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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 155 / 321
GI-4000 DB05698
biotech

A vaccine containing a heat-killed recombinant <em>Saccharomyces cerevisiae</em> yeast transfected with mutated forms of Ras, an oncogene frequently found in solid tumors, with potential immunostimulant and antitumor activity. [L112]

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GI-5005 DB05942
biotech | CAS: 1001913-27-4

GI-5005 is GlobeImmune's lead infectious disease product from its proprietary Tarmogen active immunotherapy platform for the treatment of chronic hepatitis C infection. GI-5005 is whole, heat-killed recombinant yeast genetically modified to express HCV-specif…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +5
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GI-6207 DB17532
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +17
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GI-6301 DB17533
biotech

Deskripsi belum tersedia.

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Gibberella fujikuroi Approved DB15511
biotech

Gibberella fujikuroi allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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small molecule | CAS: 77-06-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +5
Target Protein:
Arylacetamide deacetylase-like 2
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Gibberellin A4 DB07815
small molecule | CAS: 468-44-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +2
Target Protein:
Arylacetamide deacetylase-like 2
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Gildeuretinol DB18468
small molecule | CAS: 118139-36-9

Deskripsi belum tersedia.

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Giloralimab DB18862
biotech | CAS: 2226292-20-0

Giloralimab is under investigation in clinical trial NCT04807972 (Study to Evaluate Adverse Events and Change in Disease Activity When Intravenous (IV) Infusion of ABBV-927 Is Administered in Combination With IV Modified FOLFIRINOX (Mffx) With or Without IV B…

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Gilteritinib Approved DB12141
small molecule | CAS: 1254053-43-4

Gilteritinib, also known as ASP2215, is a small molecule part of the FLT3 tyrosine kinase inhibitors that presented a greater selectivity and potency when compared with other agents from this group.[A40036] It is a pyrazinecarboxamide derivative that showed h…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +16
Target Protein:
Receptor-type tyrosine-protein kinase FLT3Tyrosine-protein kinase receptor UFOALK tyrosine kinase receptor +1
Waktu ParuhThe reported median…
Vol. DistribusiThe estimated appar…
KlirensThe estimated clear…
Genetik -
Gimatecan DB06721
small molecule | CAS: 292618-32-7

Gimatecan is an orally available 7-t-butoxyiminomethyl-substituted lipophilic camptothecin derivative.

Kategori:
AlkaloidsOATP1B1/SLCO1B1 Substrates
Target Protein:
DNA topoisomerase 1
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Gimeracil Approved DB09257
small molecule | CAS: 103766-25-2

Gimeracil is an adjunct to antineoplastic therapy, used to increase the concentration and effect of the main active componets within chemotherapy regimens. Approved by the European Medicines Agency (EMA) in March 2011, Gimeracil is available in combination wi…

Kategori:
Drugs that are Mainly Renally Excreted
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]
Waktu ParuhFollowing a single …
Vol. DistribusiAlthough no intrave…
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Gimsilumab DB15280
biotech | CAS: 1648796-29-5

Gimsilumab is under investigation in clinical trial NCT01357759 (Safety and Tolerability of MORAb-022 in Healthy and Rheumatoid Arthritis Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +9
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Ginger oil Approved DB14690
biotech | CAS: 8007-08-7

Deskripsi belum tersedia.

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Gingerol DB19255
small molecule | CAS: 23513-14-6

Gingerol is under investigation in clinical trial NCT05882864 (Efficacy of Ginger Muco-bioadhesive Gel in Management of Oral Lichen Planus With Immunohistochemical Analysis).

Kategori:
AlcoholsBenzene DerivativesLipids +2
Target Protein:
Transient receptor potential cation channel subfamily A member 1
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Ginisortamab DB18863
biotech | CAS: 2390147-17-6

Ginisortamab is under investigation in clinical trial NCT04393298 (A Study to Assess the Safety, Pharmacokinetics and Anti Tumor Activity of UCB6114 Administered Intravenously to Participants With Advanced Solid Tumors).

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Ginkgo biloba Approved DB01381
biotech | CAS: 90045-36-6

_Ginkgo biloba_ extract contains a group of terpene lactones (notably, ginkgolides and diterpenes) and ginkgo flavone glycosides (notably, ginkgetin, bilobetin, and sciadopitysin) that have antioxidant and vasoactive properties.[A232389] Most of the studies t…

Kategori:
Anti-Dementia DrugsBiological ProductsBlood Circulation +27
Target Protein:
Sodium-dependent noradrenaline transporterPhospholipase A2, membrane associatedGlycine receptor subunit alpha-1 +5
Waktu ParuhUnpublished human d…
Vol. DistribusiNo data available.
KlirensNo data available.
Genetik -
biotech

Ginkgo biloba leaf oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Ginkgolide A DB06743
small molecule | CAS: 15291-75-5

Ginkgolide A is a highly active PAF antagonist cage molecule that is isolated from the leaves of the Ginkgo biloba tree. Shows potential in a wide variety of inflammatory and immunological disorders.

