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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 159 / 236
Nadolol Approved DB01203
small molecule | CAS: 42200-33-9

Nadolol is a nonselective beta adrenal receptor blocker that is used to lower blood pressure.[L7922,L7925] Nonselective beta adrenal receptor blockers may no longer be first line in the treatment of hypertension as newer generations of beta adrenal receptor b…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +30
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu ParuhThe half life of na…
Vol. DistribusiIn healthy subjects…
KlirensIn healthy subjects…
Genetik -
NADPH DB02338
small molecule | CAS: 53-57-6

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Thioredoxin reductase 1, cytoplasmicGlucose-6-phosphate 1-dehydrogenasePteridine reductase 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nafarelin Approved DB00666
small molecule | CAS: 76932-56-4

Nafarelin is a potent synthetic agonist of gonadotropin-releasing hormone with 3-(2-naphthyl)-D-alanine substitution at residue 6. Nafarelin has been used in the treatments of central precocious puberty and endometriosis.

Kategori:
Adrenal Cortex HormonesAgents Causing Muscle ToxicityAmino Acids, Peptides, and Proteins +19
Target Protein:
Gonadotropin-releasing hormone receptorPutative gonadotropin-releasing hormone II receptor
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Nafcillin Approved DB00607
small molecule | CAS: 147-52-4

A semi-synthetic antibiotic related to penicillin, Naficillin is a narrow-spectrum beta-lactam antibiotic drug. It is a beta-lactamase-resistant penicillin that is indicated for the treatment of Staphylococcal infections caused by strains that are resistant t…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +17
Target Protein:
Penicillin-binding protein 1bPenicillin-binding protein 2BPenicillin-binding protein 2a +2
Waktu ParuhThe serum half-life…
Vol. DistribusiNafcillin is report…
Klirens-
Genetik -
Nafithromycin DB16246
small molecule | CAS: 1691240-78-4

Nafithromycin is under investigation in clinical trial NCT02903836 (Phase II Study of Oral Nafithromycin in CABP).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naftazone Approved DB13680
small molecule | CAS: 15687-37-3

Deskripsi belum tersedia.

Kategori:
Capillary Stabilizing AgentsCoagulantsHematologic Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naftidrofuryl DB13588
small molecule | CAS: 31329-57-4

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCardiovascular AgentsCentral Nervous System Depressants +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naftifine Approved DB00735
small molecule | CAS: 65472-88-0

Naftifine is a synthetic, broad spectrum, antifungal agent and allylamine derivative for the topical treatment of tinea pedis, tinea cruris, and tinea corporis caused by the organisms Trichophyton rubrum, Trichophyton mentagrophytes, Trichophyton tonsurans an…

Kategori:
AlkenesAllyl CompoundsAllylamine Antifungal +7
Target Protein:
Squalene monooxygenase
Waktu ParuhApproximately 2 to …
Vol. Distribusi-
Klirens-
Genetik -
Naftopidil DB12092
small molecule | CAS: 57149-07-2

Naftopidil has been investigated for the treatment of Disorder of Urinary Stent.

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +16
Target Protein:
Alpha-1A adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nagrestipen DB12075
biotech | CAS: 166089-33-4

Nagrestipen has been used in trials studying the treatment of CANCER, Neoplasm, Metastasis, Radiation Oncology, and Neoplasm Metastasis.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsChemokines +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naldemedine Approved DB11691
small molecule | CAS: 916072-89-4

Naldemedine is an opioid receptor antagonist [FDA Label]. It is a modified form of [DB00704] to which a side chain has been added to increase molecular weight and polar surface area resulting in restricted transport across the blood brain barrier. Naldemedine…

Kategori:
Alimentary Tract and MetabolismAlkaloidsDrugs for Constipation +8
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Nalfurafine DB13471
small molecule | CAS: 152657-84-6

Deskripsi belum tersedia.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingOpiate Alkaloids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nalidixic acid Approved DB00779
small molecule | CAS: 389-08-2

Nalidixic acid is a synthetic 1,8-naphthyridine antimicrobial agent with a limited bacteriocidal spectrum. It is an inhibitor of the A subunit of bacterial DNA gyrase.

