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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 156 / 252
MEM 1003 DB05547
small molecule

MEM 10003 was under investigation in clinical trial NCT00257673 (Safety and Efficacy of MEM 1003 Versus Placebo in Patients With Mild to Moderate Alzheimer's Disease) for the treatment of Alzheimer's Disease.

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MEM 1414 DB05888
small molecule

MEM 1414 is a PDE4 inhibitor that is being evaluated for the treatment of Alzheimer’s disease. This drug candidate has completed Phase 1 clinical trials. MEM 1414 works by blocking phosphodiesterase, an enzyme that breaks down an important brain chemical, cyc…

Target Protein:
CAMP phosphodiesterase
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Memantine Approved DB01043
small molecule | CAS: 19982-08-2

Initially approved by the FDA in 2013, memantine is an N-methyl-D-aspartate (NMDA) receptor antagonist used in the management of Alzheimer's Disease (AD). It is different from many other Alzheimer's Disease medications, as it works by a different mechanism t…

Kategori:
Anti-Dementia DrugsAnti-Dyskinesia AgentsAnti-Parkinson Drugs +20
Target Protein:
Glutamate (NMDA) receptor5-hydroxytryptamine receptor 3ANeuronal acetylcholine receptor subunit alpha-7 +3
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThis drug is cleare…
Genetik -
Menadiol diphosphate Approved DB14650
small molecule | CAS: 84-98-0

Deskripsi belum tersedia.

Kategori:
DiterpenesNaphthalenesNaphthoquinones +2
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Menadione Approved DB00170
small molecule | CAS: 58-27-5

A synthetic naphthoquinone without the isoprenoid side chain and biological activity, but can be converted to active vitamin K2, menaquinone, after alkylation in vivo.

Kategori:
Antifibrinolytic AgentsBlood and Blood Forming OrgansCoagulants +45
Target Protein:
Aldehyde oxidaseVitamin K-dependent gamma-carboxylaseVitamin K epoxide reductase complex subunit 1 +8
Waktu Paruh-
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Genetik -
small molecule | CAS: 130-36-9

Deskripsi belum tersedia.

Kategori:
Antifibrinolytic AgentsCoagulantsDiet, Food, and Nutrition +15
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Menaquinone DB15381
small molecule | CAS: 1182-68-9

Menaquinone is under investigation in clinical trial NCT01533441 (Vitamin K2 Intervention in Patients With Vitamin K Antagonists).

Kategori:
CoagulantsDiet, Food, and NutritionDiterpenes +15
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Menaquinone 7 DB13075
small molecule | CAS: 2124-57-4

Menaquinone 7 is under investigation in clinical trial NCT00402974 (The Effect of Vitamin K Supplementation on Osteocalcin Carboxylation in Healthy Children).

Kategori:
CoagulantsDiterpenesHematologic Agents +9
Waktu Paruh-
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Menglytate DB15983
small molecule | CAS: 579-94-2

Deskripsi belum tersedia.

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biotech

Meningococcal (groups A, C, Y and W-135) oligosaccharide diphtheria CRM197 conjugate vaccine is used to prevent invasive meningococcal disease, which is caused by bacteria _Neisseria meningitidis_ entering the bloodstream and invading the blood-brain barrier …

Kategori:
Diphtheria VaccinesMeningococcal VaccinesVaccines
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Genetik -
biotech

Meningococcal group W-135 polysaccharide is group-specific polysaccharide antigens extracted and purified from *Neisseria meningitidis* serogroup W-135. *N. meningitidis* is a bacteria that causes endemic and epidemic diseases including meningitis and meningo…

Kategori:
Actively Acquired ImmunityInactivated Meningococcal Vaccine
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Genetik -
biotech

Deskripsi belum tersedia.

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Menthol Approved DB14123
small molecule | CAS: 1490-04-6

Deskripsi belum tersedia.