Kategori:
DiterpenesTerpenes
Target Protein:
Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2Glycine receptor subunit alpha-3 +1
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ginkgolide-B DB06744
small molecule

Deskripsi belum tersedia.

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ginkgolide-C DB06745
small molecule | CAS: 15291-76-6

Deskripsi belum tersedia.

Kategori:
DiterpenesTerpenes
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ginkgolide-J DB06746
small molecule | CAS: 107438-79-9

Deskripsi belum tersedia.

Kategori:
DiterpenesTerpenes
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ginkgolide-M DB06747
small molecule | CAS: 15291-78-8

Deskripsi belum tersedia.

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Ginseng DB01404
biotech | CAS: 50647-08-0

Ginseng is promoted as an adaptogen (a product that increases the body's resistance to stress), one which can to a certain extent be supported with reference to its anticarcinogenic and antioxidant properties. Ginseng is also known to contain phytoestrogens.

Kategori:
AngiospermsAraliaceaeBiological Products +11
Target Protein:
Aryl hydrocarbon receptorInterleukin-6Prostaglandin G/H synthase 2
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Ginsenoside B2 DB14815
small molecule | CAS: 52286-59-6

Ginsenoside B2 is under investigation in clinical trial NCT00781534 (A Clinical Trial of Ginseng in Diabetes).

Kategori:
CarbohydratesGlycosidesPanax +3
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Ginsenoside C DB06748
small molecule | CAS: 11021-13-9

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsCarbohydratesGlycosides +6
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Ginsenoside Rb1 DB06749
small molecule | CAS: 41753-43-9

Ginsenosides are a class of steroid glycosides, and triterpene saponins, found exclusively in the plant genus Panax (ginseng). Ginsenosides have been the target of research, as they are viewed as the active compounds behind the claims of ginseng's efficacy. B…

Kategori:
CarbohydratesGlycosidesOATP1B3 inhibitors +4
Target Protein:
Solute carrier organic anion transporter family member 1B3
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Ginsenoside Rd DB19256
small molecule | CAS: 52705-93-8

Ginsenoside Rd is under investigation in clinical trial NCT00815763 (Efficacy and Safety of Ginsenoside-rd for Acute Ischemic Stroke).

Kategori:
CarbohydratesGlycosidesPanax +3
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Ginsenoside Rg1 DB06750
small molecule | CAS: 22427-39-0

Ginsenosides are a class of steroid glycosides, and triterpene saponins, found exclusively in the plant genus Panax (ginseng). Ginsenosides have been the target of research, as they are viewed as the active compounds behind the claims of ginseng's efficacy. B…

Kategori:
CarbohydratesCentral Nervous System AgentsGlycosides +4
Target Protein:
Solute carrier organic anion transporter family member 1B3
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Ginsenoside Rg3 DB19257
small molecule | CAS: 14197-60-5

Ginsenoside Rg3 is under investigation in clinical trial NCT01757366 (Safety and Efficacy of Ginsenoside Rg3 in Combination With First-line Chemotherapy in Advanced Gastric Cancer).

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicCarbohydrates +5
Target Protein:
Voltage-gated inwardly rectifying potassium channel KCNH2
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Ginsenosides DB14152
small molecule | CAS: 74749-74-9

Dammarane type triterpene saponins based mainly on the aglycones, protopanaxadiol and protopanaxatriol.

Kategori:
CarbohydratesGlycosidesSaponins +2
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Giredestrant DB19125
small molecule | CAS: 1953133-47-5

Giredestrant is under investigation in clinical trial NCT06065748 (A Study to Evaluate Efficacy and Safety of Giredestrant Compared With Fulvestrant (Plus a CDK4/6 Inhibitor), in Participants With Er-positive, Her2-negative Advanced Breast Cancer Resistant to…

Kategori:
Heterocyclic Compounds, Fused-RingIndole AlkaloidsIndoles +1
Target Protein:
Estrogen receptor
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Girentuximab DB05304
biotech | CAS: 916138-87-9

Girentuximab is a monoclonal chimeric (mouse/human) antibody directed against carbonic anhydrase IX, an antigen expressed in 95% of clear cell renal cell carcinomas (RCC).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Carbonic anhydrase 9Interleukin-2
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biotech | CAS: 1011710-99-8

Girentuximab I-124 is under investigation in clinical trial NCT01762592 (REDECT 2: REnal Masses: Pivotal Trial to DEteCT Clear Cell Renal Cell Carcinoma With PET/CT).

