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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 155 / 272
KAb201 DB17210
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Kabiramide C DB03616
small molecule

Deskripsi belum tersedia.

Target Protein:
Actin, alpha skeletal muscle
Waktu Paruh-
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Kaempherol DB01852
small molecule | CAS: 520-18-3

Deskripsi belum tersedia.

Target Protein:
Polyunsaturated fatty acid 5-lipoxygenasePolyunsaturated fatty acid lipoxygenase ALOX15Aldo-keto reductase family 1 member B1 +5
Waktu Paruh-
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Kallidinogenase DB13197
biotech | CAS: 9001-01-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +17
Waktu Paruh-
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Kanamycin Approved DB01172
small molecule | CAS: 59-01-8

Kanamycin (also known as kanamycin A) is an aminoglycoside bacteriocidal antibiotic, available in oral, intravenous, and intramuscular forms, and used to treat a wide variety of infections. Kanamycin is isolated from the bacterium Streptomyces kanamyceticus a…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAminoglycoside Antibacterials +16
Target Protein:
30S ribosomal protein S1216S ribosomal RNA
Waktu Paruh2.5 hours
Vol. Distribusi-
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KAND567 DB16511
small molecule | CAS: 911715-90-7

KAND567, a small molecule, blocks the fractaline (CX3CL1) receptor, which mediates the immune system response to inflammation[L32908]. Because COVID-19 involves cytotoxic cells associated with this pathway, KAND567 is currently being tested as a treatment for…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
CX3C chemokine receptor 1
Waktu Paruh-
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Kaolin Approved DB01575
small molecule | CAS: 1332-58-7

Kaolin is a layered silicate mineral. Kaolin is used in ceramics, medicine, coated paper, as a food additive, in toothpaste, as a light diffusing material in white incandescent light bulbs, and in cosmetics. Until the early 1990s it was the active substance o…

Kategori:
Alimentary Tract and MetabolismAluminium CompoundsAluminum Silicates +11
Waktu Paruh-
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Kappadione Approved DB09332
small molecule | CAS: 131-13-5

Kappadione is a Vitamin K derivative (chemically, it is menadiol sodium diphosphate), previously approved by FDA prior to 1982 and marketed by Lilly Marketing for this drug has been discontinued and is not available in North America [L1543]. It has been found…

Target Protein:
ProthrombinCoagulation factor VIICoagulation factor IX +4
Waktu ParuhMean elimination ha…
Vol. DistribusiIn a study of rabbi…
KlirensThe plasma clearanc…
Genetik -
Karaya gum Approved DB10535
biotech | CAS: 9000-36-6

Karaya gum allergenic extract is used in allergenic testing.

Kategori:
Alimentary Tract and MetabolismBiological ProductsBiopolymers +19
Waktu Paruh-
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Kava Approved DB01322
small molecule | CAS: 9000-38-8

Deskripsi belum tersedia.

Waktu Paruh-
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KB-141 DB03176
small molecule | CAS: 219691-94-8

An anticholesteremic agent.

Kategori:
Acids, CarbocyclicBenzene DerivativesEthers +2
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
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KB109 DB16531
biotech

KB109 is a prebiotic to feed healthy bacteria for them to to outcompete multi-drug resistance organisms.

Waktu Paruh-
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KB3305 DB06349
small molecule | CAS: 639520-46-0

KB3305 is an investigational liver selective antagonist for the glucocorticoid receptor, developed by Karo Bio for the treatment of Type 2 Diabetes.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesBile Acids and Salts +11
Waktu Paruh-
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KB407 DB18223
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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KBP-COVID-19 DB15858
biotech

The KBP-201 COVID-19 Vaccine was developed by British American Tobacco’s (BAT) U.S. biotech subsidiary, Kentucky BioProcessing (KBP). KBP cloned COVID-19’s genetic sequence, identified a potential antigen, and then inserted it into tobacco plants for reproduc…

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KC706 DB05157
small molecule

KC706 is a novel anti-inflammatory drug that works by inhibiting the activity of p38 MAP kinase. KC706 holds potential to treat inflammatory conditions such as rheumatoid arthritis, psoriasis, inflammatory bowel disease and cardiovascular disease.

Target Protein:
Mitogen-activated protein kinase 14Mitogen-activated protein kinase 11Mitogen-activated protein kinase 12 +1
Waktu Paruh-
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KD3010 DB05188
small molecule | CAS: 934760-90-4

KD3010 is a small molecule peroxisome proliferator-activator receptor delta (PPAR Delta) agonist for the treatment of metabolic disorders, including obesity.

Kategori:
AmidesPPAR delta, antagonists & inhibitorsSulfones +1
Target Protein:
Peroxisome proliferator-activated receptor delta
Waktu Paruh-
Vol. Distribusi-
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KDT-3594 DB17085
small molecule

KDT-3594 is a non-ergot dopamine receptor agonist developed by Kissei Pharmaceutical.

