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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 155 / 252
biotech | CAS: 2460400-64-8

Mecbotamab vedotin is an anti-Axl humanized monoclonal antibody conjugated to monomethyl auristatin E using a cleavable linker (CAB-Axl-ADC).[A255212]

Waktu Paruh-
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Mechlorethamine Approved DB00888
small molecule | CAS: 51-75-2

A vesicant and necrotizing irritant destructive to mucous membranes, mechlorethamine is an alkylating drug. It was formerly used as a war gas. The hydrochloride is used as an antineoplastic in Hodgkin's disease and lymphomas. It causes severe gastrointestinal…

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +16
Target Protein:
DNA
Waktu Paruh15 minutes
Vol. Distribusi-
Klirens-
Genetik -
Meclinertant DB06455
small molecule | CAS: 146362-70-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Neurotensin, antagonists & inhibitors
Target Protein:
Neurotensin receptor type 1
Waktu Paruh-
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Meclizine Approved DB00737
small molecule | CAS: 569-65-3

Meclizine is a histamine H1 antagonist with antiemetic and antivertigo properties. It is used in the symptomatic treatment of motion sickness and control of vertigo associated with vestibular system diseases. It also exhibits anticholinergic, central nervous …

Kategori:
Anti-Allergic AgentsAnticholinergic AgentsAntiemetics +19
Target Protein:
Histamine H1 receptorNuclear receptor subfamily 1 group I member 3
Waktu ParuhMeclizine has a pla…
Vol. DistribusiThe volume of distr…
KlirensThere is limited da…
Genetik -
Meclocycline DB13092
small molecule | CAS: 2013-58-3

Meclocycline is under investigation in clinical trial NCT00385515 (Efficacy of SNX-1012 in the Treatment of Oral Mucositis) [L797].

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Topical UseAnti-Bacterial Agents +5
Target Protein:
30S ribosomal protein S7
Waktu ParuhHalf life estimated…
Vol. DistribusiEstimated Vd of 121…
Klirens-
Genetik -
Meclofenoxate DB13758
small molecule | CAS: 51-68-3

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicCentral Nervous System Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mecloxamine DB15790
small molecule | CAS: 5668-06-4

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Mecobalamin Approved DB03614
small molecule | CAS: 13422-55-4

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCorrinoids +4
Target Protein:
Methionine synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI-491 DB17859
biotech

MEDI-491 is a recombinant human parvovirus B19 vaccine composed of the VP1 and VP2 capsid proteins.

Waktu Paruh-
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MEDI-547 DB18360
biotech

MEDI-547 is an anti-EphA1 monoclonal antibody conjugated to mcMMAF

Kategori:
Acids, CarbocyclicAmino Acids, Peptides, and ProteinsAntibodies +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI-6469 DB15306
biotech | CAS: 1715924-11-0

MEDI-6469 is a monoclonal antibody under investigation in clinical trial NCT02205333 (A Phase 1b/2 Safety and Tolerability of MEDI6469 in Combination With Therapeutic Immune Agents or Monoclonal Antibodies).

Waktu Paruh-
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MEDI0680 DB15768
biotech

Deskripsi belum tersedia.

Kategori:
Immune Checkpoint Inhibitors
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI3506 DB16473
biotech | CAS: 2376858-66-9

Tozorakimab (MEDI3506), developed by AstraZeneca, was investigated in multiple clinical trials to evaluate its safety, tolerability, efficacy, and pharmacokinetics across various conditions. These trials include NCT03096795 (completed; healthy participants, C…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Interleukin-33
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI6012 DB14833
biotech

Recombinant human lecithin:cholesterol acyltransferase is under investigation in clinical trial NCT03578809 (A Study to Evaluate the Safety and Efficacy of MEDI6012 in Acute ST Elevation Myocardial Infarction).

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Medicago sativa pollen Approved DB10454
biotech

Medicago sativa pollen is the pollen of the Medicago sativa plant. Medicago sativa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 84082-36-0

Deskripsi belum tersedia.

Waktu Paruh-
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Medical air Approved DB09337
small molecule | CAS: 132259-10-0

Medical air is supplied by a special air compressor to patient care areas using clean outside air.

Kategori:
Medical GasesOther Miscellaneous Therapeutic Agents
Waktu Paruh-
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Genetik -
biotech

The use of the plant species _Cannabis sativa_ and _Cannabis indica_, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical conditions as a wave of legalization in North America has changed public …

Kategori:
Agents producing tachycardiaBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Inducers +51
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +38
Waktu ParuhThe half life of TH…
Vol. DistribusiAs a very lipophili…
KlirensOne study reported …
Genetik -
Medifoxamine Approved DB13219
small molecule | CAS: 32359-34-5

Medifoxamine was marketed as an atypical antidepressant, with anxiolyitc properties in France, Spain, and Morrocco in the 1990s but was later withdrawn from the market due to it causing cases of hepatotoxicity [L5461, A174976].