Kategori:
4-QuinolonesAgents that reduce seizure thresholdAnti-Bacterial Agents +19
Target Protein:
DNADNA topoisomerase 2-betaDNA topoisomerase 2-alpha
Waktu Paruh1.1 to 2.5 hours in…
Vol. Distribusi-
Klirens-
Genetik -
Nalmefene Approved DB06230
small molecule | CAS: 55096-26-9

Nalmefene, a 6-methylene analogue of [naltrexone], is an opioid receptor antagonist.[L40684] It acts as an antagonist at the mu (?)-opioid and delta (?)-opioid receptors and a partial agonist at the kappa (?)-opioid receptor.[L1024] In Europe, nalmefene or…

Kategori:
AlkaloidsAntidotesAntipruritics +18
Target Protein:
Kappa-type opioid receptorDelta-type opioid receptorMu-type opioid receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiFollowing a 1 mg pa…
KlirensThe oral clearance …
Genetik -
Nalorphine DB11490
small molecule | CAS: 62-67-9

Nalorphine is a mixed opioid agonist–antagonist. It acts at two opioid receptors—at the mu receptor it has antagonistic effects, and at the kappa receptors it exerts high-efficacy agonistic characteristics. It is used to reverse opioid overdose and (starting …

Kategori:
AlkaloidsAntidotesCentral Nervous System Agents +10
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naloxegol Approved DB09049
small molecule | CAS: 854601-70-0

Naloxegol, for "PEGylated naloxol" is a peripherally-selective opioid antagonist developed by AstraZeneca. It was approved by the FDA in September 2014 and is indicated for the treatment of opioid-induced constipation (OIC) in adult patients with chronic non?…

Kategori:
AlcoholsAlimentary Tract and MetabolismAlkaloids +24
Target Protein:
Mu-type opioid receptor
Waktu Paruh6-11 hours.
Vol. Distribusi968 to 2140 L.
KlirensFeces (68%), urine …
Genetik -
Naloxone Approved DB01183
small molecule | CAS: 465-65-6

Naloxone is an opioid antagonist medication used to block or reverse the effects of opioid drugs, particularly within the setting of drug overdoses which are rapidly becoming a leading cause of death worldwide.[A234594] More specifically, naloxone has a high …

Kategori:
Alimentary Tract and MetabolismAlkaloidsAnalgesics +27
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +4
Waktu ParuhThe mean half life …
Vol. DistribusiThe volume of distr…
KlirensThe clearance of na…
Genetik -
small molecule | CAS: 133397-81-6

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naltrexone Approved DB00704
small molecule | CAS: 16590-41-3

Derivative of noroxymorphone that is the N-cyclopropylmethyl congener of naloxone. It is a narcotic antagonist that is effective orally, longer lasting and more potent than naloxone, and has been proposed for the treatment of heroin addiction. The FDA has app…

Kategori:
Agents Causing Muscle ToxicityAlcohol DeterrentsAlimentary Tract and Metabolism +21
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Gen Terkait:
OPRM1
Waktu Paruh4 hours for naltrex…
Vol. Distribusi* 1350 L [intraveno…
Klirens* ~ 3.5 L/min [afte…
Genetik 1 Varian
Naluzotan DB05562
small molecule | CAS: 740873-06-7

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAmidesAntidepressive Agents +7
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Namilumab DB13037
biotech | CAS: 1206681-39-1

Namilumab has been used in trials studying the treatment of Plaque Psoriasis and Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Namitecan DB12124
small molecule | CAS: 372105-27-6

Namitecan has been used in trials studying the treatment of Solid Tumors.

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic Agents, Phytogenic
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nanatinostat DB15419
small molecule | CAS: 1256448-47-1

Nanatinostat is under investigation in clinical trial NCT00697879 (Safety Study of the Histone Deacetylase Inhibitor, CHR-3996, in Patients With Advanced Solid Tumours).