Kategori:
AlcoholsAntipruriticsCyclohexane Monoterpenes +9
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menthone DB15920
small molecule | CAS: 89-80-5

Deskripsi belum tersedia.

Kategori:
AlcoholsCyclohexane MonoterpenesCyclohexanes +7
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Mepenzolate Approved DB04843
small molecule | CAS: 25990-43-6

Mepenzolate is a post-ganglionic parasympathetic inhibitor. It decreases gastric acid and pepsin secretion and suppresses spontaneous contractions of the colon. Mepenzolate diminishes gastric acid and pepsin secretion. Mepenzolate also suppresses spontaneous …

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +7
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M3
Waktu Paruh-
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Meperidine Approved DB00454
small molecule | CAS: 57-42-1

A narcotic analgesic that can be used for the relief of most types of moderate to severe pain, including postoperative pain and the pain of labor. Prolonged use may lead to dependence of the morphine type; withdrawal symptoms appear more rapidly than with mor…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents that reduce seizure threshold +34
Target Protein:
Kappa-type opioid receptorGlutamate receptor ionotropic, NMDA 1Glutamate receptor ionotropic, NMDA 2B +9
Waktu ParuhInitial distributio…
Vol. DistribusiMeperidine crosses …
Klirens-
Genetik -
Mephedrone DB13108
small molecule | CAS: 1189805-46-6

Mephedrone has been investigated in Alcohol-Related Disorders and Amphetamine-Related Disorders.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +7
Waktu Paruh-
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Mephenesin Approved DB13583
small molecule | CAS: 59-47-2

Mephenesin is a synthetic cresol glyceryl ether which produces transient muscle relaxation and paralysis via central nervous system depression [A32760]. It first entered use in the 1950s.

Kategori:
AlcoholsCentral Nervous System AgentsCentral Nervous System Depressants +7
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small molecule | CAS: 533-06-2

Deskripsi belum tersedia.

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Mephenoxalone DB13754
small molecule | CAS: 70-07-5

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsCentral Nervous System DepressantsMuscle Relaxants +3
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Mephentermine Approved DB01365
small molecule | CAS: 100-92-5

A sympathomimetic agent with mainly indirect effects on adrenergic receptors. It is used to maintain blood pressure in hypotensive states, for example, following spinal anesthesia. Although the central stimulant effects of mephentermine are much less than tho…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +17
Target Protein:
Alpha adrenergic receptorD(2) dopamine receptorBeta adrenergic receptor
Waktu Paruh17 to 18 hours.
Vol. Distribusi-
Klirens-
Genetik -
Mephenytoin Approved DB00532
small molecule | CAS: 50-12-4

Mephenytoin is used for the treatment of refractory partial epilepsy. Mephenytoin is a solid. This compound belongs to the phenylhydantoins. These are heterocyclic aromatic compounds containing an imiazolidinedione moiety substituted by a phenyl group. Mephen…

Kategori:
Anti-epileptic AgentAnticonvulsantsCentral Nervous System Agents +17
Target Protein:
Sodium channel protein type 5 subunit alphaNuclear receptor subfamily 1 group I member 2
Gen Terkait:
CYP2C19 CYP2C19 CYP2C19
Waktu ParuhApproximately 7 hou…
Vol. Distribusi* 1.4 L/kg
Klirens-
Genetik 3 Varian
Mepindolol DB13530
small molecule | CAS: 23694-81-7

Mepindolol is a 2-methyl derivative of pindolol. It is a beta blocker.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +12
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
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Mepiprazole DB09197
small molecule | CAS: 20326-12-9

Mepiprazole is a minor tranquilizer with a phenylpiperazine structure. It is a pyrazolyl-alkyl-piperazine derivative. Mepiprazole mediates a weak inhibitory action on the uptake of 5-HT on hypothalamic neurons [A7816]. Mepiprazole is marketed in Spain for th…