Kategori:
AminesAntidepressive AgentsCentral Nervous System Depressants +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medium-chain triglycerides Approved DB13959
small molecule | CAS: 438544-49-1

Medium-chain triglycerides (MCTs) are triglycerides made up of a glycerol backbone and three fatty acids with an aliphatic tail of six to 12 carbon atoms. MCTs are found in natural foods, such as coconut oil, palm kernel oil, and raw coconut meat. In the body…

Kategori:
LipidsOilsParenteral Nutrition Solutions +1
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of me…
Genetik -
Medrogestone Approved DB09124
small molecule | CAS: 977-79-7

Medrogestone (INN), also known as 6,17?-dimethyl-6-dehydroprogesterone, is a progestational agent derived from 17-methylprogesterone. It was conceived as an alternative for an orally effective contraceptive option.[A31526] It was developed by Ayerst, approved…

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +10
Target Protein:
Progesterone receptor
Waktu ParuhThe half-life of me…
Vol. Distribusi-
Klirens-
Genetik -
Medronic acid Approved DB14078
small molecule | CAS: 1984-15-2

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Medroxyprogesterone acetate Approved DB00603
small molecule | CAS: 71-58-9

Medroxyprogesterone acetate (MPA) is a [progesterone] derivative that is more resistant to metabolism for improved pharmacokinetic properties.[A14848] MPA can be use to treat secondary amenorrhea, endometrial hyperplasia, abnormal uterine bleeding, osteoporos…

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +46
Target Protein:
Progesterone receptorEstrogen receptorATP-dependent translocase ABCB1 +1
Waktu ParuhOral medroxyprogest…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Medrysone Approved DB00253
small molecule | CAS: 2668-66-8

Medrysone is a corticosteroid used in ophthalmology.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +24
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mefenorex DB13852
small molecule | CAS: 17243-57-1

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAlimentary Tract and Metabolism +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mefloquine Approved DB00358
small molecule | CAS: 53230-10-7

Malaria is a protozoan disease that places an enormous burden on human health in endemic areas around the world. The 2020 World Health Organization malaria report indicates a 60% decrease in the global malaria fatality rate between 2000 to 2019.[L30618] Despi…

Kategori:
Agents Causing Muscle ToxicityAgents that reduce seizure thresholdAminoquinolines +20
Target Protein:
Fe(II)-protoporphyrin IX80S ribosomal subunitAdenosine receptor A2a
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThe systemic cleara…
Genetik -
Mefruside DB13405
small molecule | CAS: 7195-27-9

Deskripsi belum tersedia.

Kategori:
AmidesDiureticsLow-Ceiling Diuretics, Excl. Thiazides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mefuparib DB18248
small molecule | CAS: 1392502-82-7

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Megestrol Approved DB19378
small molecule | CAS: 3562-63-8

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +19
Target Protein:
Progesterone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Megestrol acetate Approved DB00351
small molecule | CAS: 595-33-5

17-Hydroxy-6-methylpregna-3,6-diene-3,20-dione. A progestational hormone used most commonly as the acetate ester. As the acetate, it is more potent than progesterone both as a progestagen and as an ovulation inhibitor. It has also been used in the palliative …

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +31
Target Protein:
Progesterone receptorGlucocorticoid receptor
Waktu Paruh34 hours
Vol. Distribusi-
Klirens-
Genetik -
Meglumine Approved DB09415
small molecule | CAS: 6284-40-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlcoholsAmino Sugars +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 133-51-7

Deskripsi belum tersedia.

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAlcoholsAmino Sugars +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meglutol DB04377
small molecule | CAS: 503-49-1

An antilipemic agent which lowers cholesterol, triglycerides, serum beta-lipoproteins and phospholipids. It acts by interfering with the enzymatic steps involved in the conversion of acetate to hydroxymethylglutaryl coenzyme A as well as inhibiting the activi…

Kategori:
Acids, AcyclicAnticholesteremic AgentsAntimetabolites +7
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meladrazine DB13272
small molecule | CAS: 13957-36-3

Deskripsi belum tersedia.

Kategori:
Drugs for Urinary Frequency and IncontinenceGenito Urinary System and Sex HormonesUrologicals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melagatran DB13616
small molecule | CAS: 159776-70-2

Deskripsi belum tersedia.

