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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
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17430 (100.0%)

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Halaman 156 / 349
Fezakinumab DB12344
biotech | CAS: 1007106-86-6

Fezakinumab has been used in trials studying the treatment of Atopic Dermatitis and Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fezolinetant Approved DB15669
small molecule | CAS: 1629229-37-3

Vasomotor symptoms (VMS), more colloquially known as hot flashes or night sweats, are some of the most common symptoms in menopause. With a median duration of 7.4 years, vasomotor symptoms are also the most common reasons why women seek treatments for menopau…

Kategori:
Cytochrome P-450 CYP1A2 SubstratesCytochrome P-450 CYP2C19 SubstratesCytochrome P-450 CYP2C9 Substrates +6
Target Protein:
Neuromedin-K receptor
Waktu ParuhThe effective half-…
Vol. DistribusiThe mean apparent v…
KlirensThe apparent cleara…
Genetik -
FF-10101-01 DB16050
small molecule | CAS: 1472797-69-5

FF-10101-01 is under investigation in clinical trial NCT03194685 (Study of FF-10101-01 in Patients With Relapsed or Refractory Acute Myeloid Leukemia).

Kategori:
Enzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FF-10501-01 DB17554
small molecule

FF-10501-01 is a novel, selective inosine monophosphate dehydrogenase (IMPDH) inhibitor with anticancer activity.[A257306] FF-10501-01 is under investigation in clinical trial NCT03486353 (A Study of FF-10501-01 in Combination With Azacitidine in Patients Wit…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
FG-2216 DB08687
small molecule | CAS: 223387-75-5

A orally active prolyl-hydroxylase inhibitor which can stabilize hypoxia-inducible transcription factor independent of oxygen availability. [A14422]

Target Protein:
Egl nine homolog 1Hypoxia-inducible factor 1-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FG-9041 DB03759
small molecule | CAS: 2379-57-9

Deskripsi belum tersedia.

Kategori:
Excitatory Amino Acid AgentsExcitatory Amino Acid AntagonistsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Glutamate receptor 1Glutamate receptor ionotropic, kainate 1Glutamate receptor ionotropic, NMDA 2B +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fiacitabine DB12901
small molecule | CAS: 69123-90-6

Fiacitabine has been used in trials studying the treatment of HIV Infections and Cytomegalovirus Infections.

Kategori:
Anti-Infective AgentsAntineoplastic AgentsAntiviral Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fialuridine DB15427
small molecule | CAS: 69123-98-4

Fialuridine is under investigation in clinical trial NCT01337466 (Biodistribution and Dosimetry Evaluation of [124I]FIAU).

Kategori:
Anti-Infective AgentsAntiviral AgentsArabinonucleosides +7
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fianlimab DB18858
biotech | CAS: 2126132-98-5

Fianlimab is under investigation in clinical trial NCT06190951 (A Trial to Learn if Fianlimab and Cemiplimab Are Safe and Work Better Than Anti-pd1 Alone in Adult Participants With Resectable Stage 3 or 4 Melanoma).

Waktu Paruh-
Vol. Distribusi-
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Fiboflapon DB06346
small molecule | CAS: 936350-00-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAsthma, drug therapyFatty Acids +4
Target Protein:
Arachidonate 5-lipoxygenase-activating protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fibrin DB16604
biotech | CAS: 9001-31-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsFibrin +1
Waktu Paruh-
Vol. Distribusi-
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Fibrinogen human Approved DB09222
biotech | CAS: 9001-32-5

Fibrinogen concentrate (human) is a hematological agent. It works by replacing a specific protein in the blood, fibrinogen (factor I), that helps with blood clotting. It is a soluble plasma glycoprotein with a molecular weight of about 340 kDa and is a physi…

Kategori:
Acute-Phase ProteinsAmino Acids, Peptides, and ProteinsBiological Factors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fibrinolysin DB05254
biotech | CAS: 9004-09-5