Kategori:
Antineoplastic AgentsAza CompoundsHistone Deacetylase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nandrolone DB13169
small molecule | CAS: 434-22-0

Nandrolone, also known as 19-nortestosterone or 19-norandrostenolone, is a synthetic anabolic-androgenic steroid (AAS) derived from testosterone.

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +16
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nandrolone decanoate Approved DB08804
small molecule | CAS: 360-70-3

Nandrolone decanoate, also known as nandrolone caprinate, is an alkylated anabolic steroid indicated in the management of anemia of renal insufficiency and as an adjunct therapy in the treatment of senile and postmenopausal osteoporosis.[A233789,A233849,L3256…

Kategori:
Anabolic AgentsAndrogensBone Density Conservation Agents +16
Target Protein:
Androgen receptorProtein c-Fos5-hydroxytryptamine 2 receptor +3
Waktu ParuhNandrolone decanoat…
Vol. Distribusi-
Klirens50 mg, 100 mg, and …
Genetik -
Nangibotide DB16247
biotech | CAS: 2014384-91-7

Nangibotide is under investigation in clinical trial NCT04055909 (Efficacy, Safety and Tolerability of Nangibotide in Patients With Septic Shock).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsFatty Acids +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Nanrilkefusp alfa is a human fusion protein consisting of the cytokine interleukin (IL)-15 and the high-affinity binding sushi+ domain of IL-15 receptor alpha (IL-15Ra).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nanvuranlat DB18250
small molecule | CAS: 1037592-40-7

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naphazoline Approved DB06711
small molecule | CAS: 835-31-4

Naphazoline is a rapid acting imidazoline sympathomimetic vasoconstrictor of ocular or nasal artierioles[L5804,L5807]. It acts to decrease congestion and is found in many over the counter (OTC) eye drops and nasal preparations[L5804,L5807]. Naphazoline was…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +17
Target Protein:
D(2) dopamine receptorAlpha-2A adrenergic receptorAlpha-1A adrenergic receptor
Waktu ParuhHalf life has not b…
Vol. DistribusiDistribution data f…
KlirensClearance data for …
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 581-75-9

Deskripsi belum tersedia.

Kategori:
ArylsulfonatesArylsulfonic AcidsNaphthalenes +3
Target Protein:
Bacterioferritin comigratory proteinL-lactate dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naphthoquine DB16249
small molecule | CAS: 173531-57-2

Naphthoquine is under investigation in clinical trial NCT01930331 (Safety, Tolerability, Pharmacokinetics and Efficacy of ARCO).

Kategori:
AminesAntimalarialsAntiparasitic Products, Insecticides and Repellents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naporafenib DB18865
small molecule | CAS: 1800398-38-2

Naporafenib is under investigation in clinical trial NCT06346067 (A Study to Assess Naporafenib (ERAS-254) Administered With Trametinib in Patients With Nras-mutant Melanoma (SEACRAFT-2)).

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
RAF proto-oncogene serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naproxen Approved DB00788
small molecule | CAS: 22204-53-1

Naproxen is classified as a nonsteroidal anti-inflammatory dug (NSAID) and was initially approved for prescription use in 1976 and then for over-the-counter (OTC) use in 1994.[A178975] It can effectively manage acute pain as well as pain related to rheumatic …

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +41
Target Protein:
Pancreatic triacylglycerol lipaseProstaglandin G/H synthase 1Prostaglandin G/H synthase 2 +1
Waktu ParuhThe elimination hal…
Vol. DistribusiNaproxen has a volu…
KlirensNaproxen is cleared…
Genetik -
biotech | CAS: 676258-98-3

Naptumomab Estafenatox has been used in trials studying the treatment of Pancreatic Cancer, Renal Cell Carcinoma, and Non-Small-Cell Lung Carcinoma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBiological Factors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naratriptan Approved DB00952
small molecule | CAS: 121679-13-8

Naratriptan is a triptan drug that is selective for the 5-hydroxytryptamine1 receptor subtype. It is typically used for the treatment of migraine headaches.

