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2279

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866 (38.0%)
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1100 (48.3%)
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Halaman 15 / 46
Duvakitug DB19444
biotech | CAS: 2750005-84-4

Duvakitug is under investigation in clinical trial NCT05668013 (A Study to Evaluate the Long-term Effect of TEV-48574 in Moderate to Severe Ulcerative Colitis or Crohn's Disease).

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Duvoglustat DB03206
small molecule | CAS: 19130-96-2

An alpha-glucosidase inhibitor with antiviral action. Derivatives of deoxynojirimycin may have anti-HIV activity.

Kategori:
AlkaloidsAmino SugarsAnti-Infective Agents +7
Target Protein:
Maltase-glucoamylaseLysosomal alpha-glucosidaseNeutral alpha-glucosidase AB +6
Waktu Paruh-
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Genetik -
Dydrogesterone Approved DB00378
small molecule | CAS: 152-62-5

A synthetic progestational hormone with no androgenic or estrogenic properties. Unlike many other progestational compounds, dydrogesterone produces no increase in temperature and does not inhibit ovulation.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +12
Target Protein:
Progesterone receptor
Waktu ParuhDydrogesterone: 5-7…
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Dynorphin DB16146
small molecule | CAS: 80448-90-4

Dynorphin is under investigation in clinical trial NCT00000244 (Effects of Dynorphin 1-13 on Heroin Addiction - 1).

Kategori:
Amino Acids, Peptides, and ProteinsNerve Tissue ProteinsNeuropeptides +4
Target Protein:
Kappa-type opioid receptorMu-type opioid receptorDelta-type opioid receptor
Waktu Paruh-
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Dyphylline Approved DB00651
small molecule | CAS: 479-18-5

Dyphylline is a theophylline derivative with broncho- and vasodilator properties. It is typically used in the management of asthma, cardiac dyspnea, and bronchitis.

Kategori:
Anti-Asthmatic AgentsAutonomic AgentsBronchodilator Agents +13
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B5'-nucleotidase3',5'-cyclic-AMP phosphodiesterase 4A +4
Waktu Paruh2 hours (range 1.8 …
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E59 DB18372
biotech

E59 is a humanized IgG1 low affinity allergic reactivity inhibiting (LARI) monoclonal antibody. It was developed by Sixal Inc.

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EB05 DB16477
biotech | CAS: 2641646-59-3

EB05, in combination with standard of care (SOC), is being investigated in clinical trial NCT04401475 to evaluate its safety and efficacy in adult hospitalized patients with COVID-19 and ARDS.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Genetik -
biotech

Ebola virus vaccine is a vaccine used to prevent Ebola virus disease caused by _Zaire ebolavirus_ in adults, prevent outbreaks, and reduce the extent of the virus spreading in case of outbreaks.[L10854] Ebola virus disease, formerly known as Ebola hemorrhagic…

Kategori:
ImmunizationImmunologic FactorsVaccines +1
Waktu ParuhThere is limited ph…
Vol. DistribusiThere is limited ph…
KlirensThere is limited ph…
Genetik -
Ecallantide Approved DB05311
biotech | CAS: 460738-38-9

Ecallantide is a potent and selective human plasma kallikrein inhibitor that is indicated for the symptomatic treatment of hereditary angioedema. Ecallantide is a recombinant 60-amino-acid protein produced in _Pichia pastoris_ yeast cells that contains three …

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +10
Target Protein:
Plasma kallikrein
Waktu ParuhFollowing subcutane…
Vol. DistribusiThe volume of distr…
KlirensPlasma clearance wa…
Genetik -
Ecamsule Approved DB09534
small molecule | CAS: 92761-26-7

Ecamsule is an organic compound which is added to many sunscreens to filter out UVA rays. It is a benzylidene camphor derivative, many of which are known for their excellent photostability. Ecamsule has been approved for use in the U.S. since 2006, but only a…

Kategori:
AcidsAcids, NoncarboxylicBicyclic Monoterpenes +12
Waktu ParuhEcamsule is not abs…
Vol. DistribusiEcamsule is intende…
KlirensEcamsule is used to…
Genetik -
Eculizumab Approved DB01257
biotech | CAS: 219685-50-4

Eculizumab is a monoclonal antibody that targets complement protein C5.[L6919,A2245] Binding to this protein prevents the activation of a complement terminal complex, which is used to treat a number of autoimmune conditions.[L6919,A2245,A2246] Eculizumab w…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Complement C5
Waktu ParuhThe half life of ec…
Vol. DistribusiThe volume of distr…
KlirensPharmacokinetic pro…
Genetik -
Edaravone Approved DB12243
small molecule | CAS: 89-25-8

