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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 159 / 252
Methylpentynol DB13733
small molecule | CAS: 77-75-8

Deskripsi belum tersedia.

Kategori:
AlcoholsCentral Nervous System DepressantsFatty Alcohols +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylphenidate Approved DB00422
small molecule | CAS: 113-45-1

Methylphenidate is a central nervous system stimulant used most commonly in the treatment of Attention-Deficit/Hyperactivity Disorder (ADHD) and for narcolepsy. Also known as the marketed products Ritalin, Concerta, or Biphentin, methylphenidate is used with …

Kategori:
Acids, CarbocyclicAgents that produce hypertensionAgents that reduce seizure threshold +17
Target Protein:
Sodium-dependent dopamine transporter5-hydroxytryptamine receptor 1ASodium-dependent noradrenaline transporter
Waktu ParuhConcerta: The half-…
Vol. DistribusiConcerta: Plasma me…
KlirensThe apparent mean s…
Genetik -
Methylphenobarbital Approved DB00849
small molecule | CAS: 115-38-8

A barbiturate that is metabolized to phenobarbital. It has been used for similar purposes, especially in epilepsy, but there is no evidence mephobarbital offers any advantage over phenobarbital.

Kategori:
Anticholinergic AgentsAnticonvulsantsBarbiturates +20
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-4 +8
Waktu Paruh34 (range 11-67) ho…
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 4206-94-4

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicCholinesterase Inhibitors +3
Target Protein:
AcetylcholinesteraseCholinesteraseEsterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylprednisolone Approved DB00959
small molecule | CAS: 83-43-2

Methylprednisolone is a [prednisolone] derivative glucocorticoid with higher potency than [prednisone].[A188811] It was first described in the literature in the late 1950s.[A188811,A188814] Methylprednisolone was granted FDA approval on 24 October 1957.[L1…

Kategori:
Adrenal Cortex HormonesAdrenalsAnti-Acne Preparations +50
Target Protein:
Glucocorticoid receptorAnnexin A1
Waktu ParuhMethylprednisolone …
Vol. DistribusiThe average volume …
KlirensThe average plasma …
Genetik -
Methylprednisolone aceponate Approved DB14643
small molecule | CAS: 86401-95-8

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2921-57-5

A water-soluble ester of methylprednisolone used for cardiac, allergic, and hypoxic emergencies.

Kategori:
Adrenal Cortex HormonesAdrenalsAnti-Inflammatory Agents +21
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylprednisone Approved DB12952
small molecule | CAS: 91523-05-6

Methylprednisone has been used in trials studying the treatment of Leukemia, Rheumatoid Arthritis, Renal Transplantation, Kidney Transplantation, and Acute Lymphocytic Leukemia, among others.

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 CYP3A4 Substrates (strength unknown) +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10605-24-0

Deskripsi belum tersedia.

Kategori:
Antianginal AgentsCardiac TherapyOrganic Nitrates +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1119361-12-4

Methylsamidorphan is under investigation in clinical trial NCT01418092 (ALK37-007: Evaluation of Safety and Efficacy of ALKS 37 (RDC-1036) in Adults With Opioid-induced Constipation (OIC)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methyltestosterone Approved DB06710
small molecule | CAS: 58-18-4

A synthetic anabolic steroid used for treating men with testosterone deficiency or similar androgen replacement therapies. Also, has antineoplastic properties and so has been used secondarily in women with advanced breast cancer. Methyltestosterone is a sched…

Kategori:
3-Oxoandrosten (4) DerivativesAnabolic AgentsAndrogens +20
Target Protein:
Androgen receptorEstrogen receptor
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 56-04-2

Deskripsi belum tersedia.

Kategori:
Antithyroid agentsHormone AntagonistsHormones, Hormone Substitutes, and Hormone Antagonists +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 59322-44-0

Deskripsi belum tersedia.

