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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 160 / 272
Letermovir Approved DB12070
small molecule | CAS: 917389-32-3

Letermovir recieved approval from the FDA on November 8th, 2017 for use in prophylaxis of cytomegalovirus (CMV) infection in allogeneic hematopoietic stem cell transplant patients.[L1021] It is the first of a new class of CMV anti-infectives called DNA termin…

Kategori:
Acids, AcyclicAnti-Infective AgentsAntiinfectives for Systemic Use +44
Target Protein:
CMV DNA Terminase Complex
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe mean steady sta…
KlirensThe mean clearance …
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LetibotulinumtoxinA Approved DB16820
biotech | CAS: 1800016-51-6

The aesthetic utility of botulinum toxin was discovered incidentally following its initial use in the treatment of facial spasmodic disorders in the early 1970s.[A249920] The first aesthetic use of botulinum toxin was reported in 1989, when [onabotulinumtoxin…

Kategori:
Acetylcholine Release InhibitorsBotulinum Toxins, Type ACentral Nervous System Depressants +2
Target Protein:
Synaptosomal-associated protein 25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letolizumab DB19072
biotech | CAS: 1450981-87-9

Letolizumab is under investigation in clinical trial NCT02273960 (Study to Evaluate Safety and Efficacy in Adult Subjects With ITP).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Letosteine DB08939
small molecule | CAS: 53943-88-7

Letosteine is a mucolytic used in the treatment of chronic bronchopneumopathies and related conditions.

Kategori:
Cough and Cold PreparationsExpectorantsRespiratory System Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letrazuril DB12663
small molecule | CAS: 103337-74-2

Letrazuril has been used in trials studying the treatment of HIV Infections and Cryptosporidiosis.

Kategori:
Nitriles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letrozole Approved DB01006
small molecule | CAS: 112809-51-5

Letrozole, or CGS 20267, is an oral non-steroidal type II aromatase inhibitor first described in the literature in 1990.[A190543,A1559,L11623,L11626] It is a third generation aromatase inhibitor like [exemestane] and [anastrozole], meaning it does not signifi…

Kategori:
Agents Causing Muscle ToxicityAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
Aromatase
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Lettuce Approved DB10539
biotech

Lettuce allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +1
Target Protein:
Bacterial leucyl aminopeptidaseCytosol aminopeptidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Leukotriene C4 DB08855
small molecule | CAS: 72025-60-6

The conjugation product of LEUKOTRIENE A4 and glutathione. It is the major arachidonic acid metabolite in macrophages and human mast cells as well as in antigen-sensitized lung tissue. It stimulates mucus secretion in the lung, and produces contractions of no…

Kategori:
Arachidonic AcidsAutacoidsBiological Factors +8
Target Protein:
Cysteinyl leukotriene receptor 1Cysteinyl leukotriene receptor 2Multidrug resistance-associated protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leukotriene D4 DB11858
small molecule | CAS: 73836-78-9

Leukotriene D4 has been used in trials studying the diagnostic of Asthma and Allergic Rhinitis.

Kategori:
Arachidonic AcidsAutacoidsBiological Factors +8
Target Protein:
Cysteinyl leukotriene receptor 1Cysteinyl leukotriene receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leupeptin DB16961
small molecule | CAS: 55123-66-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCathepsins, antagonists & inhibitorsCysteine Proteinase Inhibitors +4
Target Protein:
Plasmepsin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leuprolide Approved DB00007
biotech | CAS: 53714-56-0

Leuprolide is a synthetic 9-residue peptide analogue of gonadotropin-releasing hormone (GnRH). Unlike the endogenous decapeptide GnRH, leuprolide contains a single D-amino acid (D-leucyl) residue, which helps to increase its circulating half-life from three t…

Kategori:
Adrenal Cortex HormonesAgents Causing Muscle ToxicityAmino Acids, Peptides, and Proteins +25
Target Protein:
Gonadotropin-releasing hormone receptorProgonadoliberin-1
Waktu ParuhLeuprolide has a te…
Vol. DistribusiLeuprolide has an a…
KlirensLeuprolide administ…
Genetik -
Leuvectin DB17303
biotech

