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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 151 / 252
Lunsekimig DB19009
biotech | CAS: 2770858-49-4

Lunsekimig is under investigation in clinical trial NCT06102005 (Dose Ranging Study of Lunsekimig Compared With Placebo-control in Adult Participants With Moderate-to-severe Asthma).

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Lupeol DB12622
small molecule | CAS: 545-47-1

Lupeol has been investigated for the treatment of Acne.

Kategori:
Anti-Inflammatory AgentsPentacyclic TriterpenesTerpenes +1
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaNeutrophil elastase
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Luprostiol DB11425
small molecule | CAS: 67110-79-6

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +6
Target Protein:
Androgen receptor
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Lurasidone Approved DB08815
small molecule | CAS: 367514-87-2

Lurasidone is an atypical antipsychotic developed by Dainippon Sumitomo Pharma. It was approved by the U.S. Food and Drug Administration (FDA) for treatment of schizophrenia on October 29, 2010 and is currently pending approval for the treatment of bipolar di…

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +34
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 7 +3
Waktu Paruh40 mg dose= 18 hour…
Vol. Distribusi6173 L
Klirens3902 mL/min
Genetik -
Lurbinectedin Approved DB12674
small molecule | CAS: 497871-47-3

Lurbinectedin is a DNA alkylating agent that has been investigated in the treatment of a variety of cancers, including mesothelioma,[A214325] chronic lymphocytic leukemia (CLL),[A214328] breast cancer,[A214322] and small-cell lung cancer (SCLC).[A214310] It i…

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +12
Target Protein:
DNA
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe steady-state vo…
KlirensThe total plasma cl…
Genetik -
Lurtotecan DB12222
small molecule | CAS: 149882-10-0

Lurtotecan is under investigation in clinical trial NCT00022594 (Liposomal Lurtotecan in Treating Patients With Metastatic or Locally Recurrent Head and Neck Cancer).

Kategori:
AlkaloidsAntineoplastic Agents
Target Protein:
DNA topoisomerase 1
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Lusacomfar Alfa DB18526
biotech | CAS: 2640087-71-2

Lusacomfar Alfa is a recombinant complement factor H

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Luseogliflozin DB12214
small molecule | CAS: 898537-18-3

Luseogliflozin has been used in trials studying the treatment of Diabetes Melltius, Type 2.

Kategori:
AlcoholsAlimentary Tract and MetabolismBlood Glucose Lowering Agents +5
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Luspatercept Approved DB12281
biotech | CAS: 1373715-00-4

Luspatercept is a recombinant fusion protein comprised of a modified extracellular domain of activin receptor type IIB fused to the FC domain of human IgG1.[A187829,L42455] It was first approved for use in the United States in November 2019 under the brand na…

Kategori:
Activin ReceptorsAmino Acids, Peptides, and ProteinsAntianemia Drugs +25
Waktu ParuhThe average half-li…
Vol. DistribusiThe average apparen…
KlirensThe total apparent …
Genetik -
Lusutrombopag Approved DB13125
small molecule | CAS: 1110766-97-6

Lusutrombopag is an orally bioavailable thrombopoietin receptor (TPOR) agonist developed by Shionogi & Company (Osaka, Japan). TPOR is a regulatory target site for endogenous thrombopoietin, which acts as a primary cytokine to promote megakaryocyte proliferat…

Kategori:
Acids, CarbocyclicBCRP/ABCG2 SubstratesBlood and Blood Forming Organs +4
Target Protein:
Thrombopoietin receptor
Waktu ParuhIn healthy adult su…
Vol. DistribusiThe mean (%CV) lusu…
KlirensThe approximate mea…
Genetik -
Lusvertikimab DB18778
biotech | CAS: 2375835-91-7

Deskripsi belum tersedia.

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Luteolin DB15584
small molecule | CAS: 491-70-3

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +3
Target Protein:
Signal transducer and activator of transcription 3Lysophosphatidylcholine acyltransferase 2Lysophosphatidylcholine acyltransferase 1 +1
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Lutetium Lu 177 dotatate Approved DB13985
small molecule | CAS: 437608-50-9

A 177Lu-labeled somatostatin analog peptide, Lutetium Lu 177 dotatate belongs to an emerging form of treatments called Peptide Receptor Radionuclide Therapy (PRRT), which involves targeting tumours with molecules carrying radioactive particles that bind to sp…

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +8
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 1Somatostatin receptor type 3 +2
Waktu ParuhThe mean (± standar…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Lutetium Lu-177 Approved DB13982
small molecule | CAS: 14265-75-9

Deskripsi belum tersedia.

