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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 151 / 236
MMI-175 DB02378
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-secretase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mobocertinib Approved DB16390
small molecule | CAS: 1847461-43-1

Mobocertinib is a kinase inhibitor targeted against human epidermal growth factor receptor (EGFR). It is used specifically in the treatment of non-small cell lung cancer (NSCLC) caused by exon 20 insertion mutations in the _EGFR_ gene,[L38368] which are typic…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +15
Target Protein:
Epidermal growth factor receptor
Waktu ParuhAt steady-state, th…
Vol. DistribusiThe mean apparent v…
KlirensAt steady-state, th…
Genetik -
Mocetinostat DB11830
small molecule | CAS: 726169-73-9

Mocetinostat has been used in trials studying the treatment of Lymphoma, Urothelial Carcinoma, Relapsed and Refractory, Myelodysplastic Syndrome, and Metastatic Leiomyosarcoma, among others.

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +6
Target Protein:
Histone deacetylase 1Histone deacetylase 3Histone deacetylase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moclobemide Approved DB01171
small molecule | CAS: 71320-77-9

A reversible monoamine oxidase inhibitor (MAOI) selective for isoform A (RIMA) used to treat major depressive disorder. Most meta-analyses and most studies indicate that in the acute management of depression, moclobemide is more efficacious than placebo medic…

Kategori:
Acids, CarbocyclicAgents that produce hypertensionAgents that reduce seizure threshold +28
Target Protein:
Amine oxidase [flavin-containing] AMonoamine oxidaseAmine oxidase [flavin-containing] B
Waktu Paruh1-2 hours (4 hours …
Vol. Distribusi1-1.5 L/Kg [L1350]
KlirensClearance of 30-78 …
Genetik -
MOD-5014 DB17715
biotech

MOD-5014 is a long-acting carboxy-terminal peptide (CTP)-modified Factor IIa.[A259088] It is being investigated for the treatment of hemophilia.[L46173]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modafinil Approved DB00745
small molecule | CAS: 68693-11-8

Modafinil is a stimulant drug marketed as a 'wakefulness promoting agent' and is one of the stimulants used in the treatment of narcolepsy. Narcolepsy is caused by dysfunction of a family of wakefulness-promoting and sleep-suppressing peptides, the orexins, w…

Kategori:
Benzene DerivativesBenzhydryl CompoundsCentral Nervous System Agents +35
Target Protein:
Sodium-dependent dopamine transporterAlpha-1B adrenergic receptor
Gen Terkait:
COMT COMT
Waktu Paruh23-215 hours
Vol. Distribusi* 0.9 L/kg
Klirens-
Genetik 2 Varian
Modakafusp alfa DB16399
biotech

Modakafusp alfa is under investigation in clinical trial NCT03215030 (A Study to Investigate the Safety, Tolerability, Efficacy, Pharmacokinetics, and Immunogenicity of TAK-573 in Participants With Refractory Multiple Myeloma (MM)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moderna COVID-19 Vaccine Approved DB15654
biotech

The Moderna COVID-19 Vaccine (mRNA-1273) is a novel mRNA-based vaccine encapsulated in a lipid nanoparticle that encodes for a full-length pre-fusion stabilized spike (S) protein of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2). Coronavirus dis…

Kategori:
Biological ProductsCOVID-19 VaccinesExperimental Unapproved Treatments for COVID-19 +5
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nucleoside 2-deoxyribosyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modified vaccinia ankara Approved DB15483
biotech

Modified Vaccinia Ankara (MVA) refers to an attenuated strain of the Vaccinia virus. Vaccines using MVA are live and non-replicating, and are produced using Modified Vaccinia Ankara-Bavarian Nordic (MVA-BN).[L42660,L42670]

Kategori:
Anti-Infective AgentsAntiviral AgentsBiological Products +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2171576-44-4

Modified vaccinia virus Ankara-85A antigen is under investigation in clinical trial NCT00953927 (A Study of MVA85A in Healthy Infants).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBacterial Vaccines +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modimelanotide DB15314
small molecule | CAS: 926277-68-1

Modimelanotide is under investigation in clinical trial NCT01897519 (A Safety and Efficacy Trial of Multiple Dosing Regimens of ABT-719 for the Prevention of Acute Kidney Injury in Subjects Undergoing High Risk Surgery).

Kategori:
Pyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modipafant DB16237
small molecule | CAS: 122957-06-6

Modipafant is under investigation in clinical trial NCT02569827 (Celgosivir or Modipafant as Treatment for Adult Participants With Uncomplicated Dengue Fever in Singapore).

Kategori:
Pyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modithromycin DB16238
small molecule | CAS: 736992-12-4

Modithromycin is under investigation in clinical trial NCT00270517 (Comparative Study of EDP-420 Versus Another Antibiotic in the Treatment of Community Acquired Pneumonia).