Leuvectin (formerly known as VCL-1102) is a component of gene therapy along with cationic lipid 1,2-dimyristyloxypropyl-3-dimethyl-hydroxyethyl ammonium bromide/dioleyl-phosphatidyl-ethanolamine (DMRIE/DOPE).[A254711]

Kategori:
Biological ProductsComplex MixturesGene Transfer Techniques +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levacetylmethadol Approved DB01227
small molecule | CAS: 1477-40-3

Levacetylmethadol is a narcotic analgesic with a long onset and duration of action. It is used mainly in the treatment of narcotic dependence. Levacetylmethadol was withdrawn from use in the European Union due to its high risk of QT interval prolongation.…

Kategori:
AnalgesicsAnticholinergic AgentsCentral Nervous System Agents +20
Target Protein:
Mu-type opioid receptorNeuronal acetylcholine receptor subunit beta-4Neuronal acetylcholine receptor subunit alpha-3
Waktu Paruh2.6 days
Vol. Distribusi-
Klirens-
Genetik -
Levallorphan Approved DB00504
small molecule | CAS: 152-02-3

An opioid antagonist with properties similar to those of naloxone; in addition it also possesses some agonist properties. It should be used cautiously; levallorphan reverses severe opioid-induced respiratory depression but may exacerbate respiratory depressio…

Kategori:
AlkaloidsCentral Nervous System AgentsHeterocyclic Compounds, Fused-Ring +6
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Mu-type opioid receptor
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
Levamisole Approved DB00848
small molecule | CAS: 14769-73-4

Levamisole is an antihelminthic drug that was commonly used for the treatment of parasitic, viral, and bacterial infections. [A178117] It was manufactured by _Janssen_ and first used in 1969 as an agent to treat worm infestations[A178123] Levamisole was appro…

Kategori:
Adjuvants, ImmunologicAnthelminticsAnti-Infective Agents +10
Target Protein:
Neuronal acetylcholine receptor subunit alpha-3Alkaline phosphatase, tissue-nonspecific isozymeAlkaline phosphatase, germ cell type +4
Waktu Paruh4.4-5.6 hours (biph…
Vol. Distribusi-
Klirens-
Genetik -
Levamlodipine Approved DB09237
small molecule | CAS: 103129-82-4

Levamlodipine, also known as S-amlodipine, is a pharmacologically active enantiomer of [amlodipine], an antihypertensive medication.[L10833] Levamlodipine belongs to the dihydropyridine group of calcium channel blockers.[L10833] This medication was first mark…

Kategori:
Antiarrhythmic agentsAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +11
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1DNitric oxide synthase 3 +1
Waktu ParuhLevamlodipine has a…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Levilimab DB16387
biotech | CAS: 2035008-70-7

Levilimab is under investigation in clinical trial NCT04227366 (Study of the Efficacy and Safety of BCD-089 in Combination With Methotrexate in Patients With Active Rheumatoid Arthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levmetamfetamine Approved DB09571
small molecule | CAS: 33817-09-3

Levomethamphetamine, the L-enantiomer of methamphetamine is a sympathomimetic vasoconstrictor used in some over-the-counter (OTC) nasal decongestant inhalers in the United States.

Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Levobetaxolol Approved DB09351
small molecule | CAS: 93221-48-8

Levobetaxolol is a beta-blocker used to lower the pressure in the eye to treat conditions such as glaucoma. It was marketed as a 0.5% ophthalmic solution of levobetaxolol hydrochloride under the trade name Betaxon but has been discontinued.