Waktu Paruh-
Vol. Distribusi-
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Kebuzone DB08940
small molecule | CAS: 853-34-9

Kebuzone (also known as ketophenylbutazone ) is a non-steroidal anti-inflammatory drug.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +14
Waktu Paruh-
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Kelatorphan DB08040
small molecule | CAS: 92175-57-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsCentral Nervous System Agents +4
Target Protein:
Aminopeptidase NGlutamyl aminopeptidaseLeukotriene A-4 hydrolase
Waktu Paruh-
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KER-047 DB19111
small molecule | CAS: 2248154-85-8

KER-047 is under investigation in clinical trial NCT05927012 (A Study to Evaluate the Safety and Preliminary Efficacy of a Response-guided Dose Titration of KER-047 in the Treatment of Functional IDA (Iron Deficiency Anemia).).

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Ketamine Approved DB01221
small molecule | CAS: 6740-88-1

Ketamine is an NMDA receptor antagonist with a potent anesthetic effect.[A31869] It was developed in 1963 as a replacement for phencyclidine (PCP) by Calvin Stevens at Parke Davis Laboratories. It started being used for veterinary purposes in Belgium and in 1…

Kategori:
Agents producing tachycardiaAmino AcidsAmino Acids, Acidic +35
Target Protein:
Glutamate receptor ionotropic, NMDA 3A5-hydroxytryptamine receptor 3ANeuronal acetylcholine receptor subunit alpha-7 +11
Waktu ParuhThe reported half-l…
Vol. DistribusiThe apparent volume…
KlirensThe clearance rate …
Genetik -
Ketazolam Approved DB01587
small molecule | CAS: 27223-35-4

Ketazolam is a benzodiazepine derivative with anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant activity. Ketazolam is not approved in Canada or America.

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +16
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh26-200 hours
Vol. Distribusi-
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Ketobemidone DB06738
small molecule | CAS: 469-79-4

Ketobemidone is a powerful opioid analgesic. It also has some NMDA-antagonist properties. This makes it useful for some types of pain that don't respond well to other opioids. The most commonly cited equalisation ratio for analgesic doses is 25 mg of ketobemi…

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +20
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Waktu ParuhPlasma half-life: 2…
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small molecule | CAS: 1297537-33-7

Ketodarolutamide, a nonsteroidal antiandrogen (NSAA), is the major active metabolite of [darolutamide].

Kategori:
AntiandrogensAntiandrogens, non-steroidal
Target Protein:
Androgen receptor
Waktu Paruh-
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Ketoprofen Approved DB01009
small molecule | CAS: 22071-15-4

Ketoprofen, a propionic acid derivative, is a nonsteroidal anti-inflammatory agent (NSAIA) with analgesic and antipyretic properties.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +38
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1C-X-C chemokine receptor type 1
Waktu ParuhConventional capsul…
Vol. Distribusi-
Klirens* Oral-dose cl=6.9 …
Genetik -
Ketorolac Approved DB00465
small molecule | CAS: 74103-06-3

Ketorolac is a Non-steroidal anti-inflammatory drug (NSAID) and is commercially available as an oral tablet, injectable, nasal spray and as an ophthalmic solution.[L6358][L6508][L11055][L3674][L11070] It's analgesic properties make it a useful pain manage…

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +26
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhKetorolac trometham…
Vol. DistribusiThe apparent volume…
KlirensThe plasma clearanc…
Genetik -
Ketotifen Approved DB00920
small molecule | CAS: 34580-13-7

Ketotifen is a benzocycloheptathiophene derivative[A231204] with potent antihistaminic and mast cell stabilizing properties. It has a similar structure to some other first-generation antihistamines such as [cyproheptadine] and [azatadine].[A231204] Ketotif…

Kategori:
Anti-Allergic AgentsAnti-Asthmatic AgentsAntihistamine Drugs +15
Target Protein:
Histamine H1 receptor6-phosphogluconate dehydrogenase, decarboxylating
Waktu ParuhKetotifen clearance…
Vol. Distribusi-
Klirens-
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KF-1601 DB18297
small molecule | CAS: 2699634-21-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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KH064 DB04287
small molecule | CAS: 393569-31-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
Phospholipase A2, membrane associated
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Kidney bean Approved DB10639
biotech

Kidney bean allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
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KIN-3248 DB17587
small molecule

KIN-3248 is a small molecule that targets and inhibits oncogenic fibroblast growth factor receptors (FGFRs). It was designed to mainly target FGFR2 and FGFR3 alterations, which act as oncogenic drivers in 10-20% of cholangiocarcinoma and 20-35% of urothelial …

Target Protein:
Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3
Waktu Paruh-
Vol. Distribusi-
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Kinetin Approved DB11336
small molecule | CAS: 525-79-1

Kinetin is a cytokinin which are plant hormones promotes cell division and plant growth. It was shown to naturally exist in DNA of organisms including humans and various plants. While kinetin is used in tissue cultures to produce new plants, it is also found …

Kategori:
CytokininsGrowth SubstancesHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
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KIO-301 DB18465
small molecule | CAS: 1224953-72-3

Deskripsi belum tersedia.