Target Protein:
Trans-sialidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methyprylon Approved DB01107
small molecule | CAS: 125-64-4

Methyprylon is a sedative of the piperidinedione derivative family that was previously used for the treatment of insomnia. However, with the introduction of newer drugs with fewer side effects, such as benzodiazepines, the clinical use of methyprylon is now l…

Kategori:
Central Nervous System DepressantsHypnotics and SedativesNervous System +3
Target Protein:
GABA(A) ReceptorGamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh6-16 hours
Vol. Distribusi-
Klirens-
Genetik -
Methysergide Approved DB00247
small molecule | CAS: 361-37-5

An ergot derivative that is a congener of lysergic acid diethylamide. It antagonizes the effects of serotonin in blood vessels and gastrointestinal smooth muscle, but has few of the properties of other ergot alkaloids. Methysergide is used prophylactically i…

Kategori:
Agents that produce hypertensionAlkaloidsAnalgesics +20
Target Protein:
5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metiamide DB08805
small molecule | CAS: 34839-70-8

Metiamide is an H-2 receptor antagonist derived from burimamide. It was an intermediate product on the path to developing cimetidine.

Kategori:
Acid ReducersAmidesAnti-Ulcer Agents +8
Target Protein:
Histamine H2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meticillin Approved DB01603
small molecule | CAS: 61-32-5

One of the penicillins which is resistant to penicillinase but susceptible to a penicillin-binding protein. It is inactivated by gastric acid so administered by injection.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
MecA PBP2' (penicillin binding protein 2')Penicillin-binding protein 2aPenicillin-binding protein 1b +3
Waktu Paruh25-60 minutes
Vol. Distribusi-
Klirens-
Genetik -
Meticrane Approved DB13284
small molecule | CAS: 1084-65-7

Meticrane is a diuretic medication. It has been marketed in Japan under the trade name Arresten and is used to lower blood pressure [L5647].

Kategori:
DiureticsGenito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metildigoxin DB13401
small molecule | CAS: 30685-43-9

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsCarbohydratesCardanolides +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metipranolol Approved DB01214
small molecule | CAS: 22664-55-7

A beta-adrenergic antagonist effective for both beta-1 and beta-2 receptors. It is used as an antiarrhythmic, antihypertensive, and antiglaucoma agent.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metisazone DB13641
small molecule | CAS: 1910-68-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoclopramide Approved DB01233
small molecule | CAS: 364-62-5

Diabetic gastroparesis is a condition that causes frequent nausea and vomiting, which has a negative impact on quality of life and poses a significant burden on the healthcare system.[A184934] Metoclopramide is a dopamine antagonist used to treat nausea and v…

Kategori:
Acids, CarbocyclicAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +35
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 3AMuscarinic acetylcholine receptor M1 +1
Gen Terkait:
KCNH2 ADRA1D CYP2D6 +4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik 7 Varian
Metocurine Approved DB01336
small molecule | CAS: 5152-30-7

Dimethyltubocurarinium (INN) or metocurine (USAN), also known as dimethyltubocurarine, is a non-depolarizing muscle relaxant. Patients on chronic anticonvulsant drugs are relatively resistant to metocurine. [A2393]

Kategori:
Agents producing tachycardiaAlkaloidsAmines +18
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metocurine iodide Approved DB00416
small molecule | CAS: 7601-55-0

Metocurine iodide is a benzylisoquinolinium competitive nondepolarizing neuromuscular blocking agent. It is used as an anesthesia adjunct to induce skeletal muscle relaxation and to reduce the intensity of muscle contractions in convulsive therapy Metocurine …

Kategori:
AlkaloidsAminesAnticholinergic Agents +12
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit beta-2Neuronal acetylcholine receptor subunit alpha-2
Waktu Paruh3 to 4 hours
Vol. Distribusi-
Klirens-
Genetik -
Metolazone Approved DB00524
small molecule | CAS: 17560-51-9

A quinazoline-sulfonamide that is considered a thiazide-like diuretic which is long-acting so useful in chronic renal failure. It also tends to lower blood pressure and increase potassium loss.

