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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
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6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Halaman 160 / 252
MG-S-2525 DB18063
small molecule

Deskripsi belum tersedia.

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MG98 DB06544
biotech

MG98, a second-generation antisense oligodeoxynucleotide inhibitor of human DNMT1, was investigated in the completed clinical trial NCT00003890 for treating patients with advanced solid tumors.

Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
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MGB-BP-3 DB12892
small molecule | CAS: 1000277-08-6

Mgb Bp 3 is under investigation in clinical trial NCT02518607 (Safety, Blood Levels and Effects of MGB-BP-3).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
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MGD-024 DB17265
biotech

MGD-024 is an anti-CD123/anti-CD3 bispecific DART molecule.

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MGN-4893 DB17338
biotech

MGN-4893 is an inhibitor of microRNA-451. In February 2011, it was granted FDA orphan designation for the treatment of polycythemia vera.[L47356]

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Mibampator DB12717
small molecule | CAS: 375345-95-2

Mibampator has been used in trials studying the treatment of Alzheimer's Disease.

Kategori:
AmidesBenzene DerivativesSulfones +1
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Mibavademab DB16673
biotech | CAS: 2305770-44-7

Mibavademab is under investigation in clinical trial NCT04159415 (Study of REGN4461, a Leptin Receptor Agonist Antibody, in Patients With Generalized Lipodystrophy).

Waktu Paruh-
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Mibefradil DB01388
small molecule | CAS: 116644-53-2

Mibefradil was withdrawn from the market in 1998 because of potentially harmful interactions with other drugs.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +31
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1GVoltage-dependent T-type calcium channel subunit alpha-1HVoltage-dependent L-type calcium channel subunit alpha-1C +8
Waktu Paruh17 to 25 hours at s…
Vol. Distribusi-
Klirens-
Genetik -
Mibenratide DB15195
small molecule | CAS: 1239011-83-6

Mibenratide is under investigation in clinical trial NCT01798745 (A Study to Assess the Pharmacokinetics and Pharmacodynamics of JNJ-54452840 in Participants With Heart Failure and Anti-beta1-adrenergic Receptor Autoantibodies).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
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Micafungin Approved DB01141
small molecule | CAS: 235114-32-6

Micafungin is an antifungal drug. It belongs to the antifungal class of compounds known as echinocandins and exerts its effect by inhibiting the synthesis of 1,3-beta-D-glucan, an integral component of the fungal cell wall.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +9
Target Protein:
1,3-beta-glucan synthase component FKS11,3-beta-glucan synthase component GSC2
Waktu Paruh14-17 hours
Vol. Distribusi* 0.39 ± 0.11 L/kg …
Klirens* 0.359 +/- 0.179 m…
Genetik -
Miconazole Approved DB01110
small molecule | CAS: 22916-47-8

Miconazole is a broad-spectrum azole antifungal with some activity against Gram-positive bacteria as well.[A203636] It is widely used to treat mucosal yeast infections, including both oral and vaginal infections; although intravenous miconazole is no longer a…

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +41
Target Protein:
Lanosterol 14-alpha demethylaseNitric oxide synthase 3Nitric oxide synthase, inducible +5
Waktu ParuhMiconazole has a te…
Vol. DistribusiA 1200 mg miconazol…
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
CollagenasesEndopeptidasesEnzymes +6
Waktu Paruh-
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Microcrystalline cellulose Approved DB14158
small molecule | CAS: 9004-34-6

A polysaccharide with glucose units linked as in CELLOBIOSE. It is the chief constituent of plant fibers, cotton being the purest natural form of the substance. As a raw material, it forms the basis for many derivatives used in chromatography, ion exchange ma…

Kategori:
BiopolymersCarbohydratesCellulose +9
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Micronomicin Approved DB13274
small molecule | CAS: 52093-21-7

Micronomicin is an aminoglycoside antibiotic which is marketed in Japan, and sold under the brand names Sagamicin and Luxomicina.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +11
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Midazolam Approved DB00683
small molecule | CAS: 59467-70-8

Midazolam is a short-acting hypnotic-sedative drug with anxiolytic, muscle relaxant, anticonvulsant, sedative, hypnotic, and amnesic properties.[A173842] It belongs to a class of drugs called _benzodiazepines_. This drug is unique from others in this class du…

