Hasil Filter

15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (15718)

Halaman 158 / 315
Iberdomide DB12101
small molecule | CAS: 1323403-33-3

Iberdomide (CC-220) has been used in trials studying the treatment of Systemic Lupus Erythematosus.

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingImides +4
Target Protein:
Protein cereblon
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ibezapolstat DB16189
small molecule | CAS: 1275582-97-2

Ibezapolstat is under investigation in clinical trial NCT04247542 (ACX-362E [Ibezapolstat] for Oral Treatment of Clostridioides Difficile Infection).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingNucleic Acid Synthesis Inhibitors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IBIO-100 DB18233
biotech

IBIO-100 is a high molecular weight multimer of E3-Fc, an endostatin C-terminus and IgG1-Fc fusion protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ibipinabant DB12649
small molecule | CAS: 464213-10-3

Ibipinabant has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.

Kategori:
Agents producing tachycardiaAmidesCannabinoid Receptor Antagonists +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iboctadekin DB14920
biotech | CAS: 479198-61-3

Iboctadekin is under investigation in clinical trial NCT00500058 (A Phase I, Dose-Escalation Study to Assess the Safety and Biological Activity of Recombinant Human Interleukin-18).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ibodutant DB12042
small molecule | CAS: 522664-63-7

Ibodutant has been used in trials studying the treatment of Irritable Bowel Syndrome and Irritable Bowel Syndrome With Diarrhea.

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides +2
Target Protein:
Substance-K receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ibopamine DB13316
small molecule | CAS: 66195-31-1

Deskripsi belum tersedia.

Kategori:
Adrenergic and Dopaminergic AgentsAgents that produce hypertensionAmines +25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IBP-1118 DB18461
biotech | CAS: 2483-17-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ibrexafungerp Approved DB12471
small molecule | CAS: 1207753-03-4

Ibrexafungerp, also known as SCY-078 or MK-3118, is a novel enfumafungin derivative oral triterpene antifungal approved for the treatment of vulvovaginal candidiasis (VVC), also known as a vaginal yeast infection.[A235384,L34349] It was developed out of a nee…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiinfectives for Systemic Use +17
Target Protein:
1,3-beta-glucan synthase component GSC2GTP-binding protein RHO1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensClearance values of…
Genetik -
Ibritumomab tiuxetan Approved DB00078
biotech | CAS: 206181-63-7

Indium or yttrium conjugated murine IgG1 kappa monoclonal antibody directed against the CD20 antigen, which is found on the surface of normal and malignant B lymphocytes. Ibritumomab is produced in Chinese hamster ovary cells and is composed of two murine gam…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
B-lymphocyte antigen CD20
Waktu Paruh0.8 hours (mammalia…
Vol. DistribusiBinding observed on…
KlirensApproximately 7.2% …
Genetik -
Ibrutinib Approved DB09053
small molecule | CAS: 936563-96-1

Ibrutinib is a small molecule that acts as an irreversible potent inhibitor of Burton's tyrosine kinase. It is designated as a targeted covalent drug and presented as a promising activity in B-cell malignancies in clinical trials.[A32299] Ibrutinib was develo…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +15
Target Protein:
Tyrosine-protein kinase BTK
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensIn patients with no…
Genetik -
Ibudilast DB05266
small molecule | CAS: 50847-11-5

Ibudilast is an anti-inflammatory and neuroprotective oral agent which shows an excellent safety profile at 60 mg/day and provides significantly prolonged time-to-first relapse and attenuated brain volume shrinkage in patients with relapsing-remitting (RR) an…

Kategori:
Anti-Asthmatic AgentsAntiplatelet agentsAutonomic Agents +12
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4C +2
Waktu Paruh19 hours
Vol. Distribusi-
Klirens-
Genetik -
Ibuprofen Approved DB01050
small molecule | CAS: 15687-27-1

Ibuprofen is a non-steroidal anti-inflammatory drug (NSAID) derived from propionic acid and it is considered the first of the propionics.[A39074] The formula of ibuprofen is 2-(4-isobutylphenyl) propionic acid and its initial development was in 1960 while res…