Kategori:
Adrenergic AntagonistsAdrenergic beta-AntagonistsAgents causing hyperkalemia +3
Target Protein:
Beta-1 adrenergic receptor
Waktu ParuhThe mean half life …
Vol. Distribusi-
Klirens-
Genetik -
Levobunolol Approved DB01210
small molecule | CAS: 47141-42-4

A nonselective beta-adrenoceptor antagonist used in the treatment of glaucoma.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +22
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh20 hours
Vol. Distribusi-
Klirens-
Genetik -
Levobupivacaine Approved DB01002
small molecule | CAS: 27262-47-1

Levobupivacaine is an amino-amide local anaesthetic drug belonging to the family of n-alkylsubstituted pipecoloxylidide. It is the S-enantiomer of bupivacaine. Levobupivacaine hydrochloride is commonly marketed by AstraZeneca under the trade name Chirocaine.…

Kategori:
AmidesAminesAnesthetics +15
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh3.3 hours
Vol. Distribusi66.91 ±18.23 L [aft…
Klirens39.06 ±13.29 L/h [a…
Genetik -
Levocarnitine Approved DB00583
small molecule | CAS: 541-15-1

Constituent of striated muscle and liver. It is used therapeutically to stimulate gastric and pancreatic secretions and in the treatment of hyperlipoproteinemias.

Kategori:
Alimentary Tract and MetabolismAminesAmino Acids and Derivatives +9
Target Protein:
Carnitine O-palmitoyltransferase 1, muscle isoformXanthine dehydrogenase/oxidaseLiver carboxylesterase 1 +9
Waktu Paruh17.4 hours (elimina…
Vol. DistribusiThe steady state vo…
KlirensTotal body clearanc…
Genetik -
Levocetirizine Approved DB06282
small molecule | CAS: 130018-77-8

Levocetirizine is a selective histamine H<sub>1</sub> antagonist used to treat a variety of allergic symptoms.[A181748,A181790,L7694] It is the R enantiomer of [cetirizine].[L7694] Levocetirizine has greater affinity for the histamine H<sub>1</sub> receptor t…

Kategori:
Antihistamines for Systemic UseCentral Nervous System DepressantsCytochrome P-450 CYP3A Substrates +12
Target Protein:
Histamine H1 receptor
Waktu ParuhThe average half li…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Levodopa Approved DB01235
small molecule | CAS: 59-92-7

Levodopa is a prodrug of dopamine that is administered to patients with Parkinson's due to its ability to cross the blood-brain barrier[Label]. Levodopa can be metabolised to dopamine on either side of the blood-brain barrier and so it is generally administer…

Kategori:
AminesAmino AcidsAmino Acids, Aromatic +21
Target Protein:
D(1A) dopamine receptorD(1B) dopamine receptorD(2) dopamine receptor +2
Waktu Paruh2.3 hours for orall…
Vol. Distribusi168L for orally inh…
KlirensIntravenously admin…
Genetik -
small molecule | CAS: 99291-25-5

Levodropropizine is under investigation in clinical trial NCT01573663 (A Drug-Drug Interaction Study of Ambroxol and Levodropropizine).

Kategori:
AlcoholsAntitussive AgentsCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levofloxacin Approved DB01137
small molecule | CAS: 100986-85-4

Levofloxacin is a fluoroquinolone antibiotic and the optical S-(-) isomer of racemic [ofloxacin].[A190663] It reportedly carries 8 to 128-fold more activity against both gram-negative and gram-positive bacteria compared to R-(+)-ofloxacin[A190663] and remains…

Kategori:
4-QuinolonesAlimentary Tract and MetabolismAnti-Bacterial Agents +35
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu ParuhThe average termina…
Vol. DistribusiLevofloxacin is wid…
KlirensThe average apparen…
Genetik -
Levoketoconazole Approved DB05667
small molecule | CAS: 142128-57-2

Cushing's syndrome (CS) is underpinned by chronic hypercortisolism leading to multisystem morbidity, including effects on the cardiovascular and endocrine systems, metabolic syndrome with accompanying changes in body composition, neuropsychiatric effects, cha…