Kategori:
Adjuvants, AnesthesiaAnestheticsAnti-Anxiety Agents +27
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site +1
Waktu Paruh**Intravenous**: …
Vol. DistribusiFemale gender, old …
Klirens**Intramuscular** …
Genetik -
Midecamycin DB13456
small molecule | CAS: 35457-80-8

Midecamycin is a naturally occurring 16-membered macrolide[A33072] that fits under the category of acetoxy-substituted macrolide antibiotics. In this molecule, an acetoxy group is substituted on the position 9 of the 16-member ring and on position 4 of the te…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +12
Waktu ParuhThe half-life of mi…
Vol. DistribusiThe reported appare…
KlirensMidecamycin present…
Genetik -
Midodrine Approved DB00211
small molecule | CAS: 42794-76-3

An ethanolamine derivative that is an adrenergic alpha agonist. It is used as a vasoconstrictor agent in the treatment of hypotension.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +19
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor
Waktu ParuhThe metabolites dis…
Vol. Distribusi-
Klirens* Renal cl=385 mL/m…
Genetik -
Midomafetamine DB01454
small molecule | CAS: 42542-10-9

An N-substituted amphetamine analog. It is a widely abused drug classified as a hallucinogen and causes marked, long-lasting changes in brain serotonergic systems. It is commonly referred to as MDMA or ecstasy. It is a widely abused drug classified as a hallu…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +20
Target Protein:
Synaptic vesicular amine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter +4
Waktu Paruh6–10 (though durati…
Vol. Distribusi-
Klirens-
Genetik -
Midostaurin Approved DB06595
small molecule | CAS: 120685-11-2

Midostaurin (as Rydapt) is a multitarget kinase inhibitor for the treatment for adult patients with newly diagnosed acute myeloid leukemia (AML) who have a specific genetic mutation called FLT3. It was initially characterized as a potential broad-spectrum ant…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +53
Target Protein:
Protein kinase C gamma typeProtein kinase C alpha typeVascular endothelial growth factor receptor 2 +4
Waktu ParuhElimination half li…
Vol. DistribusiThe Vd of midostaur…
KlirensThe clearance value…
Genetik -
Mifamurtide Approved DB13615
small molecule | CAS: 83461-56-7

Mifamurtide is an immunomodulator with antitumor activity via activation of macrophages and monocytes. Also called L-MTP-PE, mifamurtide may be a liposomal form of of the active ingredient MTP-PE, which is a synthetic, less pyrogenic, and longer-acting deriva…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAmino Sugars +15
Target Protein:
Toll-like receptor 4Nucleotide-binding oligomerization domain-containing protein 2
Waktu ParuhFollowing intraveno…
Vol. DistribusiThe mean volume of …
KlirensThe clearance from …
Genetik -
Mifepristone Approved DB00834
small molecule | CAS: 84371-65-3

Mifepristone is a progestational and glucocorticoid hormone antagonist. Its inhibition of progesterone induces bleeding during the luteal phase and in early pregnancy by releasing endogenous prostaglandins from the endometrium or decidua. As a glucocorticoid …

Kategori:
Abortifacient AgentsAbortifacient Agents, SteroidalAdrenal Cortex Hormones +49
Target Protein:
Progesterone receptorGlucocorticoid receptorProstate-specific antigen +1
Waktu Paruh18 hours
Vol. Distribusi-
Klirens-
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Migalastat Approved DB05018
small molecule | CAS: 108147-54-2

Fabry disease is a rare, progressive genetic disorder characterized by a defective GLA gene that causes a deficiency in the enzyme alpha-Galactosidase A (alpha-Gal A). This enzyme is responsible for breaking down glycosphingolipid substrate that, when deficie…

Kategori:
Alimentary Tract and MetabolismAlkaloidsAlpha-Galactosidase A (alpha-Gal A) Pharmacological Chaperones +6
Target Protein:
Alpha-galactosidase A
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIn healthy voluntee…
KlirensFollowing ascending…
Genetik -
Miglustat Approved DB00419
small molecule | CAS: 72599-27-0

Miglustat, commonly marketed under the trade name Zavesca, is a drug used to treat Gaucher disease. It inhibits the enzyme glucosylceramide synthase, an essential enzyme for the synthesis of most glycosphingolipids. It is only used for patients who cannot be …

Kategori:
Alimentary Tract and MetabolismAlkaloidsAnti-HIV Agents +14
Target Protein:
Ceramide glucosyltransferase
Waktu ParuhThe effective half-…
Vol. Distribusi-
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Milademetan DB15257
small molecule | CAS: 1398568-47-2