Kategori:
AminesAnticoagulantsAntithrombins +8
Target Protein:
ProthrombinPlasminogenSerine protease 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Melanoma antigen recognized by T-cells 1 is under investigation in clinical trial NCT01748747 (Vaccine Therapy and Resiquimod in Treating Patients With Stage II-IV Melanoma That Has Been Removed By Surgery).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melarsomine DB11528
small molecule | CAS: 128470-15-5

Melarsomine is a trypanocidal agent marketed by Merial under the trade name Immiticide. It is the only FDA-approved treatment for adult heartworm infection in dogs, however, is is not approved for use in dogs with late-stage infection.

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Melatonin Approved DB01065
small molecule | CAS: 73-31-4

Melatonin is a biogenic amine that is found in animals, plants and microbes. Aaron B. Lerner of Yale University is credited for naming the hormone and for defining its chemical structure in 1958. In mammals, melatonin is produced by the pineal gland. The pin…

Kategori:
AminesAntioxidantsBiogenic Amines +21
Target Protein:
Melatonin receptor type 1AMelatonin receptor type 1BRibosyldihydronicotinamide dehydrogenase [quinone] +7
Waktu Paruh35 to 50 minutes
Vol. Distribusi-
Klirens-
Genetik -
Meldonium DB13723
small molecule | CAS: 76144-81-5

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicCardiac TherapyCardiovascular Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melengestrol DB11529
small molecule | CAS: 5633-18-1

Melengestrol is a steroidal progestin and antineoplastic agent which was never marketed. An acylated derivative, melengestrol acetate, is used as a growth promoter in animals.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCorticosteroids for Systemic Use +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2919-66-6

A 6-methyl progesterone acetate with reported glucocorticoid activity and effect on estrus.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCytochrome P-450 CYP3A Inducers +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melevodopa DB13313
small molecule | CAS: 7101-51-1

Deskripsi belum tersedia.

Kategori:
AminesAmino AcidsAmino Acids, Aromatic +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melilotus albus pollen Approved DB10858
biotech

Melilotus albus pollen is the pollen of the Melilotus albus plant. Melilotus albus pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melilotus officinalis pollen Approved DB10859
biotech

Melilotus officinalis pollen is the pollen of the Melilotus officinalis plant. Melilotus officinalis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melitracen DB13384
small molecule | CAS: 5118-29-6

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meloxicam Approved DB00814
small molecule | CAS: 71125-38-7

Meloxicam is a nonsteroidal anti-inflammatory drug (NSAID) used to relieve various types of pain, including pain caused by musculoskeletal conditions, osteoarthritis, and rheumatoid arthritis.[A190189] With a longer half-life than most other NSAIDS, it is a f…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +28
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe half-life of me…
Vol. DistribusiThe volume of distr…
KlirensAfter an oral dose,…
Genetik -
Melperone DB09224
small molecule | CAS: 3575-80-2

Melperone is an atypical antipsychotic of the butyrophenone chemical class, making it structurally related to the typical antipsychotic haloperidol. Melperone has been used for a span of greater than 30 years in the European Union [L1316]. It has been well e…

Kategori:
Antiarrhythmic agentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +17
Target Protein:
D(2) dopamine receptor
Waktu ParuhApproximately 3-4 h…
Vol. Distribusi-
Klirens-
Genetik -
Melphalan Approved DB01042
small molecule | CAS: 148-82-3

Melphalan is a nitrogen mustard or bischloroethylamine type alkylating agent.[L40928] It was first synthesized in the early 1950s by substituting L-phenylalanine for the methyl group on nitrogen mustard.[A261150, A261155] Melphalan is used in the treatment of…

Kategori:
Alkylating ActivityAlkylating DrugsAmino Acids +17
Target Protein:
DNA
Waktu ParuhIn patients given a…
Vol. DistribusiThe volume of distr…
KlirensAverage total body …
Genetik -
Melphalan flufenamide Approved DB16627
small molecule | CAS: 380449-51-4

Melphalan flufenamide, also known as melflufen or J1, is a prodrug of [melphalan].[A230123,L32173] Melphalan flufenamide is more readily uptaken by cells than melphalan, and is cleaved to the active metabolite by aminopeptidases.[A230123] _In vitro_ models sh…

Kategori:
Alkylating ActivityAlkylating DrugsAmino Acids +12
Target Protein:
DNA
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Melrilimab DB16373
biotech | CAS: 2222865-46-3

Melrilimab is under investigation in clinical trial NCT03207243 (Efficacy and Safety Study of GSK3772847 in Subjects With Moderately Severe Asthma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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