Fibrinolysin consists of two polypeptide chains, one light and one heavy, linked by a disulfide bond. The light chain has a molecular weight of approximately 27,000 Da and contains the active center of Fibrinolysin; the heavy chain has a molecular weight of a…

Kategori:
AnticoagulantsBlood and Blood Forming OrgansCardiovascular Agents +11
Target Protein:
Plasminogen activator inhibitor 1Urokinase-type plasminogen activator
Waktu ParuhAlmost completely i…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 106096-92-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsFibroblast Growth Factor 1 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fibronectin DB15150
biotech

Fibronectin is under investigation in clinical trial NCT01812239 (Vaginal Progesterone in Twins With Short Cervix).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsCarbohydrates +9
Waktu Paruh-
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Genetik -
Fica DB03384
small molecule

Deskripsi belum tersedia.

Target Protein:
Caspase-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ficlatuzumab DB11680
biotech | CAS: 1174900-84-5

Ficlatuzumab has been used in trials studying the treatment of Acute Myeloid Leukemia, Non-small Cell Lung Cancer, Mullerian Mixed Tumor of Ovary, Relapsed Acute Myeloid Leukemia, and Refractory Acute Myeloid Leukemia, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ficonalkib DB18774
small molecule | CAS: 2233574-95-1

Deskripsi belum tersedia.

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Fidanacogene elaparvovec Approved DB16783
biotech | CAS: 1954659-47-2

Fidanacogene elaparvovec is a liver-specific adeno-associated virus (AAV) vector containing a codon-optimized human coagulation FIX gene that was investigated as a potential treatment for hemophilia B.[L46691] Hemophilia B is a rare X-linked genetic disorder …

Kategori:
Adeno-associated Viral Vector TherapiesHepatotoxic Agents
Target Protein:
Coagulation factor IX (F9)
Waktu Paruh-
Vol. DistribusiIn a monkey biodist…
KlirensClearance of vector…
Genetik -
Fidarestat DB02021
small molecule | CAS: 136087-85-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsImidazoles
Target Protein:
Aldo-keto reductase family 1 member B1Aldo-keto reductase family 1 member B10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fidaxomicin Approved DB08874
small molecule | CAS: 873857-62-6

Fidaxomicin is a novel macrolide antibiotic used in the treatment of diarrhea caused by _Clostridioides_ (formerly _Clostridium_) _difficile_ in adult and pediatric patients over the age of 6 months.[L11575] Fidaxomicin is a naturally-occurring 18-member macr…

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
RNA polymerase sigma factor SigA
Waktu ParuhFollowing oral admi…
Vol. DistribusiFidaxomicin is main…
KlirensThere is limited in…
Genetik -
Fidrisertib DB18064
small molecule | CAS: 2141955-96-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Field mushroom Approved DB15605
biotech

Field mushroom allergenic extract is used in allergenic testing.

Waktu Paruh-
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Fig Approved DB10633
biotech

Fig allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Figitumumab DB11685
biotech | CAS: 943453-46-1

Figitumumab has been used in trials studying the treatment of Sarcoma, Solid Tumor, Breast Cancer, Lung Neoplasms, and Advanced Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Figopitant DB12122
small molecule | CAS: 502422-74-4

Figopitant is under investigation in clinical trial NCT02209714 (Safety, Tolerability and Pharmacodynamics After Oral Administration of BIIF 1149 BS in Healthy Male Volunteers).

Kategori:
AcetamidesAmidesBenzene Derivatives
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Filaminast DB02660
small molecule | CAS: 141184-34-1

Filaminast is a phosphodiesterase 4 inhibitor (PDE4 inhibitor). As such, has potential in the treatment of asthma and chronic obstructive pulmonary disease (COPD).