Kategori:
Adrenal Cortex HormonesAntiadrenal PreparationsAnticorticosteroids +32
Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyaseCytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial +2
Waktu ParuhLevoketoconazole ha…
Vol. DistribusiLevoketoconazole ha…
Klirens-
Genetik -
Levoleucovorin Approved DB11596
small molecule | CAS: 68538-85-2

Levoleucovorin is the enantiomerically active form of Folinic Acid (also known as 5-formyl tetrahydrofolic acid or leucovorin). Commercially available leucovorin is composed of a 1:1 racemic mixture of the dextrorotary and levorotary isomers, while levoleucov…

Kategori:
AntidotesCoenzymesCompounds used in a research, industrial, or household setting +14
Target Protein:
Serine hydroxymethyltransferase
Waktu ParuhThe mean terminal h…
Vol. DistribusiData can't be found.
KlirensData can't be found.
Genetik -
Levomefolic acid Approved DB11256
small molecule | CAS: 31690-09-2

Levomefolic acid (INN) is the metabolite of folic acid (Vitamin B9) and it is a predominant active form of folate found in foods and in the blood circulation, accounting for 98% of folates in human plasma [A19276]. It is transported across the membranes inclu…

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +10
Waktu ParuhThe mean eliminatio…
Vol. DistribusiCirculates in its f…
Klirens-
Genetik -
Levomenol Approved DB13153
small molecule | CAS: 23089-26-1

Bisabolol, or more formally ?-(?)-bisabolol or also known as levomenol, (-)-alpha-Bisabolol is found in fats and oils. (-)-alpha-Bisabolol is isolated from essential oil of Matricaria chamomilla (German chamomile) (-)-alpha-Bisabolol belongs to the family of …

Kategori:
Biological ProductsComplex MixturesLipids +7
Waktu Paruh-
Vol. DistribusiTo demonstrate the …
Klirens-
Genetik -
Levomenthol Approved DB00825
small molecule | CAS: 2216-51-5

Menthol is a covalent organic compound made synthetically or obtained from peppermint or other mint oils. Forming clear or white waxy, crystalline substance, menthol is typically solid at room temperature. (-)-Menthol is the naturally-occurring and main form …

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntipruritics +16
Target Protein:
Transient receptor potential cation channel subfamily M member 8Transient receptor potential cation channel subfamily A member 1Transient receptor potential cation channel subfamily V member 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levomethadone DB13515
small molecule | CAS: 125-58-6

Deskripsi belum tersedia.

Kategori:
Drugs Used in Addictive DisordersDrugs Used in Opioid DependenceNervous System
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levomilnacipran Approved DB08918
small molecule | CAS: 96847-54-0

Levomilnacipran is a selective serotonin and norepinephrine reuptake inhibitor (SNRI), although it is a more potent inhibitor of norepinephrine reuptake than serotonin reuptake.[A261181, A38560] Levomilnacipran is the more active 1S,2R-enantiomer in the racem…

Kategori:
Adrenergic Uptake InhibitorsAgents producing tachycardiaAntidepressive Agents +27
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporter
Waktu ParuhThe apparent termin…
Vol. DistribusiLevomilnacipran is …
KlirensFollowing oral admi…
Genetik -
small molecule | CAS: 154357-42-3

Levonadifloxacin is under investigation in clinical trial NCT03405064 (Comparative Study of Levonadifloxacin (IV and Oral) With Linezolid (IV and Oral) in Acute Bacterial Skin and Skin Structure Infections (ABSSSI)).

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levonordefrin Approved DB06707
small molecule | CAS: 829-74-3

Levonordefrin acts as a topical nasal decongestant and vasoconstrictor, most often used in dentistry.