Edaravone is a free radical scavenger and neuroprotective agent with antioxidant properties.[A254257] It has three tautomers.[A19140] Edaravone works to scavenge reactive oxygen species, which have been implicated in neurological disorders, such as amyotrophi…

Kategori:
AntioxidantsCentral Nervous System AgentsCompounds used in a research, industrial, or household setting +14
Target Protein:
Apoptosis regulator Bcl-2
Waktu ParuhThe mean terminal e…
Vol. DistribusiAfter intravenous a…
KlirensFollowing intraveno…
Genetik -
Edetic acid Approved DB00974
small molecule | CAS: 60-00-4

A chelating agent (chelating agents) that sequesters a variety of polyvalent cations. It is used in pharmaceutical manufacturing and as a food additive.

Kategori:
AcetatesAcids, AcyclicAmines +19
Target Protein:
LeadIronManganese cation
Waktu ParuhThe half life of ed…
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EDI-200 DB18188
biotech

EDI-200 is a fusion protein consisting of human immunoglobim G1 constant region Fc region fused to the human receptor binding domain of ectodysplasin-A1.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Proteins +17
Waktu Paruh-
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Edodekin alfa DB15631
biotech | CAS: 187348-17-0

Edodekin alfa is under investigation in clinical trial NCT01468896 (Cetuximab and Recombinant Interleukin-12 in Treating Patients With Squamous Cell Carcinoma of the Head and Neck That Is Recurrent, Metastatic, or Cannot Be Removed by Surgery).

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAngiogenesis Inhibitors +12
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Edoxaban Approved DB09075
small molecule | CAS: 480449-70-5

Edoxaban is a member of the Novel Oral Anti-Coagulants (NOACs) class of drugs, and is a rapidly acting, oral, selective factor Xa inhibitor. By inhibiting factor Xa, a key protein in the coagulation cascade, edoxaban prevents the stepwise amplification of pro…

Kategori:
AnticoagulantsAntithrombinsBlood and Blood Forming Organs +9
Target Protein:
Coagulation factor X
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe steady state vo…
Klirens22 L/hr
Genetik -
Efalizumab Approved DB00095
biotech | CAS: 214745-43-4

Humanized IgG1 kappa isotype monoclonal antibody that binds to human CD11a. Efalizumab has a molecular weight of approximately 150 kilodaltons and is produced in a Chinese hamster ovary mammalian cell expression system in a nutrient medium containing the anti…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Integrin alpha-XIntegrin alpha-L
Waktu Paruh5 days
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Efanesoctocog alfa Approved DB16662
biotech | CAS: 2252477-42-0

Efanesoctocog alfa (BIVV001) is a recombinant factor VIII (FVIII) analogue fusion protein used for the routine prophylaxis, perioperative management of bleeding and on-demand treatment and control of bleeding episodes in patients with hemophilia A.[L45379] Th…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +6
Target Protein:
Coagulation factor IXCoagulation factor XLow-density lipoprotein receptor-related protein 2 +1
Waktu ParuhEfanesoctocog alfa …
Vol. DistribusiEfanesoctocog alfa …
KlirensEfanesoctocog alfa …
Genetik -
biotech | CAS: 2049067-94-7

Efavaleukin alfa is a fusion protein consisting of interleukin mutein fused to the C-terminus of an immunoglobulin G Fc domain by way of a G4S linker. It is under investigation in clinical trial NCT03422627 (Safety and Efficacy of AMG 592 in Subjects With Ste…

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Efavirenz Approved DB00625
small molecule | CAS: 154598-52-4

Efavirenz (brand names Sustiva® and Stocrin®) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) and is used as part of highly active antiretroviral therapy (HAART) for the treatment of a human immunodeficiency virus (HIV) type 1. For HIV infectio…

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiinfectives for Systemic Use +52
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Gen Terkait:
CYP2B6
Waktu Paruh40-55 hours
Vol. Distribusi-
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Genetik 1 Varian
Efbemalenograstim alfa Approved DB18704
biotech | CAS: 2200269-79-8

Efbemalenograstim alfa is a long-acting recombinant fusion protein of granulocyte-colony stimulating factor (G-CSF) due to the addition of the Fc portion of human IgG2, allowing for once-per-cycle administration.[L48852,A262167] As endogenous G-CSF mediates t…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsColony-Stimulating Factors +2
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Efepoetin alfa DB19197
biotech | CAS: 1905452-78-9

Efepoetin alfa is under investigation in clinical trial NCT04155125 (A Study of Efepoetin Alfa in Treating Anaemia Associated With Chronic Kidney Diseases Patient).