Kategori:
ElementsIsotopesLanthanoid Series Elements +3
Waktu Paruh-
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biotech | CAS: 1703749-62-5

Lutetium Lu-177 vipivotide tetraxetan is a radioligand therapeutic agent. It consists of a radionuclide, [lutetium Lu-177], linked to a moiety that binds to PSMA, a transmembrane protein that is expressed in prostate cancer.[L41280] Lutetium Lu-177 vipivot…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic Uses of ChemicalsRadioactive Therapeutic Agent +6
Target Protein:
Prostate-specific antigen
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
small molecule | CAS: 321835-55-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +5
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Lutikizumab DB16224
biotech | CAS: 1791411-57-8

Lutikizumab is under investigation in clinical trial NCT02087904 (A Study Evaluating the Safety, Efficacy, and Pharmacodynamic Effects of ABT-981 in Patients With Knee Osteoarthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +6
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Lutropin alfa Approved DB00044
biotech | CAS: 152923-57-4

Lutropin alfa is a recombinant human luteinizing hormone produced in yeast with 2 subunits, alpha = 92 residues, beta = 121 residues. It is a heterodimeric glycoprotein made up of monomeric units. Lutropin alfa was the first and only recombinant human form of…

Kategori:
Genito Urinary System and Sex HormonesGonadotropinsGonadotropins and Antigonadotropins +1
Target Protein:
Lutropin-choriogonadotropic hormone receptor
Waktu ParuhBiphasic; terminal …
Vol. DistribusiThe steady state vo…
Klirens* 2 – 3 L/h [health…
Genetik -
Luvadaxistat DB16067
small molecule | CAS: 1425511-32-5

Luvadaxistat is under investigation in clinical trial NCT03214588 (Efficacy, Tolerability, and Pharmacokinetics of Multiple Doses of Oral TAK-831 in Adults With Friedreich Ataxia).

Kategori:
D-Amino Acid Oxidase Inhibitor
Target Protein:
D-amino-acid oxidase
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biotech

Luveltamab tazevibulin, formerly known as STRO-002, is novel homogeneous folate receptor alpha (FolR?) targeting antibody-drug conjugate.[A257414] It is under investigation in clinical trial NCT05200364 (A Study of STRO-002, an Anti-folate Receptor Alpha Anti…

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Luvixasertib DB19200
small molecule | CAS: 1610759-22-2

Luvixasertib is under investigation in clinical trial NCT05251714 (CFI-402257, a Potent and Selective TTK Inhibitor, in Solid Tumors and With Fulvestrant in Breast Cancer).

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Luxeptinib DB19179
small molecule | CAS: 1616428-23-9

Deskripsi belum tersedia.

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biotech

LV-SMENP-DC is a vaccine candidate being developed by Shenzhen Geno-Immune Medical Institute that comprises dendritic cells that are modified with lentiviral vector-expressing synthetic minigene which are based on domains of selected viral proteins. This vacc…

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LV305 DB17288
biotech

LV305 is a lentiviral vector encoding NY-ESO-1 gene. LV305 is an active component of CMB305 along with [G305].[L47346]

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LX-2931 DB06297
small molecule | CAS: 948840-25-3

Deskripsi belum tersedia.

Kategori:
AminesHydroxylamines
Target Protein:
Sphingosine-1-phosphate lyase 1
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LX-7101 DB16009
small molecule | CAS: 1192189-69-7

LX-7101 is under investigation in clinical trial NCT01528111 (Study to Evaluate the Safety, Tolerability, and Efficacy of LX7101 in Subjects With Primary Open-angle Glaucoma or Ocular Hypertension).

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LX1031 DB05199
small molecule

LX1031 is an orally-dosed drug candidate for irritable bowel syndrome and other gastrointestinal disorders. LX1031 was generated by Lexicon medicinal chemists, and its target was internally identified as a key control point for the regulation of peripheral se…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +3
Target Protein:
Tryptophan 5-hydroxylase 1
Waktu Paruh-
Vol. Distribusi-
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LX6171 DB05180
small molecule

LX6171 is an oral drug candidate that was generated by Lexicon medicinal chemists and is being developed to treat disorders characterized by cognitive impairment, such as Alzheimer's disease, schizophrenia or vascular dementia.

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LY-2183240 DB17035
small molecule | CAS: 874902-19-9

LY-2183240 is an inhibitor of endocannabinoid reuptake/breakdown.[A253037]

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LY-2300559 DB13016
small molecule | CAS: 889116-06-7

Ly2300559 has been used in trials studying the prevention of Migraine Headache.

Kategori:
Acids, CarbocyclicBenzene DerivativesKetones
Target Protein:
Metabotropic glutamate receptor 2Cysteinyl leukotriene receptor 1
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LY-2452473 DB12573
small molecule | CAS: 1029692-15-6

Ly2452473 is under investigation for the supportive care of Prostate Cancer. Ly2452473 has been investigated for the treatment of Erectile Dysfunction.

Kategori:
Acids, Acyclic
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LY-2584702 DB12690
small molecule | CAS: 1082949-67-4

LY2584702 has been used in trials studying the treatment of Cancer, Advanced Cancer, Renal Cell Carcinoma, Metastases, Neoplasm, and Neuroendocrine Tumors, among others.