Kategori:
LactonesPolyketides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modotuximab DB14827
biotech | CAS: 1310460-86-6

Modotuximab is under investigation in clinical trial NCT03549338 (Sym004 Versus Futuximab or Modotuximab in Patients With mCRC).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Modufolin DB12676
small molecule | CAS: 31690-11-6

Modufolin is under investigation for the treatment of Osteosarcoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moexipril Approved DB00691
small molecule | CAS: 103775-10-6

Moexipril is a non-sulfhydryl containing precursor of the active angiotensin-converting enzyme (ACE) inhibitor moexiprilat. It is used to treat high blood pressure (hypertension). It works by relaxing blood vessels, causing them to widen. Lowering high blood …

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +14
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhMoexipril eliminati…
Vol. Distribusi* 183 L
Klirens* 441 mL/min
Genetik -
Moexiprilat DB14210
small molecule | CAS: 103775-14-0

The active metabolite of the prodrug [Moexipril].

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAngiotensin-Converting Enzyme Inhibitors +2
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mogamulizumab Approved DB12498
biotech | CAS: 1159266-37-1

Mogamulizumab is a humanized monoclonal antibody (mAb) directed against CC chemokine receptor 4 (CCR4) for the treatment of Mycosis Fungoides (MF) and Sézary Syndrome (SS), the most common subtypes of cutaneous T-cell lymphoma. Cutaneous T-cell lymphomas occu…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
C-C chemokine receptor type 4
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe central volume …
KlirensClearance is 12 mL/…
Genetik -
Molibresib DB16239
small molecule | CAS: 1260907-17-2

Molibresib is under investigation in clinical trial NCT01943851 (A Dose Escalation Study to Investigate the Safety, Pharmacokinetics (PK), Pharmacodynamics (PD) and Clinical Activity of GSK525762 in Subjects With Relapsed, Refractory Hematologic Malignancies).

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Bromodomain-containing protein 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Molindone Approved DB01618
small molecule | CAS: 7416-34-4

An indole derivative effective in schizophrenia and other psychoses and possibly useful in the treatment of the aggressive type of undersocialized conduct disorder. Molindone has much lower affinity for D2 receptors than most antipsychotic agents and has a re…

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +18
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2A +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Molsidomine Approved DB09282
small molecule | CAS: 25717-80-0

Molsidomine is an orally active, long-acting vasodilator, which belongs to the class of medications known as syndnones. Interestingly, it is being studied as being a preventive measure in cerebral infarction [A31932].

Kategori:
Cardiac TherapyCardiovascular AgentsMorpholines +7
Target Protein:
Guanylate cyclase soluble subunit alpha-2
Waktu Paruh-
Vol. Distribusi98 L [L1369]
Klirensrenal excretion is …
Genetik -
Molybdate DB15878
small molecule | CAS: 14259-85-9

Deskripsi belum tersedia.

Kategori:
ElementsMetalsMetals, Heavy +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Molybdate Mo-99 DB16587
small molecule | CAS: 72826-31-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Molybdenum Approved DB11137
small molecule | CAS: 7439-98-7

Molybdenum is a chemical element with symbol Mo and atomic number 42. As it is not a naturally occuring free metal on Earth, molybdenum is found only in various oxidation states in minerals. Molybdenum is commonly used in metallurgy and other chemical applica…

Kategori:
Diet, Food, and NutritionElementsFood +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 872689-63-9

Absence of molybdenum cofactor leads to accumulation of toxic levels of sulphite and neurological damage usually leading to death within months of birth, due to the lack of active sulfite oxidase.

Kategori:
CoenzymesEnzymes and Coenzymes
Target Protein:
Aldehyde oxidoreductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1313-27-5

Deskripsi belum tersedia.

Kategori:
Air PollutantsAnionsElectrolytes +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Momelotinib Approved DB11763
small molecule | CAS: 1056634-68-4

Momelotinib is a Janus Kinase 1 (JAK1) and 2 (JAK2) inhibitor. It is a competitive inhibitor of JAK ATP binding.[A261566] First approved by the FDA on September 15, 2023,[L48206] momelotinib is used to treat myelofibrosis.[L48186] Myelofibrosis (MF) is a grou…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +24
Target Protein:
Tyrosine-protein kinase JAK1Tyrosine-protein kinase JAK2Tyrosine-protein kinase JAK3 +3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean (%CV) appa…
KlirensThe mean (%CV) clea…
Genetik -
Mometasone DB00764
small molecule | CAS: 105102-22-5

Mometasone is a corticosteroid not currently used in medical products. [Mometasone furoate] however, is still in use.