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Mepixanox DB13579
small molecule | CAS: 17854-59-0

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingRespiratory System AgentsXanthenes
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Meplazumab DB16465
biotech

Meplazumab is a humanized anti-CD147 antibody being investigated as an add-on therapy in patients with COVID-19 pneumonia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
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Mepolizumab Approved DB06612
biotech | CAS: 196078-29-2

Eosinophils are involved in inflammatory immune responses, and prolonged hypereosinophilia (typically defined as absolute eosinophil levels of 1500/mm<sup>3</sup> or more) is associated with a spectrum of diseases, including severe asthma, eosinophilic granul…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Interleukin-5
Waktu ParuhMepolizumab has a m…
Vol. DistribusiMepolizumab has a p…
KlirensMepolizumab has an …
Genetik -
MePPEP C-11 DB19280
small molecule | CAS: 1022083-25-5

Deskripsi belum tersedia.

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Genetik -
small molecule | CAS: 1106-03-2

Deskripsi belum tersedia.

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Meprobamate Approved DB00371
small molecule | CAS: 57-53-4

A carbamate with hypnotic, sedative, and some muscle relaxant properties, although in therapeutic doses reduction of anxiety rather than a direct effect may be responsible for muscle relaxation. Meprobamate has been reported to have anticonvulsant actions aga…

Kategori:
Acids, AcyclicAnti-Anxiety AgentsCarbamates +10
Target Protein:
Peptide deformylase, mitochondrialProtein kinase C epsilon typeGABA(A) Receptor +6
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Meprotixol DB13822
small molecule | CAS: 4295-63-0

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
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Meptazinol DB13478
small molecule | CAS: 54340-58-8

Deskripsi belum tersedia.

Kategori:
AnalgesicsAzepinesCentral Nervous System Agents +10
Target Protein:
Cholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mequinol Approved DB09516
small molecule | CAS: 150-76-5

Mequinol is a phenol used in various applications. It is used as an inhibitor for acrylic monomers and acrylonitirles, as a stabilizer for chlorinated hydrocarbons and ethyl cellulose, as an ultraviolet inhibitor, as a chemical intermediate in the manufacture…

Kategori:
AntioxidantsBenzene DerivativesBiological Factors +11
Waktu ParuhMequinol demonstrat…
Vol. DistribusiThe volume of distr…
KlirensReadily accessible …
Genetik -
Meradimate Approved DB11096
small molecule | CAS: 134-09-8

Meradimate, before known as menthyl anthranilate, is used in a maximal concentration of 5% in different products as a UV filter.[T200] It is currently required to be named as meradimate in all FDA approved OTC products. Meradimate is approved by the FDA and H…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +2
Waktu ParuhAs meradimate is no…
Vol. DistribusiAs meradimate is no…
KlirensAs meradimate is no…
Genetik -
Mercaptoethanol DB03345
small molecule | CAS: 60-24-2

Deskripsi belum tersedia.

Kategori:
AlcoholsSulfhydryl CompoundsSulfur Compounds
Target Protein:
Lactoylglutathione lyaseFibroblast growth factor 2M-phase inducer phosphatase 2 +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mercaptopurine Approved DB01033
small molecule | CAS: 50-44-2

An antimetabolite antineoplastic agent with immunosuppressant properties. It interferes with nucleic acid synthesis by inhibiting purine metabolism and is used, usually in combination with other drugs, in the treatment of or in remission maintenance programs …

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +20
Target Protein:
Hypoxanthine-guanine phosphoribosyltransferaseInosine-5'-monophosphate dehydrogenase 1Amidophosphoribosyltransferase +1
Gen Terkait:
TPMT TPMT TPMT
Waktu ParuhTriphasic: 45 minut…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik 3 Varian
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2Divalent-cation tolerance protein CutA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7487-94-7

Mercury chloride (HgCl2) is a highly toxic compound that volatizes slightly at ordinary temperature and appreciably at 100 degrees C. It is corrosive to mucous membranes and used as a topical antiseptic and disinfectant. Mercuric chloride was used to disinfec…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntiseptics and Disinfectants +7
Waktu Paruh-
Vol. Distribusi-
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Mercuric iodide DB04445
small molecule | CAS: 7774-29-0

Deskripsi belum tersedia.