Kategori:
Ribosomal Protein S6 Kinases, 70-kDa, antagonists & inhibitors
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LY-2599506 DB05970
small molecule | CAS: 745051-65-4

LY2599506 was under investigation in clinical trials NCT01024244 and NCT01029795 for the treatment of patients with type 2 diabetes.

Target Protein:
Hexokinase-4
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LY-2623091 DB15367
small molecule | CAS: 1162264-07-4

LY-2623091 is under investigation in clinical trial NCT02194465 (A Study of LY2623091 in Participants With High Blood Pressure).

Target Protein:
Mineralocorticoid receptor
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LY-2624803 DB15092
small molecule | CAS: 879409-35-5

LY-2624803 is under investigation in clinical trial NCT01236105 (Effect of Activated Charcoal and Time of Dose on the Pharmacokinetics of LY2624803 in Healthy Subject).

Target Protein:
Histamine H1 receptor
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LY-2811376 DB13065
small molecule | CAS: 1194044-20-6

LY2811376 has been used in trials studying the basic science of Alzheimer's Disease.

Kategori:
Sulfur Compounds
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LY-2874455 DB13022
small molecule | CAS: 1254473-64-7

LY2874455 has been used in trials studying the treatment of Advanced Cancer.

Kategori:
Heterocyclic Compounds, Fused-RingPyrazolesReceptors, Fibroblast Growth Factor, antagonists & inhibitors
Target Protein:
Fibroblast growth factor receptor 2
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LY-2881835 DB15046
small molecule | CAS: 1292290-38-0

LY-2881835 is under investigation in clinical trial NCT01358981 (A Study of LY2881835 in Healthy People and People With Diabetes).

Target Protein:
Free fatty acid receptor 1
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LY-2886721 DB12547
small molecule | CAS: 1262036-50-9

LY2886721 has been used in trials studying the basic science of Alzheimer's Disease.

Kategori:
Heterocyclic Compounds, Fused-RingPyridines
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LY-294002 DB02656
small molecule | CAS: 154447-36-6

Specific inhibitor of phosphatidylinositol 3-kinase.

Kategori:
BenzopyransEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase pim-1
Waktu Paruh-
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LY-295501 DB12574
small molecule | CAS: 150869-74-2

ILX-295501 has been used in trials studying the treatment of Ovarian Cancer, Metastatic Cancer, Fallopian Tube Cancer, and Primary Peritoneal Cavity Cancer.

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring
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LY-3039478 DB12050
small molecule | CAS: 1421438-81-4

LY3039478 has been used in trials studying the treatment and basic science of LYMPHOMA, Neoplasms, Solid Tumor, COLON CANCER, and BREAST CANCER, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Neurogenic locus notch homolog protein 4Neurogenic locus notch homolog protein 1
Waktu Paruh-
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LY-3200882 DB16064
small molecule | CAS: 1898283-02-7

LY-3200882 is under investigation in clinical trial NCT04158700 (A Study of LY3200882 and Pembrolizumab in Participants With Advanced Cancer).

Target Protein:
TGF-beta receptor type-1
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LY-3499446 DB17486
small molecule | CAS: 2409131-50-4

Deskripsi belum tersedia.

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LY-377604 DB12858
small molecule | CAS: 204592-94-9

Ly377604 has been used in trials studying the treatment of Obesity.

Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
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LY-517717 DB05713
small molecule | CAS: 313489-71-3

LY517717 is an investigational oral direct inhibitor of activated Factor Xa. It is believed to be Lilly's PMD-3112 (licensed from Amgen).

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Coagulation factor X
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LY-518674 DB12988
small molecule | CAS: 425671-29-0

LY518674 has been used in trials studying the treatment of Metabolic Syndrome X.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
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LY2140023 DB05096
small molecule

LY2140023 is an investigational drug from Lilly, which is being developed as a new treatment option for schizophrenia. LY2140023 is an oral "prodrug," meaning it is devoid of intrinsic biological activity and, once administered, is metabolized to provide the …

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
Metabotropic glutamate receptor 2Metabotropic glutamate receptor 3
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LY2181308 DB05141
small molecule

LY2181308 is investigated in clinical trials for treating solid tumors. LY2181308 is a solid. LY2181308 is directed against a molecular target called survivin. LY2181308 is known to target baculoviral IAP repeat-containing protein 5. LY2181308 is an anti-sens…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Baculoviral IAP repeat-containing protein 5
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LY2275796 DB05165
small molecule

LY2275796 is a second-generation antisense anti-cancer drug candidate for clinical development. LY2275796 targets eukaryotic initiation factor- 4E (eIF-4E), a protein involved in the translation of key growth and survival factors that drive tumor progression,…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Eukaryotic translation initiation factor 4E
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