Kategori:
AmidesAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +21
Target Protein:
Solute carrier family 12 member 3
Waktu ParuhApproximately 14 ho…
Vol. Distribusi-
Klirens-
Genetik -
Metopimazine DB13591
small molecule | CAS: 14008-44-7

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntiemeticsAntiemetics and Antinauseants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoprine DB04655
small molecule | CAS: 7761-45-7

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsFolic Acid Antagonists +1
Target Protein:
Peptide deformylase, mitochondrialHistamine N-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoprolol Approved DB00264
small molecule | CAS: 51384-51-1

Metoprolol is a selective beta-1 blocker commonly employed as the succinate and tartrate derivatives depending if the formulation is designed to be of immediate release or extended release.[A175159, L5530] The possibility of the generation of these formulatio…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-1 Receptor Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta adrenergic receptor
Gen Terkait:
ADRB1 CYP2D6 ADRB1
Waktu ParuhThe immediate relea…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik 3 Varian
Metoserpate DB11530
small molecule | CAS: 1178-28-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIndole Alkaloids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metralindole DB09306
small molecule | CAS: 54188-38-4

Metralindole, also known as Inkazan, is similar in structure and pharmacology to pirlindole. It functions as a reversible inhibitor of monoamine oxidase A. In Russia, this drug was investigated for potential antidepressant activity.

Kategori:
Heterocyclic Compounds, Fused-RingIndole AlkaloidsIndoles +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metreleptin Approved DB09046
biotech | CAS: 186018-45-1

Metreleptin, a recombinant analog of the human hormone leptin, is an orphan drug used to treat complications of leptin deficiency in people with lipodystrophy. Lipodystrophies include a range of disorders characterized by the reduction, absence, or altered di…

Kategori:
AdipokinesAlimentary Tract and MetabolismAmino Acids and Derivatives +11
Target Protein:
Leptin receptor
Waktu ParuhFollowing subcutane…
Vol. DistribusiFollowing intraveno…
KlirensThe clearance of me…
Genetik -
Metribolone DB02998
small molecule | CAS: 965-93-5

A synthetic non-aromatizable androgen and anabolic steroid. It binds strongly to the androgen receptor and has therefore also been used as an affinity label for this receptor in the prostate and in prostatic tumors.

Kategori:
EstranesEstrenesFused-Ring Compounds +1
Target Protein:
Progesterone receptorAndrogen receptorNuclear receptor coactivator 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrifonate DB11473
small molecule | CAS: 52-68-6

Metrifonate or trichlorfon is an irreversible organophosphate acetylcholinesterase inhibitor. It is a prodrug which is activated non-enzymatically into 2,2-dichlorovinyl dimethyl phosphate.

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrizamide DB01578
small molecule | CAS: 31112-62-6

Metrizamide is a solute for density gradient centrifugation offering higher maximum solution density without the problems of increased viscosity. It is also used as a resorbable, non-ionic contrast medium.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrizoic acid Approved DB09346
small molecule | CAS: 1949-45-7

Metrizoic acid is a molecule used as a contrast medium. It present a higher risk of allergic reactions due to its high osmolality. Its approval has been discontinued by the FDA. One study in 1976 demonstrated that metrizoic acid, when used for cardiac angiog…

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metronidazole Approved DB00916
small molecule | CAS: 443-48-1

Metronidazole is a commonly used antibiotic, belonging to the nitroimidazole class of antibiotics.[L3754] It is frequently used to treat gastrointestinal infections as well as trichomoniasis and giardiasis, and amebiasis which are parasitic infections.[A18103…

Kategori:
Agents that reduce seizure thresholdAlimentary Tract and MetabolismAnti-Bacterial Agents +38
Target Protein:
Oxygen-insensitive NADPH nitroreductaseAnaerobic bacterial DNAProtozoal DNA
Waktu ParuhThe elimination hal…
Vol. DistribusiMetronidazole is wi…
KlirensDose adjustments ma…
Genetik -
small molecule | CAS: 13182-89-3

Deskripsi belum tersedia.

Kategori:
ImidazolesNitro CompoundsNitroimidazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metyrapone Approved DB01011
small molecule | CAS: 54-36-4

An inhibitor of the enzyme steroid 11-beta-monooxygenase. It is used as a test of the feedback hypothalamic-pituitary mechanism in the diagnosis of cushing syndrome.