Waktu Paruh-
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Kisspeptin DB19112
biotech | CAS: 388138-21-4

Kisspeptin is under investigation in clinical trial NCT03315325 (Age-dependent Changes in the Responsiveness of Hypothalamic Pituitary Gonadal Axis in Men).

Kategori:
Amino Acids, Peptides, and ProteinsIntercellular Signaling Peptides and ProteinsNeoplasm Proteins +4
Waktu Paruh-
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Kisspeptin-10 DB16210
biotech | CAS: 374675-21-5

Kisspeptin-10 is under investigation in clinical trial NCT03771326 (KP-10 and Insulin Secretion in Men).

Kategori:
Amino Acids, Peptides, and ProteinsGenes, Tumor SuppressorIntercellular Signaling Peptides and Proteins +5
Target Protein:
KiSS-1 receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
KIT-13 DB18093
small molecule | CAS: 103628-72-4

Deskripsi belum tersedia.

Waktu Paruh-
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Kitasamycin DB09309
small molecule | CAS: 1392-21-8

Kitasamycin is a macrolide antibiotic derived from <em>Streptomyces kitasatoensis</em>.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCytochrome P-450 CYP3A Inhibitors +7
Waktu Paruh-
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KL1333 DB17622
small molecule | CAS: 1800405-30-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Kojic acid DB01759
small molecule | CAS: 501-30-4

Deskripsi belum tersedia.

Kategori:
AntioxidantsBiological FactorsCompounds used in a research, industrial, or household setting +3
Target Protein:
Tyrosinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Konjac mannan DB14963
small molecule | CAS: 37220-17-0

Konjac mannan is under investigation in clinical trial NCT01709955 (The Effects of Glucomannan on Weight Loss).

Kategori:
CarbohydratesGastrointestinal AgentsLaxatives +2
Waktu Paruh-
Vol. Distribusi-
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KOS-1584 DB05903
small molecule | CAS: 350493-61-7

KOS-1584 is a second-generation epothilone. Epothilones are anticancer agents with a taxane-like mechanism of action that have demonstrated activity in taxane-resistant tumors. KOS-1584 is a second-generation compound with increased potency, favorable tissue …

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsCytochrome P-450 CYP3A Inhibitors +6
Waktu Paruh-
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Genetik -
KOS-2187 DB05946
small molecule

KOS-2187, a novel erythromycin-based motilin agonist, or motilide, as a clinical candidate for the treatment of gastrointestinal motility disorders such as gastroparesis and gastroesophageal reflux disease (GERD).

Target Protein:
Promotilin
Waktu Paruh-
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KOSN-1724 DB13078
small molecule | CAS: 693272-98-9

KOSN-1724 is under investigation in clinical trial NCT01379287 (Dose-Escalation Safety and Pharmacokinetic Study of Iso-Fludelone in Patients With Advanced Solid Tumors).

Waktu Paruh-
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KP-1461 DB05644
small molecule | CAS: 815588-85-3

KP-1461 is a potent, non-chain-terminating, mutagenic deoxyribonucleoside analogue. Designated a DNA covert nucleoside, the drug consists of a modified base that incorporates randomly into HIV and pairs with multiple bases.

Kategori:
CarbohydratesGlycosidesNucleic Acids, Nucleotides, and Nucleosides
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
KP1237 DB18401
biotech

KP1237 is a antibody-redirecting molecule composed of two binding sites (a CD38 binder and a universal antibody binding terminus binder) connected by a linker chain.

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KRN-330 DB19075
biotech

Anti-a33 fully-human monoclonal antibody is under investigation in clinical trial NCT00838578 (Phase I/II Study of KRN330 Plus Irinotecan in Patients With Metastatic Colorectal Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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KRN-5500 DB15215
small molecule | CAS: 151276-95-8

KRN-5500 is under investigation in clinical trial NCT00002923 (KRN5500 in Treating Patients With Metastatic Solid Tumors).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +4
Waktu Paruh-
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KRN-7000 DB12232
small molecule | CAS: 158021-47-7

KRN7000 has been used in trials studying the treatment of Lung Cancer, Chronic Hepatitis C, Hepatitis B, Chronic, Unspecified Adult Solid Tumor, Protocol Specific, and Prevention of GvHD in Patients With Hematological Malignancies Undergoing AHSCT.

Kategori:
Adjuvants, ImmunologicAmidesAntineoplastic Agents +11
Waktu Paruh-
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Krypton Kr 81m Approved DB09443
small molecule | CAS: 15678-91-8

Deskripsi belum tersedia.

Kategori:
Diagnostic Radiopharmaceuticals
Waktu Paruh-
Vol. Distribusi-
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Genetik -
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