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biotech | CAS: 2026634-47-7

Efineptakin alfa (also known as NT-I7) is a long-acting human interleukin-7 (IL-7) fusion protein that promotes T-cell development, contributing to the immune response. Compared to endogenous IL-7, NT-I7 is more stable and potent, has a longer half-life, and …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
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Eflapegrastim Approved DB15001
biotech | CAS: 1384099-30-2

Febrile neutropenia (FN), defined as the co-occurrence of fever (temperature > 38 ?C) and severe neutropenia (ANC < 500 cells/mm<sup>3</sup>), is a potential side effect of myelosuppressive chemotherapy in which the patient develops an infection during a peri…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +20
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhIn patients with br…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ef…
Genetik -
biotech

Eflepedocokin alfa is a recombinant IL-22-Fc fusion protein manufactured in Chinese hamster ovary cells that is composed of 2 human interleukin 22 (IL-22) molecules linked to an immunoglobulin constant region (IgG2-Fc).[A225706, L27661] It is being developed …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +5
Waktu Paruh-
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Eflornithine Approved DB06243
small molecule | CAS: 70052-12-9

Eflornithine is an irreversible ornithine decarboxylase inhibitor originally developed as a treatment for human African trypanosomiasis.[A262829] Further research has also implicated ornithine decarboxylase in other conditions like facial hirsutism and cancer…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAmino AcidsAmino Acids, Basic +15
Target Protein:
Ornithine decarboxylase
Waktu ParuhThe terminal plasma…
Vol. DistribusiEflornithine volume…
KlirensThe clearance (CL/F…
Genetik -
biotech | CAS: 1953227-87-6

Efmarodocokin alfa is under investigation in clinical trial NCT04386616 (A Study to Evaluate the Safety and Efficacy of MSTT1041A (Astegolimab) or UTTR1147A in Patients With Severe COVID-19 Pneumonia).

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biotech | CAS: 1644543-31-6

Efmitermant alfa, a locally-acting GDF/activin ligand trap, is under investigation in clinical trial NCT03124459 (Study of ACE-083 in Patients With Charcot-marie-tooth Disease).

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Efmoroctocog alfa Approved DB11607
biotech | CAS: 1270012-79-7

Efmoroctocog alfa is a fully recombinant factor VIII-Fc fusion protein (rFVIIIFc) with an extended half-life compared with conventional factor VIII (FVIII) preparations, including recombinant FVIII (rFVIII) products such as [DB13999][A31551]. It is an antihem…

Kategori:
HemostaticsHuman Antihemophilic Factors
Target Protein:
von Willebrand factor
Waktu ParuhFollowing a single …
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Efocipegtrutide DB18194
biotech | CAS: 2513399-19-2

Efocipegtrutide is a long-acting, monomeric peptide triple agonist.

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Efprezimod alfa DB16448
biotech

CD24Fc is a biological immunomodulator originally developed to address graft-versus-host disease in stem cell transplantation in leukemia patients.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
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Efruxifermin DB19012
biotech | CAS: 2375240-92-7

Efruxifermin is under investigation in clinical trial NCT06215716 (A Study Evaluating Efruxifermin in Subjects With Non-cirrhotic Nonalcoholic Steatohepatitis (Nash)/metabolic Dysfunction-associated Steatohepatitis (MASH) and Fibrosis).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +3
Waktu Paruh-
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Genetik -
biotech | CAS: 1905448-17-0

Eftansomatropin alfa (GX-H9) comprises a recombinant human growth hormone fused to hyFc, a synthetic hybrid Fc fragment.[L48275] It is under investigation for the treatment of growth hormone deficiency.

Kategori:
Amino Acids, Peptides, and ProteinsGrowth HormoneHormones +7
Waktu Paruh-
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Eftrenonacog alfa Approved DB11608
biotech | CAS: 1270012-74-2

Eftrenonacog alfa is a long-acting recombinant fusion protein used in the treatment of hemophilia B. It is comprised of a single molecule of human factor IX (FIX) covalently linked to the constant region (Fc) domain of human IgG1 via recombinant DNA technolog…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +15
Target Protein:
IgG receptor FcRn large subunit p51
Waktu ParuhFollowing administr…
Vol. DistribusiFollowing administr…
KlirensFollowing administr…
Genetik -
Efungumab DB16151
biotech | CAS: 762260-74-2

Efungumab is under investigation in clinical trial NCT00217815 (Preliminary Study of Mycograb and Docetaxel in Advanced Breast Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
Waktu Paruh-
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Efzofitimod DB16453
biotech

Efzofitimod (ATYR1923) is a fusion protein comprised of the immuno-modulatory domain of histidyl tRNA synthetase fused to the FC region of a human antibody. It is a selective modulator of neuropilin-2 that downregulates the innate and adaptive immune response…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Neuropilin-2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
EGEN-001 DB05953
small molecule