Kategori:
AnionsAntiseptics and DisinfectantsDermatologicals +4
Target Protein:
Sulfotransferase 2A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Merestinib DB12381
small molecule | CAS: 1206799-15-6

Merestinib has been used in trials studying the treatment of Cancer, Solid Tumor, Advanced cancer, ColoRectal Cancer, and Metastatic Cancer, among others.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-RingNicotinic Acids +3
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mericitabine DB12045
small molecule | CAS: 940908-79-2

Mericitabine has been investigated for the treatment of Hepatitis C, Chronic. Mericitabine is a polymerase inhibitor being developed for the treatment of chronic hepatitis C. Mericitabine is a prodrug of PSI-6130, which demonstrated excellent potency in p…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
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Meropenem Approved DB00760
small molecule | CAS: 96036-03-2

Meropenem is a broad-spectrum carbapenem antibiotic. It is active against Gram-positive and Gram-negative bacteria. Meropenem exerts its action by penetrating bacterial cells readily and interfering with the synthesis of vital cell wall components, which lead…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacB
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Merotocin DB12932
biotech | CAS: 1190083-57-8

Merotocin has been used in trials studying the treatment of Preterm Delivery.

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Mersalyl DB09338
small molecule | CAS: 486-67-9

Mersalyl is the sodium salt form of mersalyl acid, a mercurial diuretic. It is an outdated drug, and its approval has been discontinued by the FDA. Mersalyl acid is currently replaced by less toxic non-mercury containing diuretics [L1575, L1577]. The sodium s…

Kategori:
Alkylmercury CompoundsDiureticsDrugs that are Mainly Renally Excreted +5
Target Protein:
Alkaline phosphatase, tissue-nonspecific isozymeAquaporin-1Monocarboxylate transporter 1
Waktu Paruh-
Vol. Distribusi-
KlirensThe hepatobiliary e…
Genetik -
Mertiatide DB15780
small molecule | CAS: 66516-09-4

Deskripsi belum tersedia.

Waktu Paruh-
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Mesalazine Approved DB00244
small molecule | CAS: 89-57-6

An anti-inflammatory agent, structurally related to the salicylates and non-steroidal anti-inflammatory drugs like acetylsalicylic acid, which is active in inflammatory bowel disease [A174022]. Although demonstrably effective in treating and maintaining remis…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAminosalicylate +13
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Polyunsaturated fatty acid 5-lipoxygenase +4
Waktu ParuhFor the delayed-rel…
Vol. DistribusiFor the extended-re…
KlirensThe mean (SD) renal…
Genetik -
Mescaline DB19083
small molecule | CAS: 54-04-6

Mescaline is under investigation in clinical trial NCT05933213 (Comparing Mescaline Sodium Enteric-coated Tablets vs Morte-mescaline in the Treatment of Adult Lupus Nephritis).

Kategori:
AlkaloidsAminesAntidepressive Agents +9
Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesdopetam DB16229
small molecule | CAS: 1403894-72-3

Mesdopetam is under investigation in clinical trial NCT04435431 (A Clinical Study of Mesdopetam in Patients With Parkinson's Disease Experiencing Levodopa Induced Dyskinesia).

Kategori:
AminesBenzene DerivativesDopamine Agents +4
Waktu Paruh-
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Genetik -
small molecule | CAS: 147-73-9

Deskripsi belum tersedia.

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Mesocricetus auratus skin Approved DB10605
biotech

Mesocricetus auratus skin or pelt is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Menampilkan 7751–7800 dari 12560
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