Kategori:
Agents that produce hypertensionAminesAnalgesics +23
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B +1
Gen Terkait:
GNB3
Waktu Paruh5-8 hours
Vol. Distribusi* 170 L
Klirens* 6.6 mL/min/kg
Genetik 1 Varian
biotech | CAS: 1607824-64-5

Naratuximab emtansine is under investigation in clinical trial NCT01534715 (IMGN529 in Treating Patients With Relapsed or Refractory Non-Hodgkin's Lymphoma and Chronic Lymphocytic Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Narazaciclib DB19038
small molecule | CAS: 1357470-29-1

Narazaciclib is under investigation in clinical trial NCT06351644 (On 123300 (Narazaciclib) and Dexamethasone in Patients With Relapsed And/or Refractory Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naringenin DB03467
small molecule | CAS: 480-41-1

Deskripsi belum tersedia.

Kategori:
Anti-Ulcer AgentsBCRP/ABCG2 InhibitorsBenzopyrans +9
Target Protein:
HTH-type transcriptional regulator TtgREstrogen receptorAldo-keto reductase family 1 member C1 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naringin DB16859
small molecule | CAS: 10236-47-2

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Narlaprevir DB14760
small molecule | CAS: 865466-24-6

Deskripsi belum tersedia.

Kategori:
AmidesAmino AcidsAmino Acids, Branched-Chain +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Narlumosbart DB19002
biotech | CAS: 2646587-68-8

Narlumosbart is under investigation in clinical trial NCT06314698 (Narlumosbart Compared With Denosumab in Patients With Multiple Myeloma Bone Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Narnatumab DB14964
biotech | CAS: 1188275-92-4

Narnatumab is under investigation in clinical trial NCT01119456 (A Study of IMC-RON8 in Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Naronapride DB05542
small molecule | CAS: 860174-12-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +7
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Narsoplimab DB16418
biotech | CAS: 2108782-45-0

Thrombotic microangiopathies (TMA), including thrombotic thrombocytopenic purpura and atypical hemolytic uremic syndrome, are associated with injury and dysregulation of microvascular endothelium and platelets.[A241030] Evidence increasingly points to a role …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Mannan-binding lectin serine protease 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Natalizumab Approved DB00108
biotech | CAS: 189261-10-7

Natalizumab is a recombinant humanized IgG4? monoclonal antibody that binds to ?4-integrin.[L48041] While natalizumab was originally approved by the FDA to treat multiple sclerosis in 2004, it was withdrawn from the market following multiple reports of fatal …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Integrin alpha-4Low affinity immunoglobulin gamma Fc region receptor III-BHigh affinity immunoglobulin gamma Fc receptor I +1
Waktu ParuhFollowing the repea…
Vol. DistribusiFollowing the repea…
KlirensFollowing the repea…
Genetik -
Natamycin Approved DB00826
small molecule | CAS: 7681-93-8

Amphoteric macrolide antifungal antibiotic from Streptomyces natalensis or S. chattanoogensis. It is used for a variety of fungal infections, mainly topically. [PubChem]

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
Ergosterol
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nateglinide Approved DB00731
small molecule | CAS: 105816-04-4

Nateglinide is an oral antihyperglycemic agent used for the treatment of non-insulin-dependent diabetes mellitus (NIDDM). It belongs to the meglitinide class of short-acting insulin secretagogues, which act by binding to ? cells of the pancreas to stimulate i…

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Aromatic +21
Target Protein:
ATP-binding cassette sub-family C member 8Peroxisome proliferator-activated receptor gamma
Waktu Paruh1.5 hours
Vol. Distribusi10 liters in health…
Klirens-
Genetik -
Menampilkan 7901–7950 dari 11778
Sebelumnya Halaman 159 / 236 Berikutnya