EGEN-001 is a novel non-viral vector consisting of a plasmid DNA encoding the human gene for interleukin 12 (IL-12) and a biocompatible, biodegradable delivery polymer with potential antineoplastic activity.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
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EGT-101 DB17645
biotech

EGT-101 is an adeno-associated viral vector serotype 9 (AAV9) vector-based gene therapy consisting of the human sulfamidase (SGSH) transgene. Developed by Esteve Pharmaceuticals, it is being investigated for Sanfilippo syndrome type A.[L45919]

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EGT-301 DB17649
biotech

EGT-301 is a gene therapy being investigated for Hunter Syndrome. It consists of an adeno-associated viral vector serotype 9 (AAV9) containing the human Iduronate-2-sulfatase (I2S) transgene designed to restore I2S functional deficiency in patients with Hunte…

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Genetik -
EI-001 DB17596
biotech

Deskripsi belum tersedia.

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Elacridar DB04881
small molecule | CAS: 143664-11-3

Elacridar (GW120918) is an oral bioenhancer that targets multiple drug resistance in tumors. In many cases, the appearance of multidrug resistance in cancer is due to a change in expression of protein inhibitors. As of August 2007 elacridar was not listed on …

Kategori:
BCRP/ABCG2 InhibitorsBenzocycloheptenesDrug Resistance, Multiple +3
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eladocagene exuparvovec Approved DB16780
biotech | CAS: 2098615-91-7

Eladocagene exuparvovec is a recombinant adeno-associated virus-2 (AAV2)-based gene therapy that expresses human aromatic L-amino acid decarboxylase (AADC), and it is used to treat AADC deficiency, a fatal and rare genetic disorder that causes severe disabili…

Kategori:
Adeno-associated Viral Vector TherapiesAlimentary Tract and MetabolismEnzymes +2
Waktu ParuhNot available.
Vol. DistribusiThe biodistribution…
KlirensNot available.
Genetik -
Elafin DB05161
small molecule

Elafin is a human protein that is produced naturally in the skin, lung and breast, protecting the respective tissue from destruction by the immune system. Elafin’s ability to block the activity of destructive enzymes that are involved in inflammatory reaction…

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme InhibitorsPeptides +3
Target Protein:
Neutrophil elastaseMyeloblastin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elastin (human) DB15364
biotech | CAS: 9007-58-3

Elastin (human) is under investigation in clinical trial NCT01466413 (Two Formulations of ELAPR Compared to Restylane® Vital Light Following Repeat Implants in the Upper Arm Dermis).

Kategori:
Amino Acids, Peptides, and ProteinsBiopolymersElastin +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elbasvir Approved DB11574
small molecule | CAS: 1370468-36-2

Elbasvir is a direct-acting antiviral medication used as part of combination therapy to treat chronic hepatitis C, an infectious liver disease caused by infection with hepatitis C virus (HCV). HCV is a single-stranded RNA virus that is categorized into nine d…

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +18
Target Protein:
Nonstructural protein 5A
Waktu ParuhThe geometric mean …
Vol. DistribusiElbasvir has an est…
KlirensThe clearance of el…
Genetik -
Eldelumab DB06116
biotech | CAS: 946414-98-8

MDX-1100, a fully human antibody that targets IP10 (also known as CXCL10), a chemokine expressed in association with multiple inflammatory disease indications, such as rheumatoid arthritis, inflammatory bowel disease and multiple sclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
C-X-C motif chemokine 10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eleuthero Approved DB14303
biotech

Eleuthero is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAraliaceaeBiological Products +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Elexacaftor Approved DB15444
small molecule | CAS: 2216712-66-0

Elexacaftor (previously VX-445) is a small molecule, next-generation corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) protein.[A187361] It received FDA approval in October 2019 in combination with [tezacaftor] and [ivacaftor] as the…

Kategori:
Cystic Fibrosis Transmembrane Conductance Regulator CorrectorsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +24
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Elivaldogene autotemcel Approved DB16746
biotech

Elivaldogene autotemcel is a gene therapy consisting of genetically modified autologous cells. It is used to provide functional copies of human adrenoleukodystrophy protein (ALDP) in patients with adrenoleukodystrophy,[L39491] an X-linked genetic disorder cha…

Kategori:
Alimentary Tract and MetabolismCellular and Gene TherapyVarious Alimentary Tract and Metabolism Products
Waktu ParuhAs elivaldogene aut…
Vol. DistribusiAs elivaldogene aut…
KlirensAs elivaldogene aut…
Genetik -
biotech | CAS: 1905397-73-0

Deskripsi belum tersedia.

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