Kategori:
Cytochrome P-450 CYP2A6 InhibitorsCytochrome P-450 CYP2A6 Inhibitors (strength unknown)Cytochrome P-450 CYP2E1 Inhibitors +17
Target Protein:
Cytochrome P450 11B1, mitochondrialCamphor 5-monooxygenase
Waktu Paruh1.9 ±0.7 hou…
Vol. Distribusi-
Klirens-
Genetik -
Metyrosine Approved DB00765
small molecule | CAS: 672-87-7

An inhibitor of the enzyme tyrosine 3-monooxygenase, and consequently of the synthesis of catecholamines. It is used to control the symptoms of excessive sympathetic stimulation in patients with pheochromocytoma. (Martindale, The Extra Pharmacopoeia, 30th ed)

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +6
Target Protein:
Tyrosine 3-monooxygenase
Waktu Paruh3.4 to 3.7 hours
Vol. Distribusi-
Klirens-
Genetik -
Mevalonic acid DB03518
small molecule | CAS: 150-97-0

Deskripsi belum tersedia.

Kategori:
Hydroxy Acids
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevastatin DB06693
small molecule | CAS: 73573-88-3

Mevastatin or compactin is a cholesterol-lowering agent isolated from <i>Penicillium citinium</i>. It was the first discovered agent belonging to the class of cholesterol-lowering medications known as statins. During a search for antibiotic compounds produced…

Kategori:
Agents Causing Muscle ToxicityAnti-Infective AgentsAnticholesteremic Agents +7
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevidalen DB19034
small molecule | CAS: 1638667-79-4

Mevidalen is under investigation in clinical trial NCT03305809 (A Study of LY3154207 in Participants With Dementia Due to Lewy Body Dementia (LBD) Associated With Idiopathic Parkinson's Disease (PD) or Dementia With Lewy Bodies (DLB)).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75225-51-3

Deskripsi belum tersedia.

Kategori:
Naphthalenes
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevonlerbart DB19416
biotech | CAS: 2453195-99-6

Mevonlerbart is under investigation in clinical trial NCT06602726 (A Study to Demonstrate How Well REGN1908-1909 Works in Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Cat Allergy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mexazolam DB15489
small molecule | CAS: 31868-18-5

Mexazolam (CS-386) is a benzodiazepine indicated for the treatment of anxiety with or without psychoneurotic conditions.[A184910] Mexazolam's structure is similar to that of other benzodiazepines such as [oxazolam] and [cloxazolam].[A184910] The use of benzod…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +7
Target Protein:
GABA(A) Receptor Benzodiazepine Binding SiteGABA(A) Receptor
Waktu ParuhMexazolam follows a…
Vol. Distribusi-
Klirens-
Genetik -
Mezagitamab DB16370
biotech | CAS: 2227490-52-8

Mezagitamab is under investigation in clinical trial NCT04278924 (Study to Evaluate Safety, Tolerability, and Efficacy of TAK-079 in Participants With Persistent/chronic Primary Immune Thrombocytopenia).

Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mezigdomide DB17584
small molecule | CAS: 2259648-80-9

Mezigdomide is under investigation in clinical trial NCT05372354 (A Study to Evaluate Safety, Drug Levels and Effectiveness of CC-92480 (BMS-986348) in Combination With Other Treatments in Participants With Relapsed or Refractory Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mezlocillin Approved DB00948
small molecule | CAS: 51481-65-3

Semisynthetic ampicillin-derived acylureido penicillin. It has been proposed for infections with certain anaerobes and may be useful in inner ear, bile, and CNS infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1APeptidoglycan synthase FtsIPenicillin-binding protein 3 +1
Waktu Paruh1.3 to 4.4 hours
Vol. Distribusi-
Klirens-
Genetik -
MF101 DB05052
small molecule

MF101 is a novel estrogen receptor beta (ER?) selective agonist and unlike currently available hormone therapies, does not activate the estrogen receptor alpha (ER?), known to be implicated in tumor formation. MF101 is an oral drug designed for the treatment …

Target Protein:
Estrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 7901–7950 dari 12560
Sebelumnya Halaman 159 / 252 Berikutnya