Kategori:
Adrenergic AgonistsAgents producing tachycardiaAgents that produce hypertension +9
Target Protein:
Alpha-1D adrenergic receptorAlpha-1B adrenergic receptorAlpha-1A adrenergic receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levonorgestrel Approved DB00367
small molecule | CAS: 797-63-7

Levonorgestrel (LNG) is a synthetic progestogen similar to [Progesterone] used in contraception and hormone therapy.[A181988,T659] Also known as Plan B, it is used as a single agent in emergency contraception, and as a hormonal contraceptive released from an …

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +23
Target Protein:
Progesterone receptor3-oxo-5-alpha-steroid 4-dehydrogenase 1Estrogen receptor +3
Waktu ParuhThe elimination hal…
Vol. DistribusiOne pharmacokinetic…
KlirensClearance was found…
Genetik -
small molecule | CAS: 230313-75-4

Levophencynonate is under investigation in clinical trial NCT02299804 (A Clinical Trial to Evaluate Efficacy and Safety of Levophencynonate Hydrochloride in Patient With Vertigo).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2338-37-6

Levopropoxyphene is a stereoisomer of propoxyphene in the form of 2S, 3R enantiomer. It was sold as an antitussive, but it was removed from the market in the 70s.[T133] Levopropoxyphene was developed by Lilly and FDA approved on March 21st, 1962. This drug pr…

Kategori:
Acids, AcyclicAgents that reduce seizure thresholdAntitussive Agents +3
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levosalbutamol Approved DB13139
small molecule | CAS: 34391-04-3

Levosalbutamol, or levalbuterol, is a short-acting ?2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructive pulmonary disease (COPD). [Salbutamol] has been marketed as a racemic mixture, although beta2-agonist activity resides …

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +15
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh3.3 - 4 hours
Vol. Distribusi-
Klirens-
Genetik -
Levosimendan Approved DB00922
small molecule | CAS: 141505-33-1

Levosimendan increases calcium sensitivity to myocytes by binding to troponin C in a calcium dependent manner. This increases contractility without raising calcium levels. It also relaxes vascular smooth muscle by opening adenosine triphosphate sensitive pota…

Kategori:
Antiarrhythmic agentsCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy +14
Target Protein:
Troponin C, slow skeletal and cardiac musclesATP-sensitive inward rectifier potassium channel 11ATP-sensitive inward rectifier potassium channel 8 +1
Waktu ParuhEliminination half-…
Vol. Distribusi-
Klirens-
Genetik -
Levosulpiride DB16021
small molecule | CAS: 23672-07-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntipsychotic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levothyroxine Approved DB00451
small molecule | CAS: 51-48-9

Levothyroxine is a synthetically produced form of thyroxine, a major endogenous hormone secreted by the thyroid gland.[F4633] Also known as L-thyroxine or the brand name product Synthroid, levothyroxine is used primarily to treat hypothyroidism, a condition w…

Kategori:
Agents used to treat hypothyroidismAmino AcidsAmino Acids, Aromatic +16
Target Protein:
Integrin alpha-VIntegrin beta-3Thyroid hormone receptor alpha +1
Waktu ParuhT<sub>4</sub> half-…
Vol. Distribusi-
Klirens-
Genetik -
Levotofisopam DB19073
small molecule | CAS: 82059-51-6

Levotofisopam is under investigation in clinical trial NCT01519687 (Study of Levotofisopam 50 Mg Three Times a Day (TID) Administered for 7 Days on Hyperuricemia and Gout).

Kategori:
Antidepressive AgentsBenzazepinesCentral Nervous System Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levoverbenone DB13391
small molecule | CAS: 1196-01-6

Deskripsi belum tersedia.

Kategori:
Cough and Cold PreparationsExpectorants
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levovirin DB06523
small molecule | CAS: 206269-27-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lexacalcitol DB03451
small molecule | CAS: 131875-08-6

Lexacalcitol is a solid. This compound belongs to the vitamin D and derivatives class of chemicals. These are compounds containing a secosteroid backbone, usually secoergostane or secocholestane. It is known to target the vitamin D3 receptor.

Kategori:
Antineoplastic AgentsCholestanesCholestenes +11
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lexanersen DB17933
biotech | CAS: 2073015-40-2

Lexanersen is an antisense oligonucleotide under investigation for use as a disease-modifying therapy in Huntington's disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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