase/17,20 lyase +5
Waktu ParuhKetoconazole experi…
Vol. DistribusiKetoconazole has an…
KlirensKetoconazole has an…
Genetik -
small molecule | CAS: 1297537-33-7

Ketodarolutamide, a nonsteroidal antiandrogen (NSAA), is the major active metabolite of [darolutamide].

Kategori:
AntiandrogensAntiandrogens, non-steroidal
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ketoprofen Approved DB01009
small molecule | CAS: 22071-15-4

Ketoprofen, a propionic acid derivative, is a nonsteroidal anti-inflammatory agent (NSAIA) with analgesic and antipyretic properties.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +38
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1C-X-C chemokine receptor type 1
Waktu ParuhConventional capsul…
Vol. Distribusi-
Klirens* Oral-dose cl=6.9 …
Genetik -
Ketorolac Approved DB00465
small molecule | CAS: 74103-06-3

Ketorolac is a Non-steroidal anti-inflammatory drug (NSAID) and is commercially available as an oral tablet, injectable, nasal spray and as an ophthalmic solution.[L6358][L6508][L11055][L3674][L11070] It's analgesic properties make it a useful pain manage…

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +26
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhKetorolac trometham…
Vol. DistribusiThe apparent volume…
KlirensThe plasma clearanc…
Genetik -
Ketotifen Approved DB00920
small molecule | CAS: 34580-13-7

Ketotifen is a benzocycloheptathiophene derivative[A231204] with potent antihistaminic and mast cell stabilizing properties. It has a similar structure to some other first-generation antihistamines such as [cyproheptadine] and [azatadine].[A231204] Ketotif…

Kategori:
Anti-Allergic AgentsAnti-Asthmatic AgentsAntihistamine Drugs +15
Target Protein:
Histamine H1 receptor6-phosphogluconate dehydrogenase, decarboxylating
Waktu ParuhKetotifen clearance…
Vol. Distribusi-
Klirens-
Genetik -
Keyhole limpet hemocyanin Approved DB05299
biotech

Keyhole limpet hemocyanin is an immune modulator, given as a vaccine to help the body respond to cancer. A natural protein isolated from the marine mollusc keyhole limpet. Keyhole limpet hemocyanin is an immunogenic carrier protein that, in vivo, increases an…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntigens +7
Target Protein:
Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KF-0210 DB17476
small molecule

KF-0210 is a small molecule developed by Keythera Pharmaceuticals. It is being investigated for cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KF-1601 DB18297
small molecule | CAS: 2699634-21-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KH064 DB04287
small molecule | CAS: 393569-31-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
Phospholipase A2, membrane associated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KHK2455 DB17524
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kifunensine DB02742
small molecule | CAS: 109944-15-2

Deskripsi belum tersedia.

Kategori:
Enzyme Inhibitors
Target Protein:
Alpha-mannosidase 2Endoplasmic reticulum mannosyl-oligosaccharide 1,2-alpha-mannosidaseMannosyl-oligosaccharide alpha-1,2-mannosidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KIN-3248 DB17587
small molecule

KIN-3248 is a small molecule that targets and inhibits oncogenic fibroblast growth factor receptors (FGFRs). It was designed to mainly target FGFR2 and FGFR3 alterations, which act as oncogenic drivers in 10-20% of cholangiocarcinoma and 20-35% of urothelial …

Target Protein:
Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kinetin Approved DB11336
small molecule | CAS: 525-79-1

Kinetin is a cytokinin which are plant hormones promotes cell division and plant growth. It was shown to naturally exist in DNA of organisms including humans and various plants. While kinetin is used in tissue cultures to produce new plants, it is also found …

Kategori:
CytokininsGrowth SubstancesHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KIO-301 DB18465
small molecule | CAS: 1224953-72-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kisspeptin DB19112
biotech | CAS: 388138-21-4

Kisspeptin is under investigation in clinical trial NCT03315325 (Age-dependent Changes in the Responsiveness of Hypothalamic Pituitary Gonadal Axis in Men).

Kategori:
Amino Acids, Peptides, and ProteinsIntercellular Signaling Peptides and ProteinsNeoplasm Proteins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kisspeptin-10 DB16210
biotech | CAS: 374675-21-5

Kisspeptin-10 is under investigation in clinical trial NCT03771326 (KP-10 and Insulin Secretion in Men).

Kategori:
Amino Acids, Peptides, and ProteinsGenes, Tumor SuppressorIntercellular Signaling Peptides and Proteins +5
Target Protein:
KiSS-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KIT-13 DB18093
small molecule | CAS: 103628-72-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kitasamycin DB09309
small molecule | CAS: 1392-21-8

Kitasamycin is a macrolide antibiotic derived from <em>Streptomyces kitasatoensis</em>.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KITE-222 DB17195
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KL1333 DB17622
small molecule | CAS: 1800405-30-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Kojic acid DB01759
small molecule | CAS: 501-30-4

Deskripsi belum tersedia.

Kategori:
AntioxidantsBiological FactorsCompounds used in a research, industrial, or household setting +3
Target Protein:
Tyrosinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Konjac mannan DB14963
small molecule | CAS: 37220-17-0

Konjac mannan is under investigation in clinical trial NCT01709955 (The Effects of Glucomannan on Weight Loss).

Kategori:
CarbohydratesGastrointestinal AgentsLaxatives +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
KOS-2187 DB05946
small molecule

KOS-2187, a novel erythromycin-based motilin agonist, or motilide, as a clinical candidate for the treatment of gastrointestinal motility disorders such as gastroparesis and gastroesophageal reflux disease (GERD).

Target Protein:
Promotilin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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