Kategori:
Adrenal Cortex HormonesAdrenalsAnti-Allergic Agents +29
Target Protein:
Glucocorticoid receptorProgesterone receptor
Waktu Paruh5.8 hours
Vol. Distribusi-
Klirens-
Genetik -
Mometasone furoate Approved DB14512
small molecule | CAS: 83919-23-7

Mometasone furoate is a corticosteroid drug that can be used for the treatment of asthma, rhinitis, and certain skin conditions[FDA Label][F4292,F4295]. It has a glucocorticoid receptor binding affinity 22 times stronger than [dexamethasone] and higher than m…

Kategori:
Adrenal Cortex HormonesAdrenalsAdrenergics, Inhalants +28
Target Protein:
Glucocorticoid receptorProgesterone receptor
Waktu ParuhThe terminal half l…
Vol. DistribusiSteady state volume…
KlirensThe clearance rate …
Genetik -
Monalizumab DB12824
biotech | CAS: 1228763-95-8

Monalizumab has been used in trials studying the treatment of Gynecologic Cancer, Chronic Lymphocytic Leukemia, and Squamous Cell Carcinoma of the Oral Cavity.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monastrol DB04331
small molecule | CAS: 254753-54-3

Deskripsi belum tersedia.

Kategori:
Antimitotic AgentsAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
Kinesin-like protein KIF11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monensin DB11430
small molecule | CAS: 17090-79-8

Monensin is a polyether isolated from _Streptomyces cinnamonensis_ that presents antibiotic properties. It is widely used in ruminant animal feeds.

Kategori:
Acids, AcyclicAnti-Infective AgentsAntiparasitic Agents +21
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monepantel DB18755
small molecule | CAS: 887148-69-8

Deskripsi belum tersedia.

Kategori:
AcetonitrilesNitriles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mongersen DB15019
biotech | CAS: 1443994-46-4

Mongersen is under investigation in clinical trial NCT02957474 (A Study to Evaluate the Effect of Food, Formulation Strength, and a Proton Pump Inhibitor on GED 0301 Pharmacokinetics in Healthy Adult Subjects).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesGlycoconjugatesGlycolipids +1
Target Protein:
Photosystem II protein D1 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monomethyl fumarate Approved DB14219
small molecule | CAS: 2756-87-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic AcidsImmunosuppressive Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monopotassium phosphate Approved DB09413
small molecule | CAS: 7778-77-0

Monopotassium phosphate, MKP, (also potassium dihydrogenphosphate, KDP, or monobasic potassium phosphate), KH2PO4, is a soluble salt of potassium and the dihydrogen phosphate ion. It is a source of phosphorus and potassium as well as a buffering agent. It ca…

Kategori:
AcidsAcids, NoncarboxylicAnions +15
Waktu ParuhIn healthy children…
Vol. DistribusiPotassium first ent…
KlirensPhosphates are rapi…
Genetik -
Monoxerutin DB13764
small molecule | CAS: 23869-24-1

Monoxerutin is a flavonol, a type of flavonoid.

Kategori:
Capillary Stabilizing AgentsFlavonoidsVasoprotectives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Montelukast Approved DB00471
small molecule | CAS: 158966-92-8

Montelukast was first approved for clinical use by the US FDA in 1998 as Merck's brand name Singulair.[L6301] The medication is a member of the leukotriene receptor antagonist (LTRA) category of drugs.[L6301,L6304,L6307,L6310,L6325,L6328,L6331] Although capab…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAgents to Treat Airway Disease +29
Target Protein:
Cysteinyl leukotriene receptor 1Polyunsaturated fatty acid 5-lipoxygenase
Waktu ParuhStudies have demons…
Vol. DistribusiThe steady-state vo…
KlirensThe plasma clearanc…
Genetik -
Monteplase DB12726
biotech | CAS: 156616-23-8

Monteplase has been used in trials studying the treatment of Pulmonary Embolism.

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBlood Proteins +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moperone DB13554
small molecule | CAS: 1050-79-9

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsButyrophenone DerivativesCentral Nervous System Depressants +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MOR-22 DB17790
biotech

MOR-22, a Natural human lymphoblastoid interferon-alpha, is currently being investigated to treat papillomavirus warts in the oral cavity of HIV-positive patients.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MORAb-066 DB17347
biotech

MORAb-066 is a humanized antibody directed against tissue factor (TF). It is being investigated in pancreatic cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morella cerifera pollen Approved DB10457
biotech

Morella cerifera pollen is the pollen of the Morella cerifera plant. Morella cerifera pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morin DB16770
small molecule | CAS: 480-16-0

Deskripsi belum tersedia.

Kategori:
AntioxidantsBenzopyransBiological Factors +8
Target Protein:
Estrogen receptor betaSolute carrier family 22 member 12Fatty acid synthase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morinamide DB13417
small molecule | CAS: 952-54-5

Deskripsi belum tersedia.

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsDrugs for Treatment of Tuberculosis
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morinidazole DB15098
small molecule | CAS: 92478-27-8

Morinidazole is under investigation in clinical trial NCT03380793 (A Trial to Assess the Efficacy and Safety of Morinidazole in Patients With Appendicitis).

Kategori:
ImidazolesNitro Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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