Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 152 / 236
Morniflumate DB09285
small molecule | CAS: 65847-85-0

Morniflumate is a non-steroidal anti-inflammatory drug with antipyretic properties. It is the morpholinoethyl ester of niflumic acid [L1496]. In one study, post morniflumate ingestion, physical examination and clinical symptoms of those with bronchitis show…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +14
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Polyunsaturated fatty acid 5-lipoxygenase +2
Waktu Paruh2h [L1498]
Vol. Distribusi-
Klirens45 ml/min [L1498]
Genetik -
Moroctocog alfa Approved DB13999
biotech | CAS: 284036-24-4

Moroctocog alfa, also known as BDDrFVIII (B domain deleted recombinant factor VIII), is a recombinant DNA-based drug with functional characteristics comparable to those of endogenous coagulation Factor VIII, the essential human blood clotting protein that is …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu ParuhMean terminal elimi…
Vol. DistribusiMean steady-state v…
KlirensMean clearance = 4.…
Genetik -
Moroxydine DB13597
small molecule | CAS: 3731-59-7

Deskripsi belum tersedia.

Kategori:
AmidinesAnti-Infective AgentsAntiinfectives for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morphine Approved DB00295
small molecule | CAS: 57-27-2

Morphine, the main alkaloid of opium, was first obtained from poppy seeds in 1805.[A176035] It is a potent analgesic, though its use is limited due to tolerance, withdrawal, and the risk of abuse.[A176050] Morphine is still routinely used today, though there …

Kategori:
AlkaloidsAnalgesicsAnesthetics +25
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Gen Terkait:
ABCB1 OPRM1
Waktu ParuhMorphine has a half…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik 2 Varian
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin S
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin S
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 102-77-2

Deskripsi belum tersedia.

Kategori:
Cell-mediated ImmunityHeterocyclic Compounds, Fused-RingIncreased Histamine Release +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morrhuic acid DB14087
small molecule

Morrhuic acid is a mixture of unsaturated fatty acids obtained from cod liver oil.

Kategori:
Cardiovascular AgentsCompounds used in a research, industrial, or household settingFatty Acids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Morus alba root bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morus rubra pollen Approved DB10373
biotech

Morus rubra pollen is the pollen of the Morus rubra plant. Morus rubra pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosapramine DB13676
small molecule | CAS: 89419-40-9

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosapride DB11675
small molecule | CAS: 112885-41-3

Mosapride is under investigation for the treatment and prevention of Postoperative Ileus and Gastric Peroral Endoscopic Pyloromyotomy (G-POEM). Mosapride has been investigated for the treatment and diagnostic of Constipation, Type 2 Diabetes, Functional Dyspe…

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmides +13
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Moschus berezovskii musk sac resin is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosedipimod DB12592
small molecule | CAS: 221139-79-3

Mosedipimod has been used in trials studying the supportive care and treatment of Chemotherapy-induced Neutropenia.

Kategori:
Experimental Unapproved Treatments for COVID-19Lipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosliciguat DB19425
small molecule | CAS: 2231749-54-3

Mosliciguat is under investigation in clinical trial NCT06635850 (A Phase 2 Study of Mosliciguat in PH-ILD).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Motavizumab DB06310
biotech | CAS: 677010-34-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Motesanib DB05575
small molecule | CAS: 453562-69-1

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingNicotinic Acids +3
Target Protein:
Vascular endothelial growth factor receptor 2Mast/stem cell growth factor receptor Kit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Motixafortide Approved DB14939
biotech | CAS: 664334-36-5

Motixafortide is a cyclic peptide hematopoietic stem cell mobilizer used to improve stem cell collection prior to autologous transplantation.[L48116] Hematopoietic stem cell transplantation (HSCT) is commonly employed in the context of hematologic cancers - h…

Kategori:
Amino Acids, Peptides, and ProteinsHematopoietic Stem Cell MobilizerPeptides
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhThe effective half-…
Vol. DistribusiIn a typical patien…
KlirensIn a typical patien…
Genetik -
Motolimod DB12303
small molecule | CAS: 926927-61-9

Motolimod has been used in trials studying the treatment of Lymphoma, Tongue Cancer, Ovarian Cancer, Adult Solid Neoplasm, and Fallopian Tube Cancer, among others.

Kategori:
Heterocyclic Compounds, Fused-RingToll-Like Receptor 8, agonists
Target Protein:
Toll-like receptor 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Motuporin DB04738
small molecule | CAS: 141672-08-4

Motuporin is a toxin isolated from the marine sponge Thenonella swinhoie grey.

Kategori:
Amino Acids, Peptides, and ProteinsCytotoxinsPeptides
Target Protein:
Serine/threonine-protein phosphatase PP1-gamma catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Metallo-beta-lactamase L1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moxetumomab pasudotox Approved DB12688
biotech | CAS: 1020748-57-5

CD22 is a lineage-restricted B-cell antigen that is expressed solely in on B-chronic lymphocytic leukemia, hairy cell leukemia, acute lymphocytic leukemiathe and Burkitt's lymphoma. The predecessor of Moxetumab pasudotox (MxP), named BL22, was first created b…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
B-cell receptor CD22Elongation factor 2
Waktu ParuhMxP presents a shor…
Vol. DistribusiThe mean volume of …
KlirensThe mean systemic c…
Genetik -
Moxidectin Approved DB11431
small molecule | CAS: 113507-06-5

Moxidectin is a potent, broad-spectrum endectocide (antiparasitic that is active against endo- and ecto-parasites) with activity against nematodes, insects, and acari. It was first used in cattle followed by an approved use in general animals. It is a semi-sy…