Kategori:
AminesHydroxylamines
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Filanesib DB06040
small molecule | CAS: 885060-09-3

Filanesib is a potent Kinesin Spindle Protein (KSP) inhibitor that caused marked tumor regression in preclinical models of human solid tumors and human leukemias, often leading to durable responses.

Kategori:
Antimitotic AgentsAntineoplastic AgentsMitosis Modulators +2
Target Protein:
Kinesin-like protein KIF11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Filgotinib Approved DB14845
small molecule | CAS: 1206161-97-8

Rheumatoid arthritis (RA) is a chronic, autoimmune, systemic, and inflammatory disease that causes synovial joint symptoms and can limit range of motion in severe cases.[A221451,A221456] The disease is associated with extra-articular manifestations, progressi…

Kategori:
Antineoplastic and Immunomodulating AgentsArthritis, Rheumatoid, drug therapyImmunosuppressive Agents +5
Target Protein:
Tyrosine-protein kinase JAK1
Waktu ParuhThe half-life of fi…
Vol. Distribusi-
Klirens-
Genetik -
Filgrastim Approved DB00099
biotech | CAS: 121181-53-1

Filgrastim is a short-acting recombinant, non-pegylated human granulocyte colony-stimulating factor (G-CSF) analog produced by recombinant DNA technology. It has an amino acid sequence identical to endogenous G-CSF, but it is non-glycosylated unlike the endog…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsBiological Factors +10
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhAfter intravenous a…
Vol. DistribusiAfter intravenous a…
KlirensClearance rates of …
Genetik -
Filibuvir DB11878
small molecule | CAS: 877130-28-4

Filibuvir has been used in trials studying the treatment of Hepatitis, Hepatitis C, and Chronic Hepatitis C.

Kategori:
PyransRNA Replicase, antagonists & inhibitorsRNA-Dependent RNA Polymerase, antagonists & inhibitors
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
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Filociclovir DB12438
small molecule | CAS: 632325-71-4

Filociclovir is under investigation in clinical trial NCT01433835 (Safety and Pharmacokinetics of Single Oral Doses of Filociclovir in Healthy Volunteers).

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Filorexant DB12158
small molecule | CAS: 1088991-73-4

Filorexant has been used in trials studying the prevention and treatment of Migraine, Headache, Polysomnography, Diabetic Neuropathy, Painful, and Major Depressive Disorder, Recurrent.

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Genetik -
Fimaporfin DB17253
small molecule | CAS: 1443547-43-0

Deskripsi belum tersedia.

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Fimasartan DB09279
small molecule | CAS: 247257-48-3

Fimasartan is an angiotensin II receptor antagonist (ARB) drug employed in the treatment of both hypertension and heart failure. It has been found to be safe when administered with hydrochlorothiazide (a diuretic) in clinical trials. Fimasartan was initially …

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin II receptor blockers (ARBs) and calcium channel blockers +8
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhThe half life of el…
Vol. Distribusi-
Klirens-
Genetik -
Fimepinostat DB11891
small molecule | CAS: 1339928-25-4

Fimepinostat (CUDC-907) has been used in trials studying the treatment of lymphoma, solid tumors, breast cancer, multiple myeloma, and NUT midline carcinoma, among others.

Kategori:
Antineoplastic AgentsHistone Deacetylase InhibitorsOxazines +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Finafloxacin Approved DB09047
small molecule | CAS: 209342-40-5

Finafloxacin is a fluoroquinolone antibiotic indicated in the treatment of acute otitis externa (swimmer's ear) caused by the bacteria Pseudomonas aeruginosa and Staphylococcus aureus. Finafloxacin is marketed by Novartis under the brand Xtoro™, and was appro…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Finasteride Approved DB01216
small molecule | CAS: 98319-26-7

Finasteride is a synthetic 4-azasteroid compound [L10565] and specific inhibitor of steroid Type II 5?-reductase, which is an intracellular enzyme that converts the androgen testosterone into 5?-dihydrotestosterone (DHT). It works in a similar fashion as [dut…