Milademetan is under investigation in clinical trial NCT02319369 (Safety, Tolerability and Pharmacokinetics of Milademetan Alone and With 5-Azacitidine (AZA) in Acute Myelogenous Leukemia (AML) or High-Risk Myelodysplastic Syndrome (MDS)).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Coagulation factor VIII
Waktu Paruh-
Vol. Distribusi-
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Milataxel DB12334
small molecule | CAS: 352425-37-7

Milataxel has been used in trials studying the treatment of Mesothelioma.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
Target Protein:
Tubulin beta-1 chainTubulin beta chain
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 129496-10-2

Deskripsi belum tersedia.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 802539-81-7

Milciclib Maleate is under investigation in clinical trial NCT01301391 (Study of Oral PHA-848125AC in Patients With Malignant Thymoma Previously Treated With Multiple Lines of Chemotherapy).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Cyclin-dependent kinase 2
Waktu Paruh-
Vol. Distribusi-
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Milk thistle Approved DB14375
biotech | CAS: 65666-07-1

Milk thistle is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +9
Waktu Paruh-
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Milnacipran Approved DB04896
small molecule | CAS: 92623-85-3

Milnacipran is a selective serotonin and norepinephrine reuptake inhibitor (SNRI) and like many agents in this category was originally developed for and continues to be approved and indicated for the treatment of depression [F3928, F3934, A175786, A175951]. F…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +30
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterNMDA receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThe total plasma cl…
Genetik -
Milrinone Approved DB00235
small molecule | CAS: 78415-72-2

Heart failure is a multifactorial condition that affects roughly 1-2% of the adult population. Often the result of long-term myocardial ischemia, cardiomyopathy, or other cardiac insults, heart failure results from an inability of the heart to perfuse periphe…

Kategori:
AminesAminopyridinesCardiac Stimulants Excl. Cardiac Glycosides +12
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu ParuhMilrinone administe…
Vol. DistribusiMilrinone administe…
KlirensMilrinone administe…
Genetik -
Miltefosine Approved DB09031
small molecule | CAS: 58066-85-6

Miltefosine is a broad spectrum antimicrobial, anti-leishmanial, phospholipid drug that was originally developed in the 1980s as an anti-cancer agent. It is currently the only recognized oral agent used to treat visceral, cutaneous, and mucosal forms of leish…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAminesAnti-Infective Agents +9
Target Protein:
Phospholipase A2ATP-dependent translocase ABCB1
Waktu ParuhThe primary elimina…
Vol. DistribusiRadioactivity studi…
KlirensPlasma clearance is…
Genetik -
Milvexian DB16233
small molecule | CAS: 1802425-99-5

Milvexian is under investigation in clinical trial NCT03766581 (A Study on BMS-986177 for the Prevention of a Stroke in Patients Receiving Aspirin and Clopidogrel).

Target Protein:
Coagulation factor XI
Waktu Paruh-
Vol. Distribusi-
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Mimopezil DB05520
small molecule | CAS: 180694-97-7

Mimopezil is an acetylcholinesterase (AChE) inhibitor that has demonstrated potential use in the treatment of Alzheimer's disease. Mimopezil is a pro-drug that is rapidly absorbed and converted into huperzine A.

Waktu Paruh-
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Mimosine DB01055
small molecule | CAS: 500-44-7

Mimosine is an antineoplastic alanine-substituted pyridine derivative isolated from _Leucena glauca_.

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +2
Target Protein:
Serine hydroxymethyltransferase, cytosolicC-C motif chemokine 2Tyrosinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minaprine Approved DB00805
small molecule | CAS: 25905-77-5

Minaprine is a psychotropic drug which has proved to be effective in the treatment of various depressive states. Like most antidepressants minaprine antagonizes behavioral despair. Minaprine is an amino-phenylpyridazine antidepressant reported to be relative…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +17
Target Protein:
Amine oxidase [flavin-containing] A5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2A +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mineral oil Approved DB11057
small molecule | CAS: 8042-47-5

Mineral oil, or paraffin oil, is a mixture of higher alkanes from a mineral source, such as petroleum. Petroleum mineral oil is manufactured from crude oils by vacuum distillation to produce several distillates and a residual oil that are then further refined…

Kategori:
Alimentary Tract and MetabolismBasic Ointments and ProtectantsDermatologicals +5
Waktu Paruh-
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Minigastrin DB19196
biotech | CAS: 101212-63-9

Minigastrin is under investigation in clinical trial NCT06155994 (68ga-dota-mgs5 PET/CT in Patients With Advanced Neuroendocrine Tumours).