Kategori:
Acids, CarbocyclicAgents causing angioedemaAgents causing hyperkalemia +47
Target Protein:
Prostaglandin G/H synthase 2C-X-C chemokine receptor type 2Interleukin-8 +10
Waktu ParuhThe serum half-life…
Vol. DistribusiThe apparent volume…
KlirensThe clearance rate …
Genetik -
small molecule | CAS: 64622-45-3

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicPhenylpropionates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ibutamoren DB18214
small molecule | CAS: 159634-47-6

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Growth hormone secretagogue receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ibutilide Approved DB00308
small molecule | CAS: 122647-31-8

Ibutilide is a Class III antiarrhythmic agent available in intravenous formulations. It is indicated for the conversion of acute atrial flutter and recent onset atrial fibrillation to normal sinus rhythm (NSR).

Kategori:
AmidesAntiarrhythmic agentsAntiarrhythmics, Class III +7
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit beta-1Voltage-gated inwardly rectifying potassium channel KCNH2 +7
Waktu Paruh6 hours (ranges fro…
Vol. Distribusi* 11 L/kg
Klirens* 29 mL/min/kg
Genetik -
Ibuzatrelvir DB19451
small molecule | CAS: 2755812-39-4

Ibuzatrelvir is under investigation in clinical trial NCT06679140 (A Study to Learn About a Study Medicine Called Ibuzatrelvir in Adult and Adolescent Patients With COVID-19 Who Are Not Hospitalized but Are at Risk for Severe Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IC261 DB03083
small molecule

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesHeterocyclic Compounds, Fused-RingPhenols
Target Protein:
Casein kinase I isoform alphaCasein kinase I isoform epsilonCasein kinase I isoform gamma-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IC41 DB05776
biotech

IC41 is a therapeutic peptide vaccine. It is being devloped by Intercell AG for the treatment of hepatitis C. The vaccine consists of five synthetic peptides (IPEP83, 84, 87, 89,1426) harboring HCV CD4 and CD8 T-cell epitopes and the synthetic adjuvant poly-L…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ICA-105665 DB06089
small molecule

ICA-105665 is a novel small molecule compound for the treatment of epilepsy. It is a novel opener of the KCNQ ion channel which in preclinical studies has demonstrated a broad spectrum of activity in models of epilepsy. In addition, ICA-105665 has also demon…

Target Protein:
Potassium voltage-gated channel subfamily KQT member 1Potassium voltage-gated channel subfamily KQT member 3Potassium voltage-gated channel subfamily KQT member 4 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icapamespib DB18106
small molecule | CAS: 1000999-96-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icaridin DB14074
small molecule | CAS: 119515-38-7

Icaridin, also known as Picaridin or hydroxy-ethyl isobutyl piperidine carboxylate, is a cyclic amine and a member of the piperidine chemical family. Piperidines are structural components of [piperine], which is a plant extract from the genus _Piper _, or pep…

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsect Repellents +4
Target Protein:
Odorant binding protein
Waktu ParuhThe first eliminati…
Vol. DistribusiIn a rat study, der…
KlirensThere is no availab…
Genetik -
Icariin DB12052
small molecule | CAS: 489-32-7

Icariin has been investigated for the basic science of the Pharmacokinetic Profile of Icariin in Humans.

Kategori:
BenzopyransChromonesDrugs, Chinese Herbal +3
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icaritin DB12672
small molecule | CAS: 118525-40-9

Icaritin has been used in trials studying the treatment of Solid Tumors, Metastatic Breast Cancer, and Hepatocellular Carcinoma (HCC).

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icatibant Approved DB06196
biotech | CAS: 130308-48-4

Icatibant is a synthetic decapeptide with 5 nonproteinogenic amino acid antagonist targeting the B<sub>2</sub> receptors with a similar affinity to bradykinin. It is resistant to bradykinin-cleaving enzyme degradation and has a potency of 2-3 times higher tha…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnalgesics +21
Target Protein:
B2 bradykinin receptorAminopeptidase N
Waktu ParuhFollowing subcutane…
Vol. DistribusiFollowing subcutane…
KlirensFollowing subcutane…
Genetik -
Icerguastat DB16932
small molecule | CAS: 951441-04-6

Deskripsi belum tersedia.