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +9
Target Protein:
Glutamate-gated chloride channelGABA-A gated chloride channelABC transporters
Waktu ParuhMoxidectin reporter…
Vol. DistribusiMoxidectin presents…
KlirensThe apparent cleara…
Genetik -
Moxifloxacin Approved DB00218
small molecule | CAS: 151096-09-2

Moxifloxacin is a synthetic fluoroquinolone antibiotic agent. Bayer AG developed the drug (initially called BAY 12-8039) and it is marketed worldwide (as the hydrochloride) under the brand name Avelox (in some countries also Avalox) for oral treatment.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +18
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +3
Waktu Paruh11.5-15.6 hours (si…
Vol. Distribusi* 1.7 to 2.7 L/kg
Klirens* 12 +/- 2 L/hr
Genetik -
Moxisylyte Approved DB09205
small molecule | CAS: 54-32-0

Moxisylyte, denominated as thymoxamine in the UK, is a specific and orally active ?1-adrenergic antagonist.[T45] According to the WHO, moxisylyte is approved since 1987[T91] and in the same year, it acquired the denomination of orphan product by the FDA.[L117…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +17
Target Protein:
Alpha-1D adrenergic receptorAlpha adrenergic receptor
Waktu ParuhThe half-life of mo…
Vol. DistribusiIn preclinical tria…
KlirensIn preclinical tria…
Genetik -
Moxonidine Approved DB09242
small molecule | CAS: 75438-57-2

Moxonidine is a new-generation centrally acting antihypertensive drug approved for the treatment of mild to moderate essential hypertension. It is suggested to be effective in cases where other agents such as thiazides, beta-blockers, ACE inhibitors, and calc…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +8
Target Protein:
Alpha-2C adrenergic receptorAlpha-2B adrenergic receptorAlpha-2A adrenergic receptor +1
Waktu ParuhPlasma elimination …
Vol. Distribusi1.8±0.4L/kg. [FDA l…
KlirensAdministered twice …
Genetik -
biotech

RP-L102 is a lentiviral vector carrying the Fanconi Anemia-A (FANCA) gene currently being developed by Rocket Pharmaceuticals for the treatment of Fanconi anemia type A

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mozenavir DB02102
small molecule | CAS: 174391-92-5

Deskripsi belum tersedia.

Kategori:
Amides
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MP-0250 DB17218
biotech | CAS: 1816305-70-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MP4CO DB17860
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPI-674 DB05749
small molecule

MPI-674 is an aromatase inhibitor (AI) with a well-established, multi-year chronic safety and tolerability profile. AIs are a class of drugs that reduce the amount of estrogen circulating in the body by binding to and inhibiting the enzyme aromatase, which i…

Target Protein:
Aromatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPT-0L055 DB17136
small molecule | CAS: 2069950-14-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPT0B640 DB16512
small molecule

MPT0B640 was under investigation in clinical trials NCT04526717 for COVID-19 infection and NCT04294875 for locally advanced or metastatic solid malignancies.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRG-003 DB17407
biotech

MRG-003 is a recombinant humanized anti-human epidermal growth factor receptor monoclonal antibody conjugated to monomethyl auristatin E.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRK-003 DB17015
small molecule | CAS: 623165-93-5

MRK-003 is a potent and selective ?-secretase inhibitor developed by Merck. It is the preclinical analog of [MK-0752], a drug in clinical development.[A252682]

Kategori:
Amyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme InhibitorsGamma Secretase Inhibitors and Modulators +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRK-409 DB13993
small molecule | CAS: 233275-76-8

MRK-409 is a GABA-A receptor agonist [A31972].

Kategori:
Anti-Anxiety AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-1345 DB18739
biotech

mRNA-1345 is an investigational RSV vaccine.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3351 DB17718
biotech

mRNA-3351 is a modified mRNA encoding the UGT1A1 gene. Developed by Moderna, it is currently being investigated as the treatment for Crigler-Najjar syndrome

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3705 DB17668
biotech

mRNA-3705 is an investigational mRNA encoding methylmalonic CoA mutase (MUT) enzyme. Developed by Moderna TX Inc., it is being investigated for the treatment of methylmalonic academia.[A258843]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3745 DB18554
biotech

mRNA-3745 is a lipid nanoparticle (LNP) encapsulated with nucleoside-modified, codon-optimized mRNAs encoding human glucose 6-phosphatase (G6Pase).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3927 DB17669
biotech

mRNA-3927 is an investigational mRNA therapy that consists of two mRNAs that encode for the alpha and beta subunits of the mitochondrial enzyme propionyl-CoA carboxylase (PCC) encapsulated within a lipid nanoparticle (LNP). Developed by Moderna Inc., it is be…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRT5201 DB17656
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRTX-1719 DB18016
small molecule | CAS: 2630904-44-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRx-4DP0004 DB15751
biotech

MRx-4DP0004 is a lyophilised formulation of the Bifidobacterium breve strain of commensal bacteria. It is a live biotherapeutic derived from the microbiota of a healthy human infant.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRX-I DB12796
small molecule | CAS: 1112968-42-9

MRX-I has been used in trials studying the treatment of Bacterial Infections.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRx0518 DB17523
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MS1901 DB18747
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MSX-122 DB12715
small molecule | CAS: 897657-95-3

MSX-122 has been used in trials studying the treatment of Solid Tumors.

Kategori:
Receptors, CXCR4, antagonists & inhibitors
Target Protein:
C-X-C chemokine receptor type 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MT-0169 DB17430
biotech

MT-0169 is a usion protein comprised of an enzymatically active Shiga-like toxin-I A1 subunit fused to a human single chain variable fragment with affinity for human CD38 cell surface protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MT1621 DB17970
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 7551–7600 dari 11778
Sebelumnya Halaman 152 / 236 Berikutnya