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal HormonesHormones +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minnelide DB17309
small molecule | CAS: 1254702-87-8

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +6
Target Protein:
Heat shock 70 kDa protein 1BHeat shock 70 kDa protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1254885-39-6

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minocycline Approved DB01017
small molecule | CAS: 10118-90-8

Minocycline was first described in the literacture in 1966.[A190681] It is a second generation tetracycline antibiotic that is active against gram-negative and gram-positive bacteria.[A190723] Like other semisynthetic tetracyclines, minocycline has modificati…

Kategori:
Agents Causing Muscle ToxicityAgents that produce neuromuscular block (indirect)Alimentary Tract and Metabolism +16
Target Protein:
30S ribosomal protein S930S ribosomal protein S416S ribosomal RNA +9
Waktu ParuhThe half life of mi…
Vol. DistribusiThe volume of distr…
KlirensIntravenous minocyc…
Genetik -
Minodronic acid DB06548
small molecule | CAS: 180064-38-4

Deskripsi belum tersedia.

Kategori:
OrganophosphonatesOrganophosphorus Compounds
Target Protein:
Farnesyl pyrophosphate synthaseGeranylgeranyl pyrophosphate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minoxidil Approved DB00350
small molecule | CAS: 38304-91-5

A potent direct-acting peripheral vasodilator (vasodilator agents) that reduces peripheral resistance and produces a fall in blood pressure.

Kategori:
Antihypertensive AgentsAntihypertensive Agents Indicated for HypertensionArteriolar Smooth Muscle, Agents Acting On +13
Target Protein:
ATP-sensitive inward rectifier potassium channel 1ReninProstaglandin G/H synthase 1
Waktu Paruh4.2 hours
Vol. Distribusi-
Klirens-
Genetik -
Minretumomab DB15470
biotech | CAS: 195189-17-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minzasolmin DB18961
small molecule | CAS: 1802518-92-8

Minzasolmin is under investigation in clinical trial NCT05543252 (An Extension Study to Evaluate the Long-term Efficacy, Safety and Tolerability of Minzasolmin (UCB0599) in Study Participants With Parkinson's Disease).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Miocamycin Approved DB13287
biotech | CAS: 55881-07-7

Miocamycin is a macrolide type antimicrobial [A176170]. This drug may be marketed in Japan for clinical use as it is listed in the Japanese pharmacopeia [L5737]. It has shown to be effective against several gram-positive and gram-negative microbes and may be …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MIP-1095 I-123 DB12994
small molecule | CAS: 949575-25-1

123 I Mip 1095 is under investigation in clinical trial NCT00712829 (Study to Evaluate the Safety, Pharmacokinetics, Tissue Distribution, Metabolism and Dosimetry of Two Prostate Cancer Imaging Agents).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
MIP-1095 I-131 DB14978
small molecule | CAS: 1258980-67-4

MIP-1095 I-131 is under investigation in clinical trial NCT03030885 (Use of an Experimental Radiopharmaceutical (131I-MIP-1095) in Men With Metastatic Castration-Resistant Prostate Cancer (mCRPC)).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mipicoledine DB15075
small molecule | CAS: 942149-56-6

Mipicoledine is under investigation in clinical trial NCT01048008 (Study of 4-Demethylcholesteryloxycarbonylpenclomedine (DM-CHOC-PEN) in Patients With Advanced Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mipomersen Approved DB05528
biotech | CAS: 1000120-98-8

Mipomersen sodium, which was known as the investigational drug, isis-301012, is the salt form of a synthetic phosphorothioate oligonucleotide. Mipomersen sodium prevents the formation of apo B-100, resulting in a decrease in the levels of apolipoprotein B (ap…

Kategori:
Anticholesteremic AgentsAntisense Elements (Genetics)Antisense Oligonucleotides +20
Target Protein:
Apolipoprotein B-100mRNA of ApoB-100
Waktu ParuhMipomersem has a ve…
Vol. DistribusiThe volume of distr…
KlirensClearance of mipome…
Genetik -
Mipsagargin DB11813
small molecule | CAS: 1245732-48-2

Mipsagargin has been used in trials studying the treatment of Prostate Cancer, Prostatic Neoplasms, Advanced Solid Tumors, Glioblastoma Multiforme, and Hepatocellular Carcinoma, among others.

Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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