Kategori:
AmidinesGuanidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ICG-001 DB18024
small molecule | CAS: 780757-88-2

Deskripsi belum tersedia.

Kategori:
Pyrimidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ICG-136 DB17343
biotech

ICG-136 is a compound chimeric antigen receptor (cCAR) T-cell therapy developed by iCell Gene Therapeutics. It was investigated for the treatment of acute myeloid leukemia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ICG-140 DB17344
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ichorcumab DB18930
biotech | CAS: 2589583-20-8

Ichorcumab is under investigation in clinical trial NCT03251482 (A Study to Evaluate the Safety and Efficacy of Intravenous JNJ-64179375 Versus Oral Apixaban in Participants Undergoing Elective Total Knee Replacement Surgery).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ichthammol Approved DB11341
small molecule | CAS: 8029-68-3

Ichthammol is also referred to as ammonium bituminosulfonate or ammonium bituminosulphonate. It is an ammonium salt of dark sulfonated shale oil (bituminous schists) produced via distillation of the oil followed by sulfonation and neutralization. It is availa…

Kategori:
AminesAmmonium CompoundsDermatologicals +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ICI-164384 DB03860
small molecule | CAS: 98007-99-9

Deskripsi belum tersedia.

Kategori:
AlkenesAlkynesAmides +12
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iclaprim DB06358
small molecule | CAS: 192314-93-5

Deskripsi belum tersedia.

Kategori:
Antibacterials for Systemic UseAntiinfectives for Systemic UseEnzyme Inhibitors +3
Target Protein:
Dihydrofolate reductaseDihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iclepertin DB19058
small molecule | CAS: 1421936-85-7

Iclepertin is under investigation in clinical trial NCT05211947 (A Study to Test Long-term Safety of Iclepertin in People With Schizophrenia Who Took Part in a Previous CONNEX Study).

Target Protein:
Sodium- and chloride-dependent glycine transporter 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
iCo-007 DB05268
small molecule

iCo-007 (formerly known as ISIS 13650) is a second generation antisense compound being developed by iCo for the treatment of various eye diseases caused by the formation of new blood vessels (angiogenesis) such as age-related macular degeneration (AMD) and di…

Target Protein:
RAF proto-oncogene serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icodextrin Approved DB00702
small molecule | CAS: 337376-15-5

Icodextrin is an iso-osmotic peritoneal dialysis solution containing glucose polymers. It is used primarily for ambulatory peritoneal dialysis (CAPD) of diabetic patients and automated peritoneal dialysis (APD) for patients with end-stage renal disease. It is…

Kategori:
BiopolymersCarbohydratesCompounds used in a research, industrial, or household setting +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icosabutate DB12990
small molecule | CAS: 1253909-57-7

Icosabutate is under investigation in clinical trial NCT02373176 ([14C] Icosabutate -A Phase I Absorption, Metabolism and Excretion Study).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icosapent Approved DB00159
small molecule | CAS: 10417-94-4

Important polyunsaturated fatty acid found in fish oils. It serves as the precursor for the prostaglandin-3 and thromboxane-3 families. A diet rich in eicosapentaenoic acid lowers serum lipid concentration, reduces incidence of cardiovascular disorders, preve…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +17
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Peroxisome proliferator-activated receptor gamma +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icosapent ethyl Approved DB08887
small molecule | CAS: 86227-47-6

Icosapent ethyl or ethyl eicosapentaenoic acid is a synthetic derivative of the omega-3 fatty acid eicosapentaenoic acid (EPA). It is used as an adjunct therapy for severe hypertriglyceridemia (TG levels > 500 mg/dL) and to reduce the risk of cardiovascular e…