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Giripladib DB15426
small molecule | CAS: 865200-20-0

Giripladib is under investigation in clinical trial NCT00396955 (A Study Comparing 4 Dose Regimens of PLA-695, Naproxen, and Placebo In Subjects With Osteoarthritis Of The Knee).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
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biotech | CAS: 2166101-71-7

Giroctocogene fitelparvovec is under investigation in clinical trial NCT04370054 (Study to Evaluate the Efficacy and Safety of PF-07055480 in Moderately Severe to Severe Hemophilia a Adults).

Kategori:
Adeno-associated Viral Vector Therapies
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Gisadenafil DB11902
small molecule | CAS: 334826-98-1

Gisadenafil has been investigated for the treatment of Prostatic Hyperplasia.

Kategori:
AmidesCyclic Nucleotide Phosphodiesterases, Type 5Pyrimidines +2
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase
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Gitoformate DB13537
small molecule | CAS: 10176-39-3

Deskripsi belum tersedia.

Kategori:
CarbohydratesCardanolidesCardenolides +7
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Givastomig DB18618
biotech

Givastomig is an anti-Claudin 18.2 and 4.1BB bispecific antibody.

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GIVI-MPC DB17905
biotech

GIVI-MPC is a therapy that uses human-induced pluripotent stem cell-derived myogenic progenitor cells.

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Givinostat Approved DB12645
small molecule | CAS: 497833-27-9

Givinostat is a small molecule histone deacetylase (HDAC) inhibitor. It has been investigated as a treatment for a variety of inflammatory diseases, like Crohn's disease and juvenile idiopathic arthritis, cancers like leukemia and lymphoma, as well as several…

Kategori:
Acids, AcyclicAminesAntineoplastic Agents +20
Target Protein:
Histone deacetylaseTyrosine-protein kinase JAK2Histone deacetylase 1
Waktu ParuhThe apparent plasma…
Vol. DistribusiAccording to popula…
KlirensAccording to popula…
Genetik -
Givosiran Approved DB15066
biotech | CAS: 1639325-43-1

Givosiran is a small interfering RNA (siRNA) directed towards 5-aminolevulinic acid synthase, a critical enzyme in the heme biosynthesis pathway.[L10202] It is manufactured by Alnylam Pharmaceuticals and was first approved for use in the United States in Nove…

Kategori:
Alimentary Tract and MetabolismAmino SugarsAminolevulinate Synthase 1-directed RNA Interaction +13
Target Protein:
ALAS1 mRNA5-aminolevulinate synthase, non-specific, mitochondrial
Waktu ParuhBoth givosiran and …
Vol. DistribusiThe apparent centra…
KlirensThe apparent cleara…
Genetik -
GL-0719 DB18436
biotech

Deskripsi belum tersedia.

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GL-2045 DB16971
biotech

Deskripsi belum tersedia.

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Glafenine DB08963
small molecule | CAS: 3820-67-5

An anthranilic acid derivative with analgesic properties used for the relief of all types of pain. Glafenine is withdrawn from the American market.

Kategori:
Acids, CarbocyclicAminobenzoatesAnalgesics +8
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Glasdegib Approved DB11978
small molecule | CAS: 1095173-27-5

Glasdegib, also known as PF-04449913, is a small-molecule hedgehog signaling inhibitor selected under the group of benzimidazoles. In early research, benzimidazoles attracted large interest as they represented a class of inhibitors with low molecular weight, …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Protein smoothenedSerine/threonine-protein kinase mTOR
Waktu ParuhThe reported half-l…
Vol. DistribusiGlasdegib reported …
KlirensThe clearance rate …
Genetik -
Glatiramer Approved DB05259
biotech | CAS: 28704-27-0

Glatiramer acetate is a mix of synthetic polypeptides that includes L-glutamic acid, L-alanine, L-tyrosine, and L-lysine at an average molar fraction of 0.141, 0.427, 0.095, and 0.338, respectively.[L41940] Since glatiramer acetate is a heterogeneous drug, th…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +5
Target Protein:
MHC class II protein complex
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Glecaprevir Approved DB13879
small molecule | CAS: 1365970-03-1

Glecaprevir is a direct acting antiviral agent and Hepatitis C virus (HCV) NS3/4A protease inhibitor that targets the the viral RNA replication. In combination with [DB13878], glecaprevir is a useful therapy for patients who experienced therapeutic failure fr…

Kategori:
Acids, AcyclicAmidesAmino Acids +37
Target Protein:
NS3 proteaseGenome polyprotein
Waktu ParuhThe elimination hal…
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Glecirasib DB18744
small molecule | CAS: 2657613-87-9

Deskripsi belum tersedia.

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biotech | CAS: 1182215-65-1

A conjugate of an anti-glycoprotein non-metastatic melanoma protein B mAb and monomethyl auristatin E for the treatment of melanoma and breast cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntineoplastic Agents +8
Target Protein:
Transmembrane glycoprotein NMB
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