Kategori:
5-alpha Reductase InhibitorsAdrenergic alpha-AntagonistsAdrenergic Antagonists +22
Target Protein:
3-oxo-5-alpha-steroid 4-dehydrogenase 2Polyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 1 +1
Waktu ParuhIn healthy young su…
Vol. DistribusiThe volume of distr…
KlirensIn healthy young su…
Genetik -
Finerenone Approved DB16165
small molecule | CAS: 1050477-31-0

Finerenone, or BAY 94-8862, is a mineralocorticoid receptor antagonist indicated to reduce the risk of sustained decline in glomerular filtration rate, end stage kidney disease, cardiovascular death, heart attacks, and hospitalization due to heart failure in …

Kategori:
Agents causing hyperkalemiaCytochrome P-450 CYP2C8 SubstratesCytochrome P-450 CYP3A Substrates +6
Target Protein:
Mineralocorticoid receptor
Waktu ParuhThe half life of a …
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
Fingolimod Approved DB08868
small molecule | CAS: 162359-55-9

Multiple sclerosis, or MS, is a devastating inflammatory disease that often progresses and causes severe neurological, physical, and cognitive effects.[A176474] Fingolimod is a sphingosine 1-phosphate receptor modulator for the treatment of relapsing-remittin…

Kategori:
AlcoholsAminesAmino Alcohols +16
Target Protein:
D(3) dopamine receptorSphingosine kinase 1Sphingosine 1-phosphate receptor 5 +4
Waktu ParuhThe half-life of fi…
Vol. DistribusiThe volume of distr…
KlirensFingolimod blood cl…
Genetik -
FINLAY-FR-1 DB16524
biotech

FINLAY-FR-1, also known as Soberana 01, is a vaccine candidate for COVID-19 that is being led developmentally by the Finlay Vaccine Institute[L31373]. It is currently being tested in the clinical trial RPCEC00000332 (Phase I / II, randomized, controlled, adap…

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Finotonlimab DB18859
biotech | CAS: 2350298-85-8

Finotonlimab is under investigation in clinical trial NCT04560894 (SCT-I10A Plus SCT510 Versus Sorafenib as First-line Therapy for Advanced Hepatocellular Carcinoma).

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Fipamezole DB06585
small molecule | CAS: 150586-58-6

Deskripsi belum tersedia.

Kategori:
Indenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fipaxalparant DB18124
small molecule | CAS: 1195941-38-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysophosphatidic acid receptor 1Lysophosphatidic acid receptor 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fipexide DB13790
small molecule | CAS: 34161-24-5

Deskripsi belum tersedia.

Kategori:
Nervous SystemPsychoanalepticsPsychostimulants, Agents Used for ADHD and Nootropics
Waktu Paruh-
Vol. Distribusi-
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Firategrast DB12732
small molecule | CAS: 402567-16-2

Firategrast has been used in trials studying the treatment of Multiple Sclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Firazorexton DB19440
small molecule | CAS: 2274802-95-6

Firazorexton is under investigation in clinical trial NCT04096560 (A Study of TAK-994 in Adults With Type 1 and Type 2 Narcolepsy).

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Firocoxib DB09217
small molecule | CAS: 189954-96-9

Firocoxib is a cycooxygenase-2 (COX-2) selective non-steroidal anti-inflammatory drug. It currently approved for veterinary use in dogs and horses under the brand names Equioxx and Previcox. Firocoxib was the first COX-2 inhibitor approved by the U.S. Food an…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +6
Target Protein:
Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Firsocostat DB16166
small molecule | CAS: 1434635-54-7

Firsocostat is under investigation in clinical trial NCT02781584 (Safety, Tolerability, and Efficacy of Selonsertib, Firsocostat, and Cilofexor in Adults With Nonalcoholic Steatohepatitis (NASH)).

Kategori:
Acids, AcyclicButyratesEnzyme Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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