Kategori:
Antiplatelet agentsDietary FatsDietary Fats, Unsaturated +12
Waktu ParuhThe half life of EP…
Vol. DistribusiSteady state volume…
KlirensTotal plasma cleara…
Genetik -
Icotinib DB11737
small molecule | CAS: 610798-31-7

Icotinib is a potent and specific epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI) Icotinib was approved in China by the SFDA in June, 2011 and in January 2014, Beta Pharma, Inc. was given a “May Proceed” from the US FDA to conduct a P…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCrown Compounds +16
Target Protein:
Epidermal growth factor receptor
Waktu Paruh5.5 hrs
Vol. Distribusithe volume of distr…
Klirensthe clearance was c…
Genetik -
Icrucumab DB14824
biotech | CAS: 1024603-92-6

Icrucumab is under investigation in clinical trial NCT01111604 (A Study of IMC-1121B or IMC-18F1 in Colorectal Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ICX-RHY DB05716
biotech

ICX-RHY is an investigational therapy comprised of cultured allogeneic fibroblasts. The drug was under investigation in clinical trials in the UK for the treatment of skin erosions in recessive dystrophic epidermolysis bulllosa.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idalopirdine DB11957
small molecule | CAS: 467459-31-0

Idalopirdine has been used in trials studying the treatment of Cognition, Schizophrenia, and Alzheimer's Disease.

Kategori:
AminesAntidepressive AgentsBenzene Derivatives +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idanpramine DB13276
small molecule | CAS: 25466-44-8

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal Disorders
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idarubicin Approved DB01177
small molecule | CAS: 58957-92-9

An orally administered anthracycline antineoplastic. The compound has shown activity against breast cancer, lymphomas and leukemias, together with the potential for reduced cardiac toxicity.

Kategori:
Anthracycline Topoisomerase InhibitorAnthracyclinesAnthracyclines and Related Substances +19
Target Protein:
DNA topoisomerase 2-betaDNADNA topoisomerase 2-alpha
Waktu Paruh22 hours
Vol. Distribusi-
Klirens-
Genetik -
Idarucizumab Approved DB09264
biotech | CAS: 1362509-93-0

Idarucizumab is a humanized monoclonal antibody fragment (Fab) derived from an immunoglobulin G1 isotype molecule that binds to and inactivates the oral anticoagulant dabigatran, thereby reversing its anticoagulant effect. As a direct acting oral anticoagulan…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Waktu Paruhinitial half-life: …
Vol. Distribusi8.9 L
Klirens47.0 mL/min
Genetik -
Idasanutlin DB12325
small molecule | CAS: 1229705-06-9

Idasanutlin has been used in trials studying the treatment of Neoplasms, Non-Hodgkin's Lymphoma, Leukemia, Myeloid, Acute, Recurrent Plasma Cell Myeloma, and Neoplasms, Leukemia, Acute Myeloid Leukemia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +2
Target Protein:
E3 ubiquitin-protein ligase Mdm2Receptor tyrosine-protein kinase erbB-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idazoxan DB12551
small molecule | CAS: 79944-58-4

Idazoxan has been used in trials studying the basic science of Molecular Imaging, Alzheimer Disease, and Major Depressive Disorder.

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDD-1 DB05439
biotech

Lipids promote the fusion of liposomes to cells. Eladem (IDD-1) is a therapeutic vaccine consisting of dendritophages that are loaded in vitro with tumor antigens and then reinjected into the subject. As with other monoclonal antibodies, this process stimulat…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idebenone Approved DB09081
small molecule | CAS: 58186-27-9

Idebenone is a synthetic analogue of ubiquinone (also known as Coenzyme Q10), a vital cell antioxidant and essential component of the Electron Transport Chain (ETC). It has been proposed that by interacting with the ETC, idebenone increases ATP production req…

Kategori:
AntioxidantsBenzoquinonesBiological Factors +9
Waktu Paruh-
Vol. DistribusiExperimental data h…
Klirens-
Genetik -
Menampilkan 7851–7900 dari 15718
Sebelumnya Halaman 